2R9R
| Shaker family voltage dependent potassium channel (kv1.2-kv2.1 paddle chimera channel) in association with beta subunit | 分子名称: | (1R)-2-{[(S)-{[(2S)-2,3-dihydroxypropyl]oxy}(hydroxy)phosphoryl]oxy}-1-[(hexadecanoyloxy)methyl]ethyl (9Z)-octadec-9-enoate, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, POTASSIUM ION, ... | 著者 | Long, S.B, Tao, X, Campbell, E.B, Mackinnon, R. | 登録日 | 2007-09-13 | 公開日 | 2007-11-20 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Atomic structure of a voltage-dependent K+ channel in a lipid membrane-like environment. Nature, 450, 2007
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3DD2
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2A79
| Mammalian Shaker Kv1.2 potassium channel- beta subunit complex | 分子名称: | NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, POTASSIUM ION, Potassium voltage-gated channel subfamily A member 2, ... | 著者 | Long, S.B, Campbell, E.B, MacKinnon, R. | 登録日 | 2005-07-05 | 公開日 | 2005-07-12 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Crystal structure of a mammalian voltage-dependent Shaker family K+ channel. Science, 309, 2005
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1KZO
| PROTEIN FARNESYLTRANSFERASE COMPLEXED WITH FARNESYLATED K-RAS4B PEPTIDE PRODUCT AND FARNESYL DIPHOSPHATE SUBSTRATE BOUND SIMULTANEOUSLY | 分子名称: | ACETIC ACID, FARNESYL, FARNESYL DIPHOSPHATE, ... | 著者 | Long, S.B, Casey, P.J, Beese, L.S. | 登録日 | 2002-02-07 | 公開日 | 2002-10-16 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | The Reaction Path of Protein Farnesyltransferase at Atomic Resolution Nature, 419, 2002
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1D8E
| Zinc-depleted FTase complexed with K-RAS4B peptide substrate and FPP analog. | 分子名称: | ACETATE ION, FARNESYLTRANSFERASE (ALPHA SUBUNIT), FARNESYLTRANSFERASE (BETA SUBUNIT), ... | 著者 | Long, S.B, Casey, P.J, Beese, L.S. | 登録日 | 1999-10-22 | 公開日 | 2000-03-20 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | The basis for K-Ras4B binding specificity to protein farnesyltransferase revealed by 2 A resolution ternary complex structures. Structure Fold.Des., 8, 2000
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1D8D
| CO-CRYSTAL STRUCTURE OF RAT PROTEIN FARNESYLTRANSFERASE COMPLEXED WITH A K-RAS4B PEPTIDE SUBSTRATE AND FPP ANALOG AT 2.0A RESOLUTION | 分子名称: | ACETATE ION, K-RAS4B PEPTIDE SUBSTRATE, ZINC ION, ... | 著者 | Long, S.B, Casey, P.J, Beese, L.S. | 登録日 | 1999-10-22 | 公開日 | 2000-02-09 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | The basis for K-Ras4B binding specificity to protein farnesyltransferase revealed by 2 A resolution ternary complex structures. Structure Fold.Des., 8, 2000
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1KZP
| PROTEIN FARNESYLTRANSFERASE COMPLEXED WITH A FARNESYLATED K-RAS4B PEPTIDE PRODUCT | 分子名称: | ACETIC ACID, FARNESYL, Farnesylated K-Ras4B peptide product, ... | 著者 | Long, S.B, Casey, P.J, Beese, L.S. | 登録日 | 2002-02-07 | 公開日 | 2002-10-16 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Reaction path of protein farnesyltransferase at atomic resolution Nature, 419, 2002
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1JCR
| CRYSTAL STRUCTURE OF RAT PROTEIN FARNESYLTRANSFERASE COMPLEXED WITH THE NON-SUBSTRATE TETRAPEPTIDE INHIBITOR CVFM AND FARNESYL DIPHOSPHATE SUBSTRATE | 分子名称: | ACETIC ACID, FARNESYL DIPHOSPHATE, PROTEIN FARNESYLTRANSFERASE, ... | 著者 | Long, S.B, Casey, P.J, Beese, L.S. | 登録日 | 2001-06-11 | 公開日 | 2001-11-02 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | The crystal structure of human protein farnesyltransferase reveals the basis for inhibition by CaaX tetrapeptides and their mimetics. Proc.Natl.Acad.Sci.USA, 98, 2001
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1JCQ
| CRYSTAL STRUCTURE OF HUMAN PROTEIN FARNESYLTRANSFERASE COMPLEXED WITH FARNESYL DIPHOSPHATE AND THE PEPTIDOMIMETIC INHIBITOR L-739,750 | 分子名称: | 2(S)-{2(S)-[2(R)-AMINO-3-MERCAPTO]PROPYLAMINO-3(S)-METHYL}PENTYLOXY-3-PHENYLPROPIONYLMETHIONINE SULFONE, ACETIC ACID, FARNESYL DIPHOSPHATE, ... | 著者 | Long, S.B, Casey, P.J, Beese, L.S. | 登録日 | 2001-06-11 | 公開日 | 2001-11-02 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | The crystal structure of human protein farnesyltransferase reveals the basis for inhibition by CaaX tetrapeptides and their mimetics. Proc.Natl.Acad.Sci.USA, 98, 2001
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1JCS
| CRYSTAL STRUCTURE OF RAT PROTEIN FARNESYLTRANSFERASE COMPLEXED WITH THE PEPTIDE SUBSTRATE TKCVFM AND AN ANALOG OF FARNESYL DIPHOSPHATE | 分子名称: | ACETIC ACID, PROTEIN FARNESYLTRANSFERASE, ALPHA SUBUNIT, ... | 著者 | Long, S.B, Casey, P.J, Beese, L.S. | 登録日 | 2001-06-11 | 公開日 | 2001-11-02 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | The crystal structure of human protein farnesyltransferase reveals the basis for inhibition by CaaX tetrapeptides and their mimetics. Proc.Natl.Acad.Sci.USA, 98, 2001
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7SQH
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7SQF
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6XQN
| Structure of a mitochondrial calcium uniporter holocomplex (MICU1, MICU2, MCU, EMRE) in low Ca2+ | 分子名称: | CALCIUM ION, Calcium uniporter protein, Calcium uptake protein 1, ... | 著者 | Long, S.B, Wang, C, Baradaran, R, Jacewicz, A, Delgado, B. | 登録日 | 2020-07-09 | 公開日 | 2020-07-29 | 最終更新日 | 2024-03-06 | 実験手法 | ELECTRON MICROSCOPY (3.3 Å) | 主引用文献 | Structures reveal gatekeeping of the mitochondrial Ca 2+ uniporter by MICU1-MICU2. Elife, 9, 2020
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6DNF
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6XQO
| Structure of the human MICU1-MICU2 heterodimer, calcium bound, in association with a lipid nanodisc | 分子名称: | CALCIUM ION, Calcium uptake protein 1, mitochondrial, ... | 著者 | Long, S.B, Wang, C, Baradaran, R, Jacewicz, A, Delgado, B. | 登録日 | 2020-07-09 | 公開日 | 2020-07-29 | 最終更新日 | 2024-03-06 | 実験手法 | ELECTRON MICROSCOPY (3.1 Å) | 主引用文献 | Structures reveal gatekeeping of the mitochondrial Ca 2+ uniporter by MICU1-MICU2. Elife, 9, 2020
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7SQG
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4HKR
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4HKS
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1FT2
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5T5N
| Calcium-activated chloride channel bestrophin-1 (BEST1), triple mutant: I76A, F80A, F84A; in complex with an Fab antibody fragment, chloride, and calcium | 分子名称: | CALCIUM ION, CHLORIDE ION, Fab antibody fragment, ... | 著者 | Long, S.B, Vaisey, G. | 登録日 | 2016-08-31 | 公開日 | 2016-11-30 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Distinct regions that control ion selectivity and calcium-dependent activation in the bestrophin ion channel. Proc. Natl. Acad. Sci. U.S.A., 113, 2016
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6X4S
| MCU-EMRE complex of a metazoan mitochondrial calcium uniporter | 分子名称: | CALCIUM ION, Calcium uniporter protein,Protein EMRE homolog, mitochondrial-like Protein fusion | 著者 | Long, S.B, Wang, C, Baradaran, R. | 登録日 | 2020-05-22 | 公開日 | 2020-09-02 | 最終更新日 | 2024-03-06 | 実験手法 | ELECTRON MICROSCOPY (3.5 Å) | 主引用文献 | Structure and Reconstitution of an MCU-EMRE Mitochondrial Ca 2+ Uniporter Complex. J.Mol.Biol., 432, 2020
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7MHZ
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7MHY
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1S63
| Human protein farnesyltransferase complexed with L-778,123 and FPP | 分子名称: | 4-[(5-{[4-(3-CHLOROPHENYL)-3-OXOPIPERAZIN-1-YL]METHYL}-1H-IMIDAZOL-1-YL)METHYL]BENZONITRILE, FARNESYL DIPHOSPHATE, Protein farnesyltransferase beta subunit, ... | 著者 | Long, S.B, Casey, P.J, Beese, L.S. | 登録日 | 2004-01-22 | 公開日 | 2004-07-27 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Crystallographic Analysis Reveals that Anticancer Clinical Candidate L-778,123 Inhibits Protein Farnesyltransferase and Geranylgeranyltransferase-I by Different Binding Modes. Biochemistry, 43, 2004
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3UKM
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