6KJB
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![BU of 6kjb by Molmil](/molmil-images/mine/6kjb) | wild-type apo-form E. coli ATCase holoenzyme with an unusual open conformation of R167 | 分子名称: | Aspartate carbamoyltransferase catalytic subunit, Aspartate carbamoyltransferase regulatory chain, ZINC ION | 著者 | Wang, N, Lei, Z, Zheng, J, Jia, Z.C. | 登録日 | 2019-07-22 | 公開日 | 2020-06-03 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.06 Å) | 主引用文献 | Conformational Plasticity of the Active Site Entrance inE. coliAspartate Transcarbamoylase and Its Implication in Feedback Regulation. Int J Mol Sci, 21, 2020
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5H73
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![BU of 5h73 by Molmil](/molmil-images/mine/5h73) | Crystal structure of human DHODH with 18F | 分子名称: | ACETATE ION, Dihydroorotate dehydrogenase (quinone), mitochondrial, ... | 著者 | Huang, J, Wu, D. | 登録日 | 2016-11-16 | 公開日 | 2017-07-26 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.58 Å) | 主引用文献 | Crystal structure of human DHODH with 18F at 1.58 Angstroms resolution To Be Published
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4XQ6
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4YLW
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![BU of 4ylw by Molmil](/molmil-images/mine/4ylw) | Crystal structure of human dihydroorotate dehydrogenase (DHODH) with No.33 compound | 分子名称: | Dihydroorotate dehydrogenase (quinone), mitochondrial, FLAVIN MONONUCLEOTIDE, ... | 著者 | Wu, D, Ouyang, P, Lu, W, Huang, J. | 登録日 | 2015-03-06 | 公開日 | 2016-03-09 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.79 Å) | 主引用文献 | Crystal structure of human dihydroorotate dehydrogenase (DHODH) with No.33 compound To Be Published
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6YVK
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![BU of 6yvk by Molmil](/molmil-images/mine/6yvk) | Human OMPD-domain of UMPS in complex with the substrate OMP at 1.25 Angstroms resolution, 0.71 MGy exposure | 分子名称: | GLYCEROL, OROTIDINE-5'-MONOPHOSPHATE, SULFATE ION, ... | 著者 | Tittmann, K, Rindfleisch, S, Krull, M. | 登録日 | 2020-04-28 | 公開日 | 2021-11-17 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.25 Å) | 主引用文献 | Ground-state destabilization by electrostatic repulsion is not a driving force in orotidine-5-monophosphate decarboxylase catalysis Nat Catal, 5, 2022
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6YVL
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![BU of 6yvl by Molmil](/molmil-images/mine/6yvl) | Human OMPD-domain of UMPS in complex with the substrate OMP at 1.25 Angstroms resolution, 1.42 MGy exposure | 分子名称: | GLYCEROL, OROTIDINE-5'-MONOPHOSPHATE, SULFATE ION, ... | 著者 | Tittmann, K, Rindfleisch, S, Krull, M. | 登録日 | 2020-04-28 | 公開日 | 2021-11-17 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.25 Å) | 主引用文献 | Ground-state destabilization by electrostatic repulsion is not a driving force in orotidine-5-monophosphate decarboxylase catalysis Nat Catal, 5, 2022
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6YVM
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![BU of 6yvm by Molmil](/molmil-images/mine/6yvm) | Human OMPD-domain of UMPS in complex with the substrate OMP at 1.25 Angstroms resolution, 2.13 MGy exposure | 分子名称: | GLYCEROL, OROTIDINE-5'-MONOPHOSPHATE, SULFATE ION, ... | 著者 | Tittmann, K, Rindfleisch, S, Krull, M. | 登録日 | 2020-04-28 | 公開日 | 2021-11-17 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.25 Å) | 主引用文献 | Ground-state destabilization by electrostatic repulsion is not a driving force in orotidine-5-monophosphate decarboxylase catalysis Nat Catal, 5, 2022
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6YVN
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![BU of 6yvn by Molmil](/molmil-images/mine/6yvn) | Human OMPD-domain of UMPS in complex with the substrate OMP at 1.25 Angstroms resolution, 2.84 MGy exposure | 分子名称: | GLYCEROL, OROTIDINE-5'-MONOPHOSPHATE, SULFATE ION, ... | 著者 | Tittmann, K, Rindfleisch, S, Krull, M. | 登録日 | 2020-04-28 | 公開日 | 2021-11-17 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.25 Å) | 主引用文献 | Ground-state destabilization by electrostatic repulsion is not a driving force in orotidine-5-monophosphate decarboxylase catalysis Nat Catal, 5, 2022
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6YWU
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![BU of 6ywu by Molmil](/molmil-images/mine/6ywu) | Human OMPD-domain of UMPS (K314AcK) in complex with UMP at 1.1 Angstroms resolution | 分子名称: | GLYCEROL, SULFATE ION, URIDINE-5'-MONOPHOSPHATE, ... | 著者 | Tittmann, K, Rindfleisch, S, Krull, M. | 登録日 | 2020-04-30 | 公開日 | 2022-02-23 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.1 Å) | 主引用文献 | Ground-state destabilization by electrostatic repulsion is not a driving force in orotidine-5-monophosphate decarboxylase catalysis Nat Catal, 5, 2022
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6YWT
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6YVO
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![BU of 6yvo by Molmil](/molmil-images/mine/6yvo) | Human OMPD-domain of UMPS in complex with the substrate OMP at 1.25 Angstroms resolution, 3.55 MGy exposure | 分子名称: | GLYCEROL, OROTIDINE-5'-MONOPHOSPHATE, SULFATE ION, ... | 著者 | Tittmann, K, Rindfleisch, S, Krull, M. | 登録日 | 2020-04-28 | 公開日 | 2022-02-23 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.25 Å) | 主引用文献 | Ground-state destabilization by electrostatic repulsion is not a driving force in orotidine-5-monophosphate decarboxylase catalysis Nat Catal, 5, 2022
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4RR4
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![BU of 4rr4 by Molmil](/molmil-images/mine/4rr4) | Crystal structure of human dihydroorotate dehydrogenase (DHODH) with DH03A367 | 分子名称: | 2-chloro-N-[3-(4-{[(2Z)-2-cyano-3-cyclopropyl-3-hydroxyprop-2-enoyl]amino}phenoxy)phenyl]-4-methyl-1,3-thiazole-5-carboxamide, Dihydroorotate dehydrogenase (quinone), mitochondrial, ... | 著者 | Zhu, L, Ren, X, Zhu, J, Li, H. | 登録日 | 2014-11-06 | 公開日 | 2015-11-25 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.38 Å) | 主引用文献 | Crystal structure of human dihydroorotate dehydrogenase (DHODH) with DH03A367 TO BE PUBLISHED
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4RKA
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![BU of 4rka by Molmil](/molmil-images/mine/4rka) | Crystal structure of human dihydroorotate dehydrogenase (DHODH) with DH03A347 | 分子名称: | 2-{[5-(naphthalen-1-ylmethyl)-4-oxo-4H-1lambda~4~,3-thiazol-2-yl]amino}benzoic acid, Dihydroorotate dehydrogenase (quinone), mitochondrial, ... | 著者 | Zhu, L, Ren, X, Zhu, J, Li, H. | 登録日 | 2014-10-12 | 公開日 | 2015-11-11 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.71 Å) | 主引用文献 | Crystal structure of human dihydroorotate dehydrogenase (DHODH) with DH03A347 TO BE PUBLISHED
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4RK8
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![BU of 4rk8 by Molmil](/molmil-images/mine/4rk8) | Crystal structure of human dihydroorotate dehydrogenase (DHODH) with DH03A356 | 分子名称: | 5-fluoro-2-{[(5Z)-5-(naphthalen-1-ylmethylidene)-4-oxo-4,5-dihydro-1,3-thiazol-2-yl]amino}benzoic acid, Dihydroorotate dehydrogenase (quinone), mitochondrial, ... | 著者 | Zhu, L, Ren, X, Zhu, J, Li, H. | 登録日 | 2014-10-12 | 公開日 | 2015-11-11 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.22 Å) | 主引用文献 | Crystal structure of human dihydroorotate dehydrogenase (DHODH) with DH03A356 TO BE PUBLISHED
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4WN3
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![BU of 4wn3 by Molmil](/molmil-images/mine/4wn3) | Crystal structure of Saccharomyces cerevisiae OMP synthase in complex with PRP(NH)P | 分子名称: | MAGNESIUM ION, Orotate phosphoribosyltransferase 1, [[[(2R,3R,4S,5R)-3,4-bis(oxidanyl)-5-(phosphonooxymethyl)oxolan-2-yl]oxy-oxidanyl-phosphoryl]amino]phosphonic acid | 著者 | Bang, M.B, Molich, U, Hansen, M.R, Grubmeyer, C, Harris, P. | 登録日 | 2014-10-10 | 公開日 | 2015-12-23 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Crystal structure of Saccharomyces cerevisiae OMP synthase in complex with PRP(NH)P To Be Published
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4RLI
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![BU of 4rli by Molmil](/molmil-images/mine/4rli) | Crystal structure of human dihydroorotate dehydrogenase (DHODH) with DH03A048 | 分子名称: | Dihydroorotate dehydrogenase (quinone), mitochondrial, FLAVIN MONONUCLEOTIDE, ... | 著者 | Zhu, L, Ren, X, Zhu, J, Li, H. | 登録日 | 2014-10-17 | 公開日 | 2015-11-04 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Crystal structure of human dihydroorotate dehydrogenase (DHODH) with DH03A048 TO BE PUBLISHED
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4ZMG
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![BU of 4zmg by Molmil](/molmil-images/mine/4zmg) | Crystal structure of Human Dihydroorotate Dehydrogenase (DHODH) with DH03A338 | 分子名称: | 1-(3,5-difluoro-3'-methoxybiphenyl-4-yl)-3-(1,3-thiazol-5-yl)urea, ACETATE ION, Dihydroorotate dehydrogenase (quinone), ... | 著者 | Ren, X.L, Zhu, J.S, Zhu, L.L, Li, H.L. | 登録日 | 2015-05-04 | 公開日 | 2016-05-04 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Crystal structure of Human Dihydroorotate Dehydrogenase (DHODH) with DH03A338 To Be Published
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4IGH
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![BU of 4igh by Molmil](/molmil-images/mine/4igh) | High resolution crystal structure of human dihydroorotate dehydrogenase bound with 4-quinoline carboxylic acid analog | 分子名称: | 3-[decyl(dimethyl)ammonio]propane-1-sulfonate, 6-fluoro-2-[2-methyl-4-phenoxy-5-(propan-2-yl)phenyl]quinoline-4-carboxylic acid, Dihydroorotate dehydrogenase (quinone), ... | 著者 | Deng, X, Das, P, Fontoura, B.M.A, Phillips, M.A, De Brabander, J.K. | 登録日 | 2012-12-17 | 公開日 | 2013-08-21 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.3 Å) | 主引用文献 | SAR Based Optimization of a 4-Quinoline Carboxylic Acid Analog with Potent Anti-Viral Activity. ACS MED.CHEM.LETT., 4, 2013
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4ZL1
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![BU of 4zl1 by Molmil](/molmil-images/mine/4zl1) | Crystal structure of human dihydroorotate dehydrogenase (DHODH) with 18X at 1.86 A resolution | 分子名称: | Dihydroorotate dehydrogenase (quinone), mitochondrial, FLAVIN MONONUCLEOTIDE, ... | 著者 | Huang, J, Wu, D, Ouyang, P, Lu, W, Pu, J. | 登録日 | 2015-05-01 | 公開日 | 2016-05-04 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.86 Å) | 主引用文献 | Crystal structure of human dihydroorotate dehydrogenase (DHODH) with 18XYW at 1.86 A resolution To Be Published
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6OTT
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![BU of 6ott by Molmil](/molmil-images/mine/6ott) | Structure of PurF in complex with ppApp | 分子名称: | Amidophosphoribosyltransferase, PurF, MAGNESIUM ION, ... | 著者 | Grant, R.A, Wang, B, Laub, M.T. | 登録日 | 2019-05-03 | 公開日 | 2019-11-06 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2.55 Å) | 主引用文献 | An interbacterial toxin inhibits target cell growth by synthesizing (p)ppApp. Nature, 575, 2019
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2VD6
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![BU of 2vd6 by Molmil](/molmil-images/mine/2vd6) | Human adenylosuccinate lyase in complex with its substrate N6-(1,2- Dicarboxyethyl)-AMP, and its products AMP and fumarate. | 分子名称: | 2-[9-(3,4-DIHYDROXY-5-PHOSPHONOOXYMETHYL-TETRAHYDRO-FURAN-2-YL)-9H-PURIN-6-YLAMINO]-SUCCINIC ACID, ADENOSINE MONOPHOSPHATE, ADENYLOSUCCINATE LYASE, ... | 著者 | Stenmark, P, Moche, M, Arrowsmith, C, Berglund, H, Busam, R, Collins, R, Dahlgren, L.G, Edwards, A, Flodin, S, Flores, A, Graslund, S, Hammarstrom, M, Hallberg, B.M, Holmberg-schiavone, L, Johansson, I, Kallas, A, Karlberg, T, Kotenyova, T, Lehtio, L, Nilsson, M, Nyman, T, Ogg, D, Persson, C, Sagemark, J, Sundstrom, M, Thorsell, A.G, Tresaugues, L, van den Berg, S, Weigelt, J, Welin, M, Nordlund, P, Structural Genomics Consortium (SGC) | 登録日 | 2007-09-30 | 公開日 | 2007-10-23 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Human Adenylosuccinate Lyase in Complex with its Substrate N6-(1,2-Dicarboxyethyl)-AMP, and its Products AMP and Fumarate. To be Published
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8UXF
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8WKO
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8UXL
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8UXM
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