8DW1
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![BU of 8dw1 by Molmil](/molmil-images/mine/8dw1) | Crystal structure of a host-guest complex with 5'-CTTAGTTATAACTAAG-3' | 分子名称: | DNA (5'-D(*CP*TP*TP*AP*GP*TP*TP*A)-3'), DNA (5'-D(P*TP*AP*AP*CP*TP*AP*AP*G)-3'), reverse transcriptase | 著者 | Georgiadis, M.M. | 登録日 | 2022-07-30 | 公開日 | 2023-01-11 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.849 Å) | 主引用文献 | Two distinct rotations of bithiazole DNA intercalation revealed by direct comparison of crystal structures of Co(III)•bleomycin A 2 and B 2 bound to duplex 5'-TAGTT sites. Bioorg.Med.Chem., 77, 2023
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8DVX
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![BU of 8dvx by Molmil](/molmil-images/mine/8dvx) | Structure of acetylated Pig somatic Cytochrome c (Aly39) at 1.5A | 分子名称: | Cytochrome c, HEME C, HEXACYANOFERRATE(3-) | 著者 | Edwards, B.F.P, Huettemann, M, Vaishnav, A, Brunzelle, J, Morse, P, Wan, J. | 登録日 | 2022-07-30 | 公開日 | 2023-07-19 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Cytochrome c lysine acetylation regulates cellular respiration and cell death in ischemic skeletal muscle. Nat Commun, 14, 2023
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7YNE
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8DVN
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![BU of 8dvn by Molmil](/molmil-images/mine/8dvn) | Crystal structure of LRP6 E3E4 in complex with disulfide constrained peptide E3.10 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Thakur, A.K, Liau, N.P.D, Sudhamsu, J, Hannoush, R.N. | 登録日 | 2022-07-29 | 公開日 | 2023-03-29 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.53 Å) | 主引用文献 | Synthetic Multivalent Disulfide-Constrained Peptide Agonists Potentiate Wnt1/ beta-Catenin Signaling via LRP6 Coreceptor Clustering. Acs Chem.Biol., 18, 2023
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8DVL
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![BU of 8dvl by Molmil](/molmil-images/mine/8dvl) | Crystal structure of LRP6 E3E4 in complex with disulfide constrained peptide E3.18 | 分子名称: | 1,2-ETHANEDIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Thakur, A.K, Liau, N.P.D, Sudhamsu, J, Hannoush, R.N. | 登録日 | 2022-07-29 | 公開日 | 2023-03-29 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Synthetic Multivalent Disulfide-Constrained Peptide Agonists Potentiate Wnt1/ beta-Catenin Signaling via LRP6 Coreceptor Clustering. Acs Chem.Biol., 18, 2023
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8DVM
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![BU of 8dvm by Molmil](/molmil-images/mine/8dvm) | Crystal structure of LRP6 E3E4 in complex with disulfide constrained peptide E3.6 | 分子名称: | 1,2-ETHANEDIOL, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Thakur, A.K, Liau, N.P.D, Sudhamsu, J, Hannoush, R.N. | 登録日 | 2022-07-29 | 公開日 | 2023-03-29 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Synthetic Multivalent Disulfide-Constrained Peptide Agonists Potentiate Wnt1/ beta-Catenin Signaling via LRP6 Coreceptor Clustering. Acs Chem.Biol., 18, 2023
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7YMS
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![BU of 7yms by Molmil](/molmil-images/mine/7yms) | |
8AK3
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![BU of 8ak3 by Molmil](/molmil-images/mine/8ak3) | |
8AK2
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![BU of 8ak2 by Molmil](/molmil-images/mine/8ak2) | Drosophila melanogaster UNC89 Protein Kinase Domain 1 (apo) | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, GLYCEROL, Obscurin | 著者 | Dorendorf, T, Zacharchenko, T, Mayans, O. | 登録日 | 2022-07-29 | 公開日 | 2023-03-29 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | PK1 from Drosophila obscurin is an inactive pseudokinase with scaffolding properties. Open Biology, 13, 2023
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7YMJ
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![BU of 7ymj by Molmil](/molmil-images/mine/7ymj) | Cryo-EM structure of alpha1AAR-Nb6 complex bound to tamsulosin | 分子名称: | Nb6, Tamsulosin, alpha1A-adrenergic receptor | 著者 | Toyoda, Y, Zhu, A, Yan, C, Kobilka, B.K, Liu, X. | 登録日 | 2022-07-28 | 公開日 | 2023-07-05 | 実験手法 | ELECTRON MICROSCOPY (3.35 Å) | 主引用文献 | Structural basis of alpha 1A -adrenergic receptor activation and recognition by an extracellular nanobody. Nat Commun, 14, 2023
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7YMH
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![BU of 7ymh by Molmil](/molmil-images/mine/7ymh) | Cryo-EM structure of Nb29-alpha1AAR-miniGsq complex bound to noradrenaline | 分子名称: | Nb29, Noradrenaline, alpha1A-adrenergic receptor, ... | 著者 | Toyoda, Y, Zhu, A, Yan, C, Kobilka, B.K, Liu, X. | 登録日 | 2022-07-28 | 公開日 | 2023-07-05 | 実験手法 | ELECTRON MICROSCOPY (3.52 Å) | 主引用文献 | Structural basis of alpha 1A -adrenergic receptor activation and recognition by an extracellular nanobody. Nat Commun, 14, 2023
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7YLW
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7YM8
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![BU of 7ym8 by Molmil](/molmil-images/mine/7ym8) | Cryo-EM structure of Nb29-alpha1AAR-miniGsq complex bound to oxymetazoline | 分子名称: | CHOLESTEROL HEMISUCCINATE, Oxymetazoline, alpha1A adrenergic receptor, ... | 著者 | Toyoda, Y, Zhu, A, Yan, C, Kobilka, B.K, Liu, X. | 登録日 | 2022-07-27 | 公開日 | 2023-07-05 | 実験手法 | ELECTRON MICROSCOPY (2.92 Å) | 主引用文献 | Structural basis of alpha 1A -adrenergic receptor activation and recognition by an extracellular nanobody. Nat Commun, 14, 2023
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8AJ4
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![BU of 8aj4 by Molmil](/molmil-images/mine/8aj4) | X-ray structure of lysozyme obtained upon reaction with [VIVO(malt)2] (Structure A') | 分子名称: | 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, 8,8-bis($l^{1}-oxidanyl)-2,2'-dimethyl-8,8'-spirobi[3$l^{4},7,9-trioxa-8$l^{6}-vanadabicyclo[4.3.0]nona-1(6),2,4-triene], Lysozyme, ... | 著者 | Paolillo, M, Merlino, A, Ferraro, G. | 登録日 | 2022-07-27 | 公開日 | 2022-11-23 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.22 Å) | 主引用文献 | Multiple and Variable Binding of Pharmacologically Active Bis(maltolato)oxidovanadium(IV) to Lysozyme. Inorg.Chem., 61, 2022
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8AJ3
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![BU of 8aj3 by Molmil](/molmil-images/mine/8aj3) | X-ray structure of lysozyme obtained upon reaction with [VIVO(malt)2] (Structure A) | 分子名称: | 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, 8,8,8,8-tetrakis($l^{1}-oxidanyl)-2-methyl-3,7,9-trioxa-8$l^{6}-vanadabicyclo[4.3.0]nona-1,5-diene, 8,8-bis($l^{1}-oxidanyl)-2,2'-dimethyl-8,8'-spirobi[3$l^{4},7,9-trioxa-8$l^{6}-vanadabicyclo[4.3.0]nona-1(6),2,4-triene], ... | 著者 | Paolillo, M, Merlino, A, Ferraro, G. | 登録日 | 2022-07-27 | 公開日 | 2022-11-23 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.13 Å) | 主引用文献 | Multiple and Variable Binding of Pharmacologically Active Bis(maltolato)oxidovanadium(IV) to Lysozyme. Inorg.Chem., 61, 2022
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8AJ5
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![BU of 8aj5 by Molmil](/molmil-images/mine/8aj5) | X-ray structure of lysozyme obtained upon reaction with [VIVO(malt)2] (Structure B) | 分子名称: | ACETATE ION, Lysozyme, NITRATE ION, ... | 著者 | Paolillo, M, Merlino, A, Ferraro, G. | 登録日 | 2022-07-27 | 公開日 | 2022-11-23 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.31 Å) | 主引用文献 | Multiple and Variable Binding of Pharmacologically Active Bis(maltolato)oxidovanadium(IV) to Lysozyme. Inorg.Chem., 61, 2022
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8DTN
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![BU of 8dtn by Molmil](/molmil-images/mine/8dtn) | The complex of nanobody 6101 with BCL11A ZF6 | 分子名称: | B-cell lymphoma/leukemia 11A, MAGNESIUM ION, Nanobody 6101, ... | 著者 | Yin, M, Tenglin, K, Zhai, L, Dassama, L.M, Orkin, S.H. | 登録日 | 2022-07-26 | 公開日 | 2023-02-01 | 実験手法 | X-RAY DIFFRACTION (2.199 Å) | 主引用文献 | Evolution of nanobodies specific for BCL11A. Proc.Natl.Acad.Sci.USA, 120, 2023
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8DTU
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![BU of 8dtu by Molmil](/molmil-images/mine/8dtu) | The complex of nanobody 5344N74D with BCL11A ZF6. | 分子名称: | B-cell lymphoma/leukemia 11A, Nanobody 5344N74D, ZINC ION | 著者 | Yin, M, Tenglin, K, Zhai, L, Dassama, L.M, Orkin, S.H. | 登録日 | 2022-07-26 | 公開日 | 2023-02-01 | 実験手法 | X-RAY DIFFRACTION (2.447 Å) | 主引用文献 | Evolution of nanobodies specific for BCL11A. Proc.Natl.Acad.Sci.USA, 120, 2023
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7YLK
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![BU of 7ylk by Molmil](/molmil-images/mine/7ylk) | Myoglobin containing Ir complex | 分子名称: | Myoglobin, SULFATE ION, delta-{1-([2,2'-bipyridin]-5-ylmethyl)pyrrolidine-2,5-dione}bis[2-(2,4-difluorophenyl)pyridine)]iridium(III), ... | 著者 | Lee, J.H, Song, W.J. | 登録日 | 2022-07-26 | 公開日 | 2023-03-15 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.63 Å) | 主引用文献 | Photocatalytic C-O Coupling Enzymes That Operate via Intramolecular Electron Transfer. J.Am.Chem.Soc., 145, 2023
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8DTM
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![BU of 8dtm by Molmil](/molmil-images/mine/8dtm) | Cryo-EM structure of insulin receptor (IR) bound with S597 component 2 | 分子名称: | Insulin mimetic peptide S597 component 2, Insulin receptor | 著者 | Park, J, Li, J, Mayer, J.P, Ball, K.A, Wu, J.Y, Hall, C, Accili, D, Stowell, M.H.B, Bai, X.C, Choi, E. | 登録日 | 2022-07-26 | 公開日 | 2022-09-07 | 最終更新日 | 2022-10-12 | 実験手法 | ELECTRON MICROSCOPY (3.5 Å) | 主引用文献 | Activation of the insulin receptor by an insulin mimetic peptide. Nat Commun, 13, 2022
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8DU3
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![BU of 8du3 by Molmil](/molmil-images/mine/8du3) | Crystal structure of A2AAR-StaR2-bRIL in complex with compound 21a | 分子名称: | (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, (4M)-6-bromo-4-(furan-2-yl)quinazolin-2-amine, Adenosine receptor A2a, ... | 著者 | Shiriaeva, A, Stauch, B, Han, G.W, Cherezov, V. | 登録日 | 2022-07-26 | 公開日 | 2022-08-10 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | High ligand efficiency quinazoline compounds as novel A 2A adenosine receptor antagonists. Eur.J.Med.Chem., 241, 2022
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7YL1
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![BU of 7yl1 by Molmil](/molmil-images/mine/7yl1) | |
7YKZ
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![BU of 7ykz by Molmil](/molmil-images/mine/7ykz) | Cryo-EM structure of Drg1 hexamer in the planar state treated with ADP/AMPPNP/Diazaborine | 分子名称: | 2-(TOLUENE-4-SULFONYL)-2H-BENZO[D][1,2,3]DIAZABORININ-1-OL, ADENOSINE-5'-DIPHOSPHATE, ADENOSINE-5'-TRIPHOSPHATE, ... | 著者 | Ma, C.Y, Wu, D.M, Chen, Q, Gao, N. | 登録日 | 2022-07-25 | 公開日 | 2022-12-14 | 最終更新日 | 2024-07-03 | 実験手法 | ELECTRON MICROSCOPY (4.3 Å) | 主引用文献 | Structural dynamics of AAA + ATPase Drg1 and mechanism of benzo-diazaborine inhibition. Nat Commun, 13, 2022
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8DTL
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![BU of 8dtl by Molmil](/molmil-images/mine/8dtl) | Cryo-EM structure of insulin receptor (IR) bound with S597 peptide | 分子名称: | Insulin mimetic peptide S597, Insulin receptor | 著者 | Park, J, Li, J, Mayer, J.P, Ball, K.A, Wu, J.Y, Hall, C, Accili, D, Stowell, M.H.B, Bai, X.C, Choi, E. | 登録日 | 2022-07-25 | 公開日 | 2022-09-07 | 最終更新日 | 2022-10-12 | 実験手法 | ELECTRON MICROSCOPY (5.4 Å) | 主引用文献 | Activation of the insulin receptor by an insulin mimetic peptide. Nat Commun, 13, 2022
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8AHY
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![BU of 8ahy by Molmil](/molmil-images/mine/8ahy) | |