4R7L
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![BU of 4r7l by Molmil](/molmil-images/mine/4r7l) | Structure of Human Leukotriene A4 Hydrolase in complex with inhibitor H1 | 分子名称: | ACETATE ION, GLYCEROL, IMIDAZOLE, ... | 著者 | Ouyang, P, Cui, K, Lu, W, Huang, J. | 登録日 | 2014-08-27 | 公開日 | 2015-11-25 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (1.66 Å) | 主引用文献 | Human Leukotriene A4 Hydrolase in complex with SAHA To be Published
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4E9A
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![BU of 4e9a by Molmil](/molmil-images/mine/4e9a) | Structure of Peptide Deformylase form Helicobacter Pylori in complex with inhibitor | 分子名称: | 2-phenylethyl (2E)-3-(3,4-dihydroxyphenyl)prop-2-enoate, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, COBALT (II) ION, ... | 著者 | Cui, K, Zhu, L, Lu, W, Huang, J. | 登録日 | 2012-03-20 | 公開日 | 2013-04-24 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.662 Å) | 主引用文献 | Identification of Novel Peptide Deformylase Inhibitors from Natural Products To be Published
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4CC6
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![BU of 4cc6 by Molmil](/molmil-images/mine/4cc6) | Fragment-Based Discovery of 6 Azaindazoles As Inhibitors of Bacterial DNA Ligase | 分子名称: | 2-{[2-(1H-pyrazolo[3,4-c]pyridin-3-yl)-6-(trifluoromethyl)pyridin-4-yl]amino}ethanol, DNA LIGASE, SULFATE ION | 著者 | Howard, S, Amin, N, Benowitz, A.B, Chiarparin, E, Cui, H, Deng, X, Heightman, T.D, Holmes, D.J, Hopkins, A, Huang, J, Jin, Q, Kreatsoulas, C, Martin, A.C.L, Massey, F, McCloskey, L, Mortenson, P.N, Pathuri, P, Tisi, D, Williams, P.A. | 登録日 | 2013-10-18 | 公開日 | 2014-06-18 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.01 Å) | 主引用文献 | Fragment-Based Discovery of 6-Azaindazoles as Inhibitors of Bacterial DNA Ligase. Acs Med.Chem.Lett., 4, 2013
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4CC5
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![BU of 4cc5 by Molmil](/molmil-images/mine/4cc5) | Fragment-Based Discovery of 6 Azaindazoles As Inhibitors of Bacterial DNA Ligase | 分子名称: | 2-chloranyl-6-(1H-1,2,4-triazol-3-yl)pyrazine, DNA LIGASE, SULFATE ION | 著者 | Howard, S, Amin, N, Benowitz, A.B, Chiarparin, E, Cui, H, Deng, X, Heightman, T.D, Holmes, D.J, Hopkins, A, Huang, J, Jin, Q, Kreatsoulas, C, Martin, A.C.L, Massey, F, McCloskey, L, Mortenson, P.N, Pathuri, P, Tisi, D, Williams, P.A. | 登録日 | 2013-10-18 | 公開日 | 2014-06-18 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.88 Å) | 主引用文献 | Fragment-Based Discovery of 6-Azaindazoles as Inhibitors of Bacterial DNA Ligase. Acs Med.Chem.Lett., 4, 2013
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4E9B
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![BU of 4e9b by Molmil](/molmil-images/mine/4e9b) | Structure of Peptide Deformylase form Helicobacter Pylori in complex with actinonin | 分子名称: | 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, ACTINONIN, COBALT (II) ION, ... | 著者 | Cui, K, Zhu, L, Lu, W, Huang, J. | 登録日 | 2012-03-20 | 公開日 | 2013-04-24 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Identification of Novel Peptide Deformylase Inhibitors from Natural Products To be Published
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1DT0
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![BU of 1dt0 by Molmil](/molmil-images/mine/1dt0) | CLONING, SEQUENCE, AND CRYSTALLOGRAPHIC STRUCTURE OF RECOMBINANT IRON SUPEROXIDE DISMUTASE FROM PSEUDOMONAS OVALIS | 分子名称: | FE (III) ION, SUPEROXIDE DISMUTASE | 著者 | Bond, C.J, Huang, J, Hajduk, R, Flick, K, Heath, P, Stoddard, B.L. | 登録日 | 2000-01-10 | 公開日 | 2000-12-20 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Cloning, sequence and crystallographic structure of recombinant iron superoxide dismutase from Pseudomonas ovalis. Acta Crystallogr.,Sect.D, 56, 2000
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1EMS
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![BU of 1ems by Molmil](/molmil-images/mine/1ems) | CRYSTAL STRUCTURE OF THE C. ELEGANS NITFHIT PROTEIN | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, ETHYL MERCURY ION, NIT-FRAGILE HISTIDINE TRIAD FUSION PROTEIN, ... | 著者 | Pace, H.C, Hodawadekar, S.C, Draganescu, A, Huang, J, Bieganowski, P, Pekarsky, Y, Croce, C.M, Brenner, C. | 登録日 | 2000-03-17 | 公開日 | 2000-07-20 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Crystal structure of the worm NitFhit Rosetta Stone protein reveals a Nit tetramer binding two Fhit dimers. Curr.Biol., 10, 2000
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4KN8
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![BU of 4kn8 by Molmil](/molmil-images/mine/4kn8) | Crystal structure of Bs-TpNPPase | 分子名称: | Thermostable NPPase | 著者 | Guo, Z, Wang, F, Huang, J, Gong, W, Ji, C. | 登録日 | 2013-05-09 | 公開日 | 2014-04-09 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.502 Å) | 主引用文献 | Crystal Structure of Thermostable p-nitrophenylphosphatase from Bacillus Stearothermophilus (Bs-TpNPPase) PROTEIN PEPT.LETT., 21, 2014
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2IEL
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![BU of 2iel by Molmil](/molmil-images/mine/2iel) | CRYSTAL STRUCTURE OF TT0030 from Thermus Thermophilus | 分子名称: | Hypothetical Protein TT0030 | 著者 | Zhu, J, Huang, J, Stepanyuk, G, Chen, L, Chang, J, Zhao, M, Xu, H, Liu, Z.J, Rose, J.P, Wang, B.C, Southeast Collaboratory for Structural Genomics (SECSG) | 登録日 | 2006-09-19 | 公開日 | 2006-11-14 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | CRYSTAL STRUCTURE OF TT0030 from Thermus Thermophilus AT 1.6 ANGSTROMS RESOLUTION To be Published
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3TYH
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![BU of 3tyh by Molmil](/molmil-images/mine/3tyh) | Crystal structure of oxo-cupper clusters binding to ferric binding protein from Neisseria gonorrhoeae | 分子名称: | COPPER (II) ION, FbpA protein | 著者 | Chen, W.J, Wang, H.F, Zhou, C.J, Ye, D.R, Huang, J, Tan, X.S, Zhong, W.Q. | 登録日 | 2011-09-26 | 公開日 | 2012-09-26 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Crystal structure of oxo-cupper clusters binding to ferric binding protein from Neisseria gonorrhoeae To be Published
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2JTK
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![BU of 2jtk by Molmil](/molmil-images/mine/2jtk) | |
5Z2S
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![BU of 5z2s by Molmil](/molmil-images/mine/5z2s) | Crystal structure of DUX4-HD2 domain | 分子名称: | Double homeobox protein 4 | 著者 | Dong, X, Zhang, W, Wu, H, Huang, J, Zhang, M, Wang, P, Zhang, H, Chen, Z, Chen, S, Meng, G. | 登録日 | 2018-01-03 | 公開日 | 2018-04-04 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Structural basis of DUX4/IGH-driven transactivation. Leukemia, 32, 2018
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5Z2T
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![BU of 5z2t by Molmil](/molmil-images/mine/5z2t) | Crystal structure of DNA-bound DUX4-HD2 | 分子名称: | 5'-D(*TP*TP*CP*TP*AP*AP*TP*CP*TP*AP*AP*TP*CP*TP*T)-3', 5'-D(P*AP*AP*GP*AP*TP*TP*AP*GP*AP*TP*TP*AP*GP*T)-3', Double homeobox protein 4 | 著者 | Dong, X, Zhang, W, Wu, H, Huang, J, Zhang, M, Wang, P, Zhang, H, Chen, Z, Chen, S, Meng, G. | 登録日 | 2018-01-04 | 公開日 | 2018-04-04 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.623 Å) | 主引用文献 | Structural basis of DUX4/IGH-driven transactivation. Leukemia, 32, 2018
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7DW5
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![BU of 7dw5 by Molmil](/molmil-images/mine/7dw5) | Crystal structure of DUX4 HD1-HD2 domain complexed with ERG sites | 分子名称: | BROMIDE ION, DNA (5'-D(P*CP*GP*AP*CP*TP*TP*GP*AP*TP*GP*AP*GP*AP*TP*TP*AP*GP*AP*CP*TP*G)-3'), Double homeobox protein 4-like protein 2 | 著者 | Zhang, H, Cheng, N, Li, Z, Zhang, W, Dong, X, Huang, J, Meng, G. | 登録日 | 2021-01-15 | 公開日 | 2021-11-03 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.83 Å) | 主引用文献 | DNA crosslinking and recombination-activating genes 1/2 (RAG1/2) are required for oncogenic splicing in acute lymphoblastic leukemia. Cancer Commun (Lond), 41, 2021
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7Y7Y
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![BU of 7y7y by Molmil](/molmil-images/mine/7y7y) | Cryo-EM structure of human GABA transporter GAT1 bound with nipecotic acid in NaCl solution in an inward-occluded state at 2.4 angstrom | 分子名称: | (3R)-piperidine-3-carboxylic acid, 2-acetamido-2-deoxy-beta-D-glucopyranose, CHLORIDE ION, ... | 著者 | Zhu, A, Huang, J, Kong, F, Tan, J, Lei, J, Yuan, Y, Yan, C. | 登録日 | 2022-06-22 | 公開日 | 2023-04-26 | 最終更新日 | 2023-08-16 | 実験手法 | ELECTRON MICROSCOPY (2.4 Å) | 主引用文献 | Molecular basis for substrate recognition and transport of human GABA transporter GAT1. Nat.Struct.Mol.Biol., 30, 2023
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7Y7V
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![BU of 7y7v by Molmil](/molmil-images/mine/7y7v) | Cryo-EM structure of human apo GABA transporter GAT1 in an inward-open state | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, CHLORIDE ION, Sodium- and chloride-dependent GABA transporter 1 | 著者 | Zhu, A, Huang, J, Kong, F, Tan, J, Lei, J, Yuan, Y, Yan, C. | 登録日 | 2022-06-22 | 公開日 | 2023-04-26 | 最終更新日 | 2023-08-16 | 実験手法 | ELECTRON MICROSCOPY (2.2 Å) | 主引用文献 | Molecular basis for substrate recognition and transport of human GABA transporter GAT1. Nat.Struct.Mol.Biol., 30, 2023
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7Y7Z
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![BU of 7y7z by Molmil](/molmil-images/mine/7y7z) | Cryo-EM structure of human GABA transporter GAT1 bound with tiagabine in NaCl solution in an inward-open state at 3.2 angstrom | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, CHLORIDE ION, Sodium- and chloride-dependent GABA transporter 1, ... | 著者 | Zhu, A, Huang, J, Kong, F, Tan, J, Lei, J, Yuan, Y, Yan, C. | 登録日 | 2022-06-22 | 公開日 | 2023-04-26 | 最終更新日 | 2023-11-29 | 実験手法 | ELECTRON MICROSCOPY (3.2 Å) | 主引用文献 | Molecular basis for substrate recognition and transport of human GABA transporter GAT1. Nat.Struct.Mol.Biol., 30, 2023
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7Y7W
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![BU of 7y7w by Molmil](/molmil-images/mine/7y7w) | Cryo-EM structure of human GABA transporter GAT1 bound with GABA in NaCl solution in an inward-occluded state at 2.4 angstrom | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, CHLORIDE ION, GAMMA-AMINO-BUTANOIC ACID, ... | 著者 | Zhu, A, Huang, J, Kong, F, Tan, J, Lei, J, Yuan, Y, Yan, C. | 登録日 | 2022-06-22 | 公開日 | 2023-04-26 | 最終更新日 | 2023-11-15 | 実験手法 | ELECTRON MICROSCOPY (2.4 Å) | 主引用文献 | Molecular basis for substrate recognition and transport of human GABA transporter GAT1. Nat.Struct.Mol.Biol., 30, 2023
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7JJO
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![BU of 7jjo by Molmil](/molmil-images/mine/7jjo) | Structural Basis of the Activation of Heterotrimeric Gs-protein by Isoproterenol-bound Beta1-Adrenergic Receptor | 分子名称: | Beta1-Adrenergic Receptor, Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2, Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1, ... | 著者 | Su, M, Zhu, L, Zhang, Y, Paknejad, N, Dey, R, Huang, J, Lee, M.Y, Williams, D, Jordan, K.D, Eng, E.T, Ernst, O.P, Meyerson, J.R, Hite, R.K, Walz, T, Liu, W, Huang, X.Y. | 登録日 | 2020-07-27 | 公開日 | 2020-09-02 | 最終更新日 | 2020-10-14 | 実験手法 | ELECTRON MICROSCOPY (2.6 Å) | 主引用文献 | Structural Basis of the Activation of Heterotrimeric Gs-Protein by Isoproterenol-Bound beta 1 -Adrenergic Receptor. Mol.Cell, 80, 2020
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6J3N
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![BU of 6j3n by Molmil](/molmil-images/mine/6j3n) | |
6J99
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![BU of 6j99 by Molmil](/molmil-images/mine/6j99) | |
2JZI
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![BU of 2jzi by Molmil](/molmil-images/mine/2jzi) | |
7E3M
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![BU of 7e3m by Molmil](/molmil-images/mine/7e3m) | RORgamma LBD complexed with Panaxatriol and SRC2.2 | 分子名称: | (3R,5R,6S,8R,9R,10R,12R,13R,14R,17S)-4,4,8,10,14-pentamethyl-17-[(2R)-2,6,6-trimethyloxan-2-yl]-2,3,5,6,7,9,11,12,13,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthrene-3,6,12-triol, LYS-ILE-LEU-HIS-ARG-LEU-LEU-GLN, Nuclear receptor ROR-gamma | 著者 | Liu, Z.H, Huang, J, Lu, W.Q, Tang, Y, Wu, Z.R. | 登録日 | 2021-02-09 | 公開日 | 2022-03-23 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Structure of human RORgammat LBD with SRC2.2 at 2.80 Angstroms resolution To Be Published
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7CWY
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![BU of 7cwy by Molmil](/molmil-images/mine/7cwy) | Crystal structure of a tyrosine decarboxylase from Enterococcus faecalis in complex with the cofactor PLP | 分子名称: | Decarboxylase | 著者 | Yu, X, Gong, M, Huang, J, Liu, W, Chen, C, Guo, R. | 登録日 | 2020-09-01 | 公開日 | 2021-09-01 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.59 Å) | 主引用文献 | Crystal structure of a tyrosine decarboxylase from Enterococcus faecalis in complex with the cofactor PLP to be published
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7CX0
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![BU of 7cx0 by Molmil](/molmil-images/mine/7cx0) | Crystal structure of a tyrosine decarboxylase from Enterococcus faecalis in complex with the cofactor PLP and inhibitor carbidopa | 分子名称: | CARBIDOPA, Decarboxylase, PYRIDOXAL-5'-PHOSPHATE | 著者 | Yu, X, Gong, M, Huang, J, Liu, W, Chen, C, Guo, R. | 登録日 | 2020-09-01 | 公開日 | 2021-09-01 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.66 Å) | 主引用文献 | Crystal structure of a tyrosine decarboxylase from Enterococcus faecalis in complex with the cofactor PLP and inhibitor carbidopa to be published
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