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3CX8
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BU of 3cx8 by Molmil
Crystal Structure of PDZRhoGEF rgRGS Domain in a Complex with Galpha-13 Bound to GTP-gamma-S
分子名称: 5'-GUANOSINE-DIPHOSPHATE-MONOTHIOPHOSPHATE, Guanine nucleotide-binding protein alpha-13 subunit, MAGNESIUM ION, ...
著者Sprang, S.R, Chen, Z.
登録日2008-04-23
公開日2008-10-28
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Recognition of the Activated States of Galpha13 by the rgRGS Domain of PDZRhoGEF.
Structure, 16, 2008
5WUK
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BU of 5wuk by Molmil
Crystal structure of EED [G255D] in complex with EZH2 peptide and EED226 compound
分子名称: GLYCEROL, Histone-lysine N-methyltransferase EZH2, N-(furan-2-ylmethyl)-8-(4-methylsulfonylphenyl)-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine, ...
著者Chen, Z.
登録日2016-12-19
公開日2017-05-03
実験手法X-RAY DIFFRACTION (2.03 Å)
主引用文献Split luciferase-based biosensors for characterizing EED binders
Anal. Biochem., 522, 2017
6V06
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BU of 6v06 by Molmil
Crystal structure of Beta-2 glycoprotein I purified from plasma (pB2GPI)
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-beta-D-mannopyranose-(1-6)-beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, Beta-2-glycoprotein 1, ...
著者Chen, Z, Ruben, E.A, Planer, W, Chinnaraj, M, Zuo, X, Pengo, V, Macor, P, Tedesco, F, Pozzi, N.
登録日2019-11-18
公開日2020-06-17
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献The J-elongated conformation of beta2-glycoprotein I predominates in solution: implications for our understanding of antiphospholipid syndrome.
J.Biol.Chem., 295, 2020
6V09
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BU of 6v09 by Molmil
Crystal structure of human recombinant Beta-2 glycoprotein I short tag (ST-B2GPI)
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, Beta-2-glycoprotein 1, SULFATE ION, ...
著者Chen, Z, Ruben, E.A, Planer, W, Chinnaraj, M, Zuo, X, Pengo, V, Macor, P, Tedesco, F, Pozzi, N.
登録日2019-11-18
公開日2020-06-17
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.99 Å)
主引用文献The J-elongated conformation of beta2-glycoprotein I predominates in solution: implications for our understanding of antiphospholipid syndrome.
J.Biol.Chem., 295, 2020
6DMA
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BU of 6dma by Molmil
DHD15_closed
分子名称: DHD15_closed_A, DHD15_closed_B
著者Bick, M.J, Chen, Z, Baker, D.
登録日2018-06-04
公開日2018-12-19
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (3.363 Å)
主引用文献Programmable design of orthogonal protein heterodimers.
Nature, 565, 2019
6DKM
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BU of 6dkm by Molmil
DHD131
分子名称: DHD131_A, DHD131_B
著者Bick, M.J, Chen, Z, Baker, D.
登録日2018-05-29
公開日2018-12-19
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.38 Å)
主引用文献Programmable design of orthogonal protein heterodimers.
Nature, 565, 2019
6DM9
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BU of 6dm9 by Molmil
DHD15_extended
分子名称: DHD15_extended_A, DHD15_extended_B, SULFATE ION
著者Bick, M.J, Chen, Z, Baker, D.
登録日2018-06-04
公開日2018-12-19
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献Programmable design of orthogonal protein heterodimers.
Nature, 565, 2019
6DLC
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BU of 6dlc by Molmil
Designed protein DHD1:234_A, Designed protein DHD1:234_B
分子名称: Designed protein DHD1:234_A, Designed protein DHD1:234_B
著者Bick, M.J, Chen, Z, Baker, D.
登録日2018-05-31
公開日2018-12-26
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (3.261 Å)
主引用文献Programmable design of orthogonal protein heterodimers.
Nature, 565, 2019
8D6G
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BU of 8d6g by Molmil
Nanorana parkeri saxiphilin
分子名称: PENTAETHYLENE GLYCOL, Saxiphilin
著者Zakrzewska, S, Chen, Z, Minor, D.L.
登録日2022-06-06
公開日2022-11-02
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Definition of a saxitoxin (STX) binding code enables discovery and characterization of the anuran saxiphilin family.
Proc.Natl.Acad.Sci.USA, 119, 2022
8D6O
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BU of 8d6o by Molmil
Nanorana parkeri saxiphilin:F-STX (soaked)
分子名称: (2P)-4-({6-[({[(3aS,4R,7R,10aS)-2,6-diamino-10,10-dihydroxy-3a,4,9,10-tetrahydro-3H,8H-pyrrolo[1,2-c]purin-4-yl]methoxy}carbonyl)amino]hexyl}carbamoyl)-2-{[4aP,9(9a)P]-6-hydroxy-3-oxo-3H-xanthen-9-yl}benzoic acid, PENTAETHYLENE GLYCOL, Saxiphilin
著者Zakrzewska, S, Chen, Z, Minor, D.L.
登録日2022-06-06
公開日2022-11-02
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Definition of a saxitoxin (STX) binding code enables discovery and characterization of the anuran saxiphilin family.
Proc.Natl.Acad.Sci.USA, 119, 2022
8D6M
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BU of 8d6m by Molmil
Nanorana parkeri saxiphilin:STX (co-crystal)
分子名称: PENTAETHYLENE GLYCOL, Saxiphilin, [(3aS,4R,10aS)-2,6-diamino-10,10-dihydroxy-3a,4,9,10-tetrahydro-3H,8H-pyrrolo[1,2-c]purin-4-yl]methyl carbamate
著者Zakrzewska, S, Chen, Z, Minor, D.L.
登録日2022-06-06
公開日2022-11-02
最終更新日2024-03-27
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Definition of a saxitoxin (STX) binding code enables discovery and characterization of the anuran saxiphilin family.
Proc.Natl.Acad.Sci.USA, 119, 2022
6V08
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BU of 6v08 by Molmil
Crystal structure of human recombinant Beta-2 glycoprotein I (hrB2GPI)
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Beta-2-glycoprotein 1, SULFATE ION, ...
著者Chen, Z, Ruben, E.A, Planer, W, Chinnaraj, M, Zuo, X, Pengo, V, Macor, P, Tedesco, F, Pozzi, N.
登録日2019-11-18
公開日2020-06-17
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.58 Å)
主引用文献The J-elongated conformation of beta2-glycoprotein I predominates in solution: implications for our understanding of antiphospholipid syndrome.
J.Biol.Chem., 295, 2020
6A0P
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BU of 6a0p by Molmil
Crystal structure of Usutu virus envelope protein in the pre-fusion state
分子名称: Envelope protein
著者Lu, G, Chen, Z, Ye, F, Lin, S, Yang, F, Cheng, Y.
登録日2018-06-06
公開日2018-12-26
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystal structure of Usutu virus envelope protein in the pre-fusion state
Virol. J., 15, 2018
8SYN
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BU of 8syn by Molmil
Human VPS35L/VPS29/VPS26C Complex
分子名称: VPS35 endosomal protein-sorting factor-like, Vacuolar protein sorting-associated protein 26C, Vacuolar protein sorting-associated protein 29
著者Chen, Z, Chen, B, Burstein, E, Han, Y.
登録日2023-05-25
公開日2023-11-01
最終更新日2024-07-03
実験手法ELECTRON MICROSCOPY (2.94 Å)
主引用文献Structural organization of the retriever-CCC endosomal recycling complex.
Nat.Struct.Mol.Biol., 31, 2024
8SYM
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BU of 8sym by Molmil
Human VPS29/VPS35L Complex (Locally refined map)
分子名称: VPS35 endosomal protein-sorting factor-like, Vacuolar protein sorting-associated protein 29
著者Chen, Z, Chen, B, Burstein, E, Han, Y.
登録日2023-05-25
公開日2023-11-01
最終更新日2024-07-03
実験手法ELECTRON MICROSCOPY (3.2 Å)
主引用文献Structural organization of the retriever-CCC endosomal recycling complex.
Nat.Struct.Mol.Biol., 31, 2024
8SYO
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BU of 8syo by Molmil
Human Retriever VPS35L/VPS29/VPS26C Complex (Composite Map)
分子名称: VPS35 endosomal protein-sorting factor-like, Vacuolar protein sorting-associated protein 26C, Vacuolar protein sorting-associated protein 29
著者Chen, Z, Chen, B, Burstein, E, Han, Y.
登録日2023-05-25
公開日2023-11-01
最終更新日2024-07-03
実験手法ELECTRON MICROSCOPY (2.94 Å)
主引用文献Structural organization of the retriever-CCC endosomal recycling complex.
Nat.Struct.Mol.Biol., 31, 2024
6EGC
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BU of 6egc by Molmil
Single-chain version of 2L4HC2_23 (PDB 5J0K)
分子名称: SC_2L4HC2_23
著者Bick, M.J, Chen, Z, DiMaio, F.
登録日2018-08-19
公開日2019-05-29
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.74 Å)
主引用文献Self-Assembling 2D Arrays with de Novo Protein Building Blocks.
J.Am.Chem.Soc., 141, 2019
6BB3
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BU of 6bb3 by Molmil
Lactate Dehydrogenase in complex with inhibitor 3-((2-chlorophenyl)thio)-6-(6-((4-fluorophenyl)amino)pyridin-2-yl)-4-hydroxy-6-(thiophen-3-yl)-5,6-dihydro-2H-pyran-2-one
分子名称: (6R)-3-[(2-chlorophenyl)sulfanyl]-6-{6-[(4-fluorophenyl)amino]pyridin-2-yl}-4-hydroxy-6-(thiophen-3-yl)-5,6-dihydro-2H-pyran-2-one, L-lactate dehydrogenase A chain, NICOTINAMIDE-ADENINE-DINUCLEOTIDE, ...
著者Chen, Z, Eigenbrot, C.
登録日2017-10-16
公開日2018-10-24
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structure-guided optimization and in vivo activities of hydroxylactone and hydroxylactam Inhibitors of Human Lactate Dehydrogenase
To Be Published
2KAI
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BU of 2kai by Molmil
REFINED 2.5 ANGSTROMS X-RAY CRYSTAL STRUCTURE OF THE COMPLEX FORMED BY PORCINE KALLIKREIN A AND THE BOVINE PANCREATIC TRYPSIN INHIBITOR. CRYSTALLIZATION, PATTERSON SEARCH, STRUCTURE DETERMINATION, REFINEMENT, STRUCTURE AND COMPARISON WITH ITS COMPONENTS AND WITH THE BOVINE TRYPSIN-PANCREATIC TRYPSIN INHIBITOR COMPLEX
分子名称: BOVINE PANCREATIC TRYPSIN INHIBITOR, KALLIKREIN A
著者Bode, W, Chen, Z.
登録日1984-05-21
公開日1984-07-19
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Refined 2.5 A X-ray crystal structure of the complex formed by porcine kallikrein A and the bovine pancreatic trypsin inhibitor. Crystallization, Patterson search, structure determination, refinement, structure and comparison with its components and with the bovine trypsin-pancreatic trypsin inhibitor complex
J.Mol.Biol., 164, 1983
6CQS
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BU of 6cqs by Molmil
Sediminispirochaeta smaragdinae SPS-1 metallo-beta-lactamase
分子名称: Beta-lactamase, ZINC ION
著者Page, R.C, VanPelt, J, Cheng, Z, Crowder, M.W.
登録日2018-03-16
公開日2018-08-29
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献A Noncanonical Metal Center Drives the Activity of the Sediminispirochaeta smaragdinae Metallo-beta-lactamase SPS-1.
Biochemistry, 57, 2018
5IXY
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BU of 5ixy by Molmil
Lactate Dehydrogenase in complex with hydroxylactam inhibitor compound 31: (2~{S})-5-(2-chlorophenyl)sulfanyl-2-(4-morpholin-4-ylphenyl)-4-oxidanyl-2-thiophen-3-yl-1,3-dihydropyridin-6-one
分子名称: (2~{S})-5-(2-chlorophenyl)sulfanyl-2-(4-morpholin-4-ylphenyl)-4-oxidanyl-2-thiophen-3-yl-1,3-dihydropyridin-6-one, L-lactate dehydrogenase A chain, NICOTINAMIDE-ADENINE-DINUCLEOTIDE, ...
著者Chen, Z, Eigenbrot, C.
登録日2016-03-23
公開日2016-09-14
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Cell Active Hydroxylactam Inhibitors of Human Lactate Dehydrogenase with Oral Bioavailability in Mice.
Acs Med.Chem.Lett., 7, 2016
6BCB
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BU of 6bcb by Molmil
A Complex between PH Domain of p114RhoGEF and Activated RhoA Bound to a GTP Analog
分子名称: 1,2-ETHANEDIOL, 5'-GUANOSINE-DIPHOSPHATE-MONOTHIOPHOSPHATE, MAGNESIUM ION, ...
著者Sternweis, P.C, Chen, Z.
登録日2017-10-20
公開日2017-12-13
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (1.401 Å)
主引用文献Crystal structures of the PH domains from Lbc family of RhoGEFs bound to activated RhoA GTPase.
Data Brief, 17, 2018
6BC0
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BU of 6bc0 by Molmil
A Complex between PH Domain of p190RhoGEF and Activated RhoA Bound to a GTP Analog
分子名称: 5'-GUANOSINE-DIPHOSPHATE-MONOTHIOPHOSPHATE, MAGNESIUM ION, Rho guanine nucleotide exchange factor 28, ...
著者Chen, Z, Sternweis, P.C.
登録日2017-10-20
公開日2017-12-13
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2.198 Å)
主引用文献Direct regulation of p190RhoGEF by activated Rho and Rac GTPases.
J. Struct. Biol., 202, 2018
6BC1
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A Complex between PH Domain of p190RhoGEF and Activated Rac1 Bound to a GTP Analog
分子名称: 5'-GUANOSINE-DIPHOSPHATE-MONOTHIOPHOSPHATE, MAGNESIUM ION, Ras-related C3 botulinum toxin substrate 1, ...
著者Chen, Z, Sternweis, P.C.
登録日2017-10-20
公開日2017-12-13
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Direct regulation of p190RhoGEF by activated Rho and Rac GTPases.
J. Struct. Biol., 202, 2018
6BCA
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BU of 6bca by Molmil
A Complex between PH Domain of LbcRhoGEF (AKAP-Lbc) and Activated RhoA Bound to a GTP Analog
分子名称: 5'-GUANOSINE-DIPHOSPHATE-MONOTHIOPHOSPHATE, A-kinase anchor protein 13, MAGNESIUM ION, ...
著者Sternweis, P.C, Chen, Z.
登録日2017-10-20
公開日2017-12-13
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (1.995 Å)
主引用文献Crystal structures of the PH domains from Lbc family of RhoGEFs bound to activated RhoA GTPase.
Data Brief, 17, 2018

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