7NSC
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![BU of 7nsc by Molmil](/molmil-images/mine/7nsc) | Substrate receptor scaffolding module of human CTLH E3 ubiquitin ligase | 分子名称: | Glucose-induced degradation protein 4 homolog, Glucose-induced degradation protein 8 homolog, Isoform 2 of Armadillo repeat-containing protein 8, ... | 著者 | Chrustowicz, J, Sherpa, D, Prabu, J.R, Schulman, B.A. | 登録日 | 2021-03-05 | 公開日 | 2021-05-05 | 最終更新日 | 2024-07-10 | 実験手法 | ELECTRON MICROSCOPY (3.3 Å) | 主引用文献 | GID E3 ligase supramolecular chelate assembly configures multipronged ubiquitin targeting of an oligomeric metabolic enzyme. Mol.Cell, 81, 2021
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7NS4
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![BU of 7ns4 by Molmil](/molmil-images/mine/7ns4) | Catalytic module of yeast Chelator-GID SR4 E3 ubiquitin ligase | 分子名称: | E3 ubiquitin-protein ligase RMD5, Protein FYV10, ZINC ION | 著者 | Sherpa, D, Chrustowicz, J, Prabu, J.R, Schulman, B.A. | 登録日 | 2021-03-05 | 公開日 | 2021-05-05 | 最終更新日 | 2024-07-10 | 実験手法 | ELECTRON MICROSCOPY (3.9 Å) | 主引用文献 | GID E3 ligase supramolecular chelate assembly configures multipronged ubiquitin targeting of an oligomeric metabolic enzyme. Mol.Cell, 81, 2021
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5UDH
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![BU of 5udh by Molmil](/molmil-images/mine/5udh) | HHARI/ARIH1-UBCH7~Ubiquitin | 分子名称: | E3 ubiquitin-protein ligase ARIH1, Ubiquitin C variant, Ubiquitin-conjugating enzyme E2 L3, ... | 著者 | Miller, D.J, Schulman, B.A. | 登録日 | 2016-12-27 | 公開日 | 2017-06-14 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (3.24 Å) | 主引用文献 | Structural Studies of HHARI/UbcH7Ub Reveal Unique E2Ub Conformational Restriction by RBR RING1. Structure, 25, 2017
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5V89
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![BU of 5v89 by Molmil](/molmil-images/mine/5v89) | Structure of DCN4 PONY domain bound to CUL1 WHB | 分子名称: | Cullin-1, DCN1-like protein 4 | 著者 | Guy, R.K, Schulman, B.A, Scott, D.C, Hammill, J.T. | 登録日 | 2017-03-21 | 公開日 | 2017-05-24 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Blocking an N-terminal acetylation-dependent protein interaction inhibits an E3 ligase. Nat. Chem. Biol., 13, 2017
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5V83
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![BU of 5v83 by Molmil](/molmil-images/mine/5v83) | Structure of DCN1 bound to NAcM-HIT | 分子名称: | Lysozyme,DCN1-like protein 1 chimera, N-(1-benzylpiperidin-4-yl)-N'-[3-(trifluoromethyl)phenyl]urea | 著者 | Guy, R.K, Schulman, B.A, Scott, D.C, Hammill, J.T. | 登録日 | 2017-03-21 | 公開日 | 2017-05-24 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.002 Å) | 主引用文献 | Blocking an N-terminal acetylation-dependent protein interaction inhibits an E3 ligase. Nat. Chem. Biol., 13, 2017
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4YII
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![BU of 4yii by Molmil](/molmil-images/mine/4yii) | |
8CDK
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![BU of 8cdk by Molmil](/molmil-images/mine/8cdk) | |
8CDJ
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![BU of 8cdj by Molmil](/molmil-images/mine/8cdj) | |
8C07
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![BU of 8c07 by Molmil](/molmil-images/mine/8c07) | |
8C06
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![BU of 8c06 by Molmil](/molmil-images/mine/8c06) | |
8CAF
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![BU of 8caf by Molmil](/molmil-images/mine/8caf) | N8C_Fab3b in complex with NEDD8-CUL1(WHB) | 分子名称: | Cullin-1, Fab Heavy Chain, Fab Light Chain, ... | 著者 | Duda, D.M, Yanishevski, D, Henneberg, L.T, Schulman, B.A. | 登録日 | 2023-01-24 | 公開日 | 2023-09-13 | 最終更新日 | 2023-12-06 | 実験手法 | X-RAY DIFFRACTION (2.66 Å) | 主引用文献 | Activity-based profiling of cullin-RING E3 networks by conformation-specific probes. Nat.Chem.Biol., 19, 2023
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4KBL
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![BU of 4kbl by Molmil](/molmil-images/mine/4kbl) | Structure of HHARI, a RING-IBR-RING ubiquitin ligase: autoinhibition of an Ariadne-family E3 and insights into ligation mechanism | 分子名称: | E3 ubiquitin-protein ligase ARIH1, ZINC ION | 著者 | Duda, D.M, Olszewski, J.L, Schulman, B.A. | 登録日 | 2013-04-23 | 公開日 | 2013-05-29 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (3.3 Å) | 主引用文献 | Structure of HHARI, a RING-IBR-RING Ubiquitin Ligase: Autoinhibition of an Ariadne-Family E3 and Insights into Ligation Mechanism. Structure, 21, 2013
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4KC9
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![BU of 4kc9 by Molmil](/molmil-images/mine/4kc9) | Structure of HHARI, a RING-IBR-RING ubiquitin ligase: autoinhibition of an Ariadne-family E3 and insights into ligation mechanism | 分子名称: | E3 ubiquitin-protein ligase ARIH1, ZINC ION | 著者 | Duda, D.M, Olszewski, J.L, Schulman, B.A. | 登録日 | 2013-04-24 | 公開日 | 2013-05-29 | 最終更新日 | 2013-07-03 | 実験手法 | X-RAY DIFFRACTION (3.603 Å) | 主引用文献 | Structure of HHARI, a RING-IBR-RING Ubiquitin Ligase: Autoinhibition of an Ariadne-Family E3 and Insights into Ligation Mechanism. Structure, 21, 2013
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4LCD
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![BU of 4lcd by Molmil](/molmil-images/mine/4lcd) | |
3DBL
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![BU of 3dbl by Molmil](/molmil-images/mine/3dbl) | |
3DBH
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![BU of 3dbh by Molmil](/molmil-images/mine/3dbh) | |
3DPL
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![BU of 3dpl by Molmil](/molmil-images/mine/3dpl) | |
3DBR
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![BU of 3dbr by Molmil](/molmil-images/mine/3dbr) | |
3DQV
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![BU of 3dqv by Molmil](/molmil-images/mine/3dqv) | Structural Insights into NEDD8 Activation of Cullin-RING Ligases: Conformational Control of Conjugation | 分子名称: | Cullin-5, NEDD8, Rbx1, ... | 著者 | Duda, D.M, Borg, L.A, Scott, D.C, Hunt, H.W, Hammel, M, Schulman, B.A. | 登録日 | 2008-07-09 | 公開日 | 2008-09-30 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Structural insights into NEDD8 activation of cullin-RING ligases: conformational control of conjugation. Cell(Cambridge,Mass.), 134, 2008
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2M6N
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![BU of 2m6n by Molmil](/molmil-images/mine/2m6n) | 3D solution structure of EMI1 (Early Mitotic Inhibitor 1) | 分子名称: | F-box only protein 5, ZINC ION | 著者 | Frye, J.J, Brown, N.G, Petzold, G, Watson, E.R, Royappa, G.R, Nourse, A, Jarvis, M, Kriwacki, R.W, Peters, J, Stark, H, Schulman, B.A. | 登録日 | 2013-04-06 | 公開日 | 2013-05-29 | 最終更新日 | 2024-05-01 | 実験手法 | SOLUTION NMR | 主引用文献 | Electron microscopy structure of human APC/C(CDH1)-EMI1 reveals multimodal mechanism of E3 ligase shutdown. Nat.Struct.Mol.Biol., 20, 2013
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2NVU
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![BU of 2nvu by Molmil](/molmil-images/mine/2nvu) | Structure of APPBP1-UBA3~NEDD8-NEDD8-MgATP-Ubc12(C111A), a trapped ubiquitin-like protein activation complex | 分子名称: | ADENOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, Maltose binding protein/NEDD8-activating enzyme E1 catalytic subunit chimera, ... | 著者 | Huang, D.T, Hunt, H.W, Zhuang, M, Ohi, M.D, Holton, J.M, Schulman, B.A. | 登録日 | 2006-11-13 | 公開日 | 2007-01-30 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Basis for a ubiquitin-like protein thioester switch toggling E1-E2 affinity. Nature, 445, 2007
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4P5O
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![BU of 4p5o by Molmil](/molmil-images/mine/4p5o) | |
4O1V
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![BU of 4o1v by Molmil](/molmil-images/mine/4o1v) | SPOP Promotes Tumorigenesis by Acting as a Key Regulatory Hub in Kidney Cancer | 分子名称: | Phosphatidylinositol 3,4,5-trisphosphate 3-phosphatase and dual-specificity protein phosphatase PTEN, Speckle-type POZ protein | 著者 | Calabrese, M.F, Watson, E.R, Schulman, B.A. | 登録日 | 2013-12-16 | 公開日 | 2014-04-30 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | SPOP Promotes Tumorigenesis by Acting as a Key Regulatory Hub in Kidney Cancer. Cancer Cell, 25, 2014
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4R2Y
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![BU of 4r2y by Molmil](/molmil-images/mine/4r2y) | Crystal structure of APC11 RING domain | 分子名称: | Anaphase-promoting complex subunit 11, ZINC ION | 著者 | Brown, N.G, Watson, E.R, Weissmann, F, Jarvis, M.A, Vanderlinden, R, Grace, C.R.R, Frye, J.J, Dube, P, Qiao, R, Petzold, G, Cho, S.E, Alsharif, O, Bao, J, Zheng, J, Nourse, A, Kurinov, I, Peters, J.M, Stark, H, Schulman, B.A. | 登録日 | 2014-08-13 | 公開日 | 2014-10-29 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.755 Å) | 主引用文献 | Mechanism of Polyubiquitination by Human Anaphase-Promoting Complex: RING Repurposing for Ubiquitin Chain Assembly. Mol.Cell, 56, 2014
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4RG7
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![BU of 4rg7 by Molmil](/molmil-images/mine/4rg7) | |