4QL3
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![BU of 4ql3 by Molmil](/molmil-images/mine/4ql3) | Crystal Structure of a GDP-bound G12R Oncogenic Mutant of Human GTPase KRas | 分子名称: | GTPase KRas, GUANOSINE-5'-DIPHOSPHATE, MAGNESIUM ION | 著者 | Hunter, J.C, Manandhar, A, Gurbani, D, Chen, Z, Westover, K.D. | 登録日 | 2014-06-10 | 公開日 | 2015-06-10 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.041 Å) | 主引用文献 | Biochemical and Structural Analysis of Common Cancer-Associated KRAS Mutations. Mol Cancer Res., 13, 2015
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6ATE
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![BU of 6ate by Molmil](/molmil-images/mine/6ate) | SRC kinase bound to covalent inhibitor | 分子名称: | N-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamide, Proto-oncogene tyrosine-protein kinase Src | 著者 | Gurbani, D, Westover, K.D. | 登録日 | 2017-08-28 | 公開日 | 2019-02-27 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.402 Å) | 主引用文献 | Leveraging Compound Promiscuity to Identify Targetable Cysteines within the Kinome. Cell Chem Biol, 26, 2019
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6BP1
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![BU of 6bp1 by Molmil](/molmil-images/mine/6bp1) | |
2E2J
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![BU of 2e2j by Molmil](/molmil-images/mine/2e2j) | RNA polymerase II elongation complex in 5 mM Mg+2 with GMPCPP | 分子名称: | 27-MER DNA template strand, 5'-D(P*CP*TP*GP*CP*TP*TP*AP*TP*CP*GP*GP*TP*A)-3', 5'-R(P*AP*UP*CP*GP*AP*GP*AP*GP*G)-3', ... | 著者 | Wang, D, Bushnell, D.A, Westover, K.D, Kaplan, C.D, Kornberg, R.D. | 登録日 | 2006-11-14 | 公開日 | 2006-12-12 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (3.5 Å) | 主引用文献 | Structural basis of transcription: role of the trigger loop in substrate specificity and catalysis Cell(Cambridge,Mass.), 127, 2006
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6BOF
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![BU of 6bof by Molmil](/molmil-images/mine/6bof) | |
2E2H
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![BU of 2e2h by Molmil](/molmil-images/mine/2e2h) | RNA polymerase II elongation complex at 5 mM Mg2+ with GTP | 分子名称: | 28-MER DNA template strand, 5'-D(*CP*TP*GP*CP*TP*TP*AP*TP*CP*GP*GP*TP*AP*G)-3', 5'-R(*AP*UP*CP*GP*AP*GP*AP*GP*GP*A)-3', ... | 著者 | Wang, D, Bushnell, D.A, Westover, K.D, Kaplan, C.D, Kornberg, R.D. | 登録日 | 2006-11-14 | 公開日 | 2006-12-12 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (3.95 Å) | 主引用文献 | Structural basis of transcription: role of the trigger loop in substrate specificity and catalysis Cell(Cambridge,Mass.), 127, 2006
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2E2I
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![BU of 2e2i by Molmil](/molmil-images/mine/2e2i) | RNA polymerase II elongation complex in 5 mM Mg+2 with 2'-dGTP | 分子名称: | 2'-DEOXYGUANOSINE-5'-TRIPHOSPHATE, 28-MER DNA template strand, 5'-D(*CP*TP*GP*CP*TP*TP*AP*TP*CP*GP*GP*TP*AP*G)-3', ... | 著者 | Wang, D, Bushnell, D.A, Westover, K.D, Kaplan, C.D, Kornberg, R.D. | 登録日 | 2006-11-14 | 公開日 | 2006-12-19 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (3.41 Å) | 主引用文献 | Structural basis of transcription: role of the trigger loop in substrate specificity and catalysis Cell(Cambridge,Mass.), 127, 2006
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6MQT
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![BU of 6mqt by Molmil](/molmil-images/mine/6mqt) | |
6MNX
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![BU of 6mnx by Molmil](/molmil-images/mine/6mnx) | |
6MTA
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![BU of 6mta by Molmil](/molmil-images/mine/6mta) | |
6MQN
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![BU of 6mqn by Molmil](/molmil-images/mine/6mqn) | |
6MS9
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![BU of 6ms9 by Molmil](/molmil-images/mine/6ms9) | GDP-bound KRAS P34R mutant | 分子名称: | GTPase KRas, GUANOSINE-5'-DIPHOSPHATE, MAGNESIUM ION | 著者 | Bera, A.K, Westover, K.D. | 登録日 | 2018-10-16 | 公開日 | 2020-04-15 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.49 Å) | 主引用文献 | GTP hydrolysis is modulated by Arg34 in the RASopathy-associated KRASP34R. Birth Defects Res, 112, 2020
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6MQG
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![BU of 6mqg by Molmil](/molmil-images/mine/6mqg) | |
6O36
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![BU of 6o36 by Molmil](/molmil-images/mine/6o36) | |
6O46
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![BU of 6o46 by Molmil](/molmil-images/mine/6o46) | |
2NVZ
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![BU of 2nvz by Molmil](/molmil-images/mine/2nvz) | RNA Polymerase II elongation complex with UTP, updated 11/2006 | 分子名称: | 28-MER DNA template strand, 5'-D(*CP*TP*GP*CP*TP*TP*AP*TP*CP*GP*GP*TP*AP*G)-3', 5'-R(*AP*UP*CP*GP*AP*GP*AP*GP*GP*A)-3', ... | 著者 | Wang, D, Bushnell, D.A, Westover, K.D, Kaplan, C.D, Kornberg, R.D. | 登録日 | 2006-11-14 | 公開日 | 2006-12-19 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (4.3 Å) | 主引用文献 | Structural basis of transcription: role of the trigger loop in substrate specificity and catalysis Cell(Cambridge,Mass.), 127, 2006
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2NVQ
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![BU of 2nvq by Molmil](/molmil-images/mine/2nvq) | RNA Polymerase II Elongation Complex in 150 mM Mg+2 with 2'dUTP | 分子名称: | 28-MER DNA template strand, 5'-D(*CP*TP*GP*CP*TP*TP*AP*TP*CP*GP*GP*TP*AP*G)-3', 5'-R(*AP*UP*CP*GP*AP*GP*AP*GP*GP*A)-3', ... | 著者 | Wang, D, Bushnell, D.A, Westover, K.D, Kaplan, C.D, Kornberg, R.D. | 登録日 | 2006-11-13 | 公開日 | 2006-12-12 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Structural basis of transcription: role of the trigger loop in substrate specificity and catalysis Cell(Cambridge,Mass.), 127, 2006
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2NVT
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![BU of 2nvt by Molmil](/molmil-images/mine/2nvt) | RNA Polymerase II Elongation Complex in 150 mM Mg+2 with GMPCPP | 分子名称: | 5'-D(*GP*TP*AP*CP*TP*TP*G)-3', 5'-D(P*CP*AP*AP*GP*TP*AP*CP*TP*TP*AP*CP*GP*CP*CP*TP*GP*GP*TP*CP*TP*T)-3', 5'-R(*AP*AP*GP*AP*CP*CP*AP*GP*GP*C)-3', ... | 著者 | Wang, D, Bushnell, D.A, Westover, K.D, Kaplan, C.D, Kornberg, R.D. | 登録日 | 2006-11-13 | 公開日 | 2006-12-12 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (3.36 Å) | 主引用文献 | Structural basis of transcription: role of the trigger loop in substrate specificity and catalysis Cell(Cambridge,Mass.), 127, 2006
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2NVY
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![BU of 2nvy by Molmil](/molmil-images/mine/2nvy) | RNA Polymerase II form II in 150 mM Mn+2 | 分子名称: | DNA-directed RNA polymerase II 13.6 kDa polypeptide, DNA-directed RNA polymerase II 140 kDa polypeptide, DNA-directed RNA polymerase II 45 kDa polypeptide, ... | 著者 | Wang, D, Bushnell, D.A, Westover, K.D, Kaplan, C.D, Kornberg, R.D. | 登録日 | 2006-11-13 | 公開日 | 2006-12-26 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (3.4 Å) | 主引用文献 | Structural basis of transcription: role of the trigger loop in substrate specificity and catalysis Cell(Cambridge,Mass.), 127, 2006
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2NVX
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![BU of 2nvx by Molmil](/molmil-images/mine/2nvx) | RNA polymerase II elongation complex in 5 mM Mg+2 with 2'-dUTP | 分子名称: | 28-MER DNA template strand, 5'-D(*CP*TP*GP*CP*TP*TP*AP*TP*CP*GP*GP*TP*AP*G)-3', 5'-R(*AP*UP*CP*GP*AP*GP*AP*GP*GP*A)-3', ... | 著者 | Wang, D, Bushnell, D.A, Westover, K.D, Kaplan, C.D, Kornberg, R.D. | 登録日 | 2006-11-13 | 公開日 | 2006-12-19 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (3.6 Å) | 主引用文献 | Structural basis of transcription: role of the trigger loop in substrate specificity and catalysis Cell(Cambridge,Mass.), 127, 2006
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3GTL
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![BU of 3gtl by Molmil](/molmil-images/mine/3gtl) | Backtracked RNA polymerase II complex with 13mer with G<>U mismatch | 分子名称: | DNA (28-MER), DNA (5'-D(*CP*TP*GP*CP*TP*TP*AP*TP*CP*GP*GP*TP*AP*G)-3'), DNA-directed RNA polymerase II subunit RPB1, ... | 著者 | Wang, D, Bushnell, D.A, Huang, X, Westover, K.D, Levitt, M, Kornberg, R.D. | 登録日 | 2009-03-27 | 公開日 | 2009-06-09 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (3.38 Å) | 主引用文献 | Structural basis of transcription: backtracked RNA polymerase II at 3.4 angstrom resolution. Science, 324, 2009
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3GTP
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![BU of 3gtp by Molmil](/molmil-images/mine/3gtp) | Backtracked RNA polymerase II complex with 24mer RNA | 分子名称: | DNA (28-MER), DNA (5'-D(*CP*TP*GP*CP*TP*TP*AP*TP*CP*GP*GP*TP*AP*G)-3'), DNA-directed RNA polymerase II subunit RPB1, ... | 著者 | Wang, D, Bushnell, D.A, Huang, X, Westover, K.D, Levitt, M, Kornberg, R.D. | 登録日 | 2009-03-27 | 公開日 | 2009-06-09 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (3.9 Å) | 主引用文献 | Structural basis of transcription: backtracked RNA polymerase II at 3.4 angstrom resolution. Science, 324, 2009
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3GTK
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![BU of 3gtk by Molmil](/molmil-images/mine/3gtk) | Backtracked RNA polymerase II complex with 18mer RNA | 分子名称: | DNA (29-MER), DNA (5'-D(*CP*TP*GP*CP*TP*TP*AP*TP*CP*GP*GP*TP*AP*G)-3'), DNA-directed RNA polymerase II subunit RPB1, ... | 著者 | Wang, D, Bushnell, D.A, Huang, X, Westover, K.D, Levitt, M, Kornberg, R.D. | 登録日 | 2009-03-27 | 公開日 | 2009-06-09 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (3.8 Å) | 主引用文献 | Structural basis of transcription: backtracked RNA polymerase II at 3.4 angstrom resolution. Science, 324, 2009
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3GTM
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![BU of 3gtm by Molmil](/molmil-images/mine/3gtm) | Co-complex of Backtracked RNA polymerase II with TFIIS | 分子名称: | DNA (28-MER), DNA (5'-D(*CP*TP*GP*CP*TP*TP*AP*TP*CP*GP*GP*TP*AP*G)-3'), DNA-directed RNA polymerase II subunit RPB1, ... | 著者 | Wang, D, Bushnell, D.A, Huang, X, Westover, K.D, Levitt, M, Kornberg, R.D. | 登録日 | 2009-03-27 | 公開日 | 2009-06-09 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (3.8 Å) | 主引用文献 | Structural basis of transcription: backtracked RNA polymerase II at 3.4 angstrom resolution. Science, 324, 2009
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3GTQ
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![BU of 3gtq by Molmil](/molmil-images/mine/3gtq) | Backtracked RNA polymerase II complex induced by damage | 分子名称: | DNA (5'-D(*CP*TP*AP*CP*CP*CP*AP*TP*AP*AP*CP*CP*AP*CP*AP*GP*GP*CP*TP*CP*CP*TP*CP*TP*CP*CP*AP*TP*C)-3'), DNA-directed RNA polymerase II subunit RPB1, DNA-directed RNA polymerase II subunit RPB11, ... | 著者 | Wang, D, Bushnell, D.A, Huang, X, Westover, K.D, Levitt, M, Kornberg, R.D. | 登録日 | 2009-03-27 | 公開日 | 2009-06-09 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (3.8 Å) | 主引用文献 | Structural basis of transcription: backtracked RNA polymerase II at 3.4 angstrom resolution. Science, 324, 2009
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