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6UXM
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BU of 6uxm by Molmil
Crystal structure of BAK core domain BH3-groove-dimer in complex with E. coli lipid
分子名称: 1,2-dioleoyl-sn-glycero-3-phosphoethanolamine, Bcl-2 homologous antagonist/killer
著者Cowan, A.D, Colman, P.M, Czabotar, P.E.
登録日2019-11-07
公開日2020-09-02
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.49 Å)
主引用文献BAK core dimers bind lipids and can be bridged by them.
Nat.Struct.Mol.Biol., 27, 2020
6UXR
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BU of 6uxr by Molmil
Crystal structure of BAK core domain BH3-groove-dimer in complex with LysoPC
分子名称: Bcl-2 homologous antagonist/killer, TETRAETHYLENE GLYCOL, TRIETHYLENE GLYCOL, ...
著者Cowan, A.D, Colman, P.M, Czabotar, P.E.
登録日2019-11-07
公開日2020-09-02
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献BAK core dimers bind lipids and can be bridged by them.
Nat.Struct.Mol.Biol., 27, 2020
6UXN
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BU of 6uxn by Molmil
Crystal structure of BAK core domain BH3-groove-dimer in complex with phosphatidylserine
分子名称: Bcl-2 homologous antagonist/killer, GLYCEROL, O-[(R)-{[(2R)-2,3-bis(octanoyloxy)propyl]oxy}(hydroxy)phosphoryl]-L-serine, ...
著者Cowan, A.D, Colman, P.M, Czabotar, P.E.
登録日2019-11-07
公開日2020-09-02
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.49 Å)
主引用文献BAK core dimers bind lipids and can be bridged by them.
Nat.Struct.Mol.Biol., 27, 2020
6UXO
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BU of 6uxo by Molmil
Crystal structure of BAK core domain BH3-groove-dimer in complex with DDM
分子名称: 1,2-ETHANEDIOL, ACETATE ION, Bcl-2 homologous antagonist/killer, ...
著者Cowan, A.D, Colman, P.M, Czabotar, P.E.
登録日2019-11-07
公開日2020-09-02
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (1.799 Å)
主引用文献BAK core dimers bind lipids and can be bridged by them.
Nat.Struct.Mol.Biol., 27, 2020
6UXQ
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BU of 6uxq by Molmil
Crystal structure of BAK core domain BH3-groove-dimer in complex with POPC and C8E4
分子名称: (HYDROXYETHYLOXY)TRI(ETHYLOXY)OCTANE, 1,2-ETHANEDIOL, 1-palmitoyl-2-oleoyl-sn-glycero-3-phosphocholine, ...
著者Cowan, A.D, Colman, P.M, Czabotar, P.E.
登録日2019-11-07
公開日2020-09-02
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (1.696 Å)
主引用文献BAK core dimers bind lipids and can be bridged by them.
Nat.Struct.Mol.Biol., 27, 2020
5W53
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BU of 5w53 by Molmil
Crystal structure of the erythrocyte-binding domain from Plasmodium vivax reticulocyte-binding protein 2b (PvRBP2b)
分子名称: POTASSIUM ION, Reticulocyte binding protein 2, putative, ...
著者Gruszczyk, J, Tham, W.H.
登録日2017-06-13
公開日2017-11-29
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.71 Å)
主引用文献Transferrin receptor 1 is a reticulocyte-specific receptor for Plasmodium vivax.
Science, 359, 2018
5VE6
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BU of 5ve6 by Molmil
Crystal structure of Sugen kinase 223
分子名称: Tyrosine-protein kinase SgK223
著者Patel, O, Lucet, I, Panjikar, S.
登録日2017-04-03
公開日2017-10-18
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (2.953 Å)
主引用文献Structure of SgK223 pseudokinase reveals novel mechanisms of homotypic and heterotypic association.
Nat Commun, 8, 2017
6CGA
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BU of 6cga by Molmil
Structure of the PR-DUB complex
分子名称: Polycomb protein Asx, Ubiquitin carboxyl-terminal hydrolase calypso
著者Foglizzo, M, Middleton, A.J, Day, C.L, Mace, P.D.
登録日2018-02-19
公開日2018-10-03
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (3.5 Å)
主引用文献A bidentate Polycomb Repressive-Deubiquitinase complex is required for efficient activity on nucleosomes.
Nat Commun, 9, 2018
6V0M
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BU of 6v0m by Molmil
Sterile alpha-motif from apoptosis signal-regulating kinase 3
分子名称: Mitogen-activated protein kinase kinase kinase 15
著者Trevelyan, S.J, Mace, P.D.
登録日2019-11-18
公開日2020-04-01
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Structure-based mechanism of preferential complex formation by apoptosis signal-regulating kinases.
Sci.Signal., 13, 2020
7MX3
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BU of 7mx3 by Molmil
Crystal structure of human RIPK3 complexed with GSK'843
分子名称: 1,2-ETHANEDIOL, 3-(1,3-benzothiazol-5-yl)-7-(1,3-dimethyl-1H-pyrazol-5-yl)thieno[3,2-c]pyridin-4-amine, Receptor-interacting serine/threonine-protein kinase 3
著者Davies, K.A, Czabotar, P.E.
登録日2021-05-18
公開日2021-11-24
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (3.23 Å)
主引用文献Human RIPK3 maintains MLKL in an inactive conformation prior to cell death by necroptosis.
Nat Commun, 12, 2021
5IKX
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BU of 5ikx by Molmil
Crystal structure of the alpha-esterase-7 carboxyl esterase (dimer), E3, from Lucilia cuprina
分子名称: Carboxylic ester hydrolase
著者Jackson, C, Fraser, N.
登録日2016-03-04
公開日2016-06-22
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.19 Å)
主引用文献Evolution of Protein Quaternary Structure in Response to Selective Pressure for Increased Thermostability.
J.Mol.Biol., 428, 2016
6BPC
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BU of 6bpc by Molmil
Plasmodium vivax reticulocyte binding protein 2b (PvRBP2b) bound to monoclonal antibody 4F7
分子名称: Monoclonal antibody 4F7 Fab heavy chain, Monoclonal antibody 4F7 Fab light chain, Reticulocyte binding protein 2, ...
著者Gruszczyk, J, Chan, L.J, Tham, W.H.
登録日2017-11-22
公開日2018-06-20
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.66 Å)
主引用文献Cryo-EM structure of an essential Plasmodium vivax invasion complex.
Nature, 559, 2018
6BPB
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BU of 6bpb by Molmil
Plasmodium vivax invasion blocking monoclonal antibody 4F7
分子名称: Monoclonal antibody 4F7 Fab heavy chain, Monoclonal antibody 4F7 Fab light chain
著者Gruszczyk, J, Chan, L.J, Tham, W.H.
登録日2017-11-22
公開日2018-06-20
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.87 Å)
主引用文献Cryo-EM structure of an essential Plasmodium vivax invasion complex.
Nature, 559, 2018
6BPA
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BU of 6bpa by Molmil
Plasmodium vivax reticulocyte binding protein 2b (PvRBP2b) bound to monoclonal antibody 3E9
分子名称: BROMIDE ION, Monoclonal antibody 3E9 Fab heavy chain, Monoclonal antibody 3E9 Fab light chain, ...
著者Gruszczyk, J, Chan, L.J, Tham, W.H.
登録日2017-11-22
公開日2018-06-20
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.53 Å)
主引用文献Cryo-EM structure of an essential Plasmodium vivax invasion complex.
Nature, 559, 2018
6BPD
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BU of 6bpd by Molmil
Plasmodium vivax invasion blocking monoclonal antibody 10B12
分子名称: Monoclonal antibody 10B12 Fab heavy chain, Monoclonal antibody 10B12 Fab light chain
著者Gruszczyk, J, Chan, L.J, Tham, W.H.
登録日2017-11-22
公開日2018-06-20
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.32 Å)
主引用文献Cryo-EM structure of an essential Plasmodium vivax invasion complex.
Nature, 559, 2018
6BZH
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BU of 6bzh by Molmil
Structure of mouse RIG-I tandem CARDs
分子名称: 1,2-ETHANEDIOL, CHLORIDE ION, Probable ATP-dependent RNA helicase DDX58
著者Kershaw, N.J, D'Cruz, A.A, Babon, J.J, Nicholson, S.E.
登録日2017-12-24
公開日2018-01-17
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Identification of a second binding site on the TRIM25 B30.2 domain.
Biochem. J., 475, 2018
6BPE
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BU of 6bpe by Molmil
Plasmodium vivax reticulocyte binding protein 2b (PvRBP2b) bound to monoclonal antibody 6H1
分子名称: Monoclonal antibody 6H1 Fab heavy chain, Monoclonal antibody 6H1 Fab light chain, Reticulocyte binding protein 2, ...
著者Gruszczyk, J, Chan, L.J, Tham, W.H.
登録日2017-11-22
公開日2018-06-20
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (3.34 Å)
主引用文献Cryo-EM structure of an essential Plasmodium vivax invasion complex.
Nature, 559, 2018
6C5X
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BU of 6c5x by Molmil
Crystal Structure of SOCS1 in complex with ElonginB and ElonginC
分子名称: Elongin-B, Elongin-C, GP130 peptide fragment, ...
著者Kershaw, N.J, Laktyushin, A, Babon, J.J.
登録日2018-01-17
公開日2018-05-02
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (3.105 Å)
主引用文献The molecular basis of JAK/STAT inhibition by SOCS1.
Nat Commun, 9, 2018
6D03
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BU of 6d03 by Molmil
Cryo-EM structure of a Plasmodium vivax invasion complex essential for entry into human reticulocytes; one molecule of parasite ligand.
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(2-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Gruszczyk, J, Huang, R.K, Hong, C, Yu, Z, Tham, W.H.
登録日2018-04-10
公開日2018-06-20
最終更新日2020-07-29
実験手法ELECTRON MICROSCOPY (3.68 Å)
主引用文献Cryo-EM structure of an essential Plasmodium vivax invasion complex.
Nature, 559, 2018
6D04
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BU of 6d04 by Molmil
Cryo-EM structure of a Plasmodium vivax invasion complex essential for entry into human reticulocytes; two molecules of parasite ligand, subclass 1.
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ...
著者Gruszczyk, J, Huang, R.K, Hong, C, Yu, Z, Tham, W.H.
登録日2018-04-10
公開日2018-06-20
最終更新日2020-07-29
実験手法ELECTRON MICROSCOPY (3.74 Å)
主引用文献Cryo-EM structure of an essential Plasmodium vivax invasion complex.
Nature, 559, 2018
6D05
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BU of 6d05 by Molmil
Cryo-EM structure of a Plasmodium vivax invasion complex essential for entry into human reticulocytes; two molecules of parasite ligand, subclass 2.
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ...
著者Gruszczyk, J, Huang, R.K, Hong, C, Yu, Z, Tham, W.H.
登録日2018-04-10
公開日2018-06-20
最終更新日2020-07-29
実験手法ELECTRON MICROSCOPY (3.8 Å)
主引用文献Cryo-EM structure of an essential Plasmodium vivax invasion complex.
Nature, 559, 2018
6WG7
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BU of 6wg7 by Molmil
Coordinates of NanR dimer fitted in Hexameric NanR-DNA hetero-complex cryo-EM map
分子名称: DNA (35-MER), HTH-type transcriptional repressor NanR
著者Hariprasad, V, Horne, C, Santosh, P, Amy, H, Emre, B, Rachel, N, Michael, G, Georg, R, Borries, D, Renwick, D.
登録日2020-04-05
公開日2021-03-10
最終更新日2024-03-06
実験手法ELECTRON MICROSCOPY (8.3 Å)
主引用文献Mechanism of NanR gene repression and allosteric induction of bacterial sialic acid metabolism.
Nat Commun, 12, 2021
6WFQ
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BU of 6wfq by Molmil
NanR dimer-DNA hetero-complex
分子名称: DNA (5'-D(P*GP*GP*TP*AP*TP*AP*AP*CP*AP*GP*GP*TP*AP*TP*A)-3'), DNA (5'-D(P*TP*AP*TP*AP*CP*CP*TP*GP*TP*TP*AP*TP*AP*CP*C)-3'), HTH-type transcriptional repressor NanR
著者Hariprasad, V, Horne, C, Santosh, P, Amy, H, Emre, B, Rachel, N, Michael, G, Georg, R, Borries, D, Renwick, D.
登録日2020-04-03
公開日2021-03-10
最終更新日2024-03-06
実験手法ELECTRON MICROSCOPY (3.9 Å)
主引用文献Mechanism of NanR gene repression and allosteric induction of bacterial sialic acid metabolism.
Nat Commun, 12, 2021
6VBZ
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BU of 6vbz by Molmil
Crystal structure of the rat MLKL pseudokinase domain
分子名称: MANGANESE (II) ION, Mixed lineage kinase domain-like pseudokinase
著者Davies, K.A, Czabotar, P.E.
登録日2019-12-19
公開日2020-07-08
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.192 Å)
主引用文献Distinct pseudokinase domain conformations underlie divergent activation mechanisms among vertebrate MLKL orthologues.
Nat Commun, 11, 2020
6VC0
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BU of 6vc0 by Molmil
Crystal structure of the horse MLKL pseudokinase domain
分子名称: GLYCEROL, Mixed lineage kinase domain like pseudokinase
著者Davies, K.A, Czabotar, P.E.
登録日2019-12-19
公開日2020-07-08
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.746 Å)
主引用文献Distinct pseudokinase domain conformations underlie divergent activation mechanisms among vertebrate MLKL orthologues.
Nat Commun, 11, 2020

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