6TJ0
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![BU of 6tj0 by Molmil](/molmil-images/mine/6tj0) | Crystal structure of the bacterial cellulose secretion regulator BcsE, residues 217-523, with bound c-di-GMP. | 分子名称: | 9,9'-[(2R,3R,3aS,5S,7aR,9R,10R,10aS,12S,14aR)-3,5,10,12-tetrahydroxy-5,12-dioxidooctahydro-2H,7H-difuro[3,2-d:3',2'-j][1,3,7,9,2,8]tetraoxadiphosphacyclododecine-2,9-diyl]bis(2-amino-1,9-dihydro-6H-purin-6-one), Bacterial cellulose synthesis subunit E, GLYCEROL | 著者 | Zouhir, S, Abidi, W, Krasteva, P.V. | 登録日 | 2019-11-23 | 公開日 | 2020-07-29 | 最終更新日 | 2020-08-26 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Structure and Multitasking of the c-di-GMP-Sensing Cellulose Secretion Regulator BcsE. Mbio, 11, 2020
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6YG8
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6YBB
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![BU of 6ybb by Molmil](/molmil-images/mine/6ybb) | Crystal structure of a native BcsE (217-523) - BcsR-BcsQ (R156E mutant) complex with c-di-GMP and ATP bound | 分子名称: | 9,9'-[(2R,3R,3aS,5S,7aR,9R,10R,10aS,12S,14aR)-3,5,10,12-tetrahydroxy-5,12-dioxidooctahydro-2H,7H-difuro[3,2-d:3',2'-j][1,3,7,9,2,8]tetraoxadiphosphacyclododecine-2,9-diyl]bis(2-amino-1,9-dihydro-6H-purin-6-one), ADENOSINE-5'-TRIPHOSPHATE, Bacterial cellulose secretion regulator BcsE, ... | 著者 | Abidi, W, Zouhir, S, Roche, S, Krasteva, P.V. | 登録日 | 2020-03-16 | 公開日 | 2021-02-24 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Architecture and regulation of an enterobacterial cellulose secretion system. Sci Adv, 7, 2021
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6YBU
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![BU of 6ybu by Molmil](/molmil-images/mine/6ybu) | Crystal structure of a native BcsE (349-523) RQ complex with c-di-GMP and ATP bound | 分子名称: | 9,9'-[(2R,3R,3aS,5S,7aR,9R,10R,10aS,12S,14aR)-3,5,10,12-tetrahydroxy-5,12-dioxidooctahydro-2H,7H-difuro[3,2-d:3',2'-j][1,3,7,9,2,8]tetraoxadiphosphacyclododecine-2,9-diyl]bis(2-amino-1,9-dihydro-6H-purin-6-one), ADENOSINE-5'-TRIPHOSPHATE, Bacterial cellulose secretion regulator BcsE, ... | 著者 | Abidi, W, Zouhir, S, Roche, S, Krasteva, P.V. | 登録日 | 2020-03-17 | 公開日 | 2021-02-24 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (2.49 Å) | 主引用文献 | Architecture and regulation of an enterobacterial cellulose secretion system. Sci Adv, 7, 2021
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3EOC
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![BU of 3eoc by Molmil](/molmil-images/mine/3eoc) | Cdk2/CyclinA complexed with a imidazo triazin-2-amine | 分子名称: | 5-methyl-7-phenyl-N-(3,4,5-trimethoxyphenyl)imidazo[5,1-f][1,2,4]triazin-2-amine, Cell division protein kinase 2, Cyclin-A2 | 著者 | Cheung, M, Kuntz, K, Pobanz, M, Salovich, J, Wilson, B, Andrews, W, Shewchuk, L, Epperly, A, Hassler, D, Leesnitzer, M, Smith, J, Smith, G, Lansing, T, Mook, R. | 登録日 | 2008-09-26 | 公開日 | 2008-11-04 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (3.2 Å) | 主引用文献 | Imidazo[5,1-f][1,2,4]triazin-2-amines as novel inhibitors of polo-like kinase 1. Bioorg.Med.Chem.Lett., 18, 2008
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6IC9
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6IC8
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7BAI
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7BAH
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5CM8
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5CM9
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4JGW
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3NCU
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8OS5
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![BU of 8os5 by Molmil](/molmil-images/mine/8os5) | Crystal structure of the Factor XII heavy chain reveals an interlocking dimer with a FnII to kringle domain interaction | 分子名称: | Coagulation factor XII-Mie | 著者 | Li, C, Saleem, M, Kaira, B.G, Brown, A, Wilson, C, Philippou, H, Emsley, J. | 登録日 | 2023-04-18 | 公開日 | 2024-03-27 | 実験手法 | X-RAY DIFFRACTION (3.4 Å) | 主引用文献 | Factor XII and kininogen asymmetric assembly with gC1qR/C1QBP/P32 is governed by allostery. Blood, 136, 2020
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4K6T
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![BU of 4k6t by Molmil](/molmil-images/mine/4k6t) | Crystal structure of Ad37 fiber knob in complex with trivalent sialic acid inhibitor ME0385 | 分子名称: | 1,2-ETHANEDIOL, 2,2',2''-[nitrilotris(methanediyl-1H-1,2,3-triazole-4,1-diyl)]triethanol, ACETATE ION, ... | 著者 | Stehle, T, Bauer, J. | 登録日 | 2013-04-16 | 公開日 | 2014-10-22 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Triazole linker-based trivalent sialic acid inhibitors of adenovirus type 37 infection of human corneal epithelial cells. Org.Biomol.Chem., 13, 2015
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4K6W
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![BU of 4k6w by Molmil](/molmil-images/mine/4k6w) | Crystal structure of Ad37 fiber knob in complex with trivalent sialic acid inhibitor ME0408 | 分子名称: | 1,2-ETHANEDIOL, 2,2',2''-[nitrilotris(methanediyl-1H-1,2,3-triazole-4,1-diyl)]triethanol, 3,5-dideoxy-5-(propanoylamino)-D-glycero-alpha-D-galacto-non-2-ulopyranosonic acid, ... | 著者 | Stehle, T, Bauer, J. | 登録日 | 2013-04-16 | 公開日 | 2014-10-22 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Triazole linker-based trivalent sialic acid inhibitors of adenovirus type 37 infection of human corneal epithelial cells. Org.Biomol.Chem., 13, 2015
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4K6U
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![BU of 4k6u by Molmil](/molmil-images/mine/4k6u) | Crystal structure of Ad37 fiber knob in complex with trivalent sialic acid inhibitor ME0386 | 分子名称: | 3,3',3''-[nitrilotris(methanediyl-1H-1,2,3-triazole-4,1-diyl)]tripropan-1-ol, ACETATE ION, Fiber protein, ... | 著者 | Stehle, T, Bauer, J. | 登録日 | 2013-04-16 | 公開日 | 2014-10-22 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Triazole linker-based trivalent sialic acid inhibitors of adenovirus type 37 infection of human corneal epithelial cells. Org.Biomol.Chem., 13, 2015
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4K6V
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![BU of 4k6v by Molmil](/molmil-images/mine/4k6v) | Crystal structure of Ad37 fiber knob in complex with trivalent sialic acid inhibitor ME0407 | 分子名称: | 3,3',3''-[nitrilotris(methanediyl-1H-1,2,3-triazole-4,1-diyl)]tripropan-1-ol, 3,5-dideoxy-5-(propanoylamino)-D-glycero-alpha-D-galacto-non-2-ulopyranosonic acid, ACETATE ION, ... | 著者 | Stehle, T, Bauer, J. | 登録日 | 2013-04-16 | 公開日 | 2014-10-22 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Triazole linker-based trivalent sialic acid inhibitors of adenovirus type 37 infection of human corneal epithelial cells. Org.Biomol.Chem., 13, 2015
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4XQA
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![BU of 4xqa by Molmil](/molmil-images/mine/4xqa) | CRYSTAL STRUCTURE OF AD37 FIBER KNOB IN COMPLEX WITH TRIVALENT SIALIC ACID INHIBITOR ME0462 | 分子名称: | (1-{2-[bis(2-{4-[({(6R)-5-(acetylamino)-3,5-dideoxy-6-[(1R,2R)-1,2,3-trihydroxypropyl]-beta-L-threo-hex-2-ulopyranonosyl}oxy)methyl]-1H-1,2,3-triazol-1-yl}ethyl)amino]ethyl}-1H-1,2,3-triazol-4-yl)methyl (6R)-5-(acetylamino)-3,5-dideoxy-6-[(1R,2R)-1,2,3-trihydroxypropyl]-beta-L-threo-hex-2-ulopyranosidonic acid, ACETATE ION, Fiber, ... | 著者 | Stehle, T, Liaci, A.M. | 登録日 | 2015-01-19 | 公開日 | 2015-07-29 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.4072 Å) | 主引用文献 | Triazole linker-based trivalent sialic acid inhibitors of adenovirus type 37 infection of human corneal epithelial cells. Org.Biomol.Chem., 13, 2015
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6TR8
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![BU of 6tr8 by Molmil](/molmil-images/mine/6tr8) | Corynebacterium diphtheriae methionine sulfoxide reductase B (MsrB) solution structure - reduced form | 分子名称: | Peptide-methionine (R)-S-oxide reductase, ZINC ION | 著者 | Volkov, A.N, Tossounian, M.A, Buts, L, Messens, J. | 登録日 | 2019-12-18 | 公開日 | 2020-02-05 | 最終更新日 | 2024-05-15 | 実験手法 | SOLUTION NMR | 主引用文献 | Methionine sulfoxide reductase B fromCorynebacterium diphtheriaecatalyzes sulfoxide reduction via an intramolecular disulfide cascade. J.Biol.Chem., 295, 2020
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4XQB
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![BU of 4xqb by Molmil](/molmil-images/mine/4xqb) | CRYSTAL STRUCTURE OF AD37 FIBER KNOB IN COMPLEX WITH TRIVALENT SIALIC ACID INHIBITOR ME0461 | 分子名称: | 2-(1-{2-[bis(2-{4-[2-({(6R)-5-(acetylamino)-3,5-dideoxy-6-[(1R,2R)-1,2,3-trihydroxypropyl]-beta-L-threo-hex-2-ulopyranonosyl}oxy)ethyl]-1H-1,2,3-triazol-1-yl}ethyl)amino]ethyl}-1H-1,2,3-triazol-4-yl)ethyl (6R)-5-(acetylamino)-3,5-dideoxy-6-[(1R,2R)-1,2,3-trihydroxypropyl]-beta-L-threo-hex-2-ulopyranosidonic acid, ACETATE ION, Fiber, ... | 著者 | Stehle, T, Liaci, A.M. | 登録日 | 2015-01-19 | 公開日 | 2015-07-29 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.597 Å) | 主引用文献 | Triazole linker-based trivalent sialic acid inhibitors of adenovirus type 37 infection of human corneal epithelial cells. Org.Biomol.Chem., 13, 2015
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5ZXI
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![BU of 5zxi by Molmil](/molmil-images/mine/5zxi) | Co-crystal structure of an Inhibitor in complex with human PPARdelta LBD | 分子名称: | 6-[2-({2-[4-(furan-2-yl)phenyl]-5-methyl-1H-imidazol-1-yl}methyl)phenoxy]hexanoic acid, Peroxisome proliferator-activated receptor delta | 著者 | Rani, S.T, Laxminarasimhan, A, Senaiar, R.S, Krishnamurthy, N. | 登録日 | 2018-05-21 | 公開日 | 2019-04-03 | 最終更新日 | 2024-03-27 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Selective PPAR delta Modulators Improve Mitochondrial Function: Potential Treatment for Duchenne Muscular Dystrophy (DMD). ACS Med Chem Lett, 9, 2018
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6TIK
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![BU of 6tik by Molmil](/molmil-images/mine/6tik) | Hepatitis B virus core shell--virus-like particle with NadA epitope | 分子名称: | Capsid protein,Putative adhesin/invasin,Capsid protein,Factor H-binding protein | 著者 | Roseman, A.M, Colllins, R.F, Derrick, J.P. | 登録日 | 2019-11-22 | 公開日 | 2020-04-29 | 実験手法 | ELECTRON MICROSCOPY (3.4 Å) | 主引用文献 | An assessment of the use of Hepatitis B Virus core protein virus-like particles to display heterologous antigens from Neisseria meningitidis. Vaccine, 38, 2020
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5XMX
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![BU of 5xmx by Molmil](/molmil-images/mine/5xmx) | Co-crystal structure of Inhibitor compound in complex with human PPARdelta LBD | 分子名称: | (E)-6-[2-[[[4-(furan-2-yl)phenyl]carbonyl-methyl-amino]methyl]phenoxy]-4-methyl-hex-4-enoic acid, Peroxisome proliferator-activated receptor delta | 著者 | Lakshminarasimhan, A, Rani, S.T, Senaiar, R.S, Krishnamurthy, N. | 登録日 | 2017-05-16 | 公開日 | 2018-05-23 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Novel highly selective peroxisome proliferator-activated receptor delta (PPAR delta) modulators with pharmacokinetic properties suitable for once-daily oral dosing. Bioorg. Med. Chem. Lett., 27, 2017
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3D43
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![BU of 3d43 by Molmil](/molmil-images/mine/3d43) | The crystal structure of Sph at 0.8A | 分子名称: | CALCIUM ION, Sphericase | 著者 | Almog, O. | 登録日 | 2008-05-13 | 公開日 | 2009-04-28 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (0.8 Å) | 主引用文献 | The crystal structures of the psychrophilic subtilisin S41 and the mesophilic subtilisin Sph reveal the same calcium-loaded state. Proteins, 74, 2009
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