5ACQ
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![BU of 5acq by Molmil](/molmil-images/mine/5acq) | W228A-Investigation of the impact from residues W228 and Y233 in the metallo-beta-lactamase GIM-1 | 分子名称: | BETA-LACTAMASE, ZINC ION | 著者 | Skagseth, S, Carlsen, T.J, Bjerga, G.E.K, Spencer, J, Samuelsen, O, Leiros, H.-K.S. | 登録日 | 2015-08-17 | 公開日 | 2015-12-23 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Role of Residues W228 and Y233 in the Structure and Activity of Metallo-Beta-Lactamase Gim-1. Antimicrob.Agents Chemother., 60, 2015
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5A87
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![BU of 5a87 by Molmil](/molmil-images/mine/5a87) | Crystal structure of the metallo-beta-lactamase VIM-5 | 分子名称: | GLYCEROL, METALLO-BETA-LACTAMASE VIM-5, ZINC ION | 著者 | Brem, J, Duzgun, A.O, McDonough, M.A, Schofield, C.J. | 登録日 | 2015-07-13 | 公開日 | 2015-12-23 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Comparison of Verona Integron-Borne Metallo-beta-Lactamase (VIM) Variants Reveals Differences in Stability and Inhibition Profiles. Antimicrob. Agents Chemother., 60, 2015
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5ACT
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![BU of 5act by Molmil](/molmil-images/mine/5act) | W228S-Investigation of the impact from residues W228 and Y233 in the metallo-beta-lactamase GIM-1 | 分子名称: | GIM-1 PROTEIN, ZINC ION | 著者 | Skagseth, S, Carlsen, T.J, Bjerga, G.E.K, Spencer, J, Samuelsen, O, Leiros, H.-K.S. | 登録日 | 2015-08-17 | 公開日 | 2015-12-23 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.81 Å) | 主引用文献 | Role of Residues W228 and Y233 in the Structure and Activity of Metallo-Beta-Lactamase Gim-1. Antimicrob.Agents Chemother., 60, 2015
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8R5U
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![BU of 8r5u by Molmil](/molmil-images/mine/8r5u) | |
8R5T
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![BU of 8r5t by Molmil](/molmil-images/mine/8r5t) | |
8SK2
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![BU of 8sk2 by Molmil](/molmil-images/mine/8sk2) | |
4NQ6
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![BU of 4nq6 by Molmil](/molmil-images/mine/4nq6) | Bacillus cereus Zn-dependent metallo-beta-lactamase at pH 7 complexed with compound L-CS319 | 分子名称: | (3S,5S,7aR)-5-(sulfanylmethyl)tetrahydro[1,3]thiazolo[4,3-b][1,3]thiazole-3-carboxylic acid, Beta-lactamase 2, POTASSIUM ION, ... | 著者 | Gonzalez, J.M, Gonzalez, M.M, Vila, A.J. | 登録日 | 2013-11-23 | 公開日 | 2014-11-26 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Cross-class metallo-beta-lactamase inhibition by bisthiazolidines reveals multiple binding modes. Proc. Natl. Acad. Sci. U.S.A., 113, 2016
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4LE6
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![BU of 4le6 by Molmil](/molmil-images/mine/4le6) | Crystal structure of the phosphotriesterase OPHC2 from Pseudomonas pseudoalcaligenes | 分子名称: | 1,2-ETHANEDIOL, GLYCEROL, Organophosphorus hydrolase, ... | 著者 | Gotthard, G, Hiblot, J, Chabriere, E, Elias, M. | 登録日 | 2013-06-25 | 公開日 | 2013-11-13 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Structural and Enzymatic Characterization of the Phosphotriesterase OPHC2 from Pseudomonas pseudoalcaligenes. Plos One, 8, 2013
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8SKP
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![BU of 8skp by Molmil](/molmil-images/mine/8skp) | X-ray structure of the NDM-4 beta-lactamase from Klebsiella pneumonia in complex with 1-hydroxypyridine-2(1H)-thione-6-carboxylic acid | 分子名称: | 1,2-ETHANEDIOL, 1-hydroxy-6-sulfanylidene-1,6-dihydropyridine-2-carboxylic acid, Metallo-beta-lactamase type 2, ... | 著者 | Thoden, J.B, Holden, H.M. | 登録日 | 2023-04-20 | 公開日 | 2023-08-23 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.3 Å) | 主引用文献 | Characterization of a novel inhibitor for the New Delhi metallo-beta-lactamase-4: Implications for drug design and combating bacterial drug resistance. J.Biol.Chem., 299, 2023
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8SKO
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4NQ4
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8U00
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![BU of 8u00 by Molmil](/molmil-images/mine/8u00) | Crystal structure of metallo-beta-lactamase superfamily protein from Caulobacter vibrioides | 分子名称: | 1,2-ETHANEDIOL, CHLORIDE ION, GLYCEROL, ... | 著者 | Kim, Y, Maltseva, N, Endres, M, Joachimiak, A, Center for Structural Biology of Infectious Diseases (CSBID) | 登録日 | 2023-08-28 | 公開日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Crystal structure of metallo-beta-lactamase superfamily protein from Caulobacter vibrioides To Be Published
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4O98
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![BU of 4o98 by Molmil](/molmil-images/mine/4o98) | Crystal structure of Pseudomonas oleovorans PoOPH mutant H250I/I263W | 分子名称: | ZINC ION, organophosphorus hydrolase | 著者 | Luo, X.J, Kong, X.D, Zhao, J, Chen, Q, Zhou, J.H, Xu, J.H. | 登録日 | 2014-01-02 | 公開日 | 2014-12-03 | 最終更新日 | 2017-11-22 | 実験手法 | X-RAY DIFFRACTION (2.251 Å) | 主引用文献 | Switching a newly discovered lactonase into an efficient and thermostable phosphotriesterase by simple double mutations His250Ile/Ile263Trp Biotechnol.Bioeng., 111, 2014
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4P62
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4NQ5
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![BU of 4nq5 by Molmil](/molmil-images/mine/4nq5) | Bacillus cereus Zn-dependent metallo-beta-lactamase at pH 7 complexed with compound CS319 | 分子名称: | (3R,5R,7aS)-5-(sulfanylmethyl)tetrahydro[1,3]thiazolo[4,3-b][1,3]thiazole-3-carboxylic acid, Beta-lactamase 2, POTASSIUM ION, ... | 著者 | Gonzalez, J.M, Gonzalez, M.M, Vila, A.J. | 登録日 | 2013-11-23 | 公開日 | 2014-11-26 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.29 Å) | 主引用文献 | Inhibition of metallo-lactamases with bicyclic compounds TO BE PUBLISHED
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4NQ2
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![BU of 4nq2 by Molmil](/molmil-images/mine/4nq2) | Structure of Zn(II)-bound metallo-beta-lactamse VIM-2 from Pseudomonas aeruginosa | 分子名称: | ACETATE ION, Beta-lactamase class B VIM-2, ZINC ION | 著者 | Aitha, M, Nix, J.C, Crowder, M.W, Page, R.C. | 登録日 | 2013-11-23 | 公開日 | 2014-11-12 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Biochemical, Mechanistic, and Spectroscopic Characterization of Metallo-beta-lactamase VIM-2. Biochemistry, 53, 2014
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2WRS
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![BU of 2wrs by Molmil](/molmil-images/mine/2wrs) | Crystal Structure of the Mono-Zinc Metallo-beta-lactamase VIM-4 from Pseudomonas aeruginosa | 分子名称: | BETA-LACTAMASE VIM-4, CITRATE ANION, CITRIC ACID, ... | 著者 | Lassaux, P, Hamel, M, Gulea, M, Delbruck, H, Traore, D.A.K, Mercuri, P.S, Horsfall, L, Dehareng, D, Gaumont, A.-C, Frere, J.-M, Ferrer, J.-L, Hoffmann, K, Galleni, M, Bebrone, C. | 登録日 | 2009-09-02 | 公開日 | 2010-06-23 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.79 Å) | 主引用文献 | Mercaptophosphonate Compounds as Broad-Spectrum Inhibitors of the Metallo-Beta-Lactamases. J.Med.Chem., 53, 2010
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4XUK
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3ESH
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![BU of 3esh by Molmil](/molmil-images/mine/3esh) | Crystal structure of a probable metal-dependent hydrolase from Staphylococcus aureus. Northeast Structural Genomics target ZR314 | 分子名称: | Protein similar to metal-dependent hydrolase | 著者 | Seetharaman, J, Chen, Y, Wang, H, Janjua, H, Foote, E.L, Xiao, R, Nair, R, Everett, J.K, Acton, T.B, Rost, B, Montelione, G.T, Tong, L, Hunt, J.F, Northeast Structural Genomics Consortium (NESG) | 登録日 | 2008-10-06 | 公開日 | 2008-10-28 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Crystal structure of a probable metal-dependent hydrolase from
Staphylococcus aureus. Northeast Structural Genomics target ZR314 To be Published
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2UYX
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![BU of 2uyx by Molmil](/molmil-images/mine/2uyx) | metallo-beta-lactamase (1BC2) single point mutant D120S | 分子名称: | BETA-LACTAMASE II, GLYCEROL, ZINC ION | 著者 | Larrull, L.I, Fabiane, S.M, Kowalski, J.M, Bennett, B, Sutton, B.J, Vila, A.J. | 登録日 | 2007-04-20 | 公開日 | 2007-05-08 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Asp-120 locates Zn2 for optimal metallo-beta-lactamase activity. J. Biol. Chem., 282, 2007
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2VW8
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![BU of 2vw8 by Molmil](/molmil-images/mine/2vw8) | Crystal Structure of Quinolone signal response protein pqsE from Pseudomonas aeruginosa | 分子名称: | 1,2-ETHANEDIOL, CACODYLATE ION, FE (II) ION, ... | 著者 | Carter, L.G, Johnson, K.A, Liu, H, Mcmahon, S.A, Oke, M, Naismith, J.H, White, M.F. | 登録日 | 2008-06-17 | 公開日 | 2010-07-14 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.45 Å) | 主引用文献 | The Scottish Structural Proteomics Facility: Targets, Methods and Outputs. J.Struct.Funct.Genomics, 11, 2010
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3F9O
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1KO3
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![BU of 1ko3 by Molmil](/molmil-images/mine/1ko3) | VIM-2, a Zn-beta-lactamase from Pseudomonas aeruginosa with Cys221 reduced | 分子名称: | ACETATE ION, CHLORIDE ION, HYDROXIDE ION, ... | 著者 | Garcia-Saez, I, Docquier, J.-D, Rossolini, G.M, Dideberg, O. | 登録日 | 2001-12-20 | 公開日 | 2003-09-02 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.91 Å) | 主引用文献 | The three-dimensional structure of VIM-2, a Zn-beta-lactamase from Pseudomonas aeruginosa in its reduced and oxidised form J.Mol.Biol., 375, 2008
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3FAI
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![BU of 3fai by Molmil](/molmil-images/mine/3fai) | The Di Zinc Carbapenemase CphA N220G mutant | 分子名称: | Beta-lactamase, CHLORIDE ION, GLYCEROL, ... | 著者 | Delbruck, H, Hoffmann, K.M.V. | 登録日 | 2008-11-17 | 公開日 | 2009-09-01 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | The structure of the dizinc subclass B2 metallo-beta-lactamase CphA reveals that the second inhibitory zinc ion binds in the histidine site Antimicrob.Agents Chemother., 53, 2009
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3DH8
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