7PCG
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![BU of 7pcg by Molmil](/molmil-images/mine/7pcg) | BurG (holo) in complex with cyclopropane-1,1-dicarboxylate (7): Biosynthesis of cyclopropanol rings in bacterial toxins | 分子名称: | GLYCEROL, Ketol-acid reductoisomerase, MAGNESIUM ION, ... | 著者 | Trottmann, F, Ishida, K, Ishida, M, Kries, H, Groll, M, Hertweck, C. | 登録日 | 2021-08-03 | 公開日 | 2022-08-10 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Pathogenic bacteria remodel central metabolic enzyme to build a cyclopropanol warhead. Nat.Chem., 14, 2022
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6R9M
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![BU of 6r9m by Molmil](/molmil-images/mine/6r9m) | Structure of Saccharomyces cerevisiae apo Pan2 pseudoubiquitin hydrolase-RNA exonuclease (UCH-Exo) module in complex with AAGGAA RNA | 分子名称: | AAGGAA RNA, PAN2-PAN3 deadenylation complex catalytic subunit PAN2 | 著者 | Tang, T.T.L, Stowell, J.A.W, Hill, C.H, Passmore, L.A. | 登録日 | 2019-04-03 | 公開日 | 2019-05-22 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (3.329 Å) | 主引用文献 | The intrinsic structure of poly(A) RNA determines the specificity of Pan2 and Caf1 deadenylases. Nat.Struct.Mol.Biol., 26, 2019
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6R9Q
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![BU of 6r9q by Molmil](/molmil-images/mine/6r9q) | Structure of Saccharomyces cerevisiae apo Pan2 pseudoubiquitin hydrolase-RNA exonuclease (UCH-Exo) module in complex with AACCAA RNA | 分子名称: | AACCAA, PAN2-PAN3 deadenylation complex catalytic subunit PAN2 | 著者 | Tang, T.T.L, Stowell, J.A.W, Hill, C.H, Passmore, L.A. | 登録日 | 2019-04-03 | 公開日 | 2019-05-22 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (3.079 Å) | 主引用文献 | The intrinsic structure of poly(A) RNA determines the specificity of Pan2 and Caf1 deadenylases. Nat.Struct.Mol.Biol., 26, 2019
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6R9O
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![BU of 6r9o by Molmil](/molmil-images/mine/6r9o) | Structure of Saccharomyces cerevisiae apo Pan2 pseudoubiquitin hydrolase-RNA exonuclease (UCH-Exo) module in complex with AAGGA RNA | 分子名称: | AAGGA RNA, PAN2-PAN3 deadenylation complex catalytic subunit PAN2 | 著者 | Tang, T.T.L, Stowell, J.A.W, Hill, C.H, Passmore, L.A. | 登録日 | 2019-04-03 | 公開日 | 2019-05-22 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (3.319 Å) | 主引用文献 | The intrinsic structure of poly(A) RNA determines the specificity of Pan2 and Caf1 deadenylases. Nat.Struct.Mol.Biol., 26, 2019
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6R9J
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![BU of 6r9j by Molmil](/molmil-images/mine/6r9j) | Structure of Saccharomyces cerevisiae apo Pan2 pseudoubiquitin hydrolase-RNA exonuclease (UCH-Exo) module in complex with A7 RNA | 分子名称: | A7 RNA, PAN2-PAN3 deadenylation complex catalytic subunit PAN2 | 著者 | Tang, T.T.L, Stowell, J.A.W, Hill, C.H, Passmore, L.A. | 登録日 | 2019-04-03 | 公開日 | 2019-05-22 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (3.326 Å) | 主引用文献 | The intrinsic structure of poly(A) RNA determines the specificity of Pan2 and Caf1 deadenylases. Nat.Struct.Mol.Biol., 26, 2019
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6R9P
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![BU of 6r9p by Molmil](/molmil-images/mine/6r9p) | Structure of Saccharomyces cerevisiae apo Pan2 pseudoubiquitin hydrolase-RNA exonuclease (UCH-Exo) module in complex with AAUUAA RNA | 分子名称: | AAUUAA RNA, PAN2-PAN3 deadenylation complex catalytic subunit PAN2 | 著者 | Tang, T.T.L, Stowell, J.A.W, Hill, C.H, Passmore, L.A. | 登録日 | 2019-04-03 | 公開日 | 2019-05-22 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (2.98 Å) | 主引用文献 | The intrinsic structure of poly(A) RNA determines the specificity of Pan2 and Caf1 deadenylases. Nat.Struct.Mol.Biol., 26, 2019
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6OIA
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![BU of 6oia by Molmil](/molmil-images/mine/6oia) | (1S,3S)-3-amino-4-(perfluoropropan-2-ylidene)cyclopentane-1-carboxylic acid hydrochloride, a potent inhibitor of ornithine aminotransferase | 分子名称: | (1S)-3-amino-4-[(2S)-1,1,1-trifluoro-3-oxopropan-2-yl]cyclopent-3-ene-1-carboxylic acid, GLYCEROL, Ornithine aminotransferase, ... | 著者 | Catlin, D.S, Liu, D, Moschitto, M.J, Doubleday, P.F, Kelleher, N, Silverman, R.B. | 登録日 | 2019-04-09 | 公開日 | 2019-09-18 | 最終更新日 | 2020-04-01 | 実験手法 | X-RAY DIFFRACTION (1.777 Å) | 主引用文献 | Mechanism of Inactivation of Ornithine Aminotransferase by (1S,3S)-3-Amino-4-(hexafluoropropan-2-ylidenyl)cyclopentane-1-carboxylic Acid. J.Am.Chem.Soc., 141, 2019
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6OYB
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![BU of 6oyb by Molmil](/molmil-images/mine/6oyb) | |
6OYE
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![BU of 6oye by Molmil](/molmil-images/mine/6oye) | |
6OYG
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![BU of 6oyg by Molmil](/molmil-images/mine/6oyg) | |
6OY8
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![BU of 6oy8 by Molmil](/molmil-images/mine/6oy8) | |
8F4T
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![BU of 8f4t by Molmil](/molmil-images/mine/8f4t) | Crystal structure of acetyltransferase Eis from M. tuberculosis in complex with proguanil | 分子名称: | DI(HYDROXYETHYL)ETHER, DIMETHYL SULFOXIDE, GLYCEROL, ... | 著者 | Punetha, A, Pang, A.H, Garneau-Tsodikova, S, Tsodikov, O.V. | 登録日 | 2022-11-11 | 公開日 | 2023-02-01 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.93 Å) | 主引用文献 | Discovery and Mechanistic Analysis of Structurally Diverse Inhibitors of Acetyltransferase Eis among FDA-Approved Drugs. Biochemistry, 62, 2023
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4TRF
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![BU of 4trf by Molmil](/molmil-images/mine/4trf) | |
4TRU
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![BU of 4tru by Molmil](/molmil-images/mine/4tru) | |
5XLV
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![BU of 5xlv by Molmil](/molmil-images/mine/5xlv) | Mycobacterium tuberculosis Pantothenate kinase mutant F254A | 分子名称: | 1,2-ETHANEDIOL, GLYCEROL, Pantothenate kinase, ... | 著者 | Paul, A, Kumar, P, Surolia, A, Vijayan, M. | 登録日 | 2017-05-11 | 公開日 | 2018-05-16 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Biochemical and structural studies of mutants indicate concerted movement of the dimer interface and ligand-binding region of Mycobacterium tuberculosis pantothenate kinase Acta Crystallogr F Struct Biol Commun, 73, 2017
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4LRD
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![BU of 4lrd by Molmil](/molmil-images/mine/4lrd) | Phosphopentomutase 4H11 variant | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, GLYCEROL, MANGANESE (II) ION, ... | 著者 | Birmingham, W.A, Starbird, C.A, Panosian, T.D, Nannemann, D.P, Iverson, T.M, Bachmann, B.O. | 登録日 | 2013-07-19 | 公開日 | 2013-07-31 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.78 Å) | 主引用文献 | Bioretrosynthetic construction of a didanosine biosynthetic pathway. Nat.Chem.Biol., 10, 2014
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5V70
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5UMK
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6RX5
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![BU of 6rx5 by Molmil](/molmil-images/mine/6rx5) | Trypanosoma brucei PTR1 (TbPTR1) in complex with inhibitor 1 (NMT-C0003) | 分子名称: | ACETATE ION, GLYCEROL, METHYL 1-(4-{[(2,4-DIAMINOPTERIDIN-6-YL)METHYL](METHYL)AMINO}BENZOYL)PIPERIDINE-4-CARBOXYLATE, ... | 著者 | Landi, G, Pozzi, C, Mangani, S. | 登録日 | 2019-06-07 | 公開日 | 2020-07-15 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.42 Å) | 主引用文献 | Multitarget, Selective Compound Design Yields Potent Inhibitors of a Kinetoplastid Pteridine Reductase 1. J.Med.Chem., 65, 2022
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5UZY
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5V73
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6RX0
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![BU of 6rx0 by Molmil](/molmil-images/mine/6rx0) | Trypanosoma brucei PTR1 (TbPTR1) in complex with inhibitor 3 (NMT-C0013) | 分子名称: | ACETATE ION, GLYCEROL, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, ... | 著者 | Landi, G, Pozzi, C, Mangani, S. | 登録日 | 2019-06-07 | 公開日 | 2020-07-15 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.2 Å) | 主引用文献 | Multitarget, Selective Compound Design Yields Potent Inhibitors of a Kinetoplastid Pteridine Reductase 1. J.Med.Chem., 65, 2022
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4NE2
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![BU of 4ne2 by Molmil](/molmil-images/mine/4ne2) | Pantothenamide-bound Pantothenate Kinase from Klebsiella pneumoniae | 分子名称: | (R)-N-(3-((2-(benzo[d][1,3]dioxol-5-yl)ethyl)amino)-3-oxopropyl)-2,4-dihydroxy-3,3-dimethylbutanamide, ADENOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, ... | 著者 | Hughes, S.J, Antoshchenko, T, Kim, K.P, Smil, D, Park, H.W. | 登録日 | 2013-10-28 | 公開日 | 2014-02-26 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structural characterization of a new N-substituted pantothenamide bound to pantothenate kinases from Klebsiella pneumoniae and Staphylococcus aureus. Proteins, 82, 2014
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3IRO
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![BU of 3iro by Molmil](/molmil-images/mine/3iro) | |
4NB4
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![BU of 4nb4 by Molmil](/molmil-images/mine/4nb4) | Pantothenamide-bound Pantothenate kinase from Staphylococcus aureus | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, N-[2-(1,3-benzodioxol-5-yl)ethyl]-N~3~-[(2R)-2-hydroxy-3,3-dimethyl-4-(phosphonooxy)butanoyl]-beta-alaninamide, ... | 著者 | Hughes, S.J, Antoshchenko, T, Smil, D, Park, H.W. | 登録日 | 2013-10-22 | 公開日 | 2014-03-05 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.25 Å) | 主引用文献 | Structural characterization of a new N-substituted pantothenamide bound to pantothenate kinases from Klebsiella pneumoniae and Staphylococcus aureus. Proteins, 82, 2014
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