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3DDP
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BU of 3ddp by Molmil
Structure of phosphorylated Thr160 CDK2/cyclin A in complex with the inhibitor CR8
分子名称: (2R)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9H-purin-2-yl}amino)butan-1-ol, Cell division protein kinase 2, Cyclin-A2
著者Echalier, A, Endicott, J.A.
登録日2008-06-06
公開日2008-07-22
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献CR8, a potent and selective, roscovitine-derived inhibitor of cyclin-dependent kinases.
Oncogene, 27, 2008
2KVQ
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BU of 2kvq by Molmil
Solution structure of NusE:NusG-CTD complex
分子名称: NusE, Transcription antitermination protein nusG
著者Burmann, B.M, Schweimer, K, Roesch, P.
登録日2010-03-25
公開日2010-05-05
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献A NusE:NusG complex links transcription and translation.
Science, 328, 2010
1QP9
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BU of 1qp9 by Molmil
STRUCTURE OF HAP1-PC7 COMPLEXED TO THE UAS OF CYC7
分子名称: CYP1(HAP1-PC7) ACTIVATORY PROTEIN, DNA (5'-D(*AP*CP*GP*CP*TP*AP*TP*TP*AP*TP*CP*GP*CP*TP*AP*TP*TP*AP*GP*T)-3'), DNA (5'-D(*AP*CP*TP*AP*AP*TP*AP*GP*CP*GP*AP*TP*AP*AP*TP*AP*GP*CP*GP*T)-3'), ...
著者Lukens, A, King, D, Marmorstein, R.
登録日1999-06-01
公開日2000-10-09
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Structure of HAP1-PC7 bound to DNA: implications for DNA recognition and allosteric effects of DNA-binding on transcriptional activation.
Nucleic Acids Res., 28, 2000
4BZ8
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BU of 4bz8 by Molmil
Crystal structure of Schistosoma mansoni HDAC8 complexed with J1038
分子名称: (2R)-2-methyl-3-oxo-4H-1,4-benzothiazine-6-carbohydroxamic acid, HISTONE DEACETYLASE 8, POTASSIUM ION, ...
著者Marek, M, Romier, C.
登録日2013-07-24
公開日2013-08-14
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.21 Å)
主引用文献Structural Basis for the Inhibition of Histone Deacetylase 8 (Hdac8), a Key Epigenetic Player in the Blood Fluke Schistosoma Mansoni.
Plos Pathog., 9, 2013
8SZU
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BU of 8szu by Molmil
Structure of Kdac1-Citarinostat complex from Acinetobacter baumannii
分子名称: Citarinostat, Histone deacetylase domain-containing protein, POTASSIUM ION, ...
著者Watson, P.R, Christianson, D.W.
登録日2023-05-30
公開日2023-09-06
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Structure and Function of Kdac1, a Class II Deacetylase from the Multidrug-Resistant Pathogen Acinetobacter baumannii .
Biochemistry, 62, 2023
8SZT
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BU of 8szt by Molmil
Structure of Kdac1 from Acinetobacter baumannii
分子名称: CHLORIDE ION, Histone deacetylase domain-containing protein, POTASSIUM ION, ...
著者Watson, P.R, Christianson, D.W.
登録日2023-05-30
公開日2023-09-06
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structure and Function of Kdac1, a Class II Deacetylase from the Multidrug-Resistant Pathogen Acinetobacter baumannii .
Biochemistry, 62, 2023
4BZ6
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BU of 4bz6 by Molmil
Crystal structure of Schistosoma mansoni HDAC8 complexed with SAHA
分子名称: DIMETHYLFORMAMIDE, GLYCEROL, HISTONE DEACETYLASE 8, ...
著者Marek, M, Romier, C.
登録日2013-07-24
公開日2013-08-14
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural Basis for the Inhibition of Histone Deacetylase 8 (Hdac8), a Key Epigenetic Player in the Blood Fluke Schistosoma Mansoni.
Plos Pathog., 9, 2013
5N9Q
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BU of 5n9q by Molmil
Structure of A. thaliana RCD1(468-567)
分子名称: Inactive poly [ADP-ribose] polymerase RCD1
著者Tossavainen, H, Hellman, M, Vainonen, J, Kangasjarvi, J, Permi, P.
登録日2017-02-27
公開日2018-03-14
最終更新日2024-06-19
実験手法SOLUTION NMR
主引用文献Arabidopsis RCD1 coordinates chloroplast and mitochondrial functions through interaction with ANAC transcription factors.
Elife, 8, 2019
4BZ7
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BU of 4bz7 by Molmil
Crystal structure of Schistosoma mansoni HDAC8 complexed with M344
分子名称: 4-(dimethylamino)-N-[7-(hydroxyamino)-7-oxoheptyl]benzamide, GLYCEROL, HISTONE DEACETYLASE 8, ...
著者Marek, M, Romier, C.
登録日2013-07-24
公開日2013-08-14
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献Structural Basis for the Inhibition of Histone Deacetylase 8 (Hdac8), a Key Epigenetic Player in the Blood Fluke Schistosoma Mansoni.
Plos Pathog., 9, 2013
4BZ9
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BU of 4bz9 by Molmil
Crystal structure of Schistosoma mansoni HDAC8 complexed with J1075
分子名称: 3-chlorobenzothiophene-2-carbohydroxamic acid, DIMETHYLFORMAMIDE, GLYCEROL, ...
著者Marek, M, Romier, C.
登録日2013-07-24
公開日2013-08-14
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural Basis for the Inhibition of Histone Deacetylase 8 (Hdac8), a Key Epigenetic Player in the Blood Fluke Schistosoma Mansoni.
Plos Pathog., 9, 2013
4BZ5
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BU of 4bz5 by Molmil
Crystal structure of Schistosoma mansoni HDAC8
分子名称: HISTONE DEACETYLASE 8, L(+)-TARTARIC ACID, POTASSIUM ION, ...
著者Marek, M, Romier, C.
登録日2013-07-24
公開日2013-08-14
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.785 Å)
主引用文献Structural Basis for the Inhibition of Histone Deacetylase 8 (Hdac8), a Key Epigenetic Player in the Blood Fluke Schistosoma Mansoni.
Plos Pathog., 9, 2013
3PXR
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BU of 3pxr by Molmil
Apo CDK2 crystallized from Jeffamine
分子名称: 1,2-ETHANEDIOL, Cell division protein kinase 2
著者Betzi, S, Alam, R, Schonbrunn, E.
登録日2010-12-10
公開日2011-02-16
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Discovery of a Potential Allosteric Ligand Binding Site in CDK2.
Acs Chem.Biol., 6, 2011
3PY0
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BU of 3py0 by Molmil
CDK2 in complex with inhibitor SU9516
分子名称: (3Z)-3-(1H-IMIDAZOL-5-YLMETHYLENE)-5-METHOXY-1H-INDOL-2(3H)-ONE, 1,2-ETHANEDIOL, Cell division protein kinase 2, ...
著者Betzi, S, Alam, R, Schonbrunn, E.
登録日2010-12-10
公開日2011-02-16
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Discovery of a Potential Allosteric Ligand Binding Site in CDK2.
Acs Chem.Biol., 6, 2011
3BBF
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BU of 3bbf by Molmil
Crystal structure of the NM23-H2 transcription factor complex with GDP
分子名称: 2,3-DIHYDROXY-1,4-DITHIOBUTANE, GUANOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, ...
著者Weichsel, A, Montfort, W.R.
登録日2007-11-09
公開日2008-09-23
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献NM23-H2 may play an indirect role in transcriptional activation of c-myc gene expression but does not cleave the nuclease hypersensitive element III1.
Mol.Cancer Ther., 8, 2009
8QU3
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BU of 8qu3 by Molmil
NF-YB/C Heterodimer in Complex with a 13-mer NF-YA-derived Peptide Stabilized with C8-Hydrocarbon Linker
分子名称: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, FORMIC ACID, Nuclear transcription factor Y subunit alpha, ...
著者Arbore, F, Durukan, C, Klintrot, C.I.R, Grossmann, T.N, Hennig, S.
登録日2023-10-13
公開日2024-03-20
最終更新日2024-05-15
実験手法X-RAY DIFFRACTION (1.41 Å)
主引用文献Binding Dynamics of a Stapled Peptide Targeting the Transcription Factor NF-Y.
Chembiochem, 25, 2024
8QU2
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BU of 8qu2 by Molmil
NF-YB/C Heterodimer in Complex with a 16-mer NF-YA-derived Peptide Stabilized with C8-Hydrocarbon Linker
分子名称: 1,2-ETHANEDIOL, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, FORMIC ACID, ...
著者Durukan, C, Arbore, F, Klintrot, C.I.R, Grossmann, T.N, Hennig, S.
登録日2023-10-13
公開日2024-03-20
最終更新日2024-05-15
実験手法X-RAY DIFFRACTION (1.45 Å)
主引用文献Binding Dynamics of a Stapled Peptide Targeting the Transcription Factor NF-Y.
Chembiochem, 25, 2024
3PXY
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BU of 3pxy by Molmil
CDK2 in complex with inhibitor JWS648
分子名称: 2-(4,6-diamino-1,3,5-triazin-2-yl)-4-methoxyphenol, Cell division protein kinase 2, PHOSPHATE ION
著者Han, H, Betzi, S, Alam, R, Schonbrunn, E.
登録日2010-12-10
公開日2011-02-16
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Discovery of a Potential Allosteric Ligand Binding Site in CDK2.
Acs Chem.Biol., 6, 2011
3PXQ
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BU of 3pxq by Molmil
CDK2 in complex with 3 molecules of 8-anilino-1-naphthalene sulfonate
分子名称: 1,2-ETHANEDIOL, 8-ANILINO-1-NAPHTHALENE SULFONATE, Cell division protein kinase 2
著者Betzi, S, Alam, R, Schonbrunn, E.
登録日2010-12-10
公開日2011-02-16
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Discovery of a Potential Allosteric Ligand Binding Site in CDK2.
Acs Chem.Biol., 6, 2011
3BBB
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BU of 3bbb by Molmil
Crystal structure of the NM23-H2 transcription factor complex with dinucleotide d(AG)
分子名称: DNA (5'-D(*AP*G)-3'), Nucleoside diphosphate kinase B
著者Weichsel, A, Montfort, W.R.
登録日2007-11-09
公開日2008-09-23
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (1.3 Å)
主引用文献NM23-H2 may play an indirect role in transcriptional activation of c-myc gene expression but does not cleave the nuclease hypersensitive element III1.
Mol.Cancer Ther., 8, 2009
1R4M
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BU of 1r4m by Molmil
APPBP1-UBA3-NEDD8, an E1-ubiquitin-like protein complex
分子名称: Ubiquitin-like protein NEDD8, ZINC ION, amyloid beta precursor protein-binding protein 1, ...
著者Walden, H, Podgorski, M.S, Holton, J.M, Schulman, B.A.
登録日2003-10-07
公開日2003-12-23
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献The structure of the APPBP1-UBA3-NEDD8-ATP complex reveals the basis for selective ubiquitin-like protein activation by an E1.
Mol.Cell, 12, 2003
3BBC
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BU of 3bbc by Molmil
Crystal structure of R88A mutant of the NM23-H2 transcription factor
分子名称: Nucleoside diphosphate kinase B
著者Weichsel, A, Montfort, W.R.
登録日2007-11-09
公開日2008-09-23
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献NM23-H2 may play an indirect role in transcriptional activation of c-myc gene expression but does not cleave the nuclease hypersensitive element III1.
Mol.Cancer Ther., 8, 2009
1PVH
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BU of 1pvh by Molmil
Crystal structure of leukemia inhibitory factor in complex with gp130
分子名称: IODIDE ION, Interleukin-6 receptor beta chain, Leukemia inhibitory factor
著者Boulanger, M.J, Bankovich, A.J, Kortemme, T, Baker, D, Garcia, K.C.
登録日2003-06-27
公開日2003-10-14
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Convergent mechanisms for recognition of divergent cytokines by the shared signaling receptor gp130.
Mol.Cell, 12, 2003
3PXF
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BU of 3pxf by Molmil
CDK2 in complex with two molecules of 8-anilino-1-naphthalene sulfonate
分子名称: 1,2-ETHANEDIOL, 8-ANILINO-1-NAPHTHALENE SULFONATE, Cell division protein kinase 2
著者Betzi, S, Alam, R, Schonbrunn, E.
登録日2010-12-09
公開日2011-02-16
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Discovery of a Potential Allosteric Ligand Binding Site in CDK2.
Acs Chem.Biol., 6, 2011
1R4N
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BU of 1r4n by Molmil
APPBP1-UBA3-NEDD8, an E1-ubiquitin-like protein complex with ATP
分子名称: ADENOSINE-5'-TRIPHOSPHATE, Ubiquitin-like protein NEDD8, ZINC ION, ...
著者Walden, H, Podgorski, M.S, Holton, J.M, Schulman, B.A.
登録日2003-10-07
公開日2003-12-23
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (3.6 Å)
主引用文献The structure of the APPBP1-UBA3-NEDD8-ATP complex reveals the basis for selective ubiquitin-like protein activation by an E1.
Mol.Cell, 12, 2003
2NNY
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BU of 2nny by Molmil
Crystal structure of the Ets1 dimer DNA complex.
分子名称: 5'-D(*A*CP*TP*CP*CP*AP*GP*GP*AP*AP*GP*TP*GP*CP*TP*TP*CP*CP*TP*GP*TP*CP*T)-3', 5'-D(*T*AP*GP*AP*CP*AP*GP*GP*AP*AP*GP*CP*AP*CP*TP*TP*CP*CP*TP*GP*GP*AP*G)-3', C-ets-1 protein
著者Lamber, E.P, Kachalova, G.S, Wilmanns, M.
登録日2006-10-24
公開日2008-03-04
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.58 Å)
主引用文献Regulation of the transcription factor Ets-1 by DNA-mediated homo-dimerization.
Embo J., 27, 2008

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