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3PY0

CDK2 in complex with inhibitor SU9516

Summary for 3PY0
Entry DOI10.2210/pdb3py0/pdb
Related3PXF 3PXQ 3PXR 3PXY 3PXZ 3PY1
DescriptorCell division protein kinase 2, 1,2-ETHANEDIOL, PHOSPHATE ION, ... (5 entities in total)
Functional Keywordsprotein kinase, cdk2, inhibitor, transferase-transferase inhibitor complex, transferase/transferase inhibitor
Biological sourceHomo sapiens (human)
Total number of polymer chains1
Total formula weight35159.63
Authors
Betzi, S.,Alam, R.,Schonbrunn, E. (deposition date: 2010-12-10, release date: 2011-02-16, Last modification date: 2023-09-13)
Primary citationBetzi, S.,Alam, R.,Martin, M.,Lubbers, D.J.,Han, H.,Jakkaraj, S.R.,Georg, G.I.,Schonbrunn, E.
Discovery of a Potential Allosteric Ligand Binding Site in CDK2.
Acs Chem.Biol., 6:492-501, 2011
Cited by
PubMed: 21291269
DOI: 10.1021/cb100410m
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.75 Å)
Structure validation

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