6PJH
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![BU of 6pjh by Molmil](/molmil-images/mine/6pjh) | HIV-1 Protease NL4-3 WT in Complex with LR3-28 | 分子名称: | (3R,3aS,6aR)-hexahydrofuro[2,3-b]furan-3-yl [(2S,4S,5S)-4-hydroxy-5-{[N-(methoxycarbonyl)-L-valyl]amino}-1,6-diphenylhexan-2-yl]carbamate, Protease NL4-3, SULFATE ION | 著者 | Lockbaum, G.J, Rusere, L.N, Henes, M, Kosovrasti, K, Lee, S.K, Spielvogel, E, Nalivaika, E.A, Swanstrom, R, KurtYilmaz, N, Schiffer, C.A, Ali, A. | 登録日 | 2019-06-28 | 公開日 | 2020-07-01 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Structural Analysis of Potent Hybrid HIV-1 Protease Inhibitors Containing Bis-tetrahydrofuran in a Pseudosymmetric Dipeptide Isostere. J.Med.Chem., 63, 2020
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1FB1
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![BU of 1fb1 by Molmil](/molmil-images/mine/1fb1) | CRYSTAL STRUCTURE OF HUMAN GTP CYCLOHYDROLASE I | 分子名称: | GTP CYCLOHYDROLASE I, ISOPROPYL ALCOHOL, ZINC ION | 著者 | Auerbach, G, Herrmann, A, Bracher, A, Bader, G, Gutlich, M, Fischer, M, Neukamm, M, Nar, H, Garrido-Franco, M, Richardson, J, Huber, R, Bacher, A. | 登録日 | 2000-07-14 | 公開日 | 2000-12-08 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Zinc plays a key role in human and bacterial GTP cyclohydrolase I. Proc.Natl.Acad.Sci.USA, 97, 2000
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6P13
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![BU of 6p13 by Molmil](/molmil-images/mine/6p13) | Structure of spastin AAA domain (T692A mutant) in complex with a diaminotriazole-based inhibitor (crystal form A) | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, 3-{[5-amino-1-(2-fluoro-6-methoxybenzene-1-carbonyl)-1H-1,2,4-triazol-3-yl]amino}-N-methylbenzamide, SULFATE ION, ... | 著者 | Pisa, R, Cupido, T, Kapoor, T.M. | 登録日 | 2019-05-17 | 公開日 | 2019-08-07 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Analyzing Resistance to Design Selective Chemical Inhibitors for AAA Proteins. Cell Chem Biol, 26, 2019
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1F8S
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![BU of 1f8s by Molmil](/molmil-images/mine/1f8s) | CRYSTAL STRUCTURE OF L-AMINO ACID OXIDASE FROM CALLOSELASMA RHODOSTOMA, COMPLEXED WITH THREE MOLECULES OF O-AMINOBENZOATE. | 分子名称: | 2-AMINOBENZOIC ACID, 2-acetamido-2-deoxy-beta-D-glucopyranose, FLAVIN-ADENINE DINUCLEOTIDE, ... | 著者 | Pawelek, P.D, Cheah, J, Coulombe, R, Macheroux, P, Ghisla, S, Vrielink, A. | 登録日 | 2000-07-04 | 公開日 | 2000-08-24 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | The structure of L-amino acid oxidase reveals the substrate trajectory into an enantiomerically conserved active site. EMBO J., 19, 2000
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7TPG
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![BU of 7tpg by Molmil](/molmil-images/mine/7tpg) | Single-Particle Cryo-EM Structure of the WaaL O-antigen ligase in its ligand bound state | 分子名称: | Fab Heavy (H) Chain, Fab Light (L) Chain, GERANYL DIPHOSPHATE, ... | 著者 | Ashraf, K.U, Nygaard, R, Vickery, O.N, Erramilli, S.K, Herrera, C.M, McConville, T.H, Petrou, V.I, Giacometti, S.I, Dufrisne, M.B, Nosol, K, Zinkle, A.P, Graham, C.L.B, Loukeris, M, Kloss, B, Skorupinska-Tudek, K, Swiezewska, E, Roper, D, Clarke, O.B, Uhlemann, A.C, Kossiakoff, A.A, Trent, M.S, Stansfeld, P.J, Mancia, F. | 登録日 | 2022-01-25 | 公開日 | 2022-04-06 | 最終更新日 | 2022-04-27 | 実験手法 | ELECTRON MICROSCOPY (3.23 Å) | 主引用文献 | Structural basis of lipopolysaccharide maturation by the O-antigen ligase. Nature, 604, 2022
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1FBX
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![BU of 1fbx by Molmil](/molmil-images/mine/1fbx) | CRYSTAL STRUCTURE OF ZINC-CONTAINING E.COLI GTP CYCLOHYDROLASE I | 分子名称: | CHLORIDE ION, GTP CYCLOHYDROLASE I, ZINC ION | 著者 | Auerbach, G, Herrmann, A, Bracher, A, Bader, A, Gutlich, M, Fischer, M, Neukamm, M, Nar, H, Garrido-Franco, M, Richardson, J, Huber, R, Bacher, A. | 登録日 | 2000-07-17 | 公開日 | 2001-02-14 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Zinc plays a key role in human and bacterial GTP cyclohydrolase I. Proc.Natl.Acad.Sci.USA, 97, 2000
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7TPJ
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![BU of 7tpj by Molmil](/molmil-images/mine/7tpj) | Single-Particle Cryo-EM Structure of the WaaL O-antigen ligase in its apo state | 分子名称: | Fab Heavy (H) Chain, Fab Light (L) Chain, Putative cell surface polysaccharide polymerase/ligase | 著者 | Ashraf, K.U, Nygaard, R, Vickery, O.N, Erramilli, S.K, Herrera, C.M, McConville, T.H, Petrou, V.I, Giacometti, S.I, Dufrisne, M.B, Nosol, K, Zinkle, A.P, Graham, C.L.B, Loukeris, M, Kloss, B, Skorupinska-Tudek, K, Swiezewska, E, Roper, D, Clarke, O.B, Uhlemann, A.C, Kossiakoff, A.A, Trent, M.S, Stansfeld, P.J, Mancia, F. | 登録日 | 2022-01-25 | 公開日 | 2022-04-06 | 最終更新日 | 2022-04-27 | 実験手法 | ELECTRON MICROSCOPY (3.46 Å) | 主引用文献 | Structural basis of lipopolysaccharide maturation by the O-antigen ligase. Nature, 604, 2022
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6PS1
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![BU of 6ps1 by Molmil](/molmil-images/mine/6ps1) | XFEL beta2 AR structure by ligand exchange from Alprenolol to Timolol. | 分子名称: | (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, (2S)-1-(tert-butylamino)-3-[(4-morpholin-4-yl-1,2,5-thiadiazol-3-yl)oxy]propan-2-ol, CHOLESTEROL, ... | 著者 | Ishchenko, A, Stauch, B, Han, G.W, Batyuk, A, Shiriaeva, A, Li, C, Zatsepin, N.A, Weierstall, U, Liu, W, Nango, E, Nakane, T, Tanaka, R, Tono, K, Joti, Y, Iwata, S, Moraes, I, Gati, C, Cherezov, C. | 登録日 | 2019-07-12 | 公開日 | 2019-11-13 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (3.2 Å) | 主引用文献 | Toward G protein-coupled receptor structure-based drug design using X-ray lasers. Iucrj, 6, 2019
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7U97
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![BU of 7u97 by Molmil](/molmil-images/mine/7u97) | SAAV pH 4.0 capsid structure | 分子名称: | Capsid protein | 著者 | Mietzsch, M, McKenna, R. | 登録日 | 2022-03-10 | 公開日 | 2022-04-13 | 最終更新日 | 2024-02-14 | 実験手法 | ELECTRON MICROSCOPY (2.66 Å) | 主引用文献 | Characterization of the Serpentine Adeno-Associated Virus (SAAV) Capsid Structure: Receptor Interactions and Antigenicity. J.Virol., 96, 2022
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7U95
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![BU of 7u95 by Molmil](/molmil-images/mine/7u95) | SAAV pH 6.0 capsid structure | 分子名称: | Capsid protein | 著者 | Mietzsch, M, McKenna, R. | 登録日 | 2022-03-10 | 公開日 | 2022-04-13 | 最終更新日 | 2024-02-14 | 実験手法 | ELECTRON MICROSCOPY (2.73 Å) | 主引用文献 | Characterization of the Serpentine Adeno-Associated Virus (SAAV) Capsid Structure: Receptor Interactions and Antigenicity. J.Virol., 96, 2022
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1FP7
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![BU of 1fp7 by Molmil](/molmil-images/mine/1fp7) | MONOVALENT CATION BINDING SITES IN N10-FORMYLTETRAHYDROFOLATE SYNTHETASE FROM MOORELLA THERMOACETICA | 分子名称: | FORMATE--TETRAHYDROFOLATE LIGASE, POTASSIUM ION, SULFATE ION | 著者 | Radfar, R, Leaphart, A, Brewer, J.M, Minor, W, Odom, J.D. | 登録日 | 2000-08-30 | 公開日 | 2001-08-30 | 最終更新日 | 2022-04-13 | 実験手法 | X-RAY DIFFRACTION (3.2 Å) | 主引用文献 | Cation binding and thermostability of FTHFS monovalent cation binding sites and thermostability of N10-formyltetrahydrofolate synthetase from Moorella thermoacetica. Biochemistry, 39, 2000
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1FQZ
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![BU of 1fqz by Molmil](/molmil-images/mine/1fqz) | NMR VALIDATED MODEL OF DOMAIN IIID OF HEPATITIS C VIRUS INTERNAL RIBOSOME ENTRY SITE | 分子名称: | HEPATITIS C VIRUS IRES DOMAIN IIID | 著者 | Klinck, R, Westhof, E, Walker, S, Afshar, M, Collier, A, Aboul-ela, F. | 登録日 | 2000-09-07 | 公開日 | 2001-01-17 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | A potential RNA drug target in the hepatitis C virus internal ribosomal entry site. RNA, 6, 2000
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7QVY
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![BU of 7qvy by Molmil](/molmil-images/mine/7qvy) | Cryo-EM structure of coxsackievirus A6 empty particle | 分子名称: | Capsid protein VP1, Capsid protein VP2, Capsid protein VP3 | 著者 | Buttner, C.R, Spurny, R, Fuzik, T, Plevka, P. | 登録日 | 2022-01-24 | 公開日 | 2022-09-07 | 最終更新日 | 2024-07-17 | 実験手法 | ELECTRON MICROSCOPY (2.82 Å) | 主引用文献 | Cryo-electron microscopy and image classification reveal the existence and structure of the coxsackievirus A6 virion. Commun Biol, 5, 2022
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7QVX
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![BU of 7qvx by Molmil](/molmil-images/mine/7qvx) | Cryo-EM structure of coxsackievirus A6 altered particle | 分子名称: | Capsid protein VP1, Capsid protein VP2, Capsid protein VP3 | 著者 | Buttner, C.R, Spurny, R, Fuzik, T, Plevka, P. | 登録日 | 2022-01-24 | 公開日 | 2022-09-07 | 最終更新日 | 2024-07-17 | 実験手法 | ELECTRON MICROSCOPY (2.5 Å) | 主引用文献 | Cryo-electron microscopy and image classification reveal the existence and structure of the coxsackievirus A6 virion. Commun Biol, 5, 2022
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7U96
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![BU of 7u96 by Molmil](/molmil-images/mine/7u96) | SAAV pH 5.5 capsid structure | 分子名称: | Capsid protein | 著者 | Mietzsch, M, McKenna, R. | 登録日 | 2022-03-10 | 公開日 | 2022-04-13 | 最終更新日 | 2024-02-14 | 実験手法 | ELECTRON MICROSCOPY (2.14 Å) | 主引用文献 | Characterization of the Serpentine Adeno-Associated Virus (SAAV) Capsid Structure: Receptor Interactions and Antigenicity. J.Virol., 96, 2022
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7QW9
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![BU of 7qw9 by Molmil](/molmil-images/mine/7qw9) | Cryo-EM structure of coxsackievirus A6 mature virion | 分子名称: | Capsid protein VP1, Capsid protein VP2, Capsid protein VP3, ... | 著者 | Buttner, C.R, Spurny, R, Fuzik, T, Plevka, P. | 登録日 | 2022-01-25 | 公開日 | 2022-09-07 | 最終更新日 | 2024-07-17 | 実験手法 | ELECTRON MICROSCOPY (2.68 Å) | 主引用文献 | Cryo-electron microscopy and image classification reveal the existence and structure of the coxsackievirus A6 virion. Commun Biol, 5, 2022
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7U94
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![BU of 7u94 by Molmil](/molmil-images/mine/7u94) | SAAV pH 7.4 capsid structure | 分子名称: | Capsid protein | 著者 | Mietzsch, M, McKenna, R. | 登録日 | 2022-03-10 | 公開日 | 2022-04-13 | 最終更新日 | 2024-02-14 | 実験手法 | ELECTRON MICROSCOPY (3.25 Å) | 主引用文献 | Characterization of the Serpentine Adeno-Associated Virus (SAAV) Capsid Structure: Receptor Interactions and Antigenicity. J.Virol., 96, 2022
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4YWH
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![BU of 4ywh by Molmil](/molmil-images/mine/4ywh) | CRYSTAL STRUCTURE OF AN ABC TRANSPORTER SOLUTE BINDING PROTEIN (IPR025997) FROM ACTINOBACILLUS SUCCINOGENES 130Z (Asuc_0499, TARGET EFI-511068) WITH BOUND D-XYLOSE | 分子名称: | ABC TRANSPORTER SOLUTE BINDING PROTEIN, beta-D-xylopyranose | 著者 | Vetting, M.W, Al Obaidi, N.F, Toro, R, Morisco, L.L, Benach, J, Koss, J, Wasserman, S.R, Attonito, J.D, Scott Glenn, A, Chamala, S, Chowdhury, S, Lafleur, J, Love, J, Seidel, R.D, Whalen, K.L, Gerlt, J.A, Almo, S.C, Enzyme Function Initiative (EFI) | 登録日 | 2015-03-20 | 公開日 | 2015-04-15 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.35 Å) | 主引用文献 | CRYSTAL STRUCTURE OF AN ABC TRANSPORTER SOLUTE BINDING PROTEIN (IPR025997) FROM ACTINOBACILLUS SUCCINOGENES 130Z (Asuc_0499, TARGET EFI-511068) WITH BOUND D-XYLOSE To be published
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6PJF
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![BU of 6pjf by Molmil](/molmil-images/mine/6pjf) | HIV-1 Protease NL4-3 WT in Complex with LR2-44 | 分子名称: | Protease NL4-3, SULFATE ION, methyl [(1S)-1-cyclopentyl-2-({(2S,3S,5S)-5-[({[(3R,3aS,6aR)-hexahydrofuro[2,3-b]furan-3-yl]oxy}carbonyl)amino]-3-hydroxy-1,6-diphenylhexan-2-yl}amino)-2-oxoethyl]carbamate | 著者 | Lockbaum, G.J, Rusere, L.N, Henes, M, Kosovrasti, K, Lee, S.K, Spielvogel, E, Nalivaika, E.A, Swanstrom, R, KurtYilmaz, N, Schiffer, C.A, Ali, A. | 登録日 | 2019-06-28 | 公開日 | 2020-07-01 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.94 Å) | 主引用文献 | Structural Analysis of Potent Hybrid HIV-1 Protease Inhibitors Containing Bis-tetrahydrofuran in a Pseudosymmetric Dipeptide Isostere. J.Med.Chem., 63, 2020
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4YIC
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![BU of 4yic by Molmil](/molmil-images/mine/4yic) | CRYSTAL STRUCTURE OF A TRAP TRANSPORTER SOLUTE BINDING PROTEIN (IPR025997) FROM BORDETELLA BRONCHISEPTICA RB50 (BB0280, TARGET EFI-500035) WITH BOUND PICOLINIC ACID | 分子名称: | ACETATE ION, CALCIUM ION, IMIDAZOLE, ... | 著者 | Vetting, M.W, Al Obaidi, N.F, Toro, R, Morisco, L.L, Benach, J, Koss, J, Wasserman, S.R, Attonito, J.D, Scott Glenn, A, Chamala, S, Chowdhury, S, Lafleur, J, Love, J, Seidel, R.D, Whalen, K.L, Gerlt, J.A, Almo, S.C, Enzyme Function Initiative (EFI) | 登録日 | 2015-03-01 | 公開日 | 2015-04-01 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | CRYSTAL STRUCTURE OF A TRAP TRANSPORTER SOLUTE BINDING PROTEIN (IPR025997) FROM BORDETELLA BRONCHISEPTICA RB50 (BB0280, TARGET EFI-500035) WITH BOUND PICOLINIC ACID To be published
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7QYH
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![BU of 7qyh by Molmil](/molmil-images/mine/7qyh) | |
4Y9N
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![BU of 4y9n by Molmil](/molmil-images/mine/4y9n) | PA3825-EAL Metal-Free-Apo Structure - Magnesium Co-crystallisation | 分子名称: | PA3825-EAL, PHOSPHATE ION | 著者 | Bellini, D, Horrell, S, Wagner, A, Strange, R, Walsh, M.A. | 登録日 | 2015-02-17 | 公開日 | 2016-03-09 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.92 Å) | 主引用文献 | Structure of PA3825 from P. aeruginosa bound to cyclic di-GMP and pGpG: new insights for a potential three-metal catalytic mechanism of EAL domains To Be Published
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1FCE
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![BU of 1fce by Molmil](/molmil-images/mine/1fce) | PROCESSIVE ENDOCELLULASE CELF OF CLOSTRIDIUM CELLULOLYTICUM | 分子名称: | CALCIUM ION, CELLULASE CELF, beta-D-glucopyranose-(1-4)-beta-D-glucopyranose-(1-4)-4-thio-beta-D-glucopyranose-(1-4)-methyl beta-D-glucopyranoside | 著者 | Parsiegla, G, Juy, M, Haser, R. | 登録日 | 1998-07-06 | 公開日 | 1999-07-22 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | The crystal structure of the processive endocellulase CelF of Clostridium cellulolyticum in complex with a thiooligosaccharide inhibitor at 2.0 A resolution. EMBO J., 17, 1998
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7U2R
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![BU of 7u2r by Molmil](/molmil-images/mine/7u2r) | Structure of Paenibacillus sp. J14 Apyc1 | 分子名称: | Apyc1, ZINC ION | 著者 | Hobbs, S.J, Wein, T, Lu, A, Morehouse, B.R, Schnabel, J, Sorek, R, Kranzusch, P.J. | 登録日 | 2022-02-24 | 公開日 | 2022-04-20 | 最終更新日 | 2022-06-01 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Phage anti-CBASS and anti-Pycsar nucleases subvert bacterial immunity. Nature, 605, 2022
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7QFU
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![BU of 7qfu by Molmil](/molmil-images/mine/7qfu) | Crystal Structure of AtlA catalytic domain from Enterococcus feacalis | 分子名称: | GLYCEROL, Peptidoglycan hydrolase | 著者 | Zamboni, V, Barelier, S, Dixon, R, Galley, N, Ghanem, A, Cahuzac, H, Salamaga, B, Davis, P.J, Mesnage, S, Vincent, F. | 登録日 | 2021-12-06 | 公開日 | 2022-09-21 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.45 Å) | 主引用文献 | Molecular basis for substrate recognition and septum cleavage by AtlA, the major N-acetylglucosaminidase of Enterococcus faecalis. J.Biol.Chem., 298, 2022
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