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6P13

Structure of spastin AAA domain (T692A mutant) in complex with a diaminotriazole-based inhibitor (crystal form A)

Summary for 6P13
Entry DOI10.2210/pdb6p13/pdb
DescriptorSpastin, SULFATE ION, 3-{[5-amino-1-(2-fluoro-6-methoxybenzene-1-carbonyl)-1H-1,2,4-triazol-3-yl]amino}-N-methylbenzamide, ... (5 entities in total)
Functional Keywordsinhibitor, complex, aaa protein, isomerase-isomerase inhibitor complex, isomerase/isomerase inhibitor
Biological sourceDrosophila melanogaster (Fruit fly)
Total number of polymer chains1
Total formula weight34889.61
Authors
Pisa, R.,Cupido, T.,Kapoor, T.M. (deposition date: 2019-05-17, release date: 2019-08-07, Last modification date: 2023-10-11)
Primary citationPisa, R.,Cupido, T.,Steinman, J.B.,Jones, N.H.,Kapoor, T.M.
Analyzing Resistance to Design Selective Chemical Inhibitors for AAA Proteins.
Cell Chem Biol, 26:1263-, 2019
Cited by
PubMed: 31257183
DOI: 10.1016/j.chembiol.2019.06.001
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.1 Å)
Structure validation

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