7K5K
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![BU of 7k5k by Molmil](/molmil-images/mine/7k5k) | Plasmodium vivax M17 leucyl aminopeptidase Pv-M17 | 分子名称: | CARBONATE ION, M17 leucyl aminopeptidase, putative, ... | 著者 | Malcolm, T.R, McGowan, S, Belousoff, M.J. | 登録日 | 2020-09-17 | 公開日 | 2020-12-16 | 最終更新日 | 2024-03-06 | 実験手法 | ELECTRON MICROSCOPY (2.66 Å) | 主引用文献 | Active site metals mediate an oligomeric equilibrium in Plasmodium M17 aminopeptidases. J.Biol.Chem., 296, 2020
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6EE4
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![BU of 6ee4 by Molmil](/molmil-images/mine/6ee4) | X-ray crystal structure of Pf-M1 in complex with inhibitor (6m) and catalytic zinc ion | 分子名称: | (2R)-2-[(cyclopropylacetyl)amino]-N-hydroxy-2-(3',4',5'-trifluoro[1,1'-biphenyl]-4-yl)acetamide, GLYCEROL, M1 family aminopeptidase, ... | 著者 | Drinkwater, N, McGowan, S. | 登録日 | 2018-08-13 | 公開日 | 2018-12-26 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (1.58 Å) | 主引用文献 | Hydroxamic Acid Inhibitors Provide Cross-Species Inhibition of Plasmodium M1 and M17 Aminopeptidases. J. Med. Chem., 62, 2019
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5J7C
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5KYO
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![BU of 5kyo by Molmil](/molmil-images/mine/5kyo) | Crystal Structure of CYP101J2 | 分子名称: | CYP101J2, PROTOPORPHYRIN IX CONTAINING FE | 著者 | Unterweger, B, Drinkwater, N, Dumsday, G.J, McGowan, S. | 登録日 | 2016-07-22 | 公開日 | 2017-01-04 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | X-ray crystal structure of cytochrome P450 monooxygenase CYP101J2 from Sphingobium yanoikuyae strain B2. Proteins, 85, 2017
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6EE5
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![BU of 6ee5 by Molmil](/molmil-images/mine/6ee5) | |
6NVB
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![BU of 6nvb by Molmil](/molmil-images/mine/6nvb) | Crystal structure of the inhibitor-free form of the serine protease kallikrein-4 | 分子名称: | GLYCEROL, Kallikrein-4, SULFATE ION | 著者 | Riley, B.T, Buckle, A.M, McGowan, S. | 登録日 | 2019-02-04 | 公開日 | 2019-07-17 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.636 Å) | 主引用文献 | Crystal structure of the inhibitor-free form of the serine protease kallikrein-4. Acta Crystallogr.,Sect.F, 75, 2019
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4Z0D
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![BU of 4z0d by Molmil](/molmil-images/mine/4z0d) | Crystal structure of FVO strain Plasmodium falciparum AMA1 in complex with the RON2hp [Phe2038Trp] peptide | 分子名称: | Apical membrane antigen 1, Rhoptry neck protein 2 | 著者 | Wang, G, McGowan, S, Norton, R.S, Scanlon, M.J. | 登録日 | 2015-03-26 | 公開日 | 2016-08-03 | 最終更新日 | 2020-01-08 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Structure-Activity Studies of beta-Hairpin Peptide Inhibitors of the Plasmodium falciparum AMA1-RON2 Interaction. J.Mol.Biol., 428, 2016
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4Z0E
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![BU of 4z0e by Molmil](/molmil-images/mine/4z0e) | Crystal structure of FVO strain Plasmodium falciparum AMA1 in complex with the RON2hp [Phe2038TRN] peptide | 分子名称: | Apical membrane antigen 1, Rhoptry neck protein 2 | 著者 | Wang, G, McGowan, S, Norton, R.S, Scanlon, M.J. | 登録日 | 2015-03-26 | 公開日 | 2016-08-03 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structure-Activity Studies of beta-Hairpin Peptide Inhibitors of the Plasmodium falciparum AMA1-RON2 Interaction. J.Mol.Biol., 428, 2016
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4Z0F
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![BU of 4z0f by Molmil](/molmil-images/mine/4z0f) | Crystal structure of FVO strain Plasmodium falciparum AMA1 in complex with the RON2hp [Phe2038(6CW)] peptide | 分子名称: | Apical membrane antigen 1, Rhoptry neck protein 2 | 著者 | Wang, G, McGowan, S, Norton, R.S, Scanlon, M.J. | 登録日 | 2015-03-26 | 公開日 | 2016-08-03 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Structure-Activity Studies of beta-Hairpin Peptide Inhibitors of the Plasmodium falciparum AMA1-RON2 Interaction. J.Mol.Biol., 428, 2016
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4ZY1
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4Z09
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![BU of 4z09 by Molmil](/molmil-images/mine/4z09) | Crystal structure of FVO strain Plasmodium falciparum AMA1 in complex with the RON2hp [Thr2040Ala] peptide | 分子名称: | Apical membrane antigen 1, GLYCEROL, Rhoptry neck protein 2 | 著者 | Wang, G, McGowan, S, Norton, R.S, Scanlon, M.J. | 登録日 | 2015-03-26 | 公開日 | 2016-08-03 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structure-Activity Studies of beta-Hairpin Peptide Inhibitors of the Plasmodium falciparum AMA1-RON2 Interaction. J.Mol.Biol., 428, 2016
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4ZX3
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5CDZ
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![BU of 5cdz by Molmil](/molmil-images/mine/5cdz) | Crystal structure of conserpin in the latent state | 分子名称: | Conserpin in the latent state, GLYCEROL | 著者 | Porebski, B.T, McGowan, S, Keleher, S, Buckle, A.M. | 登録日 | 2015-07-06 | 公開日 | 2016-07-20 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.449 Å) | 主引用文献 | Smoothing a rugged protein folding landscape by sequence-based redesign. Sci Rep, 6, 2016
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4X2T
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![BU of 4x2t by Molmil](/molmil-images/mine/4x2t) | X-ray crystal structure of the orally available aminopeptidase inhibitor, Tosedostat, bound to the M17 Leucyl Aminopeptidase from P. falciparum | 分子名称: | (2S)-({(2R)-2-[(1S)-1-hydroxy-2-(hydroxyamino)-2-oxoethyl]-4-methylpentanoyl}amino)(phenyl)ethanoic acid, CARBONATE ION, M17 leucyl aminopeptidase, ... | 著者 | Drinkwater, N, McGowan, S. | 登録日 | 2014-11-27 | 公開日 | 2015-02-18 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.729 Å) | 主引用文献 | X-ray crystal structures of an orally available aminopeptidase inhibitor, Tosedostat, bound to anti-malarial drug targets PfA-M1 and PfA-M17. Proteins, 83, 2015
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5CE0
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![BU of 5ce0 by Molmil](/molmil-images/mine/5ce0) | |
5CBM
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![BU of 5cbm by Molmil](/molmil-images/mine/5cbm) | Crystal structure of PfA-M17 with virtual ligand inhibitor | 分子名称: | (2S)-2-{[(R)-[(R)-amino(phenyl)methyl](hydroxy)phosphoryl]methyl}-4-methylpentanoic acid, CARBONATE ION, GLYCEROL, ... | 著者 | Ruggeri, C, Drinkwater, N, McGowan, S. | 登録日 | 2015-07-01 | 公開日 | 2015-10-07 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Identification and Validation of a Potent Dual Inhibitor of the P. falciparum M1 and M17 Aminopeptidases Using Virtual Screening. Plos One, 10, 2015
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5CDX
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4X2U
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![BU of 4x2u by Molmil](/molmil-images/mine/4x2u) | X-ray crystal structure of the orally available aminopeptidase inhibitor, Tosedostat, bound to the M1 Alanyl Aminopeptidase from P. falciparum | 分子名称: | (2S)-({(2R)-2-[(1S)-1-hydroxy-2-(hydroxyamino)-2-oxoethyl]-4-methylpentanoyl}amino)(phenyl)ethanoic acid, GLYCEROL, M1 family aminopeptidase, ... | 著者 | Drinkwater, N, McGowan, S. | 登録日 | 2014-11-27 | 公開日 | 2015-02-18 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | X-ray crystal structures of an orally available aminopeptidase inhibitor, Tosedostat, bound to anti-malarial drug targets PfA-M1 and PfA-M17. Proteins, 83, 2015
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4WVM
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![BU of 4wvm by Molmil](/molmil-images/mine/4wvm) | Stonustoxin structure | 分子名称: | Stonustoxin subunit alpha, Stonustoxin subunit beta | 著者 | Ellisdon, A.M, Panjikar, S, Whisstock, J.C, McGowan, S. | 登録日 | 2014-11-06 | 公開日 | 2015-12-02 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Stonefish toxin defines an ancient branch of the perforin-like superfamily. Proc.Natl.Acad.Sci.USA, 112, 2015
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4ZQT
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![BU of 4zqt by Molmil](/molmil-images/mine/4zqt) | Crystal structure of PfA-M1 with virtual ligand inhibitor | 分子名称: | (2R)-2-{[(R)-[(R)-amino(phenyl)methyl](hydroxy)phosphoryl]methyl}-4-methylpentanoic acid, GLYCEROL, M1 family aminopeptidase, ... | 著者 | Ruggeri, C, Drinkwater, N, McGowan, S. | 登録日 | 2015-05-11 | 公開日 | 2015-10-07 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.981 Å) | 主引用文献 | Identification and Validation of a Potent Dual Inhibitor of the P. falciparum M1 and M17 Aminopeptidases Using Virtual Screening. Plos One, 10, 2015
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4R1B
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4R1C
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4R19
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![BU of 4r19 by Molmil](/molmil-images/mine/4r19) | |
4R1A
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4R5V
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![BU of 4r5v by Molmil](/molmil-images/mine/4r5v) | |