5VQD
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![BU of 5vqd by Molmil](/molmil-images/mine/5vqd) | Beta-glucoside phosphorylase BglX | 分子名称: | Beta-glucoside phosphorylase BglX, GLYCEROL | 著者 | Patel, A, Mark, B.L. | 登録日 | 2017-05-08 | 公開日 | 2018-01-17 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Structural and mechanistic analysis of a beta-glycoside phosphorylase identified by screening a metagenomic library. J. Biol. Chem., 293, 2018
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5DN4
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5DN5
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![BU of 5dn5 by Molmil](/molmil-images/mine/5dn5) | Structure of a C-terminally truncated glycoside hydrolase domain from Salmonella typhimurium FlgJ | 分子名称: | CHLORIDE ION, IODIDE ION, Peptidoglycan hydrolase FlgJ, ... | 著者 | Zaloba, P, Bailey-Elkin, B.A, Mark, B.L. | 登録日 | 2015-09-09 | 公開日 | 2016-02-24 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (2.15 Å) | 主引用文献 | Structural and Biochemical Insights into the Peptidoglycan Hydrolase Domain of FlgJ from Salmonella typhimurium. Plos One, 11, 2016
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5FCZ
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5FD0
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4MO4
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![BU of 4mo4 by Molmil](/molmil-images/mine/4mo4) | Crystal structure of AnmK bound to AMPPCP | 分子名称: | Anhydro-N-acetylmuramic acid kinase, PHOSPHOMETHYLPHOSPHONIC ACID ADENYLATE ESTER | 著者 | Bacik, J.P, Mark, B.L. | 登録日 | 2013-09-11 | 公開日 | 2014-01-01 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.67 Å) | 主引用文献 | Conformational Itinerary of Pseudomonas aeruginosa 1,6-Anhydro-N-acetylmuramic Acid Kinase during Its Catalytic Cycle. J.Biol.Chem., 289, 2014
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4MSS
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![BU of 4mss by Molmil](/molmil-images/mine/4mss) | Crystal structure of Burkholderia cenocepacia family 3 glycoside hydrolase (NagZ) bound to (3S,4R,5R,6S)-3-acetamido-4,5,6-trihydroxyazepane | 分子名称: | Beta-hexosaminidase 1, GLYCEROL, N-[(3S,4R,5R,6S)-4,5,6-trihydroxyazepan-3-yl]acetamide | 著者 | Vadlamani, G, Mark, B.L. | 登録日 | 2013-09-18 | 公開日 | 2013-10-30 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Selective trihydroxyazepane NagZ inhibitors increase sensitivity of Pseudomonas aeruginosa to beta-lactams. Chem.Commun.(Camb.), 49, 2013
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8EHO
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![BU of 8eho by Molmil](/molmil-images/mine/8eho) | PRRSV-1 PLP2 domain bound to ubiquitin | 分子名称: | 3-AMINOPROPANE, GLYCEROL, NITRATE ION, ... | 著者 | Bailey-Elkin, B.A, Mark, B.L. | 登録日 | 2022-09-14 | 公開日 | 2023-12-06 | 最終更新日 | 2024-01-03 | 実験手法 | X-RAY DIFFRACTION (2.85 Å) | 主引用文献 | Demonstrating the importance of porcine reproductive and respiratory syndrome virus papain-like protease 2 deubiquitinating activity in viral replication by structure-guided mutagenesis. Plos Pathog., 19, 2023
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8EHN
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![BU of 8ehn by Molmil](/molmil-images/mine/8ehn) | PRRSV-1 PLP2 domain | 分子名称: | ACETATE ION, Papain-like protease 2, ZINC ION | 著者 | Bailey-Elkin, B.A, Mark, B.L. | 登録日 | 2022-09-14 | 公開日 | 2023-12-06 | 最終更新日 | 2024-01-03 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Demonstrating the importance of porcine reproductive and respiratory syndrome virus papain-like protease 2 deubiquitinating activity in viral replication by structure-guided mutagenesis. Plos Pathog., 19, 2023
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4MO5
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![BU of 4mo5 by Molmil](/molmil-images/mine/4mo5) | Crystal structure of AnmK bound to AMPPCP and anhMurNAc | 分子名称: | 2-(2-ACETYLAMINO-4-HYDROXY-6,8-DIOXA-BICYCLO[3.2.1]OCT-3-YLOXY)-PROPIONIC ACID, Anhydro-N-acetylmuramic acid kinase, MAGNESIUM ION, ... | 著者 | Bacik, J.P, Mark, B.L. | 登録日 | 2013-09-11 | 公開日 | 2014-01-01 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Conformational Itinerary of Pseudomonas aeruginosa 1,6-Anhydro-N-acetylmuramic Acid Kinase during Its Catalytic Cycle. J.Biol.Chem., 289, 2014
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8CX9
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![BU of 8cx9 by Molmil](/molmil-images/mine/8cx9) | Structure of the SARS-COV2 PLpro (C111S) in complex with a dimeric Ubv that inhibits activity by an unusual allosteric mechanism | 分子名称: | BROMIDE ION, CHLORIDE ION, Papain-like protease nsp3, ... | 著者 | Singer, A.U, Slater, C.L, Patel, A, Russel, R, Mark, B.L, Sidhu, S.S. | 登録日 | 2022-05-20 | 公開日 | 2023-01-25 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (3.5 Å) | 主引用文献 | Ubiquitin variants potently inhibit SARS-CoV-2 PLpro and viral replication via a novel site distal to the protease active site. Plos Pathog., 18, 2022
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4GYJ
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4GVH
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4GVG
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4GVF
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4GYK
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4GVI
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![BU of 4gvi by Molmil](/molmil-images/mine/4gvi) | Crystal structure of mutant (D248N) Salmonella typhimurium family 3 glycoside hydrolase (NagZ) in complex with GlcNAc-1,6-anhMurNAc | 分子名称: | 2-(2-ACETYLAMINO-4-HYDROXY-6,8-DIOXA-BICYCLO[3.2.1]OCT-3-YLOXY)-PROPIONIC ACID, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Bacik, J.P, Mark, B.L. | 登録日 | 2012-08-30 | 公開日 | 2012-12-19 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Active Site Plasticity within the Glycoside Hydrolase NagZ Underlies a Dynamic Mechanism of Substrate Distortion. Chem.Biol., 19, 2012
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4HZM
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![BU of 4hzm by Molmil](/molmil-images/mine/4hzm) | Crystal structure of Salmonella typhimurium family 3 glycoside hydrolase (NagZ) bound to N-[(3S,4R,5R,6R)-4,5-dihydroxy-6-(hydroxymethyl)piperidin-3-yl]butanamide | 分子名称: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, Beta-hexosaminidase, N-[(3S,4R,5R,6R)-4,5-dihydroxy-6-(hydroxymethyl)piperidin-3-yl]butanamide | 著者 | Bacik, J.P, Mark, B.L. | 登録日 | 2012-11-15 | 公開日 | 2013-06-19 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.45 Å) | 主引用文献 | The Development of Selective Inhibitors of NagZ: Increased Susceptibility of Gram-Negative Bacteria to beta-Lactams. Chembiochem, 14, 2013
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3QBW
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![BU of 3qbw by Molmil](/molmil-images/mine/3qbw) | Crystal structure of pseudomonas aeruginosa 1,6-anhydro-n-actetylmuramic acid kinase (ANMK) bound to adenosine diphosphate | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, Anhydro-N-acetylmuramic acid kinase, SULFATE ION | 著者 | Bacik, J.P, Martin, D.R, Mark, B.L. | 登録日 | 2011-01-14 | 公開日 | 2011-02-02 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.23 Å) | 主引用文献 | Molecular Basis of 1,6-Anhydro Bond Cleavage and Phosphoryl Transfer by Pseudomonas aeruginosa 1,6-Anhydro-N-acetylmuramic Acid Kinase. J.Biol.Chem., 286, 2011
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3QBX
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![BU of 3qbx by Molmil](/molmil-images/mine/3qbx) | Crystal structure of pseudomonas aeruginosa 1,6-anhydro-n-actetylmuramic acid kinase (ANMK) bound to 1,6-anhydro-n-actetylmuramic acid | 分子名称: | 2-(2-ACETYLAMINO-4-HYDROXY-6,8-DIOXA-BICYCLO[3.2.1]OCT-3-YLOXY)-PROPIONIC ACID, Anhydro-N-acetylmuramic acid kinase, SULFATE ION | 著者 | Bacik, J.P, Martin, D.R, Mark, B.L. | 登録日 | 2011-01-14 | 公開日 | 2011-02-02 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Molecular Basis of 1,6-Anhydro Bond Cleavage and Phosphoryl Transfer by Pseudomonas aeruginosa 1,6-Anhydro-N-acetylmuramic Acid Kinase. J.Biol.Chem., 286, 2011
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3PSE
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![BU of 3pse by Molmil](/molmil-images/mine/3pse) | Structure of a viral OTU domain protease bound to interferon-stimulated gene 15 (ISG15) | 分子名称: | 1.7.6 3-bromanylpropan-1-amine, GLYCEROL, RNA polymerase, ... | 著者 | Bacik, J.P, James, T.W, Frias-Staheli, N, Garcia-Sastre, A, Mark, B.L. | 登録日 | 2010-12-01 | 公開日 | 2011-01-19 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Structural basis for the removal of ubiquitin and interferon-stimulated gene 15 by a viral ovarian tumor domain-containing protease. Proc.Natl.Acad.Sci.USA, 108, 2011
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3PT2
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![BU of 3pt2 by Molmil](/molmil-images/mine/3pt2) | Structure of a viral OTU domain protease bound to Ubiquitin | 分子名称: | 1.7.6 3-bromanylpropan-1-amine, ACETATE ION, RNA polymerase, ... | 著者 | James, T.W, Bacik, J.P, Frias-Staheli, N, Garcia-Sastre, A, Mark, B.L. | 登録日 | 2010-12-02 | 公開日 | 2011-01-19 | 最終更新日 | 2023-05-31 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Structural basis for the removal of ubiquitin and interferon-stimulated gene 15 by a viral ovarian tumor domain-containing protease. Proc.Natl.Acad.Sci.USA, 108, 2011
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3GS6
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![BU of 3gs6 by Molmil](/molmil-images/mine/3gs6) | Vibrio Cholerea family 3 glycoside hydrolase (NagZ)in complex with N-butyryl-PUGNAc | 分子名称: | Beta-hexosaminidase, GLYCEROL, [[(3R,4R,5S,6R)-3-(BUTANOYLAMINO)-4,5-DIHYDROXY-6-(HYDROXYMETHYL)OXAN-2-YLIDENE]AMINO] N-PHENYLCARBAMATE | 著者 | Balcewich, M.D, Mark, B.L. | 登録日 | 2009-03-26 | 公開日 | 2009-06-30 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Insight into a strategy for attenuating AmpC-mediated beta-lactam resistance: structural basis for selective inhibition of the glycoside hydrolase NagZ. Protein Sci., 18, 2009
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3GSM
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![BU of 3gsm by Molmil](/molmil-images/mine/3gsm) | Vibrio cholerae family 3 glycoside hydrolase (NagZ) bound to N-Valeryl-PUGNAc | 分子名称: | Beta-hexosaminidase, GLYCEROL, [[(3R,4R,5S,6R)-4,5-dihydroxy-6-(hydroxymethyl)-3-(pentanoylamino)oxan-2-ylidene]amino] N-phenylcarbamate | 著者 | Balcewich, M.D, Mark, B.L. | 登録日 | 2009-03-27 | 公開日 | 2009-06-30 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Insight into a strategy for attenuating AmpC-mediated beta-lactam resistance: structural basis for selective inhibition of the glycoside hydrolase NagZ. Protein Sci., 18, 2009
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2GK1
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![BU of 2gk1 by Molmil](/molmil-images/mine/2gk1) | X-ray crystal structure of NGT-bound HexA | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 3AR,5R,6S,7R,7AR-5-HYDROXYMETHYL-2-METHYL-5,6,7,7A-TETRAHYDRO-3AH-PYRANO[3,2-D]THIAZOLE-6,7-DIOL, Beta-hexosaminidase subunit alpha, ... | 著者 | Lemieux, M.J, Mark, B.L, Cherney, M.M, Withers, S.G, Mahuran, D.J, James, M.N. | 登録日 | 2006-03-31 | 公開日 | 2006-05-30 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (3.25 Å) | 主引用文献 | Crystallographic Structure of Human beta-Hexosaminidase A: Interpretation of Tay-Sachs Mutations and Loss of G(M2) Ganglioside Hydrolysis. J.Mol.Biol., 359, 2006
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