5T02
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![BU of 5t02 by Molmil](/molmil-images/mine/5t02) | Structural characterisation of mutant Asp39Ala of thioesterase (NmACH) from Neisseria meningitidis | 分子名称: | Acyl-CoA hydrolase, CHLORIDE ION, COENZYME A, ... | 著者 | Khandokar, Y.B, Srivastava, P, Forwood, J.K. | 登録日 | 2016-08-15 | 公開日 | 2016-09-07 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Structural insights into GDP-mediated regulation of a bacterial acyl-CoA thioesterase. J. Biol. Chem., 292, 2017
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5SZZ
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![BU of 5szz by Molmil](/molmil-images/mine/5szz) | Novel Structural Insights into GDP-Mediated Regulation of Acyl-CoA Thioesterases | 分子名称: | Acyl-CoA hydrolase, CHLORIDE ION, COENZYME A, ... | 著者 | Khandokar, Y.B, Srivastava, P, Forwood, J.K. | 登録日 | 2016-08-15 | 公開日 | 2016-09-14 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Structural insights into GDP-mediated regulation of a bacterial acyl-CoA thioesterase. J. Biol. Chem., 292, 2017
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5SZV
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![BU of 5szv by Molmil](/molmil-images/mine/5szv) | |
5SZY
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![BU of 5szy by Molmil](/molmil-images/mine/5szy) | Novel Structural Insights into GDP-Mediated Regulation of Acyl-CoA Thioesterases | 分子名称: | Acyl-CoA hydrolase, CHLORIDE ION, COENZYME A, ... | 著者 | Khandokar, Y.B, Srivastava, P, Forwood, J.K. | 登録日 | 2016-08-15 | 公開日 | 2016-09-14 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structural insights into GDP-mediated regulation of a bacterial acyl-CoA thioesterase. J. Biol. Chem., 292, 2017
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6SDG
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![BU of 6sdg by Molmil](/molmil-images/mine/6sdg) | |
7DK1
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![BU of 7dk1 by Molmil](/molmil-images/mine/7dk1) | Crystal structure of Zinc bound SARS-CoV-2 main protease | 分子名称: | 2-[BIS-(2-HYDROXY-ETHYL)-AMINO]-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, 3C-like proteinase, CHLORIDE ION, ... | 著者 | Sonkar, K.S, Panchariya, L, Kuila, S, Khan, W.A, Arockiasamy, A. | 登録日 | 2020-11-22 | 公開日 | 2021-06-30 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.902 Å) | 主引用文献 | Zinc 2+ ion inhibits SARS-CoV-2 main protease and viral replication in vitro. Chem.Commun.(Camb.), 57, 2021
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5XMB
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![BU of 5xmb by Molmil](/molmil-images/mine/5xmb) | Mycobacterium tuberculosis Pantothenate kinase mutant F247A | 分子名称: | Pantothenate kinase, SULFATE ION | 著者 | Paul, A, Kumar, P, Surolia, A, Vijayan, M. | 登録日 | 2017-05-13 | 公開日 | 2018-05-16 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (3.2 Å) | 主引用文献 | Biochemical and structural studies of mutants indicate concerted movement of the dimer interface and ligand-binding region of Mycobacterium tuberculosis pantothenate kinase Acta Crystallogr F Struct Biol Commun, 73, 2017
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8P09
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![BU of 8p09 by Molmil](/molmil-images/mine/8p09) | 48S late-stage initiation complex with non methylated mRNA | 分子名称: | 18S ribosomal RNA, 40S ribosomal protein S11, 40S ribosomal protein S12, ... | 著者 | Guca, E, Lima, L.H.F, Boissier, F, Hashem, Y. | 登録日 | 2023-05-09 | 公開日 | 2024-03-20 | 実験手法 | ELECTRON MICROSCOPY (3.3 Å) | 主引用文献 | N 6 -methyladenosine in 5' UTR does not promote translation initiation. Mol.Cell, 84, 2024
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8P03
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![BU of 8p03 by Molmil](/molmil-images/mine/8p03) | 48S late-stage initiation complex with m6A mRNA | 分子名称: | 18S ribosomal RNA, 40S ribosomal protein S11, 40S ribosomal protein S12, ... | 著者 | Guca, E, Lima, L.H.F, Boissier, F, Hashem, Y. | 登録日 | 2023-05-09 | 公開日 | 2024-03-20 | 最終更新日 | 2024-04-24 | 実験手法 | ELECTRON MICROSCOPY (3.04 Å) | 主引用文献 | N 6 -methyladenosine in 5' UTR does not promote translation initiation. Mol.Cell, 84, 2024
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5WYE
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![BU of 5wye by Molmil](/molmil-images/mine/5wye) | |
8FTQ
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![BU of 8ftq by Molmil](/molmil-images/mine/8ftq) | Crystal structure of hRpn13 Pru domain in complex with Ubiquitin and XL44 | 分子名称: | N-(3-{[(3R)-5-fluoro-2-oxo-2,3-dihydro-1H-indol-3-yl]methyl}phenyl)-4-methoxybenzamide, Proteasomal ubiquitin receptor ADRM1, Ubiquitin | 著者 | Walters, K.J, Lu, X, Chandravanshi, M. | 登録日 | 2023-01-13 | 公開日 | 2024-03-27 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | A structure-based designed small molecule depletes hRpn13 Pru and a select group of KEN box proteins. Nat Commun, 15, 2024
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5DNI
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![BU of 5dni by Molmil](/molmil-images/mine/5dni) | Crystal structure of Methanocaldococcus jannaschii Fumarate hydratase beta subunit | 分子名称: | 1,2-ETHANEDIOL, CHLORIDE ION, DI(HYDROXYETHYL)ETHER, ... | 著者 | Jayaraman, V, Kunala, J, Balaram, H. | 登録日 | 2015-09-10 | 公開日 | 2016-09-14 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Revisiting the Burden Borne by Fumarase: Enzymatic Hydration of an Olefin. Biochemistry, 62, 2023
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3MJW
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![BU of 3mjw by Molmil](/molmil-images/mine/3mjw) | PI3 Kinase gamma with a benzofuranone inhibitor | 分子名称: | (2Z)-4,6-dihydroxy-2-[(8-methoxy-1,2,3,4-tetrahydropyrazino[1,2-a]indol-10-yl)methylidene]-1-benzofuran-3(2H)-one, Phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit gamma isoform | 著者 | Bard, J, Svenson, K. | 登録日 | 2010-04-13 | 公開日 | 2010-06-09 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.87 Å) | 主引用文献 | 5-Ureidobenzofuranone indoles as potent and efficacious inhibitors of PI3 kinase-alpha and mTOR for the treatment of breast cancer. Bioorg.Med.Chem.Lett., 20, 2010
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7WVL
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![BU of 7wvl by Molmil](/molmil-images/mine/7wvl) | |
5V3A
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![BU of 5v3a by Molmil](/molmil-images/mine/5v3a) | |
2IVX
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![BU of 2ivx by Molmil](/molmil-images/mine/2ivx) | Crystal structure of human cyclin T2 at 1.8 A resolution | 分子名称: | 1,2-ETHANEDIOL, CYCLIN-T2 | 著者 | Debreczeni, J.E, Bullock, A.N, Fedorov, O, Savitsky, P, Berridge, G, Das, S, Pike, A.C.W, Turnbull, A, Ugochukwu, E, Papagrigoriou, E, Gorrec, F, Sundstrom, M, Edwards, A, Arrowsmith, C, Weigelt, J, von Delft, F, Knapp, S. | 登録日 | 2006-06-21 | 公開日 | 2006-07-19 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | The structure of P-TEFb (CDK9/cyclin T1), its complex with flavopiridol and regulation by phosphorylation. EMBO J., 27, 2008
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7D40
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![BU of 7d40 by Molmil](/molmil-images/mine/7d40) | |
7D95
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![BU of 7d95 by Molmil](/molmil-images/mine/7d95) | |
2A3K
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![BU of 2a3k by Molmil](/molmil-images/mine/2a3k) | Crystal Structure of the Human Protein Tyrosine Phosphatase, PTPN7 (HePTP, Hematopoietic Protein Tyrosine Phosphatase) | 分子名称: | PHOSPHATE ION, protein tyrosine phosphatase, non-receptor type 7, ... | 著者 | Barr, A, Turnbull, A.P, Das, S, Eswaran, J, Debreczeni, J.E, Longmann, E, Smee, C, Burgess, N, Gileadi, O, Sundstrom, M, Arrowsmith, C, Edwards, A, von Delft, F, Knapp, S, Structural Genomics Consortium (SGC) | 登録日 | 2005-06-24 | 公開日 | 2005-07-19 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (2.55 Å) | 主引用文献 | The crystal structure of human receptor protein tyrosine phosphatase kappa phosphatase domain 1. Protein Sci., 15, 2006
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2GJT
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![BU of 2gjt by Molmil](/molmil-images/mine/2gjt) | Crystal structure of the human receptor phosphatase PTPRO | 分子名称: | CHLORIDE ION, Receptor-type tyrosine-protein phosphatase PTPRO | 著者 | Barr, A, Ugochukwu, E, Eswaran, J, Das, S, Niesen, F, Savitsky, P, Turnbull, A, Sundstrom, M, Arrowsmith, C, Edwards, A, Weigelt, J, von Delft, F, Papagrigoriou, E, Knapp, S, Structural Genomics Consortium (SGC) | 登録日 | 2006-03-31 | 公開日 | 2006-05-02 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2.15 Å) | 主引用文献 | Large-scale structural analysis of the classical human protein tyrosine phosphatome. Cell(Cambridge,Mass.), 136, 2009
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7D96
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![BU of 7d96 by Molmil](/molmil-images/mine/7d96) | |
7D97
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![BU of 7d97 by Molmil](/molmil-images/mine/7d97) | |
2JJD
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![BU of 2jjd by Molmil](/molmil-images/mine/2jjd) | Protein Tyrosine Phosphatase, Receptor Type, E isoform | 分子名称: | CHLORIDE ION, RECEPTOR-TYPE TYROSINE-PROTEIN PHOSPHATASE EPSILON | 著者 | Elkins, J.M, Ugochukwu, E, Alfano, I, Barr, A.J, Bunkoczi, G, King, O.N.F, Filippakopoulos, P, Savitsky, P, Salah, E, Pike, A, Johansson, C, Das, S, Burgess-Brown, N.A, Gileadi, O, von Delft, F, Arrowsmith, C.H, Bountra, C, Edwards, A.M, Knapp, S. | 登録日 | 2008-03-31 | 公開日 | 2008-04-08 | 最終更新日 | 2012-06-06 | 実験手法 | X-RAY DIFFRACTION (3.2 Å) | 主引用文献 | Large-Scale Structural Analysis of the Classical Human Protein Tyrosine Phosphatome. Cell(Cambridge,Mass.), 136, 2009
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2H4V
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![BU of 2h4v by Molmil](/molmil-images/mine/2h4v) | Crystal Structure of the Human Tyrosine Receptor Phosphatase Gamma | 分子名称: | 1,2-ETHANEDIOL, ACETATE ION, CHLORIDE ION, ... | 著者 | Ugochukwu, E, Barr, A, Das, S, Eswaran, J, Savitsky, P, Sundstrom, M, Edwards, A, Arrowsmith, C, Weigelt, J, Debreczeni, J, von Delft, F, Knapp, S, Structural Genomics Consortium (SGC) | 登録日 | 2006-05-25 | 公開日 | 2006-07-11 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Large-scale structural analysis of the classical human protein tyrosine phosphatome. Cell(Cambridge,Mass.), 136, 2009
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2I75
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![BU of 2i75 by Molmil](/molmil-images/mine/2i75) | Crystal Structure of Human Protein Tyrosine Phosphatase N4 (PTPN4) | 分子名称: | SULFATE ION, Tyrosine-protein phosphatase non-receptor type 4 | 著者 | Ugochukwu, E, Barr, A, Savitsky, P, Burgess, N, Das, S, Turnbull, A, von Delft, F, Sundstrom, M, Edwards, A, Arrowsmith, C, Weigelt, J, Knapp, S, Structural Genomics Consortium (SGC) | 登録日 | 2006-08-30 | 公開日 | 2006-10-17 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2.45 Å) | 主引用文献 | Large-scale structural analysis of the classical human protein tyrosine phosphatome. Cell(Cambridge,Mass.), 136, 2009
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