6SEO
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![BU of 6seo by Molmil](/molmil-images/mine/6seo) | TEAD4 bound to a FAM181B peptide | 分子名称: | Protein FAM181B, Transcriptional enhancer factor TEF-3 | 著者 | Scheufler, C, Villard, F. | 登録日 | 2019-07-30 | 公開日 | 2019-11-20 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (2.55 Å) | 主引用文献 | Identification of FAM181A and FAM181B as new interactors with the TEAD transcription factors. Protein Sci., 29, 2020
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6SEN
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![BU of 6sen by Molmil](/molmil-images/mine/6sen) | TEAD4 bound to a FAM181A peptide | 分子名称: | Protein FAM181A, SULFATE ION, Transcriptional enhancer factor TEF-3 | 著者 | Scheufler, C, Villard, F. | 登録日 | 2019-07-30 | 公開日 | 2019-11-20 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.65 Å) | 主引用文献 | Identification of FAM181A and FAM181B as new interactors with the TEAD transcription factors. Protein Sci., 29, 2020
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6D2I
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![BU of 6d2i by Molmil](/molmil-images/mine/6d2i) | JAK2 Pseudokinase V617F in complex with AT9283 | 分子名称: | 1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1H-benzimidazol-2-yl]-1H-pyrazol-4-yl}urea, Tyrosine-protein kinase | 著者 | Li, Q, Li, K, Eck, M.J. | 登録日 | 2018-04-13 | 公開日 | 2019-03-20 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (3.192 Å) | 主引用文献 | Discovery and Structural Characterization of ATP-Site Ligands for the Wild-Type and V617F Mutant JAK2 Pseudokinase Domain. ACS Chem. Biol., 14, 2019
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3SD5
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![BU of 3sd5 by Molmil](/molmil-images/mine/3sd5) | Crystal Structure of PI3K gamma with 5-(2,4-dimorpholinopyrimidin-6-yl)-4-(trifluoromethyl)pyridin-2-amine | 分子名称: | 5-[2,6-di(morpholin-4-yl)pyrimidin-4-yl]-4-(trifluoromethyl)pyridin-2-amine, Phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit gamma isoform | 著者 | Knapp, M.S, Elling, R.A. | 登録日 | 2011-06-08 | 公開日 | 2012-01-04 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (3.2 Å) | 主引用文献 | Identification and Characterization of NVP-BKM120, an Orally Available Pan-Class I PI3-Kinase Inhibitor. Mol.Cancer Ther., 11, 2012
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6Q9L
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![BU of 6q9l by Molmil](/molmil-images/mine/6q9l) | |
6Q9U
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![BU of 6q9u by Molmil](/molmil-images/mine/6q9u) | HDMX (14-111; C17S) COMPLEXED WITH COMPOUND 12 AT 2.4A; Structural states of Hdm2 and HdmX: X-ray elucidation of adaptations and binding interactions for different chemical compound classes | 分子名称: | 1,4,7,10,13,16-HEXAOXACYCLOOCTADECANE, 4-[(4~{S})-5-(5-chloranyl-2-oxidanylidene-1~{H}-pyridin-3-yl)-2-[2-(dimethylamino)-4-methoxy-pyrimidin-5-yl]-6-oxidanylidene-3-propan-2-yl-4~{H}-pyrrolo[3,4-c]pyrazol-4-yl]benzenecarbonitrile, CHLORIDE ION, ... | 著者 | Kallen, J. | 登録日 | 2018-12-18 | 公開日 | 2019-05-15 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Structural States of Hdm2 and HdmX: X-ray Elucidation of Adaptations and Binding Interactions for Different Chemical Compound Classes. Chemmedchem, 14, 2019
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6Q9O
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![BU of 6q9o by Molmil](/molmil-images/mine/6q9o) | |
6Q9Q
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![BU of 6q9q by Molmil](/molmil-images/mine/6q9q) | HDMX (14-111; C17S) COMPLEXED WITH COMPOUND 13 AT 2.1A; Structural states of Hdm2 and HdmX: X-ray elucidation of adaptations and binding interactions for different chemical compound classes | 分子名称: | 1,4,7,10,13,16-HEXAOXACYCLOOCTADECANE, 6-chloranyl-3-[3-[(1~{S})-1-(4-chlorophenyl)ethyl]-5-phenyl-imidazol-4-yl]-~{N}-[2-(4-cyclohexylpiperazin-1-yl)ethyl]-1~{H}-indole-2-carboxamide, GLYCEROL, ... | 著者 | Kallen, J. | 登録日 | 2018-12-18 | 公開日 | 2019-05-15 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Structural States of Hdm2 and HdmX: X-ray Elucidation of Adaptations and Binding Interactions for Different Chemical Compound Classes. Chemmedchem, 14, 2019
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6Q9W
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![BU of 6q9w by Molmil](/molmil-images/mine/6q9w) | X-ray structure of compound 15 bound to HdmX: Structural states of Hdm2 and HdmX: X-ray elucidation of adaptations and binding interactions for different chemical compound classes | 分子名称: | (4~{S})-4-(4-chlorophenyl)-5-[(1~{S})-1-(3-chlorophenyl)ethyl]-2-(2,4-dimethoxypyrimidin-5-yl)-3-propan-2-yl-4~{H}-pyrrolo[3,4-d]imidazol-6-one, 1,4,7,10,13,16-HEXAOXACYCLOOCTADECANE, Protein Mdm4, ... | 著者 | Kallen, J. | 登録日 | 2018-12-18 | 公開日 | 2019-05-15 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Structural States of Hdm2 and HdmX: X-ray Elucidation of Adaptations and Binding Interactions for Different Chemical Compound Classes. Chemmedchem, 14, 2019
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6Q9H
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![BU of 6q9h by Molmil](/molmil-images/mine/6q9h) | |
6Q9Y
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![BU of 6q9y by Molmil](/molmil-images/mine/6q9y) | |
6Q9S
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![BU of 6q9s by Molmil](/molmil-images/mine/6q9s) | HDMX (14-111; C17S) COMPLEXED WITH COMPOUND 14 AT 2.4A: Structural states of Hdm2 and HdmX: X-ray elucidation of adaptations and binding interactions for different chemical compound classes | 分子名称: | 1,4,7,10,13,16-HEXAOXACYCLOOCTADECANE, 3-[[6-chloranyl-3-[3-[(1~{S})-1-(2,4-dichlorophenyl)ethyl]-5-phenyl-imidazol-4-yl]-1~{H}-indol-2-yl]carbonylamino]-4-[4-(2-oxidanylidene-1,3-oxazinan-3-yl)piperidin-1-yl]benzoic acid, Protein Mdm4, ... | 著者 | Kallen, J. | 登録日 | 2018-12-18 | 公開日 | 2019-05-15 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Structural States of Hdm2 and HdmX: X-ray Elucidation of Adaptations and Binding Interactions for Different Chemical Compound Classes. Chemmedchem, 14, 2019
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6Q96
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![BU of 6q96 by Molmil](/molmil-images/mine/6q96) | |
6Q36
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![BU of 6q36 by Molmil](/molmil-images/mine/6q36) | |
6Q2X
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![BU of 6q2x by Molmil](/molmil-images/mine/6q2x) | |
6GE6
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![BU of 6ge6 by Molmil](/molmil-images/mine/6ge6) | |
6GE4
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![BU of 6ge4 by Molmil](/molmil-images/mine/6ge4) | |
6GE5
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![BU of 6ge5 by Molmil](/molmil-images/mine/6ge5) | |
6GEC
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![BU of 6gec by Molmil](/molmil-images/mine/6gec) | |
6GEI
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![BU of 6gei by Molmil](/molmil-images/mine/6gei) | |
6GE3
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![BU of 6ge3 by Molmil](/molmil-images/mine/6ge3) | |
6GEE
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![BU of 6gee by Molmil](/molmil-images/mine/6gee) | |
6GEG
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![BU of 6geg by Molmil](/molmil-images/mine/6geg) | |
6GEK
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![BU of 6gek by Molmil](/molmil-images/mine/6gek) | |
5WIN
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![BU of 5win by Molmil](/molmil-images/mine/5win) | JAK2 Pseudokinase in complex with JNJ7706621 | 分子名称: | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1H-1,2,4-triazol-3-yl}amino)benzenesulfonamide, Tyrosine-protein kinase JAK2 | 著者 | Li, Q, Eck, M.J, Li, K, Park, E. | 登録日 | 2017-07-19 | 公開日 | 2018-08-01 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2.38 Å) | 主引用文献 | Discovery and Structural Characterization of ATP-Site Ligands for the Wild-Type and V617F Mutant JAK2 Pseudokinase Domain. ACS Chem. Biol., 14, 2019
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