5XV9
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![BU of 5xv9 by Molmil](/molmil-images/mine/5xv9) | |
4WHK
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![BU of 4whk by Molmil](/molmil-images/mine/4whk) | A New Class of Peptidomimetics Targeting the Polo-box Domain of Polo-like kinase 1 | 分子名称: | C6H5(CH2)8-DERIVATIZED PEPTIDE INHIBITOR, Serine/threonine-protein kinase PLK1 | 著者 | Bang, J.K, Han, Y.H, Ahn, M.J, Lee, K.S. | 登録日 | 2014-09-23 | 公開日 | 2014-12-03 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | A new class of peptidomimetics targeting the polo-box domain of polo-like kinase 1. J.Med.Chem., 58, 2015
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4WHL
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![BU of 4whl by Molmil](/molmil-images/mine/4whl) | A New Class of Peptidomimetics Targeting the Polo-box Domain of Polo-like kinase 1 | 分子名称: | C6H5(CH2)8-DERIVATIZED PEPTIDE INHIBITOR, Serine/threonine-protein kinase PLK1 | 著者 | Bang, J.K, Han, Y.H, Ahn, M.J, Lee, K.S. | 登録日 | 2014-09-23 | 公開日 | 2014-12-03 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.71 Å) | 主引用文献 | A new class of peptidomimetics targeting the polo-box domain of polo-like kinase 1. J.Med.Chem., 58, 2015
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4WHH
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![BU of 4whh by Molmil](/molmil-images/mine/4whh) | |
2M17
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![BU of 2m17 by Molmil](/molmil-images/mine/2m17) | |
1YLA
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![BU of 1yla by Molmil](/molmil-images/mine/1yla) | Ubiquitin-conjugating enzyme E2-25 kDa (Huntington interacting protein 2) | 分子名称: | Ubiquitin-conjugating enzyme E2-25 kDa | 著者 | Choe, J, Avvakumov, G.V, Newman, E.M, Mackenzie, F, Kozieradzki, I, Bochkarev, A, Sundstrom, M, Arrowsmith, C, Edwards, A, Dhe-paganon, S, Structural Genomics Consortium (SGC) | 登録日 | 2005-01-19 | 公開日 | 2005-02-01 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Structural basis of E2-25K/UBB+1 interaction leading to proteasome inhibition and neurotoxicity J.Biol.Chem., 285, 2010
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2CKX
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![BU of 2ckx by Molmil](/molmil-images/mine/2ckx) | |
4RCP
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![BU of 4rcp by Molmil](/molmil-images/mine/4rcp) | Crystal structure of Plk1 Polo-box domain in complex with PL-2 | 分子名称: | 1,2-ETHANEDIOL, PL-2, Serine/threonine-protein kinase PLK1 | 著者 | Lee, W.C, Song, J.H, Kim, H.Y. | 登録日 | 2014-09-16 | 公開日 | 2014-11-12 | 最終更新日 | 2015-01-21 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | A new class of peptidomimetics targeting the polo-box domain of polo-like kinase 1. J.Med.Chem., 58, 2015
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4HAB
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![BU of 4hab by Molmil](/molmil-images/mine/4hab) | Crystal structure of Plk1 Polo-box domain in complex with PL-49 | 分子名称: | 3-CYCLOHEXYL-1-PROPYLSULFONIC ACID, PHOSPHATE ION, PL-49, ... | 著者 | Lee, W.C, Song, J.H, Kim, H.Y. | 登録日 | 2012-09-26 | 公開日 | 2013-04-03 | 最終更新日 | 2022-12-21 | 実験手法 | X-RAY DIFFRACTION (2.65 Å) | 主引用文献 | Development of cyclic peptomer inhibitors targeting the polo-box domain of polo-like kinase 1. Bioorg.Med.Chem., 21, 2013
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4HY2
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![BU of 4hy2 by Molmil](/molmil-images/mine/4hy2) | |
3TD5
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![BU of 3td5 by Molmil](/molmil-images/mine/3td5) | Crystal structure of OmpA-like domain from Acinetobacter baumannii in complex with L-Ala-gamma-D-Glu-m-DAP-D-Ala-D-Ala | 分子名称: | CHLORIDE ION, Outer membrane protein omp38, peptide(L-Ala-gamma-D-Glu-m-DAP-D-Ala-D-Ala) | 著者 | Park, J.S, Lee, W.C, Song, J.H, Kim, H.Y. | 登録日 | 2011-08-10 | 公開日 | 2011-10-26 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Mechanism of anchoring of OmpA protein to the cell wall peptidoglycan of the gram-negative bacterial outer membrane Faseb J., 26, 2012
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3TD4
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![BU of 3td4 by Molmil](/molmil-images/mine/3td4) | Crystal structure of OmpA-like domain from Acinetobacter baumannii in complex with diaminopimelate | 分子名称: | 2,6-DIAMINOPIMELIC ACID, Outer membrane protein omp38 | 著者 | Park, J.S, Lee, W.C, Song, J.H, Kim, H.Y. | 登録日 | 2011-08-10 | 公開日 | 2011-10-26 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.79 Å) | 主引用文献 | Mechanism of anchoring of OmpA protein to the cell wall peptidoglycan of the gram-negative bacterial outer membrane Faseb J., 26, 2012
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3TD3
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![BU of 3td3 by Molmil](/molmil-images/mine/3td3) | Crystal structure of OmpA-like domain from Acinetobacter baumannii in complex with glycine | 分子名称: | GLYCINE, Outer membrane protein omp38 | 著者 | Park, J.S, Lee, W.C, Song, J.H, Kim, H.Y. | 登録日 | 2011-08-10 | 公開日 | 2011-10-26 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (1.59 Å) | 主引用文献 | Mechanism of anchoring of OmpA protein to the cell wall peptidoglycan of the gram-negative bacterial outer membrane Faseb J., 26, 2012
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3GWJ
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![BU of 3gwj by Molmil](/molmil-images/mine/3gwj) | Crystal structure of Antheraea pernyi arylphorin | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Arylphorin, FORMIC ACID, ... | 著者 | Ryu, K.S, Lee, J.O, Kwon, T.H, Kim, S. | 登録日 | 2009-04-01 | 公開日 | 2009-05-05 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2.43 Å) | 主引用文献 | The presence of monoglucosylated N196-glycan is important for the structural stability of storage protein, arylphorin Biochem.J., 421, 2009
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3IKW
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![BU of 3ikw by Molmil](/molmil-images/mine/3ikw) | Structure of Heparinase I from Bacteroides thetaiotaomicron | 分子名称: | 1,2-ETHANEDIOL, CALCIUM ION, Heparin lyase I | 著者 | Garron, M.L, Cygler, M, Shaya, D. | 登録日 | 2009-08-06 | 公開日 | 2009-09-29 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.3 Å) | 主引用文献 | Structural snapshots of heparin depolymerization by heparin lyase I. J.Biol.Chem., 284, 2009
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3IMN
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![BU of 3imn by Molmil](/molmil-images/mine/3imn) | |
3ILR
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![BU of 3ilr by Molmil](/molmil-images/mine/3ilr) | Structure of Heparinase I from Bacteroides thetaiotaomicron in complex with tetrasaccharide product | 分子名称: | 1,2-ETHANEDIOL, 2-deoxy-6-O-sulfo-2-(sulfoamino)-alpha-D-glucopyranose-(4-1)-4-deoxy-2-O-sulfo-beta-D-erythro-hex-4-enopyranuronic acid, 4-deoxy-2-O-sulfo-beta-D-erythro-hex-4-enopyranuronic acid-(1-4)-2-deoxy-6-O-sulfo-2-(sulfoamino)-alpha-D-glucopyranose, ... | 著者 | Garron, M.L, Cygler, M, Shaya, D. | 登録日 | 2009-08-07 | 公開日 | 2009-09-29 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Structural snapshots of heparin depolymerization by heparin lyase I. J.Biol.Chem., 284, 2009
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3INA
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![BU of 3ina by Molmil](/molmil-images/mine/3ina) | Crystal structure of heparin lyase I H151A mutant complexed with a dodecasaccharide heparin | 分子名称: | 2-deoxy-6-O-sulfo-2-(sulfoamino)-alpha-D-glucopyranose-(1-4)-2-O-sulfo-alpha-L-idopyranuronic acid-(1-4)-2-deoxy-3,6-di-O-sulfo-2-(sulfoamino)-alpha-D-glucopyranose-(1-4)-2-O-sulfo-alpha-L-idopyranuronic acid-(1-4)-2-deoxy-6-O-sulfo-2-(sulfoamino)-alpha-D-glucopyranose-(1-4)-2-O-sulfo-alpha-L-idopyranuronic acid-(1-4)-2-deoxy-6-O-sulfo-2-(sulfoamino)-alpha-D-glucopyranose-(1-4)-2-O-sulfo-alpha-L-idopyranuronic acid, CALCIUM ION, Heparin lyase I | 著者 | Han, Y.H, Ryu, K.S, Kim, H.Y, Jeon, Y.H. | 登録日 | 2009-08-12 | 公開日 | 2009-09-29 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structural snapshots of heparin depolymerization by heparin lyase I J.Biol.Chem., 284, 2009
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3IN9
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![BU of 3in9 by Molmil](/molmil-images/mine/3in9) | Crystal structure of heparin lyase I complexed with disaccharide heparin | 分子名称: | 4-deoxy-2-O-sulfo-alpha-L-threo-hex-4-enopyranuronic acid-(1-4)-2-deoxy-6-O-sulfo-2-(sulfoamino)-alpha-D-glucopyranose, CALCIUM ION, Heparin lyase I | 著者 | Han, Y.H, Ryu, K.S, Kim, H.Y, Jeon, Y.H. | 登録日 | 2009-08-12 | 公開日 | 2009-09-29 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structural snapshots of heparin depolymerization by heparin lyase I J.Biol.Chem., 284, 2009
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3K9P
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![BU of 3k9p by Molmil](/molmil-images/mine/3k9p) | The crystal structure of E2-25K and ubiquitin complex | 分子名称: | Ubiquitin, Ubiquitin-conjugating enzyme E2 K | 著者 | Kang, G.B, Ko, S, Song, S.M, Lee, W, Eom, S.H. | 登録日 | 2009-10-16 | 公開日 | 2010-09-08 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Structural basis of E2-25K/UBB+1 interaction leading to proteasome inhibition and neurotoxicity J.Biol.Chem., 285, 2010
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2NX8
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![BU of 2nx8 by Molmil](/molmil-images/mine/2nx8) | |
4LKM
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![BU of 4lkm by Molmil](/molmil-images/mine/4lkm) | Crystal structure of Plk1 Polo-box domain in complex with PL-74 | 分子名称: | GLYCEROL, PL-74, SULFATE ION, ... | 著者 | Lee, W.C, Song, J.H, Kim, H.Y. | 登録日 | 2013-07-08 | 公開日 | 2013-12-11 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Exploring the binding nature of pyrrolidine pocket-dependent interactions in the polo-box domain of polo-like kinase 1 Plos One, 8, 2013
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4LKL
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![BU of 4lkl by Molmil](/molmil-images/mine/4lkl) | |
2HQO
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![BU of 2hqo by Molmil](/molmil-images/mine/2hqo) | |
2HQN
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![BU of 2hqn by Molmil](/molmil-images/mine/2hqn) | |