Loading
PDBj
メニューPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help
Search by PDB author
9FBY
DownloadVisualize
BU of 9fby by Molmil
N-TERMINAL BROMODOMAIN OF HUMAN BRD4 with (5-(4-chloro-1-((tetrahydro-2H-pyran-4-yl)methyl)-1H-imidazol-2-yl)-1,3-dimethylpyridin-2(1H)-one
分子名称: 1,2-ETHANEDIOL, 5-[4-chloranyl-1-(oxan-4-ylmethyl)imidazol-2-yl]-1,3-dimethyl-pyridin-2-one, Bromodomain-containing protein 4
著者Chung, C.
登録日2024-05-14
公開日2024-06-26
実験手法X-RAY DIFFRACTION (1.853 Å)
主引用文献Structure- and Property-Based Optimization of Efficient Pan-Bromodomain and Extra Terminal Inhibitors to Identify Oral and Intravenous Candidate I-BET787.
J.Med.Chem., 2024
1UNL
DownloadVisualize
BU of 1unl by Molmil
Structural mechanism for the inhibition of CD5-p25 from the roscovitine, aloisine and indirubin.
分子名称: CYCLIN-DEPENDENT KINASE 5, CYCLIN-DEPENDENT KINASE 5 ACTIVATOR 1, R-ROSCOVITINE
著者Mapelli, M, Crovace, C, Massimiliano, L, Musacchio, A.
登録日2003-09-10
公開日2004-11-10
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Mechanism of Cdk5/P25 Binding by Cdk Inhibitors
J.Med.Chem., 48, 2005
9FBX
DownloadVisualize
BU of 9fbx by Molmil
C-TERMINAL BROMODOMAIN OF HUMAN BRD2 WITH 5-(1-benzyl-4-chloro-1H-imidazol-2-yl)-1,3-dimethylpyridin-2(1H)-one
分子名称: 1,2-ETHANEDIOL, 2-{2-[2-(2-{2-[2-(2-ETHOXY-ETHOXY)-ETHOXY]-ETHOXY}-ETHOXY)-ETHOXY]-ETHOXY}-ETHANOL, 5-(1-benzyl-4-chloro-1H-imidazol-2-yl)-1,3-dimethylpyridin-2(1H)-one, ...
著者Chung, C.
登録日2024-05-14
公開日2024-06-26
実験手法X-RAY DIFFRACTION (1.602 Å)
主引用文献Structure- and Property-Based Optimization of Efficient Pan-Bromodomain and Extra Terminal Inhibitors to Identify Oral and Intravenous Candidate I-BET787.
J.Med.Chem., 2024
1AGX
DownloadVisualize
BU of 1agx by Molmil
REFINED CRYSTAL STRUCTURE OF ACINETOBACTER GLUTAMINASIFICANS GLUTAMINASE-ASPARAGINASE
分子名称: GLUTAMINASE-ASPARAGINASE
著者Lubkowski, J, Wlodawer, A, Housset, D, Weber, I.T, Ammon, H.L, Murphy, K.C, Swain, A.L.
登録日1994-07-13
公開日1994-12-20
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Refined crystal structure of Acinetobacter glutaminasificans glutaminase-asparaginase.
Acta Crystallogr.,Sect.D, 50, 1994
6USY
DownloadVisualize
BU of 6usy by Molmil
COAGULATION FACTOR XI CATALYTIC DOMAIN (C123S) IN COMPLEX WITH NVP-XIV936
分子名称: 1-[(2S)-2-{3-[(3S)-3-amino-2,3-dihydro-1-benzofuran-5-yl]-5-(propan-2-yl)phenyl}-2-hydroxyethyl]-1H-indole-7-carboxylic acid, Coagulation factor XIa light chain
著者Weihofen, W.A, Clark, K, Nunes, S.
登録日2019-10-28
公開日2020-07-01
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (1.26 Å)
主引用文献Structure-Based Design and Preclinical Characterization of Selective and Orally Bioavailable Factor XIa Inhibitors: Demonstrating the Power of an Integrated S1 Protease Family Approach.
J.Med.Chem., 63, 2020
6RK3
DownloadVisualize
BU of 6rk3 by Molmil
Solution structure of the ribosome Elongation Factor P (EF-P) from Staphylococcus aureus
分子名称: Elongation factor P
著者Usachev, K, Fatkhullin, B, Gabdulkhakov, A, Khusainov, I, Golubev, A, Validov, S, Yusupova, G, Yusupov, M.
登録日2019-04-30
公開日2020-03-11
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献NMR and crystallographic structural studies of the Elongation factor P from Staphylococcus aureus.
Eur.Biophys.J., 49, 2020
6RJI
DownloadVisualize
BU of 6rji by Molmil
X-ray structure of the elongation factor P of S. aureus
分子名称: Elongation factor P
著者Fatkhullin, B.F, Golubev, A.A, Gabdulkhakov, A.G, Khusainov, I.S, Validov, S.Z, Usachev, K.S, Yusupova, G, Yusupov, M.M.
登録日2019-04-27
公開日2020-04-01
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.48 Å)
主引用文献NMR and crystallographic structural studies of the Elongation factor P from Staphylococcus aureus.
Eur.Biophys.J., 49, 2020
1UNH
DownloadVisualize
BU of 1unh by Molmil
Structural mechanism for the inhibition of CDK5-p25 by roscovitine, aloisine and indirubin.
分子名称: (Z)-1H,1'H-[2,3']BIINDOLYLIDENE-3,2'-DIONE-3-OXIME, CYCLIN-DEPENDENT KINASE 5, CYCLIN-DEPENDENT KINASE 5 ACTIVATOR 1
著者Mapelli, M, Crovace, C, Massimiliano, L, Musacchio, A.
登録日2003-09-10
公開日2004-11-10
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.35 Å)
主引用文献Mechanism of Cdk5/P25 Binding by Cdk Inhibitors
J.Med.Chem., 48, 2005
1UNG
DownloadVisualize
BU of 1ung by Molmil
Structural mechanism for the inhibition of CDK5-p25 by roscovitine, aloisine and indirubin.
分子名称: 6-PHENYL[5H]PYRROLO[2,3-B]PYRAZINE, CELL DIVISION PROTEIN KINASE 5, CYCLIN-DEPENDENT KINASE 5 ACTIVATOR 1
著者Mapelli, M, Crovace, C, Massimiliano, L, Musacchio, A.
登録日2003-09-10
公開日2004-11-10
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Mechanism of Cdk5/P25 Binding by Cdk Inhibitors
J.Med.Chem., 48, 2005
8BIG
DownloadVisualize
BU of 8big by Molmil
O-Methyltransferase Plu4895 in complex with SAH
分子名称: 1,2-ETHANEDIOL, CHLORIDE ION, MAGNESIUM ION, ...
著者Huber, E.M, Groll, M.
登録日2022-11-02
公開日2023-03-08
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献A set of closely related methyltransferases for site-specific tailoring of anthraquinone pigments.
Structure, 31, 2023
8BGT
DownloadVisualize
BU of 8bgt by Molmil
O-Methyltransferase Plu4890 in complex with SAM
分子名称: GLYCEROL, Methyltransferase Plu4890, S-ADENOSYLMETHIONINE, ...
著者Huber, E.M, Groll, M.
登録日2022-10-28
公開日2023-03-08
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献A set of closely related methyltransferases for site-specific tailoring of anthraquinone pigments.
Structure, 31, 2023
8BGY
DownloadVisualize
BU of 8bgy by Molmil
O-Methyltransferase Plu4890 in complex with SAH and AQ-284a
分子名称: 1,3-dimethoxy-8-oxidanyl-anthracene-9,10-dione, CHLORIDE ION, Methyltransferase Plu4890, ...
著者Huber, E.M, Groll, M.
登録日2022-10-28
公開日2023-03-08
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献A set of closely related methyltransferases for site-specific tailoring of anthraquinone pigments.
Structure, 31, 2023
8BH0
DownloadVisualize
BU of 8bh0 by Molmil
O-Methyltransferase Plu4890 in complex with SAH and AQ-270b
分子名称: 3-methoxy-1,8-bis(oxidanyl)anthracene-9,10-dione, CHLORIDE ION, Methyltransferase Plu4890, ...
著者Huber, E.M, Groll, M.
登録日2022-10-28
公開日2023-03-08
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献A set of closely related methyltransferases for site-specific tailoring of anthraquinone pigments.
Structure, 31, 2023
8BIB
DownloadVisualize
BU of 8bib by Molmil
O-Methyltransferase Plu4890 in complex with SAH and AQ-256
分子名称: 1,3,8-tris(oxidanyl)anthracene-9,10-dione, CARBONATE ION, CHLORIDE ION, ...
著者Huber, E.M, Groll, M.
登録日2022-11-02
公開日2023-03-08
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献A set of closely related methyltransferases for site-specific tailoring of anthraquinone pigments.
Structure, 31, 2023
8BIE
DownloadVisualize
BU of 8bie by Molmil
O-Methyltransferase Plu4894 in complex with SAH
分子名称: S-ADENOSYL-L-HOMOCYSTEINE, methyltransferase Plu4894
著者Huber, E.M, Groll, M.
登録日2022-11-02
公開日2023-03-08
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献A set of closely related methyltransferases for site-specific tailoring of anthraquinone pigments.
Structure, 31, 2023
8BII
DownloadVisualize
BU of 8bii by Molmil
O-Methyltransferase Plu4895 (mutant H229N) in complex with SAH
分子名称: CHLORIDE ION, S-ADENOSYL-L-HOMOCYSTEINE, methyltransferase Plu4895 H229N mutant
著者Huber, E.M, Groll, M.
登録日2022-11-02
公開日2023-03-08
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献A set of closely related methyltransferases for site-specific tailoring of anthraquinone pigments.
Structure, 31, 2023
8BIJ
DownloadVisualize
BU of 8bij by Molmil
O-Methyltransferase Plu4894 (mutant I88M, W91L, C97Y, S142L, G146V, Y258M, L270F, S309Y) in complex with SAH
分子名称: 1,2-ETHANEDIOL, CHLORIDE ION, Methyltransferase Plu4894 mutant I88M, ...
著者Huber, E.M, Groll, M.
登録日2022-11-02
公開日2023-03-08
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.55 Å)
主引用文献A set of closely related methyltransferases for site-specific tailoring of anthraquinone pigments.
Structure, 31, 2023
8BIC
DownloadVisualize
BU of 8bic by Molmil
O-Methyltransferase Plu4891 in complex with SAH
分子名称: GLYCEROL, S-ADENOSYL-L-HOMOCYSTEINE, SODIUM ION, ...
著者Huber, E.M, Groll, M.
登録日2022-11-02
公開日2023-03-08
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献A set of closely related methyltransferases for site-specific tailoring of anthraquinone pigments.
Structure, 31, 2023
8BIR
DownloadVisualize
BU of 8bir by Molmil
O-Methyltransferase Plu4895 in complex with SAH and AQ-256
分子名称: 1,3,8-tris(oxidanyl)anthracene-9,10-dione, CHLORIDE ION, IODIDE ION, ...
著者Huber, E.M, Groll, M.
登録日2022-11-02
公開日2023-03-08
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献A set of closely related methyltransferases for site-specific tailoring of anthraquinone pigments.
Structure, 31, 2023
8BGZ
DownloadVisualize
BU of 8bgz by Molmil
O-Methyltransferase Plu4890 (mutant H229N) in complex with SAH and AQ-256
分子名称: 1,3,8-tris(oxidanyl)anthracene-9,10-dione, GLYCEROL, S-ADENOSYL-L-HOMOCYSTEINE, ...
著者Huber, E.M, Groll, M.
登録日2022-10-28
公開日2023-03-08
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献A set of closely related methyltransferases for site-specific tailoring of anthraquinone pigments.
Structure, 31, 2023
8BGX
DownloadVisualize
BU of 8bgx by Molmil
O-Methyltransferase Plu4890 in complex with SAH and AQ-270a
分子名称: 1-methoxy-3,8-bis(oxidanyl)anthracene-9,10-dione, CHLORIDE ION, GLYCEROL, ...
著者Huber, E.M, Groll, M.
登録日2022-10-28
公開日2023-03-08
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献A set of closely related methyltransferases for site-specific tailoring of anthraquinone pigments.
Structure, 31, 2023
8BIH
DownloadVisualize
BU of 8bih by Molmil
O-Methyltransferase Plu4890 in complex with SAH and AQ-284b
分子名称: 3,8-dimethoxy-1-oxidanyl-anthracene-9,10-dione, CHLORIDE ION, GLYCEROL, ...
著者Huber, E.M, Groll, M.
登録日2022-11-02
公開日2023-03-08
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献A set of closely related methyltransferases for site-specific tailoring of anthraquinone pigments.
Structure, 31, 2023
8BIF
DownloadVisualize
BU of 8bif by Molmil
O-Methyltransferase Plu4892 in complex with SAH
分子名称: 1,2-ETHANEDIOL, CHLORIDE ION, S-ADENOSYL-L-HOMOCYSTEINE, ...
著者Huber, E.M, Groll, M.
登録日2022-11-02
公開日2023-03-08
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献A set of closely related methyltransferases for site-specific tailoring of anthraquinone pigments.
Structure, 31, 2023
8BID
DownloadVisualize
BU of 8bid by Molmil
O-Methyltransferase Plu4890 (mutant H229N) in complex with SAH and AQ-270a
分子名称: 1-methoxy-3,8-bis(oxidanyl)anthracene-9,10-dione, CHLORIDE ION, GLYCEROL, ...
著者Huber, E.M, Groll, M.
登録日2022-11-02
公開日2023-03-08
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献A set of closely related methyltransferases for site-specific tailoring of anthraquinone pigments.
Structure, 31, 2023
7RSA
DownloadVisualize
BU of 7rsa by Molmil
STRUCTURE OF PHOSPHATE-FREE RIBONUCLEASE A REFINED AT 1.26 ANGSTROMS
分子名称: RIBONUCLEASE A, TERTIARY-BUTYL ALCOHOL
著者Wlodawer, A, Gilliland, G.L.
登録日1988-06-10
公開日1988-10-09
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.26 Å)
主引用文献Structure of phosphate-free ribonuclease A refined at 1.26 A.
Biochemistry, 27, 1988

221716

件を2024-06-26に公開中

PDB statisticsPDBj update infoContact PDBjnumon