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8JT9
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BU of 8jt9 by Molmil
Human VMAT2 complex with ketanserin
分子名称: 3-[2-[4-(4-fluorophenyl)carbonylpiperidin-1-yl]ethyl]-1~{H}-quinazoline-2,4-dione, Synaptic vesicular amine transporter
著者Jiang, D.H, Wu, D.
登録日2023-06-21
公開日2023-11-29
最終更新日2024-02-21
実験手法ELECTRON MICROSCOPY (2.97 Å)
主引用文献Transport and inhibition mechanisms of human VMAT2.
Nature, 626, 2024
5K8H
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BU of 5k8h by Molmil
The X-ray crystal structure of a parallel poly(rA) double helix generated by rA7 at acidic pH
分子名称: AMMONIUM ION, RNA 7-mer
著者Gleghorn, M.L, Maquat, L.E.
登録日2016-05-30
公開日2016-07-06
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.069 Å)
主引用文献Crystal structure of a poly(rA) staggered zipper at acidic pH: evidence that adenine N1 protonation mediates parallel double helix formation.
Nucleic Acids Res., 44, 2016
8H08
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BU of 8h08 by Molmil
SARS-CoV-2 BA.1 variants S ectodomain trimer in complex with neutralizing antibody 10-5B and 6-2C
分子名称: 10-5B H chain, 10-5B L chain, 2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Wang, X, Wang, Z.
登録日2022-09-28
公開日2023-05-31
実験手法ELECTRON MICROSCOPY (3.2 Å)
主引用文献Inactivated vaccine-elicited potent antibodies can broadly neutralize SARS-CoV-2 circulating variants.
Nat Commun, 14, 2023
8H07
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BU of 8h07 by Molmil
SARS-CoV-2 BA.4 variants S ectodomain trimer in complex with neutralizing antibody 10-5B and 6-2C
分子名称: 10-5B H chain, 10-5B L chain, 2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Wang, X, Wang, Z.
登録日2022-09-28
公開日2023-05-31
実験手法ELECTRON MICROSCOPY (2.9 Å)
主引用文献Inactivated vaccine-elicited potent antibodies can broadly neutralize SARS-CoV-2 circulating variants.
Nat Commun, 14, 2023
6S4Q
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BU of 6s4q by Molmil
scdSav(SASK) - Engineering Single-Chain Dimeric Streptavidin as Host for Artificial Metalloenzymes
分子名称: GLYCEROL, Streptavidin, {N-(4-{[2-(amino-kappaN)ethyl]sulfamoyl-kappaN}phenyl)-5-[(3aS,4S,6aR)-2-oxohexahydro-1H-thieno[3,4-d]imidazol-4-yl]pentanamide}(chloro)[(1,2,3,4,5-eta)-1,2,3,4,5-pentamethylcyclopentadienyl]iridium(III)
著者Rebelein, J.G.
登録日2019-06-28
公開日2019-09-25
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Breaking Symmetry: Engineering Single-Chain Dimeric Streptavidin as Host for Artificial Metalloenzymes.
J.Am.Chem.Soc., 141, 2019
6S50
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BU of 6s50 by Molmil
scdSav(SARK)mv2 - Engineering Single-Chain Dimeric Streptavidin as Host for Artificial Metalloenzymes
分子名称: GLYCEROL, SULFATE ION, Streptavidin, ...
著者Rebelein, J.G.
登録日2019-06-29
公開日2019-09-25
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Breaking Symmetry: Engineering Single-Chain Dimeric Streptavidin as Host for Artificial Metalloenzymes.
J.Am.Chem.Soc., 141, 2019
5Y6P
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BU of 5y6p by Molmil
Structure of the phycobilisome from the red alga Griffithsia pacifica
分子名称: ApcD, ApcF, LC, ...
著者Zhang, J, Ma, J.F, Liu, D.S, Sun, S, Sui, S.F.
登録日2017-08-13
公開日2017-11-15
実験手法ELECTRON MICROSCOPY (3.5 Å)
主引用文献Structure of phycobilisome from the red alga Griffithsia pacifica
Nature, 551, 2017
1I7E
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BU of 1i7e by Molmil
C-Terminal Domain Of Mouse Brain Tubby Protein bound to Phosphatidylinositol 4,5-bis-phosphate
分子名称: L-ALPHA-GLYCEROPHOSPHO-D-MYO-INOSITOL-4,5-BIS-PHOSPHATE, TUBBY PROTEIN
著者Santagata, S, Boggon, T.J, Baird, C.L, Shan, W.S, Shapiro, L.
登録日2001-03-08
公開日2001-06-27
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献G-protein signaling through tubby proteins.
Science, 292, 2001
7YUD
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BU of 7yud by Molmil
FTY720p-bound human SPNS2
分子名称: (2~{S})-2-azanyl-4-(4-octylphenyl)-2-[[oxidanyl-bis(oxidanylidene)-$l^{6}-phosphanyl]oxymethyl]butan-1-ol, NbFab L-chain, NbFab-H-chain, ...
著者He, Y, Duan, Y.
登録日2022-08-17
公開日2023-09-06
最終更新日2024-02-21
実験手法ELECTRON MICROSCOPY (2.98 Å)
主引用文献Structural basis of Sphingosine-1-phosphate transport via human SPNS2.
Cell Res., 34, 2024
7YUB
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BU of 7yub by Molmil
S1P-bound human SPNS2
分子名称: (2S,3R,4E)-2-amino-3-hydroxyoctadec-4-en-1-yl dihydrogen phosphate, NbFab-H-chain, NbFab-L-chain, ...
著者He, Y, Duan, Y.
登録日2022-08-17
公開日2023-09-06
最終更新日2024-02-21
実験手法ELECTRON MICROSCOPY (3.22 Å)
主引用文献Structural basis of Sphingosine-1-phosphate transport via human SPNS2.
Cell Res., 34, 2024
7YUF
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BU of 7yuf by Molmil
apo human SPNS2
分子名称: NbFab H-chain, NbFab L-chain, Sphingosine-1-phosphate transporter SPNS2, ...
著者He, Y, Duan, Y.
登録日2022-08-17
公開日2023-09-06
最終更新日2024-02-21
実験手法ELECTRON MICROSCOPY (3.29 Å)
主引用文献Structural basis of Sphingosine-1-phosphate transport via human SPNS2.
Cell Res., 34, 2024
6BAW
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BU of 6baw by Molmil
Structure of GRP94 with a selective resorcinylic inhibitor.
分子名称: 1,2-ETHANEDIOL, Endoplasmin, PHOSPHATE ION, ...
著者Que, N.L.S, Gewirth, D.T.
登録日2017-10-16
公開日2018-04-18
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2.703 Å)
主引用文献Structure Based Design of a Grp94-Selective Inhibitor: Exploiting a Key Residue in Grp94 To Optimize Paralog-Selective Binding.
J. Med. Chem., 61, 2018
6CEO
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BU of 6ceo by Molmil
Structure of Hsp90 NTD with a GRP94-selective resorcinylic inhibitor.
分子名称: 1,2-ETHANEDIOL, Heat shock protein HSP 90-alpha, MAGNESIUM ION, ...
著者Que, N.L.S, Gewirth, D.T.
登録日2018-02-12
公開日2018-04-18
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (1.896 Å)
主引用文献Structure Based Design of a Grp94-Selective Inhibitor: Exploiting a Key Residue in Grp94 To Optimize Paralog-Selective Binding.
J. Med. Chem., 61, 2018
6C91
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BU of 6c91 by Molmil
Structure of GRP94 with a resorcinylic inhibitor.
分子名称: 1,2-ETHANEDIOL, 5-[2-(1-benzyl-1H-imidazol-2-yl)ethyl]-4,6-dichlorobenzene-1,3-diol, Endoplasmin, ...
著者Que, N.L.S, Gewirth, D.T.
登録日2018-01-25
公開日2018-04-18
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2.895 Å)
主引用文献Structure Based Design of a Grp94-Selective Inhibitor: Exploiting a Key Residue in Grp94 To Optimize Paralog-Selective Binding.
J. Med. Chem., 61, 2018
7DAV
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BU of 7dav by Molmil
The native crystal structure of COVID-19 main protease
分子名称: COVID-19 MAIN PROTEASE
著者He, Z.S, He, B, Cao, P, Jiang, H.D, Gong, Y, Gao, X.Y.
登録日2020-10-18
公開日2021-11-03
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.77 Å)
主引用文献A comparison of Remdesivir versus gold cluster in COVID-19 animal model: A better therapeutic outcome of gold cluster.
Nano Today, 44, 2022
7DAU
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BU of 7dau by Molmil
The crystal structure of COVID-19 main protease treated by GA
分子名称: COVID-19 MAIN PROTEASE, GOLD ION
著者He, Z.S, He, B, Cao, P, Jiang, H.D, Gong, Y, Gao, X.Y.
登録日2020-10-18
公開日2021-11-03
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.72 Å)
主引用文献A comparison of Remdesivir versus gold cluster in COVID-19 animal model: A better therapeutic outcome of gold cluster.
Nano Today, 44, 2022
7DAT
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BU of 7dat by Molmil
The crystal structure of COVID-19 main protease treated by AF
分子名称: COVID-19 MAIN PROTEASE, GOLD ION
著者He, Z.S, He, B, Cao, P, Jiang, H.D, Gong, Y, Gao, X.Y.
登録日2020-10-18
公開日2021-11-03
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.75 Å)
主引用文献A comparison of Remdesivir versus gold cluster in COVID-19 animal model: A better therapeutic outcome of gold cluster.
Nano Today, 44, 2022
6K7P
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BU of 6k7p by Molmil
Crystal structure of human AFF4-THD domain
分子名称: AF4/FMR2 family member 4
著者Tang, D, Xue, Y, Li, S, Cheng, W, Duan, J, Wang, J, Qi, S.
登録日2019-06-08
公開日2020-03-11
最終更新日2024-03-27
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structural and functional insight into the effect of AFF4 dimerization on activation of HIV-1 proviral transcription.
Cell Discov, 6, 2020
8JGU
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BU of 8jgu by Molmil
Crystal structure of N-terminal domain of exopolyphosphatase from Deinococcus radiodurans
分子名称: Exopolyphosphatase, SODIUM ION
著者Zhao, Y, Dai, S.
登録日2023-05-21
公開日2024-05-15
実験手法X-RAY DIFFRACTION (1.99 Å)
主引用文献Structural Evolution of Bacterial Polyphosphate Degradation Enzyme for Phosphorus Cycling.
Adv Sci, 2024
8JGR
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BU of 8jgr by Molmil
Crystal structure of Deinococcus radiodurans exopolyphosphatase in the presence of Pi
分子名称: Exopolyphosphatase, PHOSPHATE ION, POTASSIUM ION
著者Zhao, Y, Dai, S.
登録日2023-05-21
公開日2024-05-15
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structural Evolution of Bacterial Polyphosphate Degradation Enzyme for Phosphorus Cycling.
Adv Sci, 2024
8JGW
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BU of 8jgw by Molmil
Crystal structure of Klebsiella pneumoniae exopolyphosphatase
分子名称: Exopolyphosphatase, GLYCEROL, MAGNESIUM ION, ...
著者Zhao, Y, Dai, S.
登録日2023-05-21
公開日2024-05-15
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Structural Evolution of Bacterial Polyphosphate Degradation Enzyme for Phosphorus Cycling.
Adv Sci, 2024
8JGX
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BU of 8jgx by Molmil
Crystal structure of Acinetobacter baumannii exopolyphosphatase
分子名称: Exopolyphosphatase
著者Zhao, Y, Dai, S.
登録日2023-05-21
公開日2024-05-15
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Structural Evolution of Bacterial Polyphosphate Degradation Enzyme for Phosphorus Cycling.
Adv Sci, 2024
8JGT
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BU of 8jgt by Molmil
Crystal structure of Deinococcus radiodurans exopolyphosphatase E114A mutant
分子名称: Exopolyphosphatase, MAGNESIUM ION, SULFATE ION
著者Zhao, Y, Dai, S.
登録日2023-05-21
公開日2024-05-15
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structural Evolution of Bacterial Polyphosphate Degradation Enzyme for Phosphorus Cycling.
Adv Sci, 2024
8JGP
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BU of 8jgp by Molmil
Crystal structure of Deinococcus radiodurans exopolyphosphatase complexed with pyrophosphate
分子名称: Exopolyphosphatase, MANGANESE (II) ION, PHOSPHATE ION, ...
著者Zhao, Y, Dai, S.
登録日2023-05-21
公開日2024-05-15
実験手法X-RAY DIFFRACTION (3.02 Å)
主引用文献Structural Evolution of Bacterial Polyphosphate Degradation Enzyme for Phosphorus Cycling.
Adv Sci, 2024
8JGO
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BU of 8jgo by Molmil
Crystal structure of Deinococcus radiodurans exopolyphosphatase
分子名称: Exopolyphosphatase, MAGNESIUM ION, SULFATE ION
著者Zhao, Y, Dai, S.
登録日2023-05-21
公開日2024-05-15
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structural Evolution of Bacterial Polyphosphate Degradation Enzyme for Phosphorus Cycling.
Adv Sci, 2024

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