6DBU
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![BU of 6dbu by Molmil](/molmil-images/mine/6dbu) | Cryo-EM structure of RAG in complex with 12-RSS and 23-RSS substrate DNAs | 分子名称: | CALCIUM ION, Forward strand RSS substrate DNA, Recombination activating gene 1 - MBP chimera, ... | 著者 | Wu, H, Liao, M, Ru, H, Mi, W. | 登録日 | 2018-05-03 | 公開日 | 2018-08-01 | 最終更新日 | 2024-03-13 | 実験手法 | ELECTRON MICROSCOPY (3.9 Å) | 主引用文献 | DNA melting initiates the RAG catalytic pathway. Nat. Struct. Mol. Biol., 25, 2018
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6DBI
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![BU of 6dbi by Molmil](/molmil-images/mine/6dbi) | Cryo-EM structure of RAG in complex with 12-RSS and 23-RSS nicked DNA intermediates | 分子名称: | CALCIUM ION, Forward strand of 12-RSS signal end, Forward strand of 23-RSS signal end, ... | 著者 | Wu, H, Liao, M, Ru, H, Mi, W. | 登録日 | 2018-05-03 | 公開日 | 2018-08-01 | 最終更新日 | 2024-03-13 | 実験手法 | ELECTRON MICROSCOPY (3.4 Å) | 主引用文献 | DNA melting initiates the RAG catalytic pathway. Nat. Struct. Mol. Biol., 25, 2018
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6DEF
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![BU of 6def by Molmil](/molmil-images/mine/6def) | Vps1 GTPase-BSE fusion complexed with GMPPCP | 分子名称: | MAGNESIUM ION, PHOSPHOMETHYLPHOSPHONIC ACID GUANYLATE ESTER, Vps1 GTPase-BSE | 著者 | Ford, M.G.J, Varlakhanova, N.V, Brady, T.M, Chappie, J.S, Hosford, C.J. | 登録日 | 2018-05-11 | 公開日 | 2018-08-22 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2.26 Å) | 主引用文献 | Structures of the fungal dynamin-related protein Vps1 reveal a unique, open helical architecture. J. Cell Biol., 217, 2018
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6DBJ
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![BU of 6dbj by Molmil](/molmil-images/mine/6dbj) | Cryo-EM structure of RAG in complex with 12-RSS and 23-RSS nicked DNA intermediates | 分子名称: | CALCIUM ION, Forward stand of RSS signal end, Forward strand of coding flank, ... | 著者 | Wu, H, Liao, M, Ru, H, Mi, W. | 登録日 | 2018-05-03 | 公開日 | 2018-08-01 | 最終更新日 | 2024-03-13 | 実験手法 | ELECTRON MICROSCOPY (3 Å) | 主引用文献 | DNA melting initiates the RAG catalytic pathway. Nat. Struct. Mol. Biol., 25, 2018
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6KMH
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![BU of 6kmh by Molmil](/molmil-images/mine/6kmh) | The crystal structure of CASK/Mint1 complex | 分子名称: | Amyloid-beta A4 precursor protein-binding family A member 1, CHLORIDE ION, IODIDE ION, ... | 著者 | Li, W, Feng, W. | 登録日 | 2019-07-31 | 公開日 | 2020-08-05 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | CASK modulates the assembly and function of the Mint1/Munc18-1 complex to regulate insulin secretion. Cell Discov, 6, 2020
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7XR5
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![BU of 7xr5 by Molmil](/molmil-images/mine/7xr5) | Crystal structure of imine reductase with NAPDH from Streptomyces albidoflavus | 分子名称: | 3,6,9,12,15,18,21,24,27,30,33,36,39,42,45,48,51,54,57-nonadecaoxanonapentacontane-1,59-diol, 6-phosphogluconate dehydrogenase NAD-binding, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE | 著者 | Zhang, J, Chen, R.C, Gao, S.S. | 登録日 | 2022-05-09 | 公開日 | 2022-10-19 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (1.58 Å) | 主引用文献 | Actinomycetes-derived imine reductases with a preference towards bulky amine substrates. Commun Chem, 5, 2022
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1B4P
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![BU of 1b4p by Molmil](/molmil-images/mine/1b4p) | CRYSTAL STRUCTURES OF CLASS MU CHIMERIC GST ISOENZYMES M1-2 AND M2-1 | 分子名称: | L-gamma-glutamyl-S-[(9S,10S)-10-hydroxy-9,10-dihydrophenanthren-9-yl]-L-cysteinylglycine, PROTEIN (GLUTATHIONE S-TRANSFERASE), SULFATE ION | 著者 | Xiao, G, Chen, J, Armstrong, R.N, Gilliland, G.L. | 登録日 | 1998-12-26 | 公開日 | 2003-07-08 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Crystal Structures of Class MU Chimeric GST Isoenzymes M1-2 and M2-1 To be Published
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8BSL
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![BU of 8bsl by Molmil](/molmil-images/mine/8bsl) | Human GLS in complex with compound 12 | 分子名称: | Glutaminase kidney isoform, mitochondrial, ~{N}-[5-[[(3~{R})-1-(5-azanyl-1,3,4-thiadiazol-2-yl)pyrrolidin-3-yl]amino]-1,3,4-thiadiazol-2-yl]-2-phenyl-ethanamide | 著者 | Debreczeni, J.E. | 登録日 | 2022-11-25 | 公開日 | 2023-01-18 | 最終更新日 | 2024-06-19 | 実験手法 | X-RAY DIFFRACTION (2.38 Å) | 主引用文献 | Discovery of a Thiadiazole-Pyridazine-Based Allosteric Glutaminase 1 Inhibitor Series That Demonstrates Oral Bioavailability and Activity in Tumor Xenograft Models. J Med Chem, 62, 2019
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6VBQ
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6VBO
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![BU of 6vbo by Molmil](/molmil-images/mine/6vbo) | |
6VBP
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7RE9
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![BU of 7re9 by Molmil](/molmil-images/mine/7re9) | TCR mimic antibody (Fab fragment) | 分子名称: | DI(HYDROXYETHYL)ETHER, Fab heavy chain, Fab light chain | 著者 | Dasgupta, M, Baker, B.M. | 登録日 | 2021-07-12 | 公開日 | 2022-07-27 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.77 Å) | 主引用文献 | Validation and promise of a TCR mimic antibody for cancer immunotherapy of hepatocellular carcinoma. Sci Rep, 12, 2022
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7RE8
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![BU of 7re8 by Molmil](/molmil-images/mine/7re8) | |
7RE7
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![BU of 7re7 by Molmil](/molmil-images/mine/7re7) | |
6OLU
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![BU of 6olu by Molmil](/molmil-images/mine/6olu) | RIAM RA-PH core structure in the P212121 space group | 分子名称: | Amyloid beta A4 precursor protein-binding family B member 1-interacting protein | 著者 | Wu, J. | 登録日 | 2019-04-17 | 公開日 | 2020-04-22 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Phosphorylation of RIAM by src promotes integrin activation by unmasking the PH domain of RIAM. Structure, 29, 2021
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6O6H
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![BU of 6o6h by Molmil](/molmil-images/mine/6o6h) | RIAM cc-RA-PH structure in the P21212 space group | 分子名称: | Amyloid beta A4 precursor protein-binding family B member 1-interacting protein | 著者 | Wu, J. | 登録日 | 2019-03-06 | 公開日 | 2020-09-02 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Phosphorylation of RIAM by Src Promotes Integrin Activation by Unmasking the PH Domain of RIAM. Structure, 2020
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6SB1
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![BU of 6sb1 by Molmil](/molmil-images/mine/6sb1) | Crystal structure of murine perforin-2 P2 domain crystal form 1 | 分子名称: | CHLORIDE ION, GLYCEROL, Macrophage-expressed gene 1 protein | 著者 | Ni, T, Ginger, L, Gilbert, R.J.C. | 登録日 | 2019-07-18 | 公開日 | 2020-02-05 | 最終更新日 | 2020-02-26 | 実験手法 | X-RAY DIFFRACTION (2.05 Å) | 主引用文献 | Structure and mechanism of bactericidal mammalian perforin-2, an ancient agent of innate immunity. Sci Adv, 6, 2020
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6SB3
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6SB4
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![BU of 6sb4 by Molmil](/molmil-images/mine/6sb4) | Crystal structure of murine perforin-2 P2 domain crystal form 2 | 分子名称: | Macrophage-expressed gene 1 protein | 著者 | Ni, T, Yu, X, Ginger, L, Gilbert, R.J.C. | 登録日 | 2019-07-18 | 公開日 | 2020-02-05 | 最終更新日 | 2020-02-26 | 実験手法 | X-RAY DIFFRACTION (3.17 Å) | 主引用文献 | Structure and mechanism of bactericidal mammalian perforin-2, an ancient agent of innate immunity. Sci Adv, 6, 2020
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6SB5
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5U1F
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![BU of 5u1f by Molmil](/molmil-images/mine/5u1f) | Initial contact of HIV-1 Env with CD4: Cryo-EM structure of BG505 DS-SOSIP trimer in complex with CD4 and antibody PGT145 | 分子名称: | BG505 DS-SOSIP gp120, BG505 SOSIP gp41, PGT145 heavy chain, ... | 著者 | Acharya, P, Kwong, P.D, Potter, C.S, Carragher, B. | 登録日 | 2016-11-28 | 公開日 | 2017-02-22 | 最終更新日 | 2018-10-03 | 実験手法 | ELECTRON MICROSCOPY (6.8 Å) | 主引用文献 | Quaternary contact in the initial interaction of CD4 with the HIV-1 envelope trimer. Nat. Struct. Mol. Biol., 24, 2017
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8JT6
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![BU of 8jt6 by Molmil](/molmil-images/mine/8jt6) | 5-HT1A-Gi in complex with compound (R)-IHCH-7179 | 分子名称: | 1-(4-fluorophenyl)-4-[(7R)-2,5,11-triazatetracyclo[7.6.1.0^2,7.0^12,16]hexadeca-1(15),9,12(16),13-tetraen-5-yl]butan-1-one, CHOLESTEROL, Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2, ... | 著者 | Chen, Z, Xu, P, Huang, S, Xu, H.E, Wang, S. | 登録日 | 2023-06-21 | 公開日 | 2024-02-28 | 最終更新日 | 2024-05-08 | 実験手法 | ELECTRON MICROSCOPY (3 Å) | 主引用文献 | Flexible scaffold-based cheminformatics approach for polypharmacological drug design. Cell, 187, 2024
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2QN1
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![BU of 2qn1 by Molmil](/molmil-images/mine/2qn1) | Glycogen Phosphorylase b in complex with asiatic acid | 分子名称: | Glycogen phosphorylase, muscle form, asiatic acid | 著者 | Zographos, S.E, Leonidas, D.D, Alexacou, K.-M, Hayes, J, Oikonomakos, N.G. | 登録日 | 2007-07-17 | 公開日 | 2008-06-03 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.401 Å) | 主引用文献 | Naturally occurring pentacyclic triterpenes as inhibitors of glycogen phosphorylase: synthesis, structure-activity relationships, and X-ray crystallographic studies J.Med.Chem., 51, 2008
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2QN2
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![BU of 2qn2 by Molmil](/molmil-images/mine/2qn2) | Glycogen Phosphorylase b in complex with Maslinic Acid | 分子名称: | Glycogen phosphorylase, muscle form, maslinic acid | 著者 | Zographos, S.E, Leonidas, D.D, Alexacou, K.-M, Hayes, J, Oikonomakos, N.G. | 登録日 | 2007-07-17 | 公開日 | 2008-06-03 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.698 Å) | 主引用文献 | Naturally occurring pentacyclic triterpenes as inhibitors of glycogen phosphorylase: synthesis, structure-activity relationships, and X-ray crystallographic studies J.Med.Chem., 51, 2008
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6NNJ
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