1W96
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![BU of 1w96 by Molmil](/molmil-images/mine/1w96) | Crystal Structure of Biotin Carboxylase Domain of Acetyl-coenzyme A Carboxylase from Saccharomyces cerevisiae in Complex with Soraphen A | Descriptor: | ACETYL-COENZYME A CARBOXYLASE, SORAPHEN A | Authors: | Shen, Y, Volrath, S.L, Weatherly, S.C, Elich, T.D, Tong, L. | Deposit date: | 2004-10-06 | Release date: | 2005-01-04 | Last modified: | 2024-05-08 | Method: | X-RAY DIFFRACTION (1.8 Å) | Cite: | A Mechanism for the Potent Inhibition of Eukaryotic Acetyl-Coenzyme a Carboxylase by Soraphen A, a Macrocyclic Polyketide Natural Product Mol.Cell, 16, 2004
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4WZ8
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3K8X
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![BU of 3k8x by Molmil](/molmil-images/mine/3k8x) | Crystal structure of the carboxyltransferase domain of acetyl-coenzyme A carboxylase in complex with tepraloxydim | Descriptor: | (5S)-2-[(1E)-N-{[(2E)-3-chloroprop-2-en-1-yl]oxy}propanimidoyl]-3-hydroxy-5-(tetrahydro-2H-pyran-4-yl)cyclohex-2-en-1-one, Acetyl-CoA carboxylase | Authors: | Xiang, S, Callaghan, M.M, Watson, K.G, Tong, L. | Deposit date: | 2009-10-15 | Release date: | 2009-12-01 | Last modified: | 2024-02-21 | Method: | X-RAY DIFFRACTION (2.3 Å) | Cite: | A different mechanism for the inhibition of the carboxyltransferase domain of acetyl-coenzyme A carboxylase by tepraloxydim. Proc.Natl.Acad.Sci.USA, 106, 2009
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5CTE
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![BU of 5cte by Molmil](/molmil-images/mine/5cte) | |
5CTB
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![BU of 5ctb by Molmil](/molmil-images/mine/5ctb) | |
3TVU
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![BU of 3tvu by Molmil](/molmil-images/mine/3tvu) | Crystal Structure of the humanized carboxyltransferase domain of yeast Acetyl-coA caroxylase in complex with compound 3 | Descriptor: | 4-({4-[(2-methylquinolin-6-yl)methyl]piperidin-1-yl}carbonyl)-2-phenylquinoline, Acetyl-CoA carboxylase | Authors: | Rajamohan, F, Marr, E, Reyes, A, Landro, J.A, Anderson, M.D, Corbett, J.W, Dirico, K.J, Harwood, J.H, Tu, M, Vajdos, F.F. | Deposit date: | 2011-09-20 | Release date: | 2011-10-19 | Last modified: | 2023-09-13 | Method: | X-RAY DIFFRACTION (2.4 Å) | Cite: | Structure-guided Inhibitor Design for Human Acetyl-coenzyme A Carboxylase by Interspecies Active Site Conversion. J.Biol.Chem., 286, 2011
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3H0S
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![BU of 3h0s by Molmil](/molmil-images/mine/3h0s) | |
3H0Q
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1UYR
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![BU of 1uyr by Molmil](/molmil-images/mine/1uyr) | |
5CS0
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![BU of 5cs0 by Molmil](/molmil-images/mine/5cs0) | |
1UYT
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![BU of 1uyt by Molmil](/molmil-images/mine/1uyt) | Acetyl-CoA carboxylase carboxyltransferase domain | Descriptor: | ACETYL-COA CARBOXYLASE | Authors: | Zhang, H, Tweel, B, Tong, L. | Deposit date: | 2004-03-02 | Release date: | 2004-03-29 | Last modified: | 2024-05-08 | Method: | X-RAY DIFFRACTION (2.5 Å) | Cite: | Molecular Basis for the Inhibition of the Carboxyltransferase Domain of Acetyl-Coenzyme-A Carboxylase by Haloxyfop and Diclofop. Proc.Natl.Acad.Sci.USA, 101, 2004
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1W93
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![BU of 1w93 by Molmil](/molmil-images/mine/1w93) | Crystal Structure of Biotin Carboxylase Domain of Acetyl-Coenzyme A Carboxylase from Saccharomyces cerevisiae | Descriptor: | ACETYL-COENZYME A CARBOXYLASE | Authors: | Shen, Y, Volrath, S.L, Weatherly, S.C, Elich, T.D, Tong, L. | Deposit date: | 2004-10-05 | Release date: | 2005-01-04 | Last modified: | 2024-05-08 | Method: | X-RAY DIFFRACTION (2.5 Å) | Cite: | A Mechanism for the Potent Inhibition of Eukaryotic Acetyl-Coenzyme a Carboxylase by Soraphen A, a Macrocyclic Polyketide Natural Product Mol.Cell, 16, 2004
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1UYV
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![BU of 1uyv by Molmil](/molmil-images/mine/1uyv) | |
5CTC
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3TZ3
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![BU of 3tz3 by Molmil](/molmil-images/mine/3tz3) | Crystal Structure of the humanized carboxyltransferase domain of yeast Acetyl-coA caroxylase in complex with compound 2 | Descriptor: | 6-{[1-(anthracen-9-ylcarbonyl)piperidin-4-yl]methyl}-2-methylquinoline, Acetyl-CoA carboxylase | Authors: | Rajamohan, F, Marr, E, Reyes, A, Landro, J.A, Anderson, M.D, Corbett, J.W, Dirico, K.J, Harwood, J.H, Tu, M, Vajdos, F.F. | Deposit date: | 2011-09-26 | Release date: | 2011-10-19 | Last modified: | 2023-09-13 | Method: | X-RAY DIFFRACTION (2.7 Å) | Cite: | Structure-guided Inhibitor Design for Human Acetyl-coenzyme A Carboxylase by Interspecies Active Site Conversion. J.Biol.Chem., 286, 2011
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1OD4
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![BU of 1od4 by Molmil](/molmil-images/mine/1od4) | Acetyl-CoA Carboxylase Carboxyltransferase Domain | Descriptor: | ACETYL-COENZYME A CARBOXYLASE, ADENINE | Authors: | Zhang, H, Yang, Z, Shen, Y, Tong, L. | Deposit date: | 2003-02-12 | Release date: | 2003-04-03 | Last modified: | 2018-06-13 | Method: | X-RAY DIFFRACTION (2.7 Å) | Cite: | Crystal structure of the carboxyltransferase domain of acetyl-coenzyme A carboxylase. Science, 299, 2003
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1OD2
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![BU of 1od2 by Molmil](/molmil-images/mine/1od2) | Acetyl-CoA Carboxylase Carboxyltransferase Domain | Descriptor: | ACETYL COENZYME *A, ACETYL-COENZYME A CARBOXYLASE, ADENINE | Authors: | Zhang, H, Yang, Z, Shen, Y, Tong, L. | Deposit date: | 2003-02-12 | Release date: | 2003-04-03 | Last modified: | 2018-06-13 | Method: | X-RAY DIFFRACTION (2.7 Å) | Cite: | Crystal structure of the carboxyltransferase domain of acetyl-coenzyme A carboxylase. Science, 299, 2003
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3TV5
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![BU of 3tv5 by Molmil](/molmil-images/mine/3tv5) | Crystal Structure of the humanized carboxyltransferase domain of yeast Acetyl-coA caroxylase in complex with compound 1 | Descriptor: | (3R)-1'-(9-ANTHRYLCARBONYL)-3-(MORPHOLIN-4-YLCARBONYL)-1,4'-BIPIPERIDINE, Acetyl-CoA carboxylase | Authors: | Rajamohan, F, Marr, E, Reyes, A, Landro, J.A, Anderson, M.D, Corbett, J.W, Dirico, K.J, Harwood, J.H, Tu, M, Vajdos, F.F. | Deposit date: | 2011-09-19 | Release date: | 2011-10-19 | Last modified: | 2023-09-13 | Method: | X-RAY DIFFRACTION (2.8 Å) | Cite: | Structure-guided Inhibitor Design for Human Acetyl-coenzyme A Carboxylase by Interspecies Active Site Conversion. J.Biol.Chem., 286, 2011
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3TVW
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![BU of 3tvw by Molmil](/molmil-images/mine/3tvw) | Crystal Structure of the humanized carboxyltransferase domain of yeast Acetyl-coA caroxylase in complex with compound 4 | Descriptor: | Acetyl-CoA carboxylase, [4-(2H-chromen-3-ylmethyl)piperazin-1-yl]-[3-(1H-pyrazol-5-yl)phenyl]methanone | Authors: | Rajamohan, F, Marr, E, Reyes, A, Landro, J.A, Anderson, M.D, Corbett, J.W, Dirico, K.J, Harwood, J.H, Tu, M, Vajdos, F.F. | Deposit date: | 2011-09-20 | Release date: | 2011-10-19 | Last modified: | 2023-09-13 | Method: | X-RAY DIFFRACTION (2.8 Å) | Cite: | Structure-guided Inhibitor Design for Human Acetyl-coenzyme A Carboxylase by Interspecies Active Site Conversion. J.Biol.Chem., 286, 2011
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1UYS
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3H0J
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3PGQ
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![BU of 3pgq by Molmil](/molmil-images/mine/3pgq) | Crystal Structure of the Carboxyltransferase Domain of S. cerevisiae Acetyl CoA Carboxylase in Complex with Pinoxaden | Descriptor: | 8-(2-ethenyl-6-ethyl-4-methylphenyl)tetrahydro-7H-pyrazolo[1,2-d][1,4,5]oxadiazepine-7,9(8H)-dione, Acetyl-CoA carboxylase | Authors: | Tong, L, Yu, L.P.C, Kim, Y.S. | Deposit date: | 2010-11-02 | Release date: | 2010-12-22 | Last modified: | 2024-02-21 | Method: | X-RAY DIFFRACTION (2.8 Å) | Cite: | Mechanism for the inhibition of the carboxyltransferase domain of acetyl-coenzyme A carboxylase by pinoxaden. Proc.Natl.Acad.Sci.USA, 107, 2010
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1W2X
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![BU of 1w2x by Molmil](/molmil-images/mine/1w2x) | Crystal structure of the carboxyltransferase domain of acetyl- coenzyme A carboxylase in complex with CP-640186 | Descriptor: | (3R)-1'-(9-ANTHRYLCARBONYL)-3-(MORPHOLIN-4-YLCARBONYL)-1,4'-BIPIPERIDINE, ACETYL-COA CARBOXYLASE | Authors: | Zhang, H, Tweel, B, Li, J, Tong, L. | Deposit date: | 2004-07-09 | Release date: | 2004-09-09 | Last modified: | 2024-05-08 | Method: | X-RAY DIFFRACTION (2.8 Å) | Cite: | Crystal Structure of the Carboxyltransferase Domain of Acetyl-Coenzyme a Carboxylase in Complex with Cp-640186 Structure, 12, 2004
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4WYO
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![BU of 4wyo by Molmil](/molmil-images/mine/4wyo) | |
5TRC
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![BU of 5trc by Molmil](/molmil-images/mine/5trc) | |