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2GEJ
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Crystal Structure of phosphatidylinositol mannosyltransferase (PimA) from Mycobacterium smegmatis in complex with GDP-Man
分子名称: GUANOSINE-5'-DIPHOSPHATE-ALPHA-D-MANNOSE, PHOSPHATIDYLINOSITOL MANNOSYLTRANSFERASE (PimA)
著者Guerin, M.E, Buschiazzo, A, Kordulakova, J, Jackson, M, Alzari, P.M.
登録日2006-03-20
公開日2007-04-03
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Molecular recognition and interfacial catalysis by the essential phosphatidylinositol mannosyltransferase PimA from mycobacteria.
J.Biol.Chem., 282, 2007
1UPJ
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HIV-1 PROTEASE COMPLEX WITH U095438 [3-[1-(4-BROMOPHENYL) ISOBUTYL]-4-HYDROXYCOUMARIN
分子名称: 3-[1-(4-BROMO-PHENYL)-2-METHYL-PROPYL]-4-HYDROXY-CHROMEN-2-ONE, HIV-1 PROTEASE
著者Watenpaugh, K.D, Mulichak, A.M, Janakiraman, M.N.
登録日1996-03-04
公開日1996-10-14
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.22 Å)
主引用文献Structure-based design of novel HIV protease inhibitors: carboxamide-containing 4-hydroxycoumarins and 4-hydroxy-2-pyrones as potent nonpeptidic inhibitors.
J.Med.Chem., 38, 1995
1BWB
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HIV-1 PROTEASE (V82F/I84V) DOUBLE MUTANT COMPLEXED WITH SD146 OF DUPONT PHARMACEUTICALS
分子名称: PROTEIN (HIV-1 PROTEASE), [4R-(4ALPHA,5ALPHA,6ALPHA,7ALPHA)]-3,3'-{{TETRAHYDRO-5,6-DIHYDROXY-2-OXO-4,7-BIS(PHENYLMETHYL)-1H-1,3-DIAZEPINE-1,3(2H)-DIYL]BIS(METHYLENE)]BIS[N-1H-BENZIMIDAZOL-2-YLBENZAMIDE]
著者Ala, P, Chang, C.H.
登録日1998-09-22
公開日1998-09-30
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Counteracting HIV-1 protease drug resistance: structural analysis of mutant proteases complexed with XV638 and SD146, cyclic urea amides with broad specificities.
Biochemistry, 37, 1998
4APF
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Crystal structure of the human KLHL11-Cul3 complex at 3.1A resolution
分子名称: CULLIN 3, KELCH-LIKE PROTEIN 11
著者Canning, P, Cooper, C.D.O, Krojer, T, Vollmar, M, Ugochukwu, E, Muniz, J.R.C, Ayinampudi, V, Savitsky, P, Arrowsmith, C.H, Edwards, A.M, Bountra, C, von Delft, F, Bullock, A.N, Structural Genomics Consortium (SGC)
登録日2012-04-02
公開日2012-05-09
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Structural Basis for Cul3 Assembly with the Btb-Kelch Family of E3 Ubiquitin Ligases.
J.Biol.Chem., 288, 2013
3LWW
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Structure of an open and closed conformation of Human Importin Beta bound to the Snurportin1 IBB-domain trapped in the same crystallographic asymmetric unit
分子名称: Importin subunit beta-1, Snurportin-1
著者Bhardwaj, A, Cingolani, G.
登録日2010-02-24
公開日2010-06-02
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (3.15 Å)
主引用文献Conformational selection in the recognition of the snurportin importin beta binding domain by importin beta.
Biochemistry, 49, 2010
4ARR
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Crystal structure of the N-terminal domain of Drosophila Toll receptor with the magic triangle I3C
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 5-amino-2,4,6-triiodobenzene-1,3-dicarboxylic acid, TOLL RECEPTOR, ...
著者Gangloff, M, Gay, N.J.
登録日2012-04-26
公開日2013-02-27
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Liesegang-Like Patterns of Toll Crystals Grown in Gel.
J.Appl.Crystallogr., 46, 2013
1BV7
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COUNTERACTING HIV-1 PROTEASE DRUG RESISTANCE: STRUCTURAL ANALYSIS OF MUTANT PROTEASES COMPLEXED WITH XV638 AND SD146, CYCLIC UREA AMIDES WITH BROAD SPECIFICITIES
分子名称: PROTEIN (HIV-1 PROTEASE), [4R-(4ALPHA,5ALPHA,6BETA,7BETA)]-3,3'-[[TETRAHYDRO-5,6-DIHYDROXY-2-OXO-4,7-BIS(PHENYLMETHYL)-1H-1,3-DIAZEPINE-1,3(2H)-D IYL] BIS(METHYLENE)]BIS[N-2-THIAZOLYLBENZAMIDE]
著者Ala, P, Chang, C.H.
登録日1998-09-22
公開日1998-09-30
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Counteracting HIV-1 protease drug resistance: structural analysis of mutant proteases complexed with XV638 and SD146, cyclic urea amides with broad specificities.
Biochemistry, 37, 1998
2GEK
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Crystal Structure of phosphatidylinositol mannosyltransferase (PimA) from Mycobacterium smegmatis in complex with GDP
分子名称: GUANOSINE-5'-DIPHOSPHATE, PHOSPHATIDYLINOSITOL MANNOSYLTRANSFERASE (PimA)
著者Guerin, M.E, Buschiazzo, A, Kordulakova, J, Jackson, M, Alzari, P.M.
登録日2006-03-20
公開日2007-04-03
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Molecular recognition and interfacial catalysis by the essential phosphatidylinositol mannosyltransferase PimA from mycobacteria.
J.Biol.Chem., 282, 2007
2K4T
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Solution structure of human VDAC-1 in LDAO micelles
分子名称: Voltage-dependent anion-selective channel protein 1
著者Hiller, S, Garces, R.G, Malia, T.J, Orekhov, V.Y, Colombini, M, Wagner, G.
登録日2008-06-17
公開日2008-09-09
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of the integral human membrane protein VDAC-1 in detergent micelles.
Science, 321, 2008
1NHG
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CRYSTAL STRUCTURE ANALYSIS OF PLASMODIUM FALCIPARUM ENOYL-ACYL-CARRIER-PROTEIN REDUCTASE WITH TRICLOSAN
分子名称: NICOTINAMIDE-ADENINE-DINUCLEOTIDE, TRICLOSAN, enoyl-acyl carrier reductase
著者Perozzo, R, Kuo, M, Sidhu, A.S, Valiyaveettil, J.T, Bittman, R, Jacobs Jr, W.R, Fidock, D.A, Sacchettini, J.C.
登録日2002-12-19
公開日2003-02-25
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.43 Å)
主引用文献Structural Elucidation of the Specificity of the Antibacterial Agent Triclosan for Malarial Enoyl Acyl Carrier Protein Reductase
J.Biol.Chem., 277, 2002
1NHW
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Crystal Structure Analysis of Plasmodium falciparum enoyl-acyl-carrier-protein reductase
分子名称: 2-(2,4-DICHLORO-PHENYLAMINO)-PHENOL, NICOTINAMIDE-ADENINE-DINUCLEOTIDE, enoyl-acyl carrier reductase
著者Perozzo, R, Kuo, M, Sidhu, A.S, Valiyaveettil, J.T, Bittman, R, Jacobs Jr, W.R, Fidock, D.A, Sacchettini, J.C.
登録日2002-12-19
公開日2003-02-25
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.35 Å)
主引用文献Structural Elucidation of the Specificity of the Antibacterial Agent Triclosan for Malarial Enoyl Acyl Carrier Protein Reductase Year
J.Biol.Chem., 277, 2002
2GPB
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COMPARISON OF THE BINDING OF GLUCOSE AND GLUCOSE-1-PHOSPHATE DERIVATIVES TO T-STATE GLYCOGEN PHOSPHORYLASE B
分子名称: GLYCOGEN PHOSPHORYLASE B, PYRIDOXAL-5'-PHOSPHATE, alpha-D-glucopyranose
著者Martin, J.L, Johnson, L.N.
登録日1990-06-04
公開日1992-10-15
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Comparison of the binding of glucose and glucose 1-phosphate derivatives to T-state glycogen phosphorylase b.
Biochemistry, 29, 1990
1WQJ
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Structural Basis for the Regulation of Insulin-Like Growth Factors (IGFs) by IGF Binding Proteins (IGFBPs)
分子名称: Insulin-like growth factor IB, Insulin-like growth factor binding protein 4
著者Siwanowicz, I, Popowicz, G.M, Wisniewska, M, Huber, R, Kuenkele, K.P, Lang, K, Engh, R.A, Holak, T.A.
登録日2004-09-29
公開日2005-03-01
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Structural basis for the regulation of insulin-like growth factors by IGF binding proteins
Structure, 13, 2005
2KIQ
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Solution structure of the FF Domain 2 of human transcription elongation factor CA150
分子名称: Transcription elongation regulator 1
著者Zeng, J, Boyles, J, Tripathy, C, Yan, A, Zhou, P, Donald, B.R.
登録日2009-05-07
公開日2009-07-28
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献High-resolution protein structure determination starting with a global fold calculated from exact solutions to the RDC equations.
J.Biomol.Nmr, 45, 2009
2SBL
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BU of 2sbl by Molmil
THE THREE-DIMENSIONAL STRUCTURE OF AN ARACHIDONIC ACID 15-LIPOXYGENASE
分子名称: FE (III) ION, LIPOXYGENASE-1
著者Amzel, L.M, Boyington, J.C.
登録日1993-07-22
公開日1995-02-27
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献The three-dimensional structure of an arachidonic acid 15-lipoxygenase.
Science, 260, 1993
2BDZ
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Mexicain from Jacaratia mexicana
分子名称: Mexicain, N-[N-[1-HYDROXYCARBOXYETHYL-CARBONYL]LEUCYLAMINO-BUTYL]-GUANIDINE
著者Gavira, J.A, Oliver-Salvador, M.C, Gonzalez-Ramirez, L.A, Soriano-Garcia, M, Garcia-Ruiz, J.M.
登録日2005-10-21
公開日2006-10-03
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Crystallographic structure of Mexicain from Jacaratia mexicana
To be Published
1BXZ
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CRYSTAL STRUCTURE OF A THERMOPHILIC ALCOHOL DEHYDROGENASE SUBSTRATE COMPLEX FROM THERMOANAEROBACTER BROCKII
分子名称: 2-BUTANOL, CHLORIDE ION, MAGNESIUM ION, ...
著者Li, C, Heatwole, J, Soelaiman, S, Shoham, M.
登録日1998-10-09
公開日2000-02-18
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.99 Å)
主引用文献Crystal structure of a thermophilic alcohol dehydrogenase substrate complex suggests determinants of substrate specificity and thermostability.
Proteins, 37, 1999
1BWX
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THE SOLUTION STRUCTURE OF HUMAN PARATHYROID HORMONE FRAGMENT 1-39, NMR, 10 STRUCTURES
分子名称: PARATHYROID HORMONE
著者Marx, U.C, Roesch, P, Adermann, K, Bayer, P, Forssmann, W.-G.
登録日1998-09-29
公開日2000-01-14
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Solution structures of human parathyroid hormone fragments hPTH(1-34) and hPTH(1-39) and bovine parathyroid hormone fragment bPTH(1-37).
Biochem.Biophys.Res.Commun., 267, 2000
2PDA
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BU of 2pda by Molmil
CRYSTAL STRUCTURE OF THE COMPLEX BETWEEN PYRUVATE-FERREDOXIN OXIDOREDUCTASE FROM DESULFOVIBRIO AFRICANUS AND PYRUVATE.
分子名称: CALCIUM ION, IRON/SULFUR CLUSTER, MAGNESIUM ION, ...
著者Chabriere, E, Charon, M.H.
登録日1998-11-10
公開日1999-04-23
最終更新日2024-10-16
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Crystal structures of the key anaerobic enzyme pyruvate:ferredoxin oxidoreductase, free and in complex with pyruvate.
Nat.Struct.Biol., 6, 1999
4AUO
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Crystal structure of MMP-1(E200A) in complex with a triple-helical collagen peptide
分子名称: CALCIUM ION, INTERSTITIAL COLLAGENASE, TRIPLE-HELICAL COLLAGEN PEPTIDE, ...
著者Manka, S.W, Carafoli, F, Visse, R, Bihan, D, Raynal, N, Farndale, R.W, Murphy, G, Enghild, J.J, Hohenester, E, Nagase, H.
登録日2012-05-18
公開日2012-07-11
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Structural Insights Into Triple-Helical Collagen Cleavage by Matrix Metalloproteinase 1
Proc.Natl.Acad.Sci.USA, 109, 2012
1HYK
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AGOUTI-RELATED PROTEIN (87-132) (AC-AGRP(87-132))
分子名称: AGOUTI RELATED PROTEIN
著者Bolin, K.A, Anderson, D.J, Trulson, J.A, Thompson, D.A, Wilken, J, Kent, S.B.H, Millhauser, G.L.
登録日2001-01-19
公開日2001-02-07
最終更新日2022-02-23
実験手法SOLUTION NMR
主引用文献NMR structure of a minimized human agouti related protein prepared by total chemical synthesis.
FEBS Lett., 451, 1999
4BIW
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Crystal structure of CpxAHDC (hexagonal form)
分子名称: MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, SENSOR PROTEIN CPXA, ...
著者Mechaly, A.E, Sassoon, N, Betton, J.M, Alzari, P.M.
登録日2013-04-13
公開日2014-02-12
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.85 Å)
主引用文献Segmental Helical Motions and Dynamical Asymmetry Modulate Histidine Kinase Autophosphorylation.
Plos Biol., 12, 2014
4BIY
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Crystal structure of CpxAHDC (monoclinic form 2)
分子名称: ADENOSINE-5'-DIPHOSPHATE, SENSOR PROTEIN CPXA, SULFATE ION
著者Mechaly, A.E, Sassoon, N, Betton, J.M, Alzari, P.M.
登録日2013-04-13
公開日2014-02-12
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (3.3 Å)
主引用文献Segmental Helical Motions and Dynamical Asymmetry Modulate Histidine Kinase Autophosphorylation.
Plos Biol., 12, 2014
2OX9
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Mouse Scavenger Receptor C-type Lectin carbohydrate-recognition domain.
分子名称: CALCIUM ION, Collectin placenta 1, alpha-L-fucopyranose-(1-3)-[beta-D-galactopyranose-(1-4)]2-acetamido-2-deoxy-beta-D-glucopyranose
著者Weis, W.I, Feinberg, H, Drickamer, K, Taylor, M.E.
登録日2007-02-20
公開日2007-04-03
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Scavenger receptor C-type lectin binds to the leukocyte cell surface glycan Lewis(x) by a novel mechanism.
J.Biol.Chem., 282, 2007
2RDV
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RUBREDOXIN FROM DESULFOVIBRIO VULGARIS MIYAZAKI F, MONOCLINIC CRYSTAL FORM
分子名称: FE (III) ION, RUBREDOXIN
著者Higuchi, Y, Yasuoka, N.
登録日1998-10-07
公開日1999-05-18
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structure determination of rubredoxin from Desulfovibrio vulgaris Miyazaki F in two crystal forms.
Acta Crystallogr.,Sect.D, 55, 1999

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