8V6M
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![BU of 8v6m by Molmil](/molmil-images/mine/8v6m) | Inactivated-state cryo-EM structure of human TRPV3 in presence of tetrahydrocannabivarin (THCV) in cNW30 nanodiscs | 分子名称: | (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate, SODIUM ION, Tetrahydrocannabivarin, ... | 著者 | Nadezhdin, K.D, Neuberger, A, Sobolevsky, A.I. | 登録日 | 2023-12-01 | 公開日 | 2024-04-17 | 最終更新日 | 2024-05-08 | 実験手法 | ELECTRON MICROSCOPY (3.63 Å) | 主引用文献 | TRPV3 activation by different agonists accompanied by lipid dissociation from the vanilloid site. Sci Adv, 10, 2024
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8WR2
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![BU of 8wr2 by Molmil](/molmil-images/mine/8wr2) | Crystal Structure of Human Pyridoxal Kinase with bound Luteolin | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, 2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4H-chromen-4-one, DIMETHYL SULFOXIDE, ... | 著者 | Fan, J, Zhu, Y. | 登録日 | 2023-10-12 | 公開日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (1.94 Å) | 主引用文献 | Discovery and characterization of natural product luteolin as an effective inhibitor of human pyridoxal kinase. Bioorg.Chem., 143, 2024
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8W0C
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8V6L
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![BU of 8v6l by Molmil](/molmil-images/mine/8v6l) | Open-state cryo-EM structure of human TRPV3 in presence of tetrahydrocannabivarin (THCV) in cNW30 nanodiscs | 分子名称: | (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate, SODIUM ION, Tetrahydrocannabivarin, ... | 著者 | Nadezhdin, K.D, Neuberger, A, Sobolevsky, A.I. | 登録日 | 2023-12-01 | 公開日 | 2024-04-17 | 最終更新日 | 2024-05-08 | 実験手法 | ELECTRON MICROSCOPY (3.68 Å) | 主引用文献 | TRPV3 activation by different agonists accompanied by lipid dissociation from the vanilloid site. Sci Adv, 10, 2024
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8U5Z
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![BU of 8u5z by Molmil](/molmil-images/mine/8u5z) | Structure of Mango II variant aptamer bound to T01-7M-B | 分子名称: | 2-[(E)-(1,7-dimethylquinolin-4(1H)-ylidene)methyl]-3-{2,16-dioxo-20-[(3aR,4S,6aR)-2-oxohexahydro-1H-thieno[3,4-d]imidazol-4-yl]-6,9,12-trioxa-3,15-diazaicosan-1-yl}-1,3-benzothiazol-3-ium, Mango II variant, POTASSIUM ION, ... | 著者 | Passalacqua, L.F.M, Ferre-D'Amare, A.R. | 登録日 | 2023-09-13 | 公開日 | 2024-03-27 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Structure of Mango II variant aptamer bound to T01-7M-B To Be Published
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8YBG
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![BU of 8ybg by Molmil](/molmil-images/mine/8ybg) | |
7Q0E
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![BU of 7q0e by Molmil](/molmil-images/mine/7q0e) | Human Carbonic Anhydrase II in complex with Methyl 2-(benzenesulfonyl)-4-chloro-5-sulfamoylbenzoate | 分子名称: | BICINE, Carbonic anhydrase 2, DIMETHYL SULFOXIDE, ... | 著者 | Paketuryte-Latve, V, Smirnov, A, Manakova, E, Grazulis, S. | 登録日 | 2021-10-14 | 公開日 | 2022-01-12 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.3 Å) | 主引用文献 | Methyl 2-Halo-4-Substituted-5-Sulfamoyl-Benzoates as High Affinity and Selective Inhibitors of Carbonic Anhydrase IX. Int J Mol Sci, 23, 2021
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8VFA
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![BU of 8vfa by Molmil](/molmil-images/mine/8vfa) | Ternary DNA Polymerase Beta bound to DNA containing primer terminal dC base-paired with FapydG | 分子名称: | DNA (5'-D(*CP*CP*GP*AP*CP*CP*(FAP)P*CP*GP*CP*AP*TP*CP*AP*GP*C)-3'), DNA (5'-D(*GP*CP*TP*GP*AP*TP*GP*CP*GP*C)-3'), DNA (5'-D(P*GP*TP*CP*GP*G)-3'), ... | 著者 | Oden, P.N, Ryan, B.J, Freudenthal, B.D. | 登録日 | 2023-12-21 | 公開日 | 2024-05-08 | 最終更新日 | 2024-06-05 | 実験手法 | X-RAY DIFFRACTION (2.05 Å) | 主引用文献 | Biochemical and structural characterization of Fapy•dG replication by Human DNA polymerase beta. Nucleic Acids Res., 52, 2024
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8U3C
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![BU of 8u3c by Molmil](/molmil-images/mine/8u3c) | TRPV1 in nanodisc bound with PI-Br4 bound in Conformation 2 (monomer) | 分子名称: | (2S)-2-[(9,10-dibromooctadecanoyl)oxy]-3-{[(S)-hydroxy{[(1S,2R,3R,4S,5S,6R)-2,3,4,5,6-pentahydroxycyclohexyl]oxy}phosphoryl]oxy}propyl (9R,10S)-9,10-dibromooctadecanoate, 1,2-DIACYL-GLYCEROL-3-SN-PHOSPHATE, 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, ... | 著者 | Arnold, W.R, Julius, D, Cheng, Y. | 登録日 | 2023-09-07 | 公開日 | 2024-05-08 | 最終更新日 | 2024-05-15 | 実験手法 | ELECTRON MICROSCOPY (2.3 Å) | 主引用文献 | Structural basis of TRPV1 modulation by endogenous bioactive lipids. Nat.Struct.Mol.Biol., 2024
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8VJ2
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8V9I
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![BU of 8v9i by Molmil](/molmil-images/mine/8v9i) | 1-deoxy-D-xylulose 5-phosphate synthase (DXPS) from Deinococcus radiodurans with D-phenylalanine-derived triazole acetylphosphonate (D-PheTrAP) bound | 分子名称: | 1-deoxy-D-xylulose-5-phosphate synthase, 2-HYDROXY BUTANE-1,4-DIOL, 3-[(4-amino-2-methylpyrimidin-5-yl)methyl]-2-{(1S)-1-[(S)-(2-{1-[(1R)-1-carboxy-2-phenylethyl]-1H-1,2,3-triazol-4-yl}ethoxy)(hydroxy)phosphoryl]-1-hydroxyethyl}-5-(2-{[(S)-hydroxy(phosphonooxy)phosphoryl]oxy}ethyl)-4-methyl-1,3-thiazol-3-ium, ... | 著者 | Chen, P.Y.-T, Drennan, C.L. | 登録日 | 2023-12-08 | 公開日 | 2024-04-24 | 実験手法 | X-RAY DIFFRACTION (1.981 Å) | 主引用文献 | Potent Inhibition of E. coli DXP Synthase by a gem -Diaryl Bisubstrate Analog. Acs Infect Dis., 10, 2024
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8TKB
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![BU of 8tkb by Molmil](/molmil-images/mine/8tkb) | |
7PEN
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![BU of 7pen by Molmil](/molmil-images/mine/7pen) | |
7SI5
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![BU of 7si5 by Molmil](/molmil-images/mine/7si5) | CRYSTAL STRUCTURE OF EED WITH MRTX-1919 | 分子名称: | (4R)-8-(1,3-dimethyl-1H-pyrazol-5-yl)-5-{[(5-fluoro-2,3-dihydro-1-benzofuran-4-yl)methyl]amino}imidazo[1,2-c]pyrimidine-2-carbonitrile, 1,2-ETHANEDIOL, FORMIC ACID, ... | 著者 | Gunn, R.J, Burns, A.C, Lawson, J.D, Marx, M.A. | 登録日 | 2021-10-12 | 公開日 | 2022-11-09 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | CRYSTAL STRUCTURE OF EED WITH MRTX-1919 TO BE PUBLISHED
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8YRC
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![BU of 8yrc by Molmil](/molmil-images/mine/8yrc) | |
8WFU
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![BU of 8wfu by Molmil](/molmil-images/mine/8wfu) | |
8VF9
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![BU of 8vf9 by Molmil](/molmil-images/mine/8vf9) | Binary DNA Polymerase Beta bound to DNA containing primer terminal dA base-paired with FapydG | 分子名称: | DNA (5'-D(*CP*CP*GP*AP*CP*CP*(FAP)P*CP*GP*CP*AP*TP*CP*AP*GP*C)-3'), DNA (5'-D(*GP*CP*TP*GP*AP*TP*GP*CP*GP*A)-3'), DNA (5'-D(P*GP*TP*CP*GP*G)-3'), ... | 著者 | Oden, P.N, Ryan, B.J, Freudenthal, B.D. | 登録日 | 2023-12-21 | 公開日 | 2024-05-08 | 最終更新日 | 2024-06-05 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Biochemical and structural characterization of Fapy•dG replication by Human DNA polymerase beta. Nucleic Acids Res., 52, 2024
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7PU0
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![BU of 7pu0 by Molmil](/molmil-images/mine/7pu0) | |
9B7F
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![BU of 9b7f by Molmil](/molmil-images/mine/9b7f) | S_SAD structure of HEWL using lossless default compression | 分子名称: | 1,2-ETHANEDIOL, CHLORIDE ION, Lysozyme C, ... | 著者 | Jakoncic, J, Bernstein, H.J, Soares, A.S, Horvat, K. | 登録日 | 2024-03-27 | 公開日 | 2024-04-10 | 実験手法 | X-RAY DIFFRACTION (1.65 Å) | 主引用文献 | Investigation of fast and efficient lossless compression algorithms for macromolecular crystallography experiments To Be Published
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8WUG
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![BU of 8wug by Molmil](/molmil-images/mine/8wug) | The Crystal Structure of JMJD2D from Biortus. | 分子名称: | 1,2-ETHANEDIOL, DI(HYDROXYETHYL)ETHER, Lysine-specific demethylase 4D, ... | 著者 | Wang, F, Cheng, W, Yuan, Z, Lin, D, Guo, S. | 登録日 | 2023-10-20 | 公開日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | The Crystal Structure of JMJD2D from Biortus. To Be Published
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8VMP
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7PFR
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![BU of 7pfr by Molmil](/molmil-images/mine/7pfr) | |
8VMS
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![BU of 8vms by Molmil](/molmil-images/mine/8vms) | |
8WFW
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![BU of 8wfw by Molmil](/molmil-images/mine/8wfw) | |
8VMZ
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![BU of 8vmz by Molmil](/molmil-images/mine/8vmz) | |