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2HK3
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Crystal structure of mevalonate diphosphate decarboxylase from Staphylococcus aureus (orthorhombic form)
分子名称: Diphosphomevalonate decarboxylase
著者Byres, E, Hunter, W.N.
登録日2006-07-03
公開日2007-06-12
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal Structures of Trypanosoma brucei and Staphylococcus aureus Mevalonate Diphosphate Decarboxylase Inform on the Determinants of Specificity and Reactivity
J.Mol.Biol., 371, 2007
2HKE
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Mevalonate diphosphate decarboxylase from Trypanosoma brucei
分子名称: Diphosphomevalonate decarboxylase, putative, SULFATE ION
著者Byres, E, Alphey, M.S, Hunter, W.N.
登録日2006-07-04
公開日2007-06-12
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Crystal Structures of Trypanosoma brucei and Staphylococcus aureus Mevalonate Diphosphate Decarboxylase Inform on the Determinants of Specificity and Reactivity
J.Mol.Biol., 371, 2007
2HK2
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Crystal structure of mevalonate diphosphate decarboxylase from Staphylococcus aureus (monoclinic form)
分子名称: Diphosphomevalonate decarboxylase
著者Byres, E, Hunter, W.N.
登録日2006-07-03
公開日2007-06-12
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal Structures of Trypanosoma brucei and Staphylococcus aureus Mevalonate Diphosphate Decarboxylase Inform on the Determinants of Specificity and Reactivity
J.Mol.Biol., 371, 2007
2V2V
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IspE in complex with ligand
分子名称: 4-DIPHOSPHOCYTIDYL-2C-METHYL-D-ERYTHRITOL KINASE, 5'-[(1H-BENZIMIDAZOL-2-YLACETYL)AMINO]-5'-DEOXYCYTIDINE, BROMIDE ION, ...
著者Alphey, M.S, Hunter, W.N.
登録日2007-06-07
公開日2007-06-19
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Synthesis and Characterization of Cytidine Derivatives that Inhibit the Kinase Ispe of the Non-Mevalonate Pathway for Isoprenoid Biosynthesis.
Chemmedchem, 3, 2008
2V2Z
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IspE in complex with ADP and CDPME
分子名称: 4-DIPHOSPHOCYTIDYL-2-C-METHYL-D-ERYTHRITOL, 4-DIPHOSPHOCYTIDYL-2C-METHYL-D-ERYTHRITOL KINASE, ADENOSINE-5'-DIPHOSPHATE, ...
著者Sgraja, T, Alphey, M.S, Hunter, W.N.
登録日2007-06-08
公開日2007-06-19
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献Characterization of Aquifex Aeolicus 4-Diphosphocytidyl-2C-Methyl-D-Erythritol Kinase -Ligand Recognition in a Template for Antimicrobial Drug Discovery.
FEBS J., 275, 2008
2V2Q
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IspE in complex with ligand
分子名称: 4-AMINO-1-(5-{[3-(1H-BENZIMIDAZOL-2-YL)PROPANOYL]AMINO}-5-DEOXY-ALPHA-L-LYXOFURANOSYL)PYRIMIDIN-2(1H)-ONE, 4-DIPHOSPHOCYTIDYL-2-C-METHYL-D-ERYTHRITOL KINASE, BROMIDE ION, ...
著者Alphey, M.S, Hunter, W.N.
登録日2007-06-06
公開日2007-06-19
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Synthesis and Characterization of Cytidine Derivatives that Inhibit the Kinase Ispe of the Non-Mevalonate Pathway for Isoprenoid Biosynthesis.
Chemmedchem, 3, 2008
2V34
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IspE in complex with cytidine and ligand
分子名称: 4-AMINO-1-BETA-D-RIBOFURANOSYL-2(1H)-PYRIMIDINONE, 4-DIPHOSPHOCYTIDYL-2C-METHYL-D-ERYTHRITOL KINASE, CHLORIDE ION, ...
著者Sgraja, T, Alphey, M.S, Hunter, W.N.
登録日2007-06-11
公開日2007-06-26
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Characterization of Aquifex Aeolicus 4-Diphosphocytidyl-2C-Methyl-D-Erythritol Kinase -Ligand Recognition in a Template for Antimicrobial Drug Discovery.
FEBS J., 275, 2008
2V8P
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IspE in complex with ADP and CDP
分子名称: 4-DIPHOSPHOCYTIDYL-2-C-METHYL-D-ERYTHRITOL KINASE, ADENOSINE-5'-DIPHOSPHATE, CHLORIDE ION, ...
著者Sgraja, T, Alphey, M.S, Hunter, W.N.
登録日2007-08-13
公開日2007-08-21
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Characterization of Aquifex Aeolicus 4-Diphosphocytidyl-2C-Methyl-D-Erythritol Kinase -Ligand Recognition in a Template for Antimicrobial Drug Discovery.
FEBS J., 275, 2008
2R42
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The Biochemical and Structural Basis for feedback Inhibition of Mevalonate Kinase and Isoprenoid Metabolism
分子名称: MAGNESIUM ION, Mevalonate kinase, S-[(2E,6E)-3,7,11-TRIMETHYLDODECA-2,6,10-TRIENYL] TRIHYDROGEN THIODIPHOSPHATE
著者Fu, Z, Voynova, N.E, Miziorko, H.M, Kim, J.P.
登録日2007-08-30
公開日2008-06-24
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Biochemical and Structural Basis for Feedback Inhibition of Mevalonate Kinase and Isoprenoid Metabolism.
Biochemistry, 47, 2008
2R3V
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The Biochemical and Structural Basis for Feedback Inhibition of Mevalonate Kinase and Isoprenoid Metabolism
分子名称: Mevalonate kinase
著者Fu, Z, Voynova, N.E, Miziorko, H.M, Kim, J.P.
登録日2007-08-30
公開日2008-06-24
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Biochemical and Structural Basis for Feedback Inhibition of Mevalonate Kinase and Isoprenoid Metabolism.
Biochemistry, 47, 2008
3F0N
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Mus Musculus Mevalonate Pyrophosphate Decarboxylase
分子名称: MEVALONATE PYROPHOSPHATE DECARBOXYLASE, PHOSPHATE ION
著者Walker, J.R, Davis, T, Vesterberg, A, Li, Y, Bountra, C, Weigelt, J, Arrowsmith, C.H, Edwards, A.M, Bochkarev, A, Dhe-Paganon, S, Structural Genomics Consortium (SGC)
登録日2008-10-25
公開日2008-11-25
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structure of Mus Musculus Mevalonate Pyrophosphate Decarboxylase
To be Published
2VF3
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Aquifex aeolicus IspE in complex with ligand
分子名称: 4-DIPHOSPHOCYTIDYL-2C-METHYL-D-ERYTHRITOL KINASE, BROMIDE ION, CHLORIDE ION, ...
著者Alphey, M.S, Hunter, W.N.
登録日2007-10-30
公開日2008-11-25
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Inhibitors of the Kinase Ispe: Structure-Activity Relationships and Co-Crystal Structure Analysis.
Org.Biomol.Chem., 6, 2008
3D4J
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Crystal structure of Human mevalonate diphosphate decarboxylase
分子名称: Diphosphomevalonate decarboxylase, SULFATE ION
著者Voynova, N.E, Fu, Z, Battaile, K, Herdendorf, T.J, Kim, J.-J.P, Miziorko, H.M.
登録日2008-05-14
公開日2008-12-16
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Human mevalonate diphosphate decarboxylase: characterization, investigation of the mevalonate diphosphate binding site, and crystal structure.
Arch.Biochem.Biophys., 480, 2008
3HUL
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Structure of putative homoserine kinase thrB from Listeria monocytogenes
分子名称: Homoserine kinase, SULFATE ION
著者Ramagopal, U.A, Toro, R, Burley, S.K, Almo, S.C, New York SGX Research Center for Structural Genomics (NYSGXRC)
登録日2009-06-15
公開日2009-07-14
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.19 Å)
主引用文献Structure of putative homoserine kinase thrB from Listeria monocytogenes
To be published
3GON
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Streptococcus pneumoniae Phosphomevalonate Kinase in Complex with Phosphomevalonate and AMPPNP
分子名称: (3R)-3-HYDROXY-3-METHYL-5-(PHOSPHONOOXY)PENTANOIC ACID, MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, ...
著者Andreassi, J.L, Bilder, P.W, Vetting, M.W, Roderick, S.L, Leyh, T.S.
登録日2009-03-19
公開日2009-07-21
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structure of the ternary complex of phosphomevalonate kinase: the enzyme and its family
Biochemistry, 48, 2009
3K17
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Crystal structure of a Lin0012 protein from Listeria innocua
分子名称: Lin0012 protein, TRIETHYLENE GLYCOL
著者Palani, K, Burley, S.K, Swaminathan, S, New York SGX Research Center for Structural Genomics (NYSGXRC)
登録日2009-09-25
公開日2009-10-06
最終更新日2021-02-10
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Crystal structure of a Lin0012 protein from Listeria innocua
To be Published
3K85
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Crystal structure of a D-glycero-D-manno-heptose 1-phosphate kinase from Bacteriodes thetaiotaomicron
分子名称: D-glycero-D-manno-heptose 1-phosphate kinase
著者Palani, K, Kumaran, D, Burley, S.K, Swaminathan, S, New York SGX Research Center for Structural Genomics (NYSGXRC)
登録日2009-10-13
公開日2009-12-08
最終更新日2021-02-10
実験手法X-RAY DIFFRACTION (2.28 Å)
主引用文献Crystal structure of a D-glycero-D-manno-heptose 1-phosphate kinase from Bacteriodes thetaiotaomicron
To be Published
3LTO
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BU of 3lto by Molmil
Crystal structure of a mevalonate diphosphate decarboxylase from Legionella pneumophila
分子名称: Mevalonate diphosphate decarboxylase, SULFATE ION
著者Palani, K, Burley, S.K, Swaminathan, S, New York SGX Research Center for Structural Genomics (NYSGXRC)
登録日2010-02-16
公開日2010-02-23
最終更新日2021-02-10
実験手法X-RAY DIFFRACTION (2.27 Å)
主引用文献Crystal structure of a mevalonate diphosphate decarboxylase from Legionella pneumophila
To be Published
2WW4
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a triclinic crystal form of E. coli 4-diphosphocytidyl-2C-methyl-D- erythritol kinase
分子名称: 4-DIPHOSPHOCYTIDYL-2C-METHYL-D-ERYTHRITOL KINASE, ADENOSINE-5'-DIPHOSPHATE, GLYCEROL
著者Kalinowska-Tluscik, J, Miallau, L, Gabrielsen, M, Leonard, G.A, McSweeney, S.M, Hunter, W.N.
登録日2009-10-21
公開日2010-03-09
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献A Triclinic Crystal Form of Escherichia Coli 4-Diphosphocytidyl-2C-Methyl-D-Erythritol Kinase and Reassessment of the Quaternary Structure.
Acta Crystallogr.,Sect.F, 66, 2010
3QT7
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Crystal structure of Staphylococcus epidermidis mevalonate diphosphate decarboxylase complexed with inhibitor 6-FMVAPP
分子名称: (3R)-3-(fluoromethyl)-3-hydroxy-5-{[(S)-hydroxy(phosphonooxy)phosphoryl]oxy}pentanoic acid, Mevalonate diphosphate decarboxylase
著者Barta, M.L, Skaff, A.D, McWhorter, W.J, Miziorko, H.M, Geisbrecht, B.V.
登録日2011-02-22
公開日2011-05-11
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.199 Å)
主引用文献Crystal structures of Staphylococcus epidermidis mevalonate diphosphate decarboxylase bound to inhibitory analogs reveal new insight into substrate binding and catalysis.
J.Biol.Chem., 286, 2011
3QT6
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Crystal structure of Staphylococcus epidermidis mevalonate diphosphate decarboxylase complexed with inhibitor DPGP
分子名称: 1-({[(S)-hydroxy(phosphonooxy)phosphoryl]oxy}acetyl)-L-proline, Mevalonate diphosphate decarboxylase
著者Barta, M.L, Skaff, A.D, McWhorter, W.J, Miziorko, H.M, Geisbrecht, B.V.
登録日2011-02-22
公開日2011-05-11
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.047 Å)
主引用文献Crystal structures of Staphylococcus epidermidis mevalonate diphosphate decarboxylase bound to inhibitory analogs reveal new insight into substrate binding and catalysis.
J.Biol.Chem., 286, 2011
3QT8
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Crystal structure of mutant S192A Staphylococcus epidermidis mevalonate diphosphate decarboxylase complexed with inhibitor 6-FMVAPP
分子名称: (3R)-3-(fluoromethyl)-3-hydroxy-5-{[(S)-hydroxy(phosphonooxy)phosphoryl]oxy}pentanoic acid, GLYCEROL, Mevalonate diphosphate decarboxylase
著者Barta, M.L, Skaff, A.D, McWhorter, W.J, Miziorko, H.M, Geisbrecht, B.V.
登録日2011-02-22
公開日2011-05-11
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Crystal structures of Staphylococcus epidermidis mevalonate diphosphate decarboxylase bound to inhibitory analogs reveal new insight into substrate binding and catalysis.
J.Biol.Chem., 286, 2011
3QT5
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Crystal structure of Staphylococcus epidermidis mevalonate diphosphate decarboxylase
分子名称: Mevalonate diphosphate decarboxylase
著者Barta, M.L, Skaff, A.D, McWhorter, W.J, Miziorko, H.M, Geisbrecht, B.V.
登録日2011-02-22
公開日2011-05-11
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.848 Å)
主引用文献Crystal structures of Staphylococcus epidermidis mevalonate diphosphate decarboxylase bound to inhibitory analogs reveal new insight into substrate binding and catalysis.
J.Biol.Chem., 286, 2011
3PYG
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Mycobacterium tuberculosis 4-diphosphocytidyl-2-C-methyl-D-erythritol kinase (IspE) in complex with ADP
分子名称: 4-diphosphocytidyl-2-C-methyl-D-erythritol kinase, ADENOSINE-5'-DIPHOSPHATE
著者Shan, S, Chen, X.H, Liu, T, Zhao, H.C, Rao, Z.H, Lou, Z.Y.
登録日2010-12-13
公開日2012-01-25
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (1.99 Å)
主引用文献The Structural Basis for anti-TB Drug Discovery targeting of 4-diphosphocytidyl-2-C-methyl-D-erythritol kinase (IspE) from Mycobacterium tuberculosis
To be Published
3PYE
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Mycobacterium tuberculosis 4-diphosphocytidyl-2-C-methyl-D-erythritol kinase (IspE) in complex with CDPME
分子名称: 4-DIPHOSPHOCYTIDYL-2-C-METHYL-D-ERYTHRITOL, 4-diphosphocytidyl-2-C-methyl-D-erythritol kinase
著者Shan, S, Chen, X.H, Liu, T, Zhao, H.C, Rao, Z.H, Lou, Z.Y.
登録日2010-12-13
公開日2012-01-25
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献The Structural Basis for anti-TB Drug Discovery targeting of 4-diphosphocytidyl-2-C-methyl-D-erythritol kinase (IspE) from Mycobacterium tuberculosis
To be Published

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