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9BBI
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BU of 9bbi by Molmil
Co-crystal structure of human DDB1 bound to fragment UB028669
分子名称: 3-([1,3]oxazolo[4,5-b]pyridin-2-yl)aniline, DNA damage-binding protein 1, L(+)-TARTARIC ACID, ...
著者Zeng, H, Dong, A, Frommlet, A, Seitova, A, Loppnau, P, Ackloo, S, Arrowsmith, C.H, Edwards, A.M, Halabelian, L, Structural Genomics Consortium (SGC)
登録日2024-04-05
公開日2024-06-12
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Co-crystal structure of human DDB1 bound to fragment UB028669
To be published
2FS6
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BU of 2fs6 by Molmil
Crystal Structure of Apo-Cellular Retinoic Acid Binding Protein Type II At 1.35 Angstroms Resolution
分子名称: ACETATE ION, CHLORIDE ION, Cellular retinoic acid-binding protein 2, ...
著者Vaezeslami, S, Geiger, J.H.
登録日2006-01-21
公開日2006-09-19
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.35 Å)
主引用文献The structure of Apo-wild-type cellular retinoic acid binding protein II at 1.4 A and its relationship to ligand binding and nuclear translocation.
J.Mol.Biol., 363, 2006
9BB1
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BU of 9bb1 by Molmil
Backbone Modification in the GA Module of Protein PAB: Wild-type Sequence
分子名称: Peptostreptococcal albumin-binding protein
著者Lin, Y, Horne, W.S.
登録日2024-04-05
公開日2024-06-05
実験手法SOLUTION NMR
主引用文献Backbone Modification in a Protein Hydrophobic Core.
Chemistry, 2024
9EP4
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BU of 9ep4 by Molmil
Structure of Integrator subcomplex INTS5/8/15
分子名称: Integrator complex subunit 15, Integrator complex subunit 5, Integrator complex subunit 8
著者Razew, M, Galej, W.P.
登録日2024-03-17
公開日2024-06-12
実験手法ELECTRON MICROSCOPY (3.2 Å)
主引用文献Structural basis of the Integrator complex assembly and association with transcription factors.
Mol.Cell, 2024
1MFL
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BU of 1mfl by Molmil
The Structure of ERBIN PDZ domain bound to the Carboxy-terminal tail of the ErbB2 Receptor
分子名称: Erb-B2 INTERACTING PROTEIN, PHOSPHORYLATED Erb-B2 carboxyl-terminal fragment.
著者Birrane, G, Chung, J, Ladias, J.A.
登録日2002-08-12
公開日2003-01-21
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.88 Å)
主引用文献Novel mode of ligand recognition by the erbin PDZ domain
J.Biol.Chem., 278, 2003
9BZB
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BU of 9bzb by Molmil
Crystal structure of metallo-hydrolase-like_MBL-fold protein from Salmonella typhimurium LT2
分子名称: 1,2-ETHANEDIOL, FORMIC ACID, SULFATE ION, ...
著者Kim, Y, Maltseva, N, Endres, M, Joachimiak, A, Center for Structural Biology of Infectious Diseases (CSBID)
登録日2024-05-24
公開日2024-06-05
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Crystal structure of metallo-hydrolase-like_MBL-fold protein from Salmonella typhimurium LT2
To Be Published
2G80
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BU of 2g80 by Molmil
Crystal structure of UTR4 protein (Unknown transcript 4 protein) (yel038w) from Saccharomyces cerevisiae at 2.28 A resolution
分子名称: 2-{2-[2-(2-{2-[2-(2-ETHOXY-ETHOXY)-ETHOXY]-ETHOXY}-ETHOXY)-ETHOXY]-ETHOXY}-ETHANOL, GLYCEROL, MAGNESIUM ION, ...
著者Joint Center for Structural Genomics (JCSG)
登録日2006-03-01
公開日2006-03-28
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.28 Å)
主引用文献Crystal structure of UTR4 protein (Unknown transcript 4 protein) (yel038w) from Saccharomyces cerevisiae at 2.28 A resolution
To be published
9BCZ
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BU of 9bcz by Molmil
Chicken 1-phosphatidylinositol 4,5-bisphosphate phosphodiesterase zeta-1 (PLCZ1) in complex with calcium and phosphorylated threonine
分子名称: 1-phosphatidylinositol 4,5-bisphosphate phosphodiesterase zeta-1, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, CALCIUM ION, ...
著者Edwards, M.M, Dong, A, Theo-Emegano, N, Seitova, A, Loppnau, P, Leung, R, Li, H, Ilyassov, O, Edwards, A.M, Arrowsmith, C.H, Structural Genomics Consortium, Structural Genomics Consortium (SGC)
登録日2024-04-10
公開日2024-05-15
実験手法X-RAY DIFFRACTION (1.99 Å)
主引用文献Chicken 1-phosphatidylinositol 4,5-bisphosphate phosphodiesterase zeta-1 (PLCZ1) in complex with calcium and phosphorylated threonine
To be published
2FSY
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BU of 2fsy by Molmil
Bacteriophage HK97 Pepsin-treated Expansion Intermediate IV
分子名称: major capsid protein
著者Gan, L, Speir, J.A, Conway, J.F, Lander, G, Cheng, N, Firek, B.A, Hendrix, R.W, Duda, R.L, Liljas, L, Johnson, J.E.
登録日2006-01-23
公開日2006-02-07
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (3.8 Å)
主引用文献Capsid Conformational Sampling in HK97 Maturation Visualized by X-Ray Crystallography and Cryo-EM.
Structure, 14, 2006
1MFT
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BU of 1mft by Molmil
Crystal Structure Of Four-Helix Bundle Model
分子名称: Four-helix bundle model, ZINC ION
著者Lahr, S.J, Stayrook, S.E, North, B, Kaplan, J, Geremia, S, DeGrado, W.
登録日2002-08-13
公開日2004-01-20
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Analysis and Design of Turns in alpha-Helical Hairpins
J.Mol.Biol., 346, 2005
2G8J
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BU of 2g8j by Molmil
Calpain 1 proteolytic core in complex with SNJ-1945, a alpha-ketoamide-type inhibitor.
分子名称: ((1S)-1-((((1S)-1-BENZYL-3-(CYCLOPROPYLAMINO)-2,3-DIOXOPROPYL)AMINO)CARBONYL)-3-METHYLBUTYL)CARBAMIC ACID 5-METHOXY-3-OXAPENTYL ESTER, CALCIUM ION, Calpain-1 catalytic subunit
著者Cuerrier, D, Moldoveanu, T, Davies, P.L, Campbell, R.L.
登録日2006-03-02
公開日2006-06-06
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.61 Å)
主引用文献Calpain Inhibition by alpha-Ketoamide and Cyclic Hemiacetal Inhibitors Revealed by X-ray Crystallography
Biochemistry, 45, 2006
9EQK
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BU of 9eqk by Molmil
WWP1 WW2-2,3-linker-WW3-WW4-HECT (WWP1-2L34H) with ordered WW2 domain
分子名称: NEDD4-like E3 ubiquitin-protein ligase WWP1
著者Dudey, A.P, Hemmings, A.M.
登録日2024-03-21
公開日2024-05-15
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Expanding the Inhibitor Space of the WWP1 and WWP2 HECT E3 Ligases
To Be Published
9EY3
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BU of 9ey3 by Molmil
The FK1 domain of FKBP51 in complex with (3S,11S,11aS)-12-((3,5-dichlorophenyl)sulfonyl)-5-oxo-11-vinyldecahydro-1H-6,10-epiminopyrrolo[1,2-a]azonine-3-carboxylic acid
分子名称: (1~{S},4~{S},7~{S},8~{S},9~{R})-13-[3,5-bis(chloranyl)phenyl]sulfonyl-8-ethenyl-2-oxidanylidene-3,13-diazatricyclo[7.3.1.0^{3,7}]tridecane-4-carboxylic acid, Peptidyl-prolyl cis-trans isomerase FKBP5
著者Meyners, C, Krajczy, P, Hausch, F.
登録日2024-04-09
公開日2024-06-12
実験手法X-RAY DIFFRACTION (1.16 Å)
主引用文献Structure-Based Design of Ultrapotent Tricyclic Ligands for FK506-Binding proteins.
Chemistry, 2024
9FA4
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BU of 9fa4 by Molmil
Structure of the Integrator arm module containing subunits INTS10/13/14/15 (state 1)
分子名称: Integrator complex subunit 10, Integrator complex subunit 13, Integrator complex subunit 14, ...
著者Razew, M, Galej, W.P.
登録日2024-05-10
公開日2024-06-12
実験手法ELECTRON MICROSCOPY (4 Å)
主引用文献Structural basis of the Integrator complex assembly and association with transcription factors.
Mol.Cell, 2024
8Y95
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BU of 8y95 by Molmil
Structure of NET-NE in Occluded state
分子名称: CHLORIDE ION, Noradrenaline, SODIUM ION, ...
著者Zhang, H, Xu, H.E, Jiang, Y.
登録日2024-02-06
公開日2024-05-29
最終更新日2024-07-03
実験手法ELECTRON MICROSCOPY (3.24 Å)
主引用文献Dimerization and antidepressant recognition at noradrenaline transporter.
Nature, 630, 2024
9BRT
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BU of 9brt by Molmil
Intact V-ATPase State 1 and synaptophysin complex in mouse brain isolated synaptic vesicles
分子名称: Renin receptor cytoplasmic fragment, Ribonuclease kappa, Synaptophysin, ...
著者Wang, C, Jiang, W, Yang, K, Wang, X, Guo, Q, Brunger, A.T.
登録日2024-05-11
公開日2024-06-19
実験手法ELECTRON MICROSCOPY (4.3 Å)
主引用文献Structure and topography of the synaptic V-ATPase-synaptophysin complex.
Nature, 2024
9BOL
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BU of 9bol by Molmil
Crystal structure of the complex between VHL, ElonginB, ElonginC, and compound 5
分子名称: (4R)-1-[(2S)-2-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-3,3-dimethylbutanoyl]-4-hydroxy-N-{[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl}-L-prolinamide, 1,2-ETHANEDIOL, CHLORIDE ION, ...
著者Murray, J.M, Wu, H, Fuhrmann, J, Fairbrother, W.J, DiPasquale, A.
登録日2024-05-03
公開日2024-05-29
実験手法X-RAY DIFFRACTION (1.99 Å)
主引用文献Potency-enhanced peptidomimetic VHL ligands with improved oral bioavailability
To Be Published
9BVS
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BU of 9bvs by Molmil
NMR structure of TLP-1 in solution
分子名称: Temporin-1Tl
著者Jia, R, McShan, A.C.
登録日2024-05-20
公開日2024-06-05
実験手法SOLUTION NMR
主引用文献Design and Development of Temporin L Analogues to Inhibit the Main Protease of SARS-CoV-2
To Be Published
9EOU
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BU of 9eou by Molmil
Crystal Structure of the b1b2 domains from Human Neuropilin-1 in complex with a peptide.
分子名称: Neuropilin-1, Osteopontin
著者Caing-Carlsson, R, Duelli, A, Walse, B.
登録日2024-03-15
公開日2024-06-26
実験手法X-RAY DIFFRACTION (1.55 Å)
主引用文献Identification of an osteopontin-derived peptide that binds neuropilin-1 and activates vascular repair responses and angiogenesis.
Pharmacol Res, 205, 2024
9C8S
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BU of 9c8s by Molmil
CryoEM structure of Cryptococcus neoformans H99 Acetyl-CoA Synthetase in complex with adenosine-5'-ethylphosphate
分子名称: 5'-O-[(S)-ethoxy(hydroxy)phosphoryl]adenosine, Acetyl-coenzyme A synthetase
著者Xu, Z, Schnicker, N.J, Jezeski, A.J, Krysan, D.J.
登録日2024-06-12
公開日2024-07-03
実験手法ELECTRON MICROSCOPY (2.37 Å)
主引用文献CryoEM structure of Cryptococcus neoformans H99 Acetyl-CoA Synthetase in complex with adenosine-5'-ethylphosphate
To Be Published
7LYV
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BU of 7lyv by Molmil
Crystal structure of the HCMV pentamer-specific antibody 1-103
分子名称: 1-103 Fab Heavy Chain, 1-103 Fab Light Chain
著者Wrapp, D, Jones, H.G, McLellan, J.S.
登録日2021-03-08
公開日2021-08-11
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structural basis for HCMV Pentamer recognition by neuropilin 2 and neutralizing antibodies.
Sci Adv, 8, 2022
9BRB
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BU of 9brb by Molmil
Synaptic Vesicle V-ATPase with synaptophysin and SidK, State 1
分子名称: ATPase H+-transporting V1 subunit D, ATPase, H+ transporting, ...
著者Coupland, C.E, Rubinstein, J.L.
登録日2024-05-11
公開日2024-06-26
最終更新日2024-07-03
実験手法ELECTRON MICROSCOPY (3.6 Å)
主引用文献High-resolution electron cryomicroscopy of V-ATPase in native synaptic vesicles.
Science, 2024
9FEF
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BU of 9fef by Molmil
Cryo-EM structure of Trypanosoma cruzi (MDH)4-PEX5 complex
分子名称: Peroxisome targeting signal 1 receptor, malate dehydrogenase
著者Lipinski, O, Sonani, R.R, Blat, A, Jemiola-Rzeminska, M, Patel, S.N, Sood, T, Dubin, G.
登録日2024-05-19
公開日2024-05-29
実験手法ELECTRON MICROSCOPY (2.98 Å)
主引用文献Cryo-EM structure of Trypanosoma cruzi (MDH)4-PEX5 complex
To Be Published
9BZN
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BU of 9bzn by Molmil
High resolution structure of class A Beta-lactamase from Bordetella bronchiseptica RB50
分子名称: FORMIC ACID, SULFATE ION, class A Beta-lactamase, ...
著者Maltseva, N, Kim, Y, Endres, M, Joachimiak, A, Center for Structural Biology of Infectious Diseases (CSBID)
登録日2024-05-24
公開日2024-06-12
実験手法X-RAY DIFFRACTION (1.05 Å)
主引用文献High resolution structure of class A Beta-lactamase from Bordetella bronchiseptica RB50
To Be Published
9B55
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Ubiquitin E2-Ub-E3 HECT tetrahedral transthiolation intermediate mimic - state 1
分子名称: 4-aminobutanenitrile, E3 ubiquitin-protein ligase pub2, Ubiquitin, ...
著者Kochanczyk, T, Lima, C.D.
登録日2024-03-22
公開日2024-06-05
実験手法ELECTRON MICROSCOPY (3.23 Å)
主引用文献Structural basis for transthiolation intermediates in the ubiquitin pathway
To be published

222415

件を2024-07-10に公開中

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