7TCP
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![BU of 7tcp by Molmil](/molmil-images/mine/7tcp) | Structure of Xenopus KCNQ1-CaM | 分子名称: | CALCIUM ION, Calmodulin-1, Potassium voltage-gated channel subfamily KQT member 1 | 著者 | Willegems, K, Kyriakis, E, Van Petegem, F, Eldstrom, J, Fedida, D. | 登録日 | 2021-12-27 | 公開日 | 2022-07-06 | 最終更新日 | 2024-02-28 | 実験手法 | ELECTRON MICROSCOPY (3.84 Å) | 主引用文献 | Structural and electrophysiological basis for the modulation of KCNQ1 channel currents by ML277. Nat Commun, 13, 2022
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7TJ8
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![BU of 7tj8 by Molmil](/molmil-images/mine/7tj8) | Cryo-EM structure of the human Nax channel in complex with beta3 solved in nanodiscs | 分子名称: | (1S)-2-{[(2-AMINOETHOXY)(HYDROXY)PHOSPHORYL]OXY}-1-[(PALMITOYLOXY)METHYL]ETHYL STEARATE, (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate, 2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Noland, C.L, Kschonsak, M, Ciferri, C, Payandeh, J. | 登録日 | 2022-01-14 | 公開日 | 2022-03-30 | 実験手法 | ELECTRON MICROSCOPY (3.2 Å) | 主引用文献 | Structure-guided unlocking of Na X reveals a non-selective tetrodotoxin-sensitive cation channel. Nat Commun, 13, 2022
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7TJ9
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![BU of 7tj9 by Molmil](/molmil-images/mine/7tj9) | Cryo-EM structure of the human Nax channel in complex with beta3 solved in GDN | 分子名称: | (1S)-2-{[(2-AMINOETHOXY)(HYDROXY)PHOSPHORYL]OXY}-1-[(PALMITOYLOXY)METHYL]ETHYL STEARATE, (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate, 2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Noland, C.L, Kschonsak, M, Ciferri, C, Payandeh, J. | 登録日 | 2022-01-14 | 公開日 | 2022-03-30 | 実験手法 | ELECTRON MICROSCOPY (2.9 Å) | 主引用文献 | Structure-guided unlocking of Na X reveals a non-selective tetrodotoxin-sensitive cation channel. Nat Commun, 13, 2022
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7UKD
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![BU of 7ukd by Molmil](/molmil-images/mine/7ukd) | Human Kv4.2-KChIP2 channel complex in an inactivated state, class 2, transmembrane region | 分子名称: | POTASSIUM ION, Potassium voltage-gated channel subfamily D member 2 | 著者 | Zhao, H, Dai, Y, Lee, C.H. | 登録日 | 2022-04-01 | 公開日 | 2022-06-29 | 最終更新日 | 2024-02-14 | 実験手法 | ELECTRON MICROSCOPY (2.88 Å) | 主引用文献 | Activation and closed-state inactivation mechanisms of the human voltage-gated K V 4 channel complexes. Mol.Cell, 82, 2022
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7UKC
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![BU of 7ukc by Molmil](/molmil-images/mine/7ukc) | Human Kv4.2-KChIP2 channel complex in an inactivated state, class 1, transmembrane region | 分子名称: | POTASSIUM ION, Potassium voltage-gated channel subfamily D member 2 | 著者 | Zhao, H, Dai, Y, Lee, C.H. | 登録日 | 2022-04-01 | 公開日 | 2022-06-29 | 最終更新日 | 2024-02-14 | 実験手法 | ELECTRON MICROSCOPY (3 Å) | 主引用文献 | Activation and closed-state inactivation mechanisms of the human voltage-gated K V 4 channel complexes. Mol.Cell, 82, 2022
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7UKF
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![BU of 7ukf by Molmil](/molmil-images/mine/7ukf) | Human Kv4.2-KChIP2 channel complex in a putative resting state, transmembrane region | 分子名称: | MERCURY (II) ION, POTASSIUM ION, Potassium voltage-gated channel subfamily D member 2 | 著者 | Zhao, H, Dai, Y, Lee, C.H. | 登録日 | 2022-04-01 | 公開日 | 2022-06-29 | 最終更新日 | 2024-02-14 | 実験手法 | ELECTRON MICROSCOPY (3.02 Å) | 主引用文献 | Activation and closed-state inactivation mechanisms of the human voltage-gated K V 4 channel complexes. Mol.Cell, 82, 2022
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7UK5
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![BU of 7uk5 by Molmil](/molmil-images/mine/7uk5) | |
7UKE
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![BU of 7uke by Molmil](/molmil-images/mine/7uke) | |
7UKH
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![BU of 7ukh by Molmil](/molmil-images/mine/7ukh) | Human Kv4.2-KChIP2-DPP6 channel complex in an open state, intracellular region | 分子名称: | CALCIUM ION, Isoform 2 of Kv channel-interacting protein 2, Potassium voltage-gated channel subfamily D member 2, ... | 著者 | Zhao, H, Dai, Y, Lee, C.H. | 登録日 | 2022-04-01 | 公開日 | 2022-06-29 | 最終更新日 | 2024-02-14 | 実験手法 | ELECTRON MICROSCOPY (2.33 Å) | 主引用文献 | Activation and closed-state inactivation mechanisms of the human voltage-gated K V 4 channel complexes. Mol.Cell, 82, 2022
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8DFL
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![BU of 8dfl by Molmil](/molmil-images/mine/8dfl) | |
8DDV
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![BU of 8ddv by Molmil](/molmil-images/mine/8ddv) | Cryo-EM structure of TRPM3 ion channel in the presence of PIP2, state4 | 分子名称: | (3beta,14beta,17beta,25R)-3-[4-methoxy-3-(methoxymethyl)butoxy]spirost-5-en, 1,2-DIACYL-GLYCEROL-3-SN-PHOSPHATE, SODIUM ION, ... | 著者 | Zhao, C, MacKinnon, R. | 登録日 | 2022-06-19 | 公開日 | 2022-11-02 | 最終更新日 | 2024-06-12 | 実験手法 | ELECTRON MICROSCOPY (3.2 Å) | 主引用文献 | Structural and functional analyses of a GPCR-inhibited ion channel TRPM3. Neuron, 111, 2023
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8DDQ
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![BU of 8ddq by Molmil](/molmil-images/mine/8ddq) | cryo-EM structure of TRPM3 ion channel in the presence of soluble Gbg, focused on channel | 分子名称: | (3beta,14beta,17beta,25R)-3-[4-methoxy-3-(methoxymethyl)butoxy]spirost-5-en, 1,2-DIACYL-GLYCEROL-3-SN-PHOSPHATE, SODIUM ION, ... | 著者 | Zhao, C, MacKinnon, R. | 登録日 | 2022-06-18 | 公開日 | 2022-11-02 | 最終更新日 | 2024-06-12 | 実験手法 | ELECTRON MICROSCOPY (2.7 Å) | 主引用文献 | Structural and functional analyses of a GPCR-inhibited ion channel TRPM3. Neuron, 111, 2023
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8DDS
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![BU of 8dds by Molmil](/molmil-images/mine/8dds) | cryo-EM structure of TRPM3 ion channel in the presence of PIP2, state1 | 分子名称: | (3beta,14beta,17beta,25R)-3-[4-methoxy-3-(methoxymethyl)butoxy]spirost-5-en, 1,2-DIACYL-GLYCEROL-3-SN-PHOSPHATE, SODIUM ION, ... | 著者 | Zhao, C, MacKinnon, R. | 登録日 | 2022-06-18 | 公開日 | 2022-11-02 | 最終更新日 | 2024-06-12 | 実験手法 | ELECTRON MICROSCOPY (3.5 Å) | 主引用文献 | Structural and functional analyses of a GPCR-inhibited ion channel TRPM3. Neuron, 111, 2023
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8DDR
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![BU of 8ddr by Molmil](/molmil-images/mine/8ddr) | cryo-EM structure of TRPM3 ion channel in the absence of PIP2 | 分子名称: | (3beta,14beta,17beta,25R)-3-[4-methoxy-3-(methoxymethyl)butoxy]spirost-5-en, 1,2-DIACYL-GLYCEROL-3-SN-PHOSPHATE, SODIUM ION, ... | 著者 | Zhao, C, MacKinnon, R. | 登録日 | 2022-06-18 | 公開日 | 2022-11-02 | 最終更新日 | 2024-06-12 | 実験手法 | ELECTRON MICROSCOPY (3.2 Å) | 主引用文献 | Structural and functional analyses of a GPCR-inhibited ion channel TRPM3. Neuron, 111, 2023
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8E4P
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![BU of 8e4p by Molmil](/molmil-images/mine/8e4p) | Mouse TRPM8 structure determined in the ligand- and PI(4,5)P2-free condition, Class I , C0 state | 分子名称: | CHOLESTEROL HEMISUCCINATE, Transient receptor potential cation channel subfamily M member 8 | 著者 | Yin, Y, Zhang, F, Feng, S, Butay, K.J, Borgnia, M.J, Im, W, Lee, S.-Y. | 登録日 | 2022-08-18 | 公開日 | 2022-10-26 | 最終更新日 | 2024-06-12 | 実験手法 | ELECTRON MICROSCOPY (3.59 Å) | 主引用文献 | Activation mechanism of the mouse cold-sensing TRPM8 channel by cooling agonist and PIP 2. Science, 378, 2022
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8E4L
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![BU of 8e4l by Molmil](/molmil-images/mine/8e4l) | The open state mouse TRPM8 structure in complex with the cooling agonist C3, AITC, and PI(4,5)P2 | 分子名称: | 3-isothiocyanatoprop-1-ene, CALCIUM ION, Transient receptor potential cation channel subfamily M member 8, ... | 著者 | Yin, Y, Zhang, F, Feng, S, Butay, K.J, Borgnia, M.J, Im, W, Lee, S.-Y. | 登録日 | 2022-08-18 | 公開日 | 2022-10-26 | 実験手法 | ELECTRON MICROSCOPY (3.32 Å) | 主引用文献 | Activation mechanism of the mouse cold-sensing TRPM8 channel by cooling agonist and PIP 2. Science, 378, 2022
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8E4M
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![BU of 8e4m by Molmil](/molmil-images/mine/8e4m) | The intermediate C2-state mouse TRPM8 structure in complex with the cooling agonist C3 and PI(4,5)P2 | 分子名称: | CALCIUM ION, Transient receptor potential cation channel subfamily M member 8, [(2R)-2-octanoyloxy-3-[oxidanyl-[(1R,2R,3S,4R,5R,6S)-2,3,6-tris(oxidanyl)-4,5-diphosphonooxy-cyclohexyl]oxy-phosphoryl]oxy-propyl] octanoate, ... | 著者 | Yin, Y, Zhang, F, Feng, S, Butay, K.J, Borgnia, M.J, Im, W, Lee, S.-Y. | 登録日 | 2022-08-18 | 公開日 | 2022-10-26 | 最終更新日 | 2024-06-12 | 実験手法 | ELECTRON MICROSCOPY (3.44 Å) | 主引用文献 | Activation mechanism of the mouse cold-sensing TRPM8 channel by cooling agonist and PIP 2. Science, 378, 2022
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8E4O
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![BU of 8e4o by Molmil](/molmil-images/mine/8e4o) | The closed C1-state mouse TRPM8 structure in complex with putative PI(4,5)P2 | 分子名称: | Transient receptor potential cation channel subfamily M member 8, [(2R)-2-octanoyloxy-3-[oxidanyl-[(1R,2R,3S,4R,5R,6S)-2,3,6-tris(oxidanyl)-4,5-diphosphonooxy-cyclohexyl]oxy-phosphoryl]oxy-propyl] octanoate | 著者 | Yin, Y, Zhang, F, Feng, S, Butay, K.J, Borgnia, M.J, Im, W, Lee, S.-Y. | 登録日 | 2022-08-18 | 公開日 | 2022-10-26 | 実験手法 | ELECTRON MICROSCOPY (3.43 Å) | 主引用文献 | Activation mechanism of the mouse cold-sensing TRPM8 channel by cooling agonist and PIP 2. Science, 378, 2022
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8E4Q
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![BU of 8e4q by Molmil](/molmil-images/mine/8e4q) | The closed C0-state flycatcher TRPM8 structure in complex with PI(4,5)P2 | 分子名称: | Transient receptor potential cation channel subfamily M member 8, [(2R)-2-octanoyloxy-3-[oxidanyl-[(1R,2R,3S,4R,5R,6S)-2,3,6-tris(oxidanyl)-4,5-diphosphonooxy-cyclohexyl]oxy-phosphoryl]oxy-propyl] octanoate | 著者 | Yin, Y, Zhang, F, Feng, S, Butay, K.J, Borgnia, M.J, Im, W, Lee, S.-Y. | 登録日 | 2022-08-18 | 公開日 | 2022-10-26 | 最終更新日 | 2024-06-12 | 実験手法 | ELECTRON MICROSCOPY (3.51 Å) | 主引用文献 | Activation mechanism of the mouse cold-sensing TRPM8 channel by cooling agonist and PIP 2. Science, 378, 2022
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8ED7
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![BU of 8ed7 by Molmil](/molmil-images/mine/8ed7) | cryo-EM structure of TRPM3 ion channel in apo state | 分子名称: | (3beta,14beta,17beta,25R)-3-[4-methoxy-3-(methoxymethyl)butoxy]spirost-5-en, Transient receptor potential cation channel, subfamily M, ... | 著者 | Zhao, C, MacKinnon, R. | 登録日 | 2022-09-03 | 公開日 | 2022-11-02 | 最終更新日 | 2023-01-18 | 実験手法 | ELECTRON MICROSCOPY (3.7 Å) | 主引用文献 | Structural and functional analyses of a GPCR-inhibited ion channel TRPM3. Neuron, 111, 2023
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8ED9
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![BU of 8ed9 by Molmil](/molmil-images/mine/8ed9) | cryo-EM structure of TRPM3 ion channel in the presence with PIP2 and PregS, state 2 | 分子名称: | (3beta,14beta,17beta,25R)-3-[4-methoxy-3-(methoxymethyl)butoxy]spirost-5-en, 1,2-DIACYL-GLYCEROL-3-SN-PHOSPHATE, SODIUM ION, ... | 著者 | Zhao, C, MacKinnon, R. | 登録日 | 2022-09-03 | 公開日 | 2022-11-09 | 最終更新日 | 2023-01-18 | 実験手法 | ELECTRON MICROSCOPY (3.4 Å) | 主引用文献 | Structural and functional analyses of a GPCR-inhibited ion channel TRPM3. Neuron, 111, 2023
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8E4N
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![BU of 8e4n by Molmil](/molmil-images/mine/8e4n) | The closed C1-state mouse TRPM8 structure in complex with PI(4,5)P2 | 分子名称: | Transient receptor potential cation channel subfamily M member 8, [(2R)-2-octanoyloxy-3-[oxidanyl-[(1R,2R,3S,4R,5R,6S)-2,3,6-tris(oxidanyl)-4,5-diphosphonooxy-cyclohexyl]oxy-phosphoryl]oxy-propyl] octanoate | 著者 | Yin, Y, Zhang, F, Feng, S, Butay, K.J, Borgnia, M.J, Im, W, Lee, S.-Y. | 登録日 | 2022-08-18 | 公開日 | 2022-10-26 | 実験手法 | ELECTRON MICROSCOPY (3.07 Å) | 主引用文献 | Activation mechanism of the mouse cold-sensing TRPM8 channel by cooling agonist and PIP 2. Science, 378, 2022
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8ED8
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![BU of 8ed8 by Molmil](/molmil-images/mine/8ed8) | cryo-EM structure of TRPM3 ion channel in the presence of PIP2 and PregS, state 1 | 分子名称: | (3beta,14beta,17beta,25R)-3-[4-methoxy-3-(methoxymethyl)butoxy]spirost-5-en, 1,2-DIACYL-GLYCEROL-3-SN-PHOSPHATE, SODIUM ION, ... | 著者 | Zhao, C, MacKinnon, R. | 登録日 | 2022-09-03 | 公開日 | 2022-11-02 | 最終更新日 | 2023-01-18 | 実験手法 | ELECTRON MICROSCOPY (3.2 Å) | 主引用文献 | Structural and functional analyses of a GPCR-inhibited ion channel TRPM3. Neuron, 111, 2023
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8EAR
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![BU of 8ear by Molmil](/molmil-images/mine/8ear) | Structure of the full-length IP3R1 channel determined in the presence of Calcium/IP3/ATP | 分子名称: | (9R,11S)-9-({[(1S)-1-HYDROXYHEXADECYL]OXY}METHYL)-2,2-DIMETHYL-5,7,10-TRIOXA-2LAMBDA~5~-AZA-6LAMBDA~5~-PHOSPHAOCTACOSANE-6,6,11-TRIOL, ADENOSINE-5'-TRIPHOSPHATE, CALCIUM ION, ... | 著者 | Fan, G, Baker, M.R, Terry, L.E, Arige, V, Chen, M, Seryshev, A.B, Baker, M.L, Ludtke, S.J, Yule, D.I, Serysheva, I.I. | 登録日 | 2022-08-29 | 公開日 | 2022-11-23 | 実験手法 | ELECTRON MICROSCOPY (3.5 Å) | 主引用文献 | Conformational motions and ligand-binding underlying gating and regulation in IP 3 R channel. Nat Commun, 13, 2022
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8EAQ
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![BU of 8eaq by Molmil](/molmil-images/mine/8eaq) | Structure of the full-length IP3R1 channel determined at high Ca2+ | 分子名称: | (9R,11S)-9-({[(1S)-1-HYDROXYHEXADECYL]OXY}METHYL)-2,2-DIMETHYL-5,7,10-TRIOXA-2LAMBDA~5~-AZA-6LAMBDA~5~-PHOSPHAOCTACOSANE-6,6,11-TRIOL, CALCIUM ION, Inositol 1,4,5-trisphosphate receptor type 1, ... | 著者 | Fan, G, Baker, M.R, Terry, L.E, Arige, V, Chen, M, Seryshev, A.B, Baker, M.L, Ludtke, S.J, Yule, D.I, Serysheva, I.I. | 登録日 | 2022-08-29 | 公開日 | 2022-11-23 | 実験手法 | ELECTRON MICROSCOPY (3.26 Å) | 主引用文献 | Conformational motions and ligand-binding underlying gating and regulation in IP 3 R channel. Nat Commun, 13, 2022
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