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6QDV
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BU of 6qdv by Molmil
Human post-catalytic P complex spliceosome
分子名称: 116 kDa U5 small nuclear ribonucleoprotein component, ADENOSINE-5'-TRIPHOSPHATE, ATP-dependent RNA helicase DHX8, ...
著者Fica, S.M, Oubridge, C, Wilkinson, M.E, Newman, A.J, Nagai, K.
登録日2019-01-03
公開日2019-02-20
最終更新日2024-11-13
実験手法ELECTRON MICROSCOPY (3.3 Å)
主引用文献A human postcatalytic spliceosome structure reveals essential roles of metazoan factors for exon ligation.
Science, 363, 2019
5XJC
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BU of 5xjc by Molmil
Cryo-EM structure of the human spliceosome just prior to exon ligation at 3.6 angstrom
分子名称: 116 kDa U5 small nuclear ribonucleoprotein component, ADENOSINE-5'-DIPHOSPHATE, ADENOSINE-5'-TRIPHOSPHATE, ...
著者Zhang, X, Yan, C, Hang, J, Finci, I.L, Lei, J, Shi, Y.
登録日2017-04-30
公開日2017-07-05
最終更新日2024-11-20
実験手法ELECTRON MICROSCOPY (3.6 Å)
主引用文献An Atomic Structure of the Human Spliceosome
Cell, 169, 2017
5I3C
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BU of 5i3c by Molmil
Crystal structure of E.coli purine nucleoside phosphorylase with acycloguanosine
分子名称: 9-HYROXYETHOXYMETHYLGUANINE, Purine nucleoside phosphorylase DeoD-type, SULFATE ION
著者Timofeev, V.I, Abramchik, Y.A, Esipov, R.S, Kuranova, I.P.
登録日2016-02-10
公開日2017-02-22
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.32 Å)
主引用文献Crystal structure of Escherichia coli purine nucleoside phosphorylase complexed with acyclovir.
Acta Crystallogr F Struct Biol Commun, 74, 2018
5IU6
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BU of 5iu6 by Molmil
Crystal structure of E.coli purine nucleoside phosphorylase with 7-deazahypoxanthine
分子名称: 7H-pyrrolo[2,3-d]pyrimidin-4-ol, Purine nucleoside phosphorylase DeoD-type, SULFATE ION
著者Timofeev, V.I, Abramchik, Y.A, Esipov, R.S, Kuranova, I.P.
登録日2016-03-17
公開日2017-04-05
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.51 Å)
主引用文献Crystal structure of Escherichia coli purine nucleoside phosphorylase in complex with 7-deazahypoxanthine.
Acta Crystallogr F Struct Biol Commun, 74, 2018
6PX1
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BU of 6px1 by Molmil
Set2 bound to nucleosome
分子名称: DNA (149-MER), Histone H2B 1.1, Histone H3, ...
著者Halic, M, Bilokapic, S.
登録日2019-07-24
公開日2019-08-28
最終更新日2025-05-21
実験手法ELECTRON MICROSCOPY (3.3 Å)
主引用文献Nucleosome and ubiquitin position Set2 to methylate H3K36.
Nat Commun, 10, 2019
5Z57
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BU of 5z57 by Molmil
Cryo-EM structure of the human activated spliceosome (late Bact) at 6.5 angstrom
分子名称: 116 kDa U5 small nuclear ribonucleoprotein component, ALANINE, BUD13 homolog, ...
著者Zhang, X, Yan, C, Zhan, X, Li, L, Lei, J, Shi, Y.
登録日2018-01-17
公開日2018-09-19
最終更新日2024-10-30
実験手法ELECTRON MICROSCOPY (6.5 Å)
主引用文献Structure of the human activated spliceosome in three conformational states.
Cell Res., 28, 2018
6NZO
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BU of 6nzo by Molmil
Set2 bound to nucleosome
分子名称: DNA (149-MER), Histone H2B 1.1, Histone H3, ...
著者Halic, M, Bilokapic, S.
登録日2019-02-14
公開日2019-08-28
最終更新日2025-06-04
実験手法ELECTRON MICROSCOPY (3.8 Å)
主引用文献Nucleosome and ubiquitin position Set2 to methylate H3K36.
Nat Commun, 10, 2019
6PX3
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BU of 6px3 by Molmil
Set2 bound to nucleosome
分子名称: DNA (145-MER), Histone H2B 1.1, Histone H3, ...
著者Halic, M, Bilokapic, S.
登録日2019-07-24
公開日2019-08-28
最終更新日2025-05-28
実験手法ELECTRON MICROSCOPY (4.1 Å)
主引用文献Nucleosome and ubiquitin position Set2 to methylate H3K36.
Nat Commun, 10, 2019
5IFK
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BU of 5ifk by Molmil
Purine nucleoside phosphorylase
分子名称: HYPOXANTHINE, Purine nucleoside phosphorylase
著者Thakur, K.G, Priyanka, A.
登録日2016-02-26
公開日2017-03-01
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (1.967 Å)
主引用文献Functional and Structural Characterization of Purine Nucleoside Phosphorylase from Kluyveromyces lactis and Its Potential Applications in Reducing Purine Content in Food
PLoS ONE, 11, 2016
5Z56
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BU of 5z56 by Molmil
cryo-EM structure of a human activated spliceosome (mature Bact) at 5.1 angstrom.
分子名称: 116 kDa U5 small nuclear ribonucleoprotein component, BUD13 homolog, Cell division cycle 5-like protein, ...
著者Zhang, X, Yan, C, Zhan, X, Li, L, Lei, J, Shi, Y.
登録日2018-01-17
公開日2018-09-19
最終更新日2024-11-13
実験手法ELECTRON MICROSCOPY (5.1 Å)
主引用文献Structure of the human activated spliceosome in three conformational states.
Cell Res., 28, 2018
5Z58
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BU of 5z58 by Molmil
Cryo-EM structure of a human activated spliceosome (early Bact) at 4.9 angstrom.
分子名称: 116 kDa U5 small nuclear ribonucleoprotein component, BUD13 homolog, Cell division cycle 5-like protein, ...
著者Zhang, X, Yan, C, Zhan, X, Li, L, Lei, J, Shi, Y.
登録日2018-01-17
公開日2018-09-19
最終更新日2024-11-06
実験手法ELECTRON MICROSCOPY (4.9 Å)
主引用文献Structure of the human activated spliceosome in three conformational states.
Cell Res., 28, 2018
5UGF
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BU of 5ugf by Molmil
Crystal structure of human purine nucleoside phosphorylase (F159Y) mutant complexed with DADMe-ImmG and phosphate
分子名称: 2-amino-7-{[(3R,4R)-3-hydroxy-4-(hydroxymethyl)pyrrolidin-1-yl]methyl}-3,5-dihydro-4H-pyrrolo[3,2-d]pyrimidin-4-one, PHOSPHATE ION, Purine nucleoside phosphorylase
著者Harijan, R.K, Cameron, S.A, Bonanno, J.B, Almo, S.C, Schramm, V.L.
登録日2017-01-08
公開日2017-06-21
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Catalytic-site design for inverse heavy-enzyme isotope effects in human purine nucleoside phosphorylase.
Proc. Natl. Acad. Sci. U.S.A., 114, 2017
7OOZ
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BU of 7ooz by Molmil
Purine nucleoside phosphorylase(DeoD-type) from H. pylori with 6-benzyloxo-2-chloropurine
分子名称: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, 6-benzyloxo-2-chloropurine, GLYCEROL, ...
著者Narczyk, M, Stefanic, Z.
登録日2021-05-28
公開日2022-05-04
最終更新日2024-11-20
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Interactions of 2,6-substituted purines with purine nucleoside phosphorylase from Helicobacter pylori in solution and in the crystal, and the effects of these compounds on cell cultures of this bacterium.
J Enzyme Inhib Med Chem, 37, 2022
7OP9
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BU of 7op9 by Molmil
Purine nucleoside phosphorylase(DeoD-type) from H. pylori with 2,6-dichloropurine
分子名称: 2,6-bis(chloranyl)-7H-purine, IMIDAZOLE, MAGNESIUM ION, ...
著者Narczyk, M, Stefanic, Z.
登録日2021-05-31
公開日2022-05-04
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Interactions of 2,6-substituted purines with purine nucleoside phosphorylase from Helicobacter pylori in solution and in the crystal, and the effects of these compounds on cell cultures of this bacterium.
J Enzyme Inhib Med Chem, 37, 2022
7OPA
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BU of 7opa by Molmil
Purine nucleoside phosphorylase(DeoD-type) from H. pylori with 6-benzylthiopurine
分子名称: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, 6-benzylthio-2-chloropurine, GLYCEROL, ...
著者Narczyk, M, Stefanic, Z.
登録日2021-05-31
公開日2022-05-04
最終更新日2024-11-06
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Interactions of 2,6-substituted purines with purine nucleoside phosphorylase from Helicobacter pylori in solution and in the crystal, and the effects of these compounds on cell cultures of this bacterium.
J Enzyme Inhib Med Chem, 37, 2022
7OOY
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BU of 7ooy by Molmil
Purine nucleoside phosphorylase(DeoD-type) from H. pylori with 6-benzylthio-2-chloropurine
分子名称: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, 6-benzylthio-2-chloropurine, GLYCEROL, ...
著者Narczyk, M, Stefanic, Z.
登録日2021-05-28
公開日2022-05-04
最終更新日2024-11-20
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Interactions of 2,6-substituted purines with purine nucleoside phosphorylase from Helicobacter pylori in solution and in the crystal, and the effects of these compounds on cell cultures of this bacterium.
J Enzyme Inhib Med Chem, 37, 2022
5YZG
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BU of 5yzg by Molmil
The Cryo-EM Structure of Human Catalytic Step I Spliceosome (C complex) at 4.1 angstrom resolution
分子名称: 116 kDa U5 small nuclear ribonucleoprotein component, ADENOSINE-5'-DIPHOSPHATE, ADENOSINE-5'-TRIPHOSPHATE, ...
著者Zhan, X, Yan, C, Zhang, X, Lei, J, Shi, Y.
登録日2017-12-14
公開日2018-08-08
最終更新日2024-10-23
実験手法ELECTRON MICROSCOPY (4.1 Å)
主引用文献Structure of a human catalytic step I spliceosome
Science, 359, 2018
8TZI
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BU of 8tzi by Molmil
Human equilibrative nucleoside transporter-1, JH-ENT-01 bound
分子名称: (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, 3-[4-[3-[3,4-dimethoxy-5-[[4-[oxidanyl(oxidanylidene)-$l^{4}-azanyl]phenyl]methoxy]phenyl]carbonyloxypropyl]-1,4-diazepan-1-yl]propyl 3,4,5-trimethoxybenzoate, Equilibrative nucleoside transporter 1
著者Wright, N.J, Lee, S.Y.
登録日2023-08-26
公開日2024-08-28
最終更新日2025-03-12
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Design of an equilibrative nucleoside transporter subtype 1 inhibitor for pain relief.
Nat Commun, 15, 2024
8PKI
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BU of 8pki by Molmil
Cryo-EM structure of NR5A2-nucleosome complex SHL+5.5
分子名称: DNA, Histone H2A, Histone H2B type 1-C/E/G, ...
著者Kobayashi, W, Sappler, A, Bollschweiler, D, Kummecke, M, Basquin, J, Arslantas, E, Ruangroengkulrith, S, Hornberger, R, Duderstadt, K, Tachibana, K.
登録日2023-06-26
公開日2024-02-28
最終更新日2024-05-29
実験手法ELECTRON MICROSCOPY (2.58 Å)
主引用文献Nucleosome-bound NR5A2 structure reveals pioneer factor mechanism by DNA minor groove anchor competition.
Nat.Struct.Mol.Biol., 31, 2024
8W7H
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BU of 8w7h by Molmil
Purine Nucleoside Phosphorylase in complex with MMV000848
分子名称: (2R)-1-(9H-carbazol-9-yl)-3-(cyclopentylamino)propan-2-ol, 1,2-ETHANEDIOL, PHOSPHATE ION, ...
著者Chung, Z, Lin, J.Q, Lescar, J.
登録日2023-08-30
公開日2024-01-17
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Identification and structural validation of purine nucleoside phosphorylase from Plasmodium falciparum as a target of MMV000848.
J.Biol.Chem., 300, 2023
7ZLW
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BU of 7zlw by Molmil
NME1 in complex with ADP
分子名称: ADENOSINE-5'-DIPHOSPHATE, Nucleoside diphosphate kinase A
著者Garcia-Saez, I, Iuso, D, Khochbin, S, Petosa, C.
登録日2022-04-15
公開日2023-08-09
最終更新日2024-10-16
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Nucleoside diphosphate kinases 1 and 2 regulate a protective liver response to a high-fat diet.
Sci Adv, 9, 2023
7ZTK
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BU of 7ztk by Molmil
NME1 in complex with CoA
分子名称: COENZYME A, Nucleoside diphosphate kinase A
著者Garcia-Saez, I, Iuso, D, Khochbin, S, Petosa, C.
登録日2022-05-10
公開日2023-08-09
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Nucleoside diphosphate kinases 1 and 2 regulate a protective liver response to a high-fat diet.
Sci Adv, 9, 2023
9FXE
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BU of 9fxe by Molmil
D204N mutant of Purine Nucleoside Phosphorylase from E.coli in complex with N2,3-etheno-2-aminopurine
分子名称: N,2,3-etheno-2-aminopurine, PHOSPHATE ION, Purine nucleoside phosphorylase DeoD-type
著者Narczyk, M, Stachelska-Wierzchowska, A, Wierzchowski, J.
登録日2024-07-01
公開日2024-10-30
実験手法X-RAY DIFFRACTION (2.12 Å)
主引用文献Interaction of Tri-Cyclic Nucleobase Analogs with Enzymes of Purine Metabolism: Xanthine Oxidase and Purine Nucleoside Phosphorylase.
Int J Mol Sci, 25, 2024
9FPE
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BU of 9fpe by Molmil
Wild type Purine Nucleoside Phosphorylase from E.coli in complex with N2,3-etheno-2-aminopurine
分子名称: GLYCEROL, N,2,3-etheno-2-aminopurine, PHOSPHATE ION, ...
著者Narczyk, M, Krystian, M, Stachelska-Wierzchowska, A, Wierzchowski, J.
登録日2024-06-13
公開日2024-10-30
実験手法X-RAY DIFFRACTION (1.35 Å)
主引用文献Interaction of Tri-Cyclic Nucleobase Analogs with Enzymes of Purine Metabolism: Xanthine Oxidase and Purine Nucleoside Phosphorylase.
Int J Mol Sci, 25, 2024
8PKJ
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BU of 8pkj by Molmil
Cryo-EM structure of the nucleosome containing Nr5a2 motif at SHL+5.5
分子名称: DNA, Histone H2A, Histone H2B, ...
著者Kobayashi, W, Sappler, A, Bollschweiler, D, Kummecke, M, Basquin, J, Arslantas, E, Ruangroengkulrith, S, Hornberger, R, Duderstadt, K, Tachibana, K.
登録日2023-06-26
公開日2024-02-28
最終更新日2024-05-29
実験手法ELECTRON MICROSCOPY (2.5 Å)
主引用文献Nucleosome-bound NR5A2 structure reveals pioneer factor mechanism by DNA minor groove anchor competition.
Nat.Struct.Mol.Biol., 31, 2024

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件を2025-07-09に公開中

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