8TZI
Human equilibrative nucleoside transporter-1, JH-ENT-01 bound
Summary for 8TZI
Entry DOI | 10.2210/pdb8tzi/pdb |
Descriptor | Equilibrative nucleoside transporter 1, (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, 3-[4-[3-[3,4-dimethoxy-5-[[4-[oxidanyl(oxidanylidene)-$l^{4}-azanyl]phenyl]methoxy]phenyl]carbonyloxypropyl]-1,4-diazepan-1-yl]propyl 3,4,5-trimethoxybenzoate, ... (4 entities in total) |
Functional Keywords | adenosine transport, adenosine reuptake inhibitor, nucleoside, hent1, equilibrative nucleoside transporter, slc29, transport protein-inhibitor complex, transport protein/inhibitor |
Biological source | Homo sapiens (human) |
Total number of polymer chains | 1 |
Total formula weight | 51729.74 |
Authors | |
Primary citation | Wright, N.J.,Lee, S.Y. Rational ENT1 inhibition as a pathway for neuropathic pain relief To Be Published, |
Experimental method | X-RAY DIFFRACTION (2.7 Å) |
Structure validation
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