8RWZ
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![BU of 8rwz by Molmil](/molmil-images/mine/8rwz) | Open non-crosslinked structure Brd4BD2-MZ1-(NEDD8)-CRL2VHL | 分子名称: | (2~{S},4~{R})-1-[(2~{S})-2-[2-[2-[2-[2-[2-[(9~{S})-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.0^{2,6}]trideca-2(6),4,7,10,12-pentaen-9-yl]ethanoylamino]ethoxy]ethoxy]ethoxy]ethanoylamino]-3,3-dimethyl-butanoyl]-~{N}-[[4-(4-methyl-2,3-dihydro-1,3-thiazol-5-yl)phenyl]methyl]-4-oxidanyl-pyrrolidine-2-carboxamide, Bromodomain-containing protein 4, Cullin-2, ... | 著者 | Ciulli, A, Crowe, C, Nakacone, M.A. | 登録日 | 2024-02-05 | 公開日 | 2024-03-06 | 実験手法 | ELECTRON MICROSCOPY (4 Å) | 主引用文献 | Open non-crosslinked structure Brd4BD2-MZ1-(NEDD8)-CRL2VHL To Be Published
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8ST7
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![BU of 8st7 by Molmil](/molmil-images/mine/8st7) | |
8ST9
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8ST8
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4UEL
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![BU of 4uel by Molmil](/molmil-images/mine/4uel) | UCH-L5 in complex with ubiquitin-propargyl bound to the RPN13 DEUBAD domain | 分子名称: | POLYUBIQUITIN-B, PROTEASOMAL UBIQUITIN RECEPTOR ADRM1, UBIQUITIN CARBOXYL-TERMINAL HYDROLASE ISOZYME L5 | 著者 | Sahtoe, D.D, Van Dijk, W.J, El Oualid, F, Ekkebus, R, Ovaa, H, Sixma, T.K. | 登録日 | 2014-12-18 | 公開日 | 2015-03-04 | 最終更新日 | 2019-04-03 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Mechanism of Uch-L5 Activation and Inhibition by Deubad Domains in Rpn13 and Ino80G. Mol.Cell, 57, 2015
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4UF6
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![BU of 4uf6 by Molmil](/molmil-images/mine/4uf6) | UCH-L5 in complex with ubiquitin-propargyl bound to an activating fragment of INO80G | 分子名称: | NUCLEAR FACTOR RELATED TO KAPPA-B-BINDING PROTEIN, POLYUBIQUITIN-B, UBIQUITIN CARBOXYL-TERMINAL HYDROLASE ISOZYME L5 | 著者 | Sahtoe, D.D, Van Dijk, W.J, El Oualid, F, Ekkebus, R, Ovaa, H, Sixma, T.K. | 登録日 | 2014-12-23 | 公開日 | 2015-03-04 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (3.69 Å) | 主引用文献 | Mechanism of Uch-L5 Activation and Inhibition by Deubad Domains in Rpn13 and Ino80G. Mol.Cell, 57, 2015
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4W9K
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![BU of 4w9k by Molmil](/molmil-images/mine/4w9k) | pVHL:EloB:EloC in complex with (2S,4R)-1-((S)-2-((S)-2-acetamido-3-phenylpropanamido)-3,3-dimethylbutanoyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide (ligand 14) | 分子名称: | N-acetyl-L-phenylalanyl-3-methyl-L-valyl-(4R)-4-hydroxy-N-[4-(4-methyl-1,3-thiazol-5-yl)benzyl]-L-prolinamide, Transcription elongation factor B polypeptide 1, Transcription elongation factor B polypeptide 2, ... | 著者 | Gadd, M.S, Galdeano, C, van Molle, I, Ciulli, A. | 登録日 | 2014-08-27 | 公開日 | 2014-09-10 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Structure-Guided Design and Optimization of Small Molecules Targeting the Protein-Protein Interaction between the von Hippel-Lindau (VHL) E3 Ubiquitin Ligase and the Hypoxia Inducible Factor (HIF) Alpha Subunit with in Vitro Nanomolar Affinities. J.Med.Chem., 57, 2014
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4W9I
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![BU of 4w9i by Molmil](/molmil-images/mine/4w9i) | pVHL:EloB:EloC in complex with (2S,4R)-1-((2S,4R)-1-acetyl-4-hydroxypyrrolidine-2-carbonyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide (ligand 10) | 分子名称: | (4R)-1-acetyl-4-hydroxy-L-prolyl-(4R)-4-hydroxy-N-[4-(4-methyl-1,3-thiazol-5-yl)benzyl]-L-prolinamide, Transcription elongation factor B polypeptide 1, Transcription elongation factor B polypeptide 2, ... | 著者 | Gadd, M.S, Soares, P, Galdeano, C, van Molle, I, Ciulli, A. | 登録日 | 2014-08-27 | 公開日 | 2014-09-10 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Structure-Guided Design and Optimization of Small Molecules Targeting the Protein-Protein Interaction between the von Hippel-Lindau (VHL) E3 Ubiquitin Ligase and the Hypoxia Inducible Factor (HIF) Alpha Subunit with in Vitro Nanomolar Affinities. J.Med.Chem., 57, 2014
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8EBN
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![BU of 8ebn by Molmil](/molmil-images/mine/8ebn) | |
8EBS
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8EBV
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8EBW
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8EFW
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8EFX
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1NBF
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![BU of 1nbf by Molmil](/molmil-images/mine/1nbf) | Crystal structure of a UBP-family deubiquitinating enzyme in isolation and in complex with ubiquitin aldehyde | 分子名称: | Ubiquitin aldehyde, Ubiquitin carboxyl-terminal hydrolase 7 | 著者 | Hu, M, Li, P, Li, M, Li, W, Yao, T, Wu, J.-W, Gu, W, Cohen, R.E, Shi, Y. | 登録日 | 2002-12-02 | 公開日 | 2003-01-07 | 最終更新日 | 2018-10-03 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Crystal structure of a UBP-family deubiquitinating enzyme in isolation and in complex with ubiquitin aldehyde Cell(Cambridge,Mass.), 111, 2002
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1Q0W
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![BU of 1q0w by Molmil](/molmil-images/mine/1q0w) | Solution structure of Vps27 amino-terminal UIM-ubiquitin complex | 分子名称: | Ubiquitin, Vacuolar protein sorting-associated protein VPS27 | 著者 | Swanson, K.A, Kang, R.S, Stamenova, S.D, Hicke, L, Radhakrishnan, I. | 登録日 | 2003-07-17 | 公開日 | 2003-10-07 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution Structure of Vps27 UIM-Ubiquitin Complex Important for Endosomal Sorting and Receptor Downregulation Embo J., 22, 2003
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1P9D
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1OTR
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![BU of 1otr by Molmil](/molmil-images/mine/1otr) | Solution Structure of a CUE-Ubiquitin Complex | 分子名称: | Ubiquitin, protein Cue2 | 著者 | Kang, R.S, Daniels, C.M, Salerno, W.J, Radhakrishnan, I. | 登録日 | 2003-03-22 | 公開日 | 2003-06-24 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution Structure of a CUE-Ubiquitin Complex Reveals a Conserved Mode
of Ubiquitin Binding Cell(Cambridge,Mass.), 113, 2003
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1P3Q
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![BU of 1p3q by Molmil](/molmil-images/mine/1p3q) | Mechanism of Ubiquitin Recognition by the CUE Domain of VPS9 | 分子名称: | Ubiquitin, Vacuolar protein sorting-associated protein VPS9 | 著者 | Prag, G, Misra, S, Jones, E.A, Ghirlando, R, Davies, B.A, Horazdovsky, B.F, Hurley, J.H. | 登録日 | 2003-04-18 | 公開日 | 2003-06-24 | 最終更新日 | 2021-11-10 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Mechanism of Ubiquitin Recognition by the CUE Domain of Vps9p. Cell(Cambridge,Mass.), 113, 2003
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1OQY
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![BU of 1oqy by Molmil](/molmil-images/mine/1oqy) | Structure of the DNA repair protein hHR23a | 分子名称: | UV excision repair protein RAD23 homolog A | 著者 | Walters, K.J, Lech, P.J, Goh, A.M, Wang, Q, Howley, P.M. | 登録日 | 2003-03-11 | 公開日 | 2003-10-21 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | DNA-repair protein hHR23a alters its protein structure upon binding proteasomal subunit S5a Proc.Natl.Acad.Sci.USA, 100, 2003
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2RR9
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![BU of 2rr9 by Molmil](/molmil-images/mine/2rr9) | The solution structure of the K63-Ub2:tUIMs complex | 分子名称: | Putative uncharacterized protein UIMC1, ubiquitin | 著者 | Sekiyama, N, Jee, J, Isogai, S, Akagi, K, Huang, T, Ariyoshi, M, Tochio, H, Shirakawa, M. | 登録日 | 2010-06-16 | 公開日 | 2011-07-06 | 最終更新日 | 2011-07-13 | 実験手法 | SOLUTION NMR | 主引用文献 | The solution structure of the K63-Ub2:tUIMs complex To be Published
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4RF1
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![BU of 4rf1 by Molmil](/molmil-images/mine/4rf1) | Crystal structure of the Middle-East respiratory syndrome coronavirus papain-like protease in complex with ubiquitin (space group P63) | 分子名称: | 3-AMINOPROPANE, ORF1ab protein, S-1,2-PROPANEDIOL, ... | 著者 | Bailey-Elkin, B.A, Johnson, G.G, Mark, B.L. | 登録日 | 2014-09-24 | 公開日 | 2014-10-22 | 最終更新日 | 2015-01-14 | 実験手法 | X-RAY DIFFRACTION (2.15 Å) | 主引用文献 | Crystal Structure of the Middle East Respiratory Syndrome Coronavirus (MERS-CoV) Papain-like Protease Bound to Ubiquitin Facilitates Targeted Disruption of Deubiquitinating Activity to Demonstrate Its Role in Innate Immune Suppression. J.Biol.Chem., 289, 2014
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4RF0
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![BU of 4rf0 by Molmil](/molmil-images/mine/4rf0) | Crystal structure of the Middle-East respiratory syndrome coronavirus papain-like protease in complex with ubiquitin (space group P6522) | 分子名称: | 3-AMINOPROPANE, ORF1ab protein, SULFATE ION, ... | 著者 | Bailey-Elkin, B.A, Johnson, G.G, Mark, B.L. | 登録日 | 2014-09-24 | 公開日 | 2014-10-22 | 最終更新日 | 2015-01-14 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Crystal Structure of the Middle East Respiratory Syndrome Coronavirus (MERS-CoV) Papain-like Protease Bound to Ubiquitin Facilitates Targeted Disruption of Deubiquitinating Activity to Demonstrate Its Role in Innate Immune Suppression. J.Biol.Chem., 289, 2014
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4P4H
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4S1Z
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![BU of 4s1z by Molmil](/molmil-images/mine/4s1z) | Crystal structure of TRABID NZF1 in complex with K29 linked di-Ubiquitin | 分子名称: | Ubiquitin, Ubiquitin thioesterase ZRANB1, ZINC ION | 著者 | Kristariyanto, Y.A, Abdul Rehman, S.A, Campbell, D.G, Morrice, N.A, Johnson, C, Toth, R, Kulathu, Y. | 登録日 | 2015-01-16 | 公開日 | 2015-04-08 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (3.03 Å) | 主引用文献 | K29-selective ubiquitin binding domain reveals structural basis of specificity and heterotypic nature of k29 polyubiquitin. Mol.Cell, 58, 2015
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