7TW9
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1JI7
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![BU of 1ji7 by Molmil](/molmil-images/mine/1ji7) | Crystal Structure of TEL SAM Polymer | 分子名称: | ETS-RELATED PROTEIN TEL1, SULFATE ION | 著者 | Kim, C.A, Phillips, M.L, Kim, W, Gingery, M, Tran, H.H, Robinson, M.A, Faham, S, Bowie, J.U. | 登録日 | 2001-06-29 | 公開日 | 2002-07-03 | 最終更新日 | 2022-12-21 | 実験手法 | X-RAY DIFFRACTION (1.45 Å) | 主引用文献 | Polymerization of the SAM domain of TEL in leukemogenesis and transcriptional repression. EMBO J., 20, 2001
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7TDY
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![BU of 7tdy by Molmil](/molmil-images/mine/7tdy) | The ubiquitin-associated domain of human thirty-eight negative kinase 1, flexibly fused to the 1TEL crystallization chaperone via a 2-glycine linker and crystallized at low protein concentration | 分子名称: | FORMIC ACID, Transcription factor ETV6,Non-receptor tyrosine-protein kinase TNK1 | 著者 | Nawarathnage, S, Bunn, D.R, Stewart, C, Doukev, T, Moody, J.D. | 登録日 | 2022-01-03 | 公開日 | 2023-01-11 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.53 Å) | 主引用文献 | Fusion crystallization reveals the behavior of both the 1TEL crystallization chaperone and the TNK1 UBA domain. Structure, 31, 2023
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7TW8
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8FRJ
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![BU of 8frj by Molmil](/molmil-images/mine/8frj) | Structure of nsp14 N7-MethylTransferase domain fused with TELSAM bound to SGC0946 | 分子名称: | 5-bromo-7-{5-[(3-{[(4-tert-butylphenyl)carbamoyl]amino}propyl)(propan-2-yl)amino]-5-deoxy-beta-D-ribofuranosyl}-7H-pyrrolo[2,3-d]pyrimidin-4-amine, Transcription factor ETV6,Guanine-N7 methyltransferase nsp14 chimera, ZINC ION | 著者 | Kottur, J, Aggarwal, A.K. | 登録日 | 2023-01-07 | 公開日 | 2023-07-26 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.57 Å) | 主引用文献 | Structures of SARS-CoV-2 N7-methyltransferase with DOT1L and PRMT7 inhibitors provide a platform for new antivirals. Plos Pathog., 19, 2023
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8FT8
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![BU of 8ft8 by Molmil](/molmil-images/mine/8ft8) | The von Willebrand factor A domain of human capillary morphogenesis gene II, flexibly fused to the 1TEL crystallization chaperone, Thr-Val linker variant, SUMO tag-free preparation | 分子名称: | CHLORIDE ION, GLYCEROL, POTASSIUM ION, ... | 著者 | Gajjar, P.L, Litchfield, C.M, Callahan, M, Redd, N, Doukov, T, Moody, J.D. | 登録日 | 2023-01-11 | 公開日 | 2023-03-01 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Increasing the bulk of the 1TEL-target linker and retaining the 10×His tag in a 1TEL-CMG2-vWa construct improves crystal order and diffraction limits. Acta Crystallogr D Struct Biol, 79, 2023
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8FRK
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7TW7
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8THA
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![BU of 8tha by Molmil](/molmil-images/mine/8tha) | 1TEL, non-compressed, double-helical crystal form | 分子名称: | Transcription factor ETV6,Activated CDC42 kinase 1 | 著者 | Smith, C.P, Wilson, E.W, Pedroza Romo, M.J, Averett, J.C, Moody, J.D. | 登録日 | 2023-07-14 | 公開日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (1.68 Å) | 主引用文献 | 1TEL, non-compressed, double-helical crystal form To Be Published
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7JU2
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![BU of 7ju2 by Molmil](/molmil-images/mine/7ju2) | Crystal structure of the monomeric ETV6 PNT domain | 分子名称: | FORMIC ACID, Transcription factor ETV6 | 著者 | Gerak, C.A.N, Kolesnikov, M, Murphy, M.E.P, McIntosh, L.P. | 登録日 | 2020-08-19 | 公開日 | 2021-01-20 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.85002184 Å) | 主引用文献 | Biophysical characterization of the ETV6 PNT domain polymerization interfaces. J.Biol.Chem., 296, 2021
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7T8J
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![BU of 7t8j by Molmil](/molmil-images/mine/7t8j) | The ubiquitin-associated domain of human thirty-eight negative kinase-1 flexibly fused to the 1TEL crystallization chaperone via a GSGG linker | 分子名称: | CHLORIDE ION, Transcription factor ETV6,Non-receptor tyrosine-protein kinase TNK1 | 著者 | Soleimani, S, Pedroza Romo, M.J, Smith, T, Brown, S, Doukov, T, Moody, J.D. | 登録日 | 2021-12-16 | 公開日 | 2022-12-21 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.89 Å) | 主引用文献 | Fusion crystallization reveals the behavior of both the 1TEL crystallization chaperone and the TNK1 UBA domain. Structure, 31, 2023
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8FZU
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![BU of 8fzu by Molmil](/molmil-images/mine/8fzu) | The von Willebrand factor A domain of human capillary morphogenesis gene II, flexibly fused to the 1TEL crystallization chaperone, Thr-Val linker variant, Expressed with SUMO tag | 分子名称: | POTASSIUM ION, SULFATE ION, Transcription factor ETV6,Anthrax toxin receptor 2 | 著者 | Gajjar, P.L, Litchfield, C.M, Callahan, M, Redd, N, Doukov, T, Lebedev, A, Moody, J.D. | 登録日 | 2023-01-30 | 公開日 | 2023-07-19 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Increasing the bulk of the 1TEL-target linker and retaining the 10×His tag in a 1TEL-CMG2-vWa construct improves crystal order and diffraction limits. Acta Crystallogr D Struct Biol, 79, 2023
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7U4Z
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7U4W
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![BU of 7u4w by Molmil](/molmil-images/mine/7u4w) | The ubiquitin-associated domain of human thirty-eight negative kinase-1 flexibly fused to the 1TEL crystallization chaperone via a 2-glycine linker and crystallized at traditional protein concentration | 分子名称: | Transcription factor ETV6,Non-receptor tyrosine-protein kinase TNK1 | 著者 | Nawarathnage, S, Pedroza Romo, M.J, Smith, T, Bunn, D, Stewart, C, Doukov, T, Moody, J.D. | 登録日 | 2022-03-01 | 公開日 | 2023-03-08 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Fusion crystallization reveals the behavior of both the 1TEL crystallization chaperone and the TNK1 UBA domain. Structure, 31, 2023
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8E1F
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![BU of 8e1f by Molmil](/molmil-images/mine/8e1f) | Sterile Alpha Motif Domain of Human Translocation ETS Leukemia, Non-Polymer Crystal Form | 分子名称: | CHLORIDE ION, MAGNESIUM ION, SULFATE ION, ... | 著者 | Wilson, E, Nawarathnage, S, Stewart, C, Brown, S, Bezzant, B, Bunn, D, Towne, N, Pedroza Romo, M.J, Moody, J.D. | 登録日 | 2022-08-10 | 公開日 | 2022-09-14 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.16 Å) | 主引用文献 | Sterile Alpha Motif Domain of Human Translocation ETS Leukemia, Non-Polymer Crystal Form To Be Published
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5L0P
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1LKY
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![BU of 1lky by Molmil](/molmil-images/mine/1lky) | Structure of the wild-type TEL-SAM polymer | 分子名称: | SULFATE ION, TRANSCRIPTION FACTOR ETV6 | 著者 | Tran, H.H, Kim, C.A, Faham, S, Bowie, J.U. | 登録日 | 2002-04-26 | 公開日 | 2002-06-12 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Native interface of the SAM domain polymer of TEL. BMC STRUCT.BIOL., 2, 2002
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8BWU
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![BU of 8bwu by Molmil](/molmil-images/mine/8bwu) | Crystal structure of SARS-CoV-2 nsp14 methyltransferase domain in complex with the SS148 inhibitor | 分子名称: | (2~{S})-2-azanyl-4-[[(2~{S},3~{S},4~{R},5~{R})-5-(4-azanyl-5-cyano-pyrrolo[2,3-d]pyrimidin-7-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methylsulfanyl]butanoic acid, Transcription factor ETV6,Proofreading exoribonuclease nsp14, ZINC ION | 著者 | Konkolova, E, Klima, M, Boura, E, Jin, J, Kaniskan, H.U, Han, Y, Vedadi, M. | 登録日 | 2022-12-07 | 公開日 | 2023-10-11 | 最終更新日 | 2024-06-26 | 実験手法 | X-RAY DIFFRACTION (2.36 Å) | 主引用文献 | Application of established computational techniques to identify potential SARS-CoV-2 Nsp14-MTase inhibitors in low data regimes Digit Discov, 2024
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2QAR
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2QB0
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2QB1
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8FT6
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![BU of 8ft6 by Molmil](/molmil-images/mine/8ft6) | The von Willebrand factor A domain of human capillary morphogenesis gene II, flexibly fused to the 1TEL crystallization chaperone, Ala-Ala linker variant, SUMO tag-free preparation. | 分子名称: | CITRIC ACID, IODIDE ION, SULFATE ION, ... | 著者 | Gajjar, P.L, Litchfield, C.M, Callahan, M, Redd, N, Doukov, T, Moody, J.D. | 登録日 | 2023-01-11 | 公開日 | 2023-03-22 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.62 Å) | 主引用文献 | Increasing the bulk of the 1TEL-target linker and retaining the 10×His tag in a 1TEL-CMG2-vWa construct improves crystal order and diffraction limits. Acta Crystallogr D Struct Biol, 79, 2023
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7N1O
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![BU of 7n1o by Molmil](/molmil-images/mine/7n1o) | The von Willebrand factor A domain of human capillary morphogenesis gene II, flexibly fused to the 1TEL crystallization chaperone | 分子名称: | CHLORIDE ION, MAGNESIUM ION, Transcription factor ETV6,Isoform 4 of Anthrax toxin receptor 2 | 著者 | Mathis, M.H, Bezzant, B.D, Ramirez, D.T, Sarath Nawarathnage, S.D, Doukov, T, Moody, J.D. | 登録日 | 2021-05-27 | 公開日 | 2021-06-09 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.77 Å) | 主引用文献 | Crystals of TELSAM-target protein fusions that exhibit minimal crystal contacts and lack direct inter-TELSAM contacts. Open Biology, 12, 2022
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8FZ3
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![BU of 8fz3 by Molmil](/molmil-images/mine/8fz3) | Sterile Alpha Motif of Human Translocation ETS Leukemia, Non-Polymer Crystal Form | 分子名称: | CHLORIDE ION, PHOSPHATE ION, Transcription factor ETV6, ... | 著者 | Averett, J.C, Nawarathnage, S.D, Moody, J.D. | 登録日 | 2023-01-27 | 公開日 | 2023-03-29 | 最終更新日 | 2024-05-22 | 実験手法 | X-RAY DIFFRACTION (2.784 Å) | 主引用文献 | Sterile Alpha Motif of Human Translocation ETS Leukemia, Non-Polymer Crystal Form, With Disordered Human ACK1 UBA Domain Fused to C-terminus To Be Published
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7N2B
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![BU of 7n2b by Molmil](/molmil-images/mine/7n2b) | A DARPin semi-rigidly fused to the 3TEL crystallization chaperone | 分子名称: | Transcription factor ETV6,Transcription factor ETV6,Transcription factor ETV6,3TEL-rigid-DARPin | 著者 | Sarath Nawarathange, S.D, Gajjar, P, Bunn, D, Stewart, C, Doukov, T, Moody, J.D. | 登録日 | 2021-05-28 | 公開日 | 2021-06-09 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (3.221 Å) | 主引用文献 | Crystals of TELSAM-target protein fusions that exhibit minimal crystal contacts and lack direct inter-TELSAM contacts. Open Biology, 12, 2022
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