7N9C
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7N9E
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7N9B
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7N9A
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8TLM
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![BU of 8tlm by Molmil](/molmil-images/mine/8tlm) | Structure of a class A GPCR/Fab complex | 分子名称: | C-C chemokine receptor type 8, Green fluorescent protein fusion, Fab heavy chain, ... | 著者 | Sun, D, Johnson, M, Masureel, M. | 登録日 | 2023-07-27 | 公開日 | 2023-12-20 | 実験手法 | ELECTRON MICROSCOPY (2.9 Å) | 主引用文献 | Structural basis of antibody inhibition and chemokine activation of the human CC chemokine receptor 8. Nat Commun, 14, 2023
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8U1U
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![BU of 8u1u by Molmil](/molmil-images/mine/8u1u) | Structure of a class A GPCR/agonist complex | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, C-C motif chemokine 1,C-C chemokine receptor type 8,EGFP fusion protein, Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2, ... | 著者 | Sun, D, Johnson, M, Masureel, M. | 登録日 | 2023-09-02 | 公開日 | 2023-12-20 | 実験手法 | ELECTRON MICROSCOPY (3.1 Å) | 主引用文献 | Structural basis of antibody inhibition and chemokine activation of the human CC chemokine receptor 8. Nat Commun, 14, 2023
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6Q0X
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8W0S
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![BU of 8w0s by Molmil](/molmil-images/mine/8w0s) | Human EBP complexed with compound 3a | 分子名称: | 1-methyl-8-[(oxan-4-yl)methyl]-3-[4-(trifluoromethyl)phenyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione, 3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase | 著者 | Sun, D, Masureel, M. | 登録日 | 2024-02-14 | 公開日 | 2024-06-19 | 実験手法 | ELECTRON MICROSCOPY (2.8 Å) | 主引用文献 | Discovery and Optimization of Selective Brain-Penetrant EBP Inhibitors that Enhance Oligodendrocyte Formation. J.Med.Chem., 67, 2024
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8W0R
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![BU of 8w0r by Molmil](/molmil-images/mine/8w0r) | Human EBP complexed with compound 1 | 分子名称: | 1-methyl-1'-[(oxan-4-yl)methyl]-5-(trifluoromethyl)spiro[indole-2,4'-piperidin]-3(1H)-one, 3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase | 著者 | Sun, D, Masureel, M. | 登録日 | 2024-02-14 | 公開日 | 2024-06-19 | 実験手法 | ELECTRON MICROSCOPY (2.8 Å) | 主引用文献 | Discovery and Optimization of Selective Brain-Penetrant EBP Inhibitors that Enhance Oligodendrocyte Formation. J.Med.Chem., 67, 2024
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8U31
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![BU of 8u31 by Molmil](/molmil-images/mine/8u31) | Crystal structure of PD-1 in complex with a Fab | 分子名称: | Fab heavy chain, Fab light chain, GLYCEROL, ... | 著者 | Sun, D, Masureel, M. | 登録日 | 2023-09-07 | 公開日 | 2024-06-19 | 実験手法 | X-RAY DIFFRACTION (2.73 Å) | 主引用文献 | Structure- and machine learning-guided engineering demonstrate that a non-canonical disulfide in an anti-PD-1 rabbit antibody does not impede antibody developability. Mabs, 16, 2024
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8U32
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![BU of 8u32 by Molmil](/molmil-images/mine/8u32) | Crystal structure of PD-1 in complex with a Fab | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Fab heavy chain, Fab light chain, ... | 著者 | Sun, D, Masureel, M. | 登録日 | 2023-09-07 | 公開日 | 2024-06-19 | 実験手法 | X-RAY DIFFRACTION (2.51 Å) | 主引用文献 | Structure- and machine learning-guided engineering demonstrate that a non-canonical disulfide in an anti-PD-1 rabbit antibody does not impede antibody developability. Mabs, 16, 2024
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1MG2
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![BU of 1mg2 by Molmil](/molmil-images/mine/1mg2) | MUTATION OF ALPHA PHE55 OF METHYLAMINE DEHYDROGENASE ALTERS THE REORGANIZATION ENERGY AND ELECTRONIC COUPLING FOR ITS ELECTRON TRANSFER REACTION WITH AMICYANIN | 分子名称: | Amicyanin, COPPER (II) ION, CYTOCHROME C-L, ... | 著者 | Sun, D, Chen, Z.W, Mathews, F.S, Davidson, V.L. | 登録日 | 2002-08-14 | 公開日 | 2002-12-11 | 最終更新日 | 2021-10-27 | 実験手法 | X-RAY DIFFRACTION (2.25 Å) | 主引用文献 | MUTATION OF AlPHA PHE55 OF METHYLAMINE DEHYDROGENASE ALTERS THE REORGANIZATION ENERGY AND ELECTRONIC COUPLING FOR ITS ELECTRON TRANSFER REACTION WITH AMICYANIN Biochemistry, 41, 2002
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1MG3
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![BU of 1mg3 by Molmil](/molmil-images/mine/1mg3) | MUTATION OF ALPHA PHE55 OF METHYLAMINE DEHYDROGENASE ALTERS THE REORGANIZATION ENERGY AND ELECTRONIC COUPLING FOR ITS ELECTRON TRANSFER REACTION WITH AMICYANIN | 分子名称: | Amicyanin, COPPER (II) ION, CYTOCHROME C-L, ... | 著者 | Sun, D, Chen, Z.W, Mathews, F.S, Davidson, V.L. | 登録日 | 2002-08-14 | 公開日 | 2002-12-11 | 最終更新日 | 2021-10-27 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | MUTATION OF ALPHA PHE55 OF METHYLAMINE DEHYDROGENASE ALTERS THE REORGANIZATION ENERGY AND ELECTRONIC COUPLING FOR ITS ELECTRON TRANSFER REACTION WITH AMICYANIN Biochemistry, 41, 2002
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3K8T
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![BU of 3k8t by Molmil](/molmil-images/mine/3k8t) | Structure of eukaryotic rnr large subunit R1 complexed with designed adp analog compound | 分子名称: | 2'-DEOXYGUANOSINE-5'-TRIPHOSPHATE, 2'-deoxy-2'-(2-hydroxyethyl)adenosine 5'-(trihydrogen diphosphate), GLYCEROL, ... | 著者 | Sun, D, Xu, H, Dealwis, C, Lee, R.E. | 登録日 | 2009-10-14 | 公開日 | 2010-03-02 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Structure-Based Design, Synthesis, and Evaluation of 2'-(2-Hydroxyethyl)-2'-deoxyadenosine and the 5'-Diphosphate Derivative as Ribonucleotide Reductase Inhibitors Chemmedchem, 4, 2009
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1XGF
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1S0H
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3HW9
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![BU of 3hw9 by Molmil](/molmil-images/mine/3hw9) | Cation selective pathway of OmpF porin revealed by anomalous x-ray diffraction | 分子名称: | CHLORIDE ION, HEXAETHYLENE GLYCOL, Outer membrane protein F, ... | 著者 | Balasundaresan, D, Raychaudhury, S, Blachowicz, L, Roux, B. | 登録日 | 2009-06-17 | 公開日 | 2009-12-08 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.61 Å) | 主引用文献 | Cation-selective pathway of OmpF porin revealed by anomalous X-ray diffraction. J.Mol.Biol., 396, 2010
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3HWB
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![BU of 3hwb by Molmil](/molmil-images/mine/3hwb) | Cation selective pathway of OmpF porin revealed by anomalous diffraction | 分子名称: | HEXAETHYLENE GLYCOL, Outer membrane protein F, RUBIDIUM ION | 著者 | Balasundaresan, D, Raychaudhury, S, Blachowicz, L, Roux, B. | 登録日 | 2009-06-17 | 公開日 | 2009-12-08 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Cation-selective pathway of OmpF porin revealed by anomalous X-ray diffraction. J.Mol.Biol., 396, 2010
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4LSI
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![BU of 4lsi by Molmil](/molmil-images/mine/4lsi) | Ion selectivity of OmpF porin soaked in 0.3M KBr | 分子名称: | (HYDROXYETHYLOXY)TRI(ETHYLOXY)OCTANE, BROMIDE ION, DI(HYDROXYETHYL)ETHER, ... | 著者 | Balasundaresan, D, Blachowicz, L, Roux, B. | 登録日 | 2013-07-22 | 公開日 | 2013-10-23 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.089 Å) | 主引用文献 | A structural study of ion permeation in OmpF porin from anomalous X-ray diffraction and molecular dynamics simulations. J.Am.Chem.Soc., 135, 2013
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4LSE
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![BU of 4lse by Molmil](/molmil-images/mine/4lse) | Ion selectivity of OmpF porin soaked in 0.2M NaBr | 分子名称: | (HYDROXYETHYLOXY)TRI(ETHYLOXY)OCTANE, BROMIDE ION, DI(HYDROXYETHYL)ETHER, ... | 著者 | Balasundaresan, D, Blachowicz, L, Roux, B. | 登録日 | 2013-07-22 | 公開日 | 2013-10-23 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | A structural study of ion permeation in OmpF porin from anomalous X-ray diffraction and molecular dynamics simulations. J.Am.Chem.Soc., 135, 2013
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4LSH
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4LSF
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7NA8
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![BU of 7na8 by Molmil](/molmil-images/mine/7na8) | Structures of human ghrelin receptor-Gi complexes with ghrelin and a synthetic agonist | 分子名称: | 1-(methanesulfonyl)-1'-(2-methyl-L-alanyl-O-benzyl-D-seryl)-1,2-dihydrospiro[indole-3,4'-piperidine], Antibody fragment, CHOLESTEROL, ... | 著者 | Liu, H, Sun, D, Sun, J, Zhang, C. | 登録日 | 2021-06-20 | 公開日 | 2021-12-15 | 実験手法 | ELECTRON MICROSCOPY (2.7 Å) | 主引用文献 | Structural basis of human ghrelin receptor signaling by ghrelin and the synthetic agonist ibutamoren Nat Commun, 12, 2021
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7NA7
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![BU of 7na7 by Molmil](/molmil-images/mine/7na7) | Structures of human ghrelin receptor-Gi complexes with ghrelin and a synthetic agonist | 分子名称: | Antibody fragment, CHOLESTEROL, Ghrelin-27, ... | 著者 | Liu, H, Sun, D, Sun, J, Zhang, C. | 登録日 | 2021-06-20 | 公開日 | 2021-12-15 | 実験手法 | ELECTRON MICROSCOPY (2.7 Å) | 主引用文献 | Structural basis of human ghrelin receptor signaling by ghrelin and the synthetic agonist ibutamoren Nat Commun, 12, 2021
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1D0E
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![BU of 1d0e by Molmil](/molmil-images/mine/1d0e) | CRYSTAL STRUCTURES OF THE N-TERMINAL FRAGMENT FROM MOLONEY MURINE LEUKEMIA VIRUS REVERSE TRANSCRIPTASE COMPLEXED WITH NUCLEIC ACID: FUNCTIONAL IMPLICATIONS FOR TEMPLATE-PRIMER BINDING TO THE FINGERS DOMAIN | 分子名称: | 5'-D(*TP*TP*TP*CP*AP*TP*GP*CP*AP*TP*G)-3', REVERSE TRANSCRIPTASE | 著者 | Najmudin, S, Cote, M.L, Sun, D, Yohannan, S, Montano, S.P, Gu, J, Georgiadis, M.M. | 登録日 | 1999-09-09 | 公開日 | 2000-04-04 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Crystal structures of an N-terminal fragment from Moloney murine leukemia virus reverse transcriptase complexed with nucleic acid: functional implications for template-primer binding to the fingers domain J.Mol.Biol., 296, 2000
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