8JJN
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8K5U
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8FZR
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4HKA
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2LJV
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![BU of 2ljv by Molmil](/molmil-images/mine/2ljv) | Solution structure of Rhodostomin G50L mutant | 分子名称: | Disintegrin rhodostomin | 著者 | Chuang, W, Shiu, J, Chen, C, Chen, Y, Chang, Y, Huang, C. | 登録日 | 2011-09-29 | 公開日 | 2012-10-03 | 最終更新日 | 2023-06-14 | 実験手法 | SOLUTION NMR | 主引用文献 | Design of Integrin AlphaVbeta3-Specific Disintegrin for Cancer Therapy To be Published
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7DUC
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![BU of 7duc by Molmil](/molmil-images/mine/7duc) | Crystal Structure of cyto WalK | 分子名称: | Sensor protein kinase WalK, ZINC ION | 著者 | Huang, W. | 登録日 | 2021-01-08 | 公開日 | 2022-01-19 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.56 Å) | 主引用文献 | Crystal Structure of cyto WalK To Be Published
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7DUD
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![BU of 7dud by Molmil](/molmil-images/mine/7dud) | Crystal Structure of erWalK | 分子名称: | Sensor protein kinase WalK | 著者 | Huang, W. | 登録日 | 2021-01-08 | 公開日 | 2022-01-19 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Crystal Structure of erWalK To Be Published
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2JTC
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![BU of 2jtc by Molmil](/molmil-images/mine/2jtc) | 3D structure and backbone dynamics of SPE B | 分子名称: | Streptopain | 著者 | Chuang, W, Wang, C, Houng, H, Chen, C, Wang, P. | 登録日 | 2007-07-26 | 公開日 | 2008-08-26 | 最終更新日 | 2024-05-29 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure and backbone dynamics of streptopain: insight into diverse substrate specificity. J.Biol.Chem., 284, 2009
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2M75
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2M7H
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2M7F
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2KIU
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6E53
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![BU of 6e53 by Molmil](/molmil-images/mine/6e53) | Structure of TERT in complex with a novel telomerase inhibitor | 分子名称: | MAGNESIUM ION, RNA/DNA hairpin, Telomerase reverse transcriptase, ... | 著者 | Hernandez-Sanchez, W, Huang, W, Plucinsky, B, Garcia-Vazquez, N, Berdis, A.J, Skordalakes, E, Taylor, D.J. | 登録日 | 2018-07-19 | 公開日 | 2019-03-27 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | A non-natural nucleotide uses a specific pocket to selectively inhibit telomerase activity. Plos Biol., 17, 2019
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1EAP
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![BU of 1eap by Molmil](/molmil-images/mine/1eap) | CRYSTAL STRUCTURE OF A CATALYTIC ANTIBODY WITH A SERINE PROTEASE ACTIVE SITE | 分子名称: | IGG2B-KAPPA 17E8 FAB (HEAVY CHAIN), IGG2B-KAPPA 17E8 FAB (LIGHT CHAIN), PHENYL[1-(N-SUCCINYLAMINO)PENTYL]PHOSPHONATE | 著者 | Zhou, G.W, Guo, J, Huang, W, Scanlan, T.S, Fletterick, R.J. | 登録日 | 1994-08-10 | 公開日 | 1994-12-20 | 最終更新日 | 2024-06-05 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Crystal structure of a catalytic antibody with a serine protease active site. Science, 265, 1994
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1ONR
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![BU of 1onr by Molmil](/molmil-images/mine/1onr) | STRUCTURE OF TRANSALDOLASE B | 分子名称: | TRANSALDOLASE B | 著者 | Jia, J, Huang, W, Lindqvist, Y, Schneider, G. | 登録日 | 1996-08-13 | 公開日 | 1997-03-12 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (1.87 Å) | 主引用文献 | Crystal structure of transaldolase B from Escherichia coli suggests a circular permutation of the alpha/beta barrel within the class I aldolase family. Structure, 4, 1996
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8IR4
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![BU of 8ir4 by Molmil](/molmil-images/mine/8ir4) | Crystal structure of the SLF1 BRCT domain in complex with a Rad18 peptide containing pS442 | 分子名称: | CHLORIDE ION, ISOPROPYL ALCOHOL, MAGNESIUM ION, ... | 著者 | Xiang, S, Huang, W, Qiu, F. | 登録日 | 2023-03-17 | 公開日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.62 Å) | 主引用文献 | Structural insights into Rad18 targeting by the SLF1 BRCT domains. J.Biol.Chem., 299, 2023
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8IR2
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![BU of 8ir2 by Molmil](/molmil-images/mine/8ir2) | Crystal structure of the SLF1 BRCT domain in complex with a Rad18 peptide containing pS442 and pS444 | 分子名称: | CHLORIDE ION, ISOPROPYL ALCOHOL, MAGNESIUM ION, ... | 著者 | Xiang, S, Huang, W, Qiu, F. | 登録日 | 2023-03-17 | 公開日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Structural insights into Rad18 targeting by the SLF1 BRCT domains. J.Biol.Chem., 299, 2023
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6UP7
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![BU of 6up7 by Molmil](/molmil-images/mine/6up7) | neurotensin receptor and arrestin2 complex | 分子名称: | ARG-ARG-PRO-TYR-ILE-LEU, Beta-arrestin-1, Neurotensin receptor type 1, ... | 著者 | Qu, Q.H, Huang, W, Masureel, M, Janetzko, J, Kobilka, B.K, Skiniotis, G. | 登録日 | 2019-10-16 | 公開日 | 2020-02-26 | 最終更新日 | 2020-06-17 | 実験手法 | ELECTRON MICROSCOPY (4.2 Å) | 主引用文献 | Structure of the neurotensin receptor 1 in complex with beta-arrestin 1. Nature, 579, 2020
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1XDO
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1XDP
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![BU of 1xdp by Molmil](/molmil-images/mine/1xdp) | Crystal Structure of the E.coli Polyphosphate Kinase in complex with AMPPNP | 分子名称: | ADENOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, Polyphosphate kinase | 著者 | Zhu, Y, Huang, W, Lee, S.S, Xu, W. | 登録日 | 2004-09-07 | 公開日 | 2005-06-21 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Crystal structure of a polyphosphate kinase and its implications for polyphosphate synthesis Embo Rep., 6, 2005
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8YRF
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1AFR
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1D2L
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3EZR
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![BU of 3ezr by Molmil](/molmil-images/mine/3ezr) | CDK-2 with indazole inhibitor 17 bound at its active site | 分子名称: | 3-methoxy-4-{3-[4-(4-methylpiperazin-1-yl)-1H-benzimidazol-2-yl]-1H-indazol-6-yl}aniline, Cell division protein kinase 2 | 著者 | Kiefer, J.R, Day, J.E, Caspers, N.L, Mathis, K.J, Kretzmer, K.K, Weinberg, R.A, Reitz, B.A, Stegeman, R.A, Trujillo, J.I, Huang, W, Thorarensen, A, Xing, L, Wrightstone, A, Christine, L, Compton, R, Li, X. | 登録日 | 2008-10-23 | 公開日 | 2009-02-03 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | 2-(6-Phenyl-1H-indazol-3-yl)-1H-benzo[d]imidazoles: Design and synthesis of a potent and isoform selective PKC-zeta inhibitor Bioorg.Med.Chem.Lett., 19, 2009
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3F5X
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![BU of 3f5x by Molmil](/molmil-images/mine/3f5x) | CDK-2-Cyclin complex with indazole inhibitor 9 bound at its active site | 分子名称: | 4-{3-[7-(4-methylpiperazin-1-yl)-1H-benzimidazol-2-yl]-1H-indazol-6-yl}aniline, Cell division protein kinase 2, Cyclin-A2, ... | 著者 | Kiefer, J.R, Day, J.E, Caspers, N.L, Mathis, K.J, Kretzmer, K.K, Weinberg, R.A, Reitz, B.A, Stegeman, R.A, Trujillo, J.I, Huang, W, Thorarensen, A, Xing, L, Wrightstone, A, Christine, L, Compton, R, Li, X. | 登録日 | 2008-11-04 | 公開日 | 2009-02-03 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | 2-(6-Phenyl-1H-indazol-3-yl)-1H-benzo[d]imidazoles: Design and synthesis of a potent and isoform selective PKC-zeta inhibitor. Bioorg.Med.Chem.Lett., 19, 2009
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