3SZE
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![BU of 3sze by Molmil](/molmil-images/mine/3sze) | Crystal structure of the passenger domain of the E. coli autotransporter EspP | 分子名称: | Serine protease espP | 著者 | Khan, S, Mian, H.S, Sandercock, L.E, Battaile, K.P, Lam, R, Chirgadze, N.Y, Pai, E.F. | 登録日 | 2011-07-18 | 公開日 | 2011-10-12 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Crystal Structure of the Passenger Domain of the Escherichia coli Autotransporter EspP. J.Mol.Biol., 413, 2011
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3R3X
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![BU of 3r3x by Molmil](/molmil-images/mine/3r3x) | Crystal Structure of the Fluoroacetate Dehalogenase RPA1163 - Asp110Asn/Bromoacetate | 分子名称: | CALCIUM ION, CHLORIDE ION, Fluoroacetate dehalogenase, ... | 著者 | Chan, P.W.Y, Yakunin, A.F, Edwards, E.A, Pai, E.F. | 登録日 | 2011-03-16 | 公開日 | 2011-05-04 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Mapping the reaction coordinates of enzymatic defluorination. J.Am.Chem.Soc., 133, 2011
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3RIJ
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![BU of 3rij by Molmil](/molmil-images/mine/3rij) | Epitope backbone grafting by computational design for improved presentation of linear epitopes on scaffold proteins | 分子名称: | GLYCEROL, SC_2cx5 | 著者 | Azoitei, M.L, Ban, Y.A, Julien, J.P, Bryson, S, Schroeter, A, Kalyuzhniy, O, Porter, J.R, Adachi, Y, Baker, D, Szabo, E, Pai, E.F, Schief, W.R. | 登録日 | 2011-04-13 | 公開日 | 2011-11-09 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Computational design of high-affinity epitope scaffolds by backbone grafting of a linear epitope. J.Mol.Biol., 415, 2012
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3R3U
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![BU of 3r3u by Molmil](/molmil-images/mine/3r3u) | Crystal Structure of the Fluoroacetate Dehalogenase RPA1163 - WT/apo | 分子名称: | CHLORIDE ION, Fluoroacetate dehalogenase, NICKEL (II) ION | 著者 | Chan, P.W.Y, Yakunin, A.F, Edwards, E.A, Pai, E.F. | 登録日 | 2011-03-16 | 公開日 | 2011-05-04 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Mapping the reaction coordinates of enzymatic defluorination. J.Am.Chem.Soc., 133, 2011
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3R41
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![BU of 3r41 by Molmil](/molmil-images/mine/3r41) | Crystal Structure of the Fluoroacetate Dehalogenase RPA1163 - His280Asn/apo | 分子名称: | CALCIUM ION, CHLORIDE ION, Fluoroacetate dehalogenase | 著者 | Chan, P.W.Y, Yakunin, A.F, Edwards, E.A, Pai, E.F. | 登録日 | 2011-03-17 | 公開日 | 2011-05-04 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.05 Å) | 主引用文献 | Mapping the reaction coordinates of enzymatic defluorination. J.Am.Chem.Soc., 133, 2011
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2MWN
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![BU of 2mwn by Molmil](/molmil-images/mine/2mwn) | Talin-F3 / RIAM N-terminal Peptide complex | 分子名称: | Amyloid beta A4 precursor protein-binding family B member 1-interacting protein, Talin-1 | 著者 | Yang, J, Zhu, L, Zhang, H, Hirbawi, J, Fukuda, K, Dwivedi, P, Liu, J, Byzova, T, Plow, E.F, Wu, J, Qin, J. | 登録日 | 2014-11-13 | 公開日 | 2014-12-17 | 最終更新日 | 2024-05-15 | 実験手法 | SOLUTION NMR | 主引用文献 | Conformational activation of talin by RIAM triggers integrin-mediated cell adhesion. Nat Commun, 5, 2014
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2NNI
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![BU of 2nni by Molmil](/molmil-images/mine/2nni) | CYP2C8dH complexed with montelukast | 分子名称: | Cytochrome P450 2C8, MONTELUKAST, PALMITIC ACID, ... | 著者 | Schoch, G.A, Yano, J.K, Stout, C.D, Johnson, E.F. | 登録日 | 2006-10-24 | 公開日 | 2007-10-23 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Determinants of cytochrome P450 2C8 substrate binding: structures of complexes with montelukast, troglitazone, felodipine, and 9-cis-retinoic acid. J.Biol.Chem., 283, 2008
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3S9Y
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![BU of 3s9y by Molmil](/molmil-images/mine/3s9y) | Crystal Structure of P. falciparum orotidine 5'-monophosphate decarboxylase complexed with 5-fluoro-6-amino-UMP in space group P21, produced from 5-fluoro-6-azido-UMP | 分子名称: | 6-amino-5-fluorouridine 5'-(dihydrogen phosphate), DI(HYDROXYETHYL)ETHER, HEXAETHYLENE GLYCOL, ... | 著者 | Liu, Y, Kotra, L.P, Pai, E.F. | 登録日 | 2011-06-02 | 公開日 | 2012-04-18 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Structure-activity relationships of orotidine-5'-monophosphate decarboxylase inhibitors as anticancer agents. J.Med.Chem., 52, 2009
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2NNH
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![BU of 2nnh by Molmil](/molmil-images/mine/2nnh) | CYP2C8dH complexed with 2 molecules of 9-cis retinoic acid | 分子名称: | (9cis)-retinoic acid, Cytochrome P450 2C8, PALMITIC ACID, ... | 著者 | Schoch, G.A, Yano, J.K, Stout, C.D, Johnson, E.F. | 登録日 | 2006-10-24 | 公開日 | 2007-10-23 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Determinants of cytochrome P450 2C8 substrate binding: structures of complexes with montelukast, troglitazone, felodipine, and 9-cis-retinoic acid. J.Biol.Chem., 283, 2008
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3SSJ
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3R3Z
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![BU of 3r3z by Molmil](/molmil-images/mine/3r3z) | Crystal Structure of the Fluoroacetate Dehalogenase RPA1163 - WT/Glycolate | 分子名称: | Fluoroacetate dehalogenase, GLYCOLIC ACID, NICKEL (II) ION | 著者 | Chan, P.W.Y, Yakunin, A.F, Edwards, E.A, Pai, E.F. | 登録日 | 2011-03-16 | 公開日 | 2011-05-04 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Mapping the reaction coordinates of enzymatic defluorination. J.Am.Chem.Soc., 133, 2011
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1AVT
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![BU of 1avt by Molmil](/molmil-images/mine/1avt) | SUBTILISIN CARLSBERG D-PARA-CHLOROPHENYL-1-ACETAMIDO BORONIC ACID INHIBITOR COMPLEX | 分子名称: | SODIUM ION, SUBTILISIN CARLSBERG, TYPE VIII | 著者 | Stoll, V.S, Eger, B.T, Hynes, R.C, Martichonok, V, Jones, J.B, Pai, E.F. | 登録日 | 1997-09-19 | 公開日 | 1998-03-25 | 最終更新日 | 2023-08-02 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Differences in binding modes of enantiomers of 1-acetamido boronic acid based protease inhibitors: crystal structures of gamma-chymotrypsin and subtilisin Carlsberg complexes. Biochemistry, 37, 1998
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3RZ4
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1CXV
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![BU of 1cxv by Molmil](/molmil-images/mine/1cxv) | STRUCTURE OF RECOMBINANT MOUSE COLLAGENASE-3 (MMP-13) | 分子名称: | 2-{4-[4-(4-CHLORO-PHENOXY)-BENZENESULFONYL]-TETRAHYDRO-PYRAN-4-YL}-N-HYDROXY-ACETAMIDE, CALCIUM ION, PROTEIN (COLLAGENASE-3), ... | 著者 | Botos, I, Meyer, E, Swanson, S.M, Lemaitre, V, Eeckhout, Y, Meyer, E.F. | 登録日 | 1999-08-30 | 公開日 | 2000-08-30 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structure of recombinant mouse collagenase-3 (MMP-13). J.Mol.Biol., 292, 1999
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2O4D
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![BU of 2o4d by Molmil](/molmil-images/mine/2o4d) | Crystal Structure of a hypothetical protein from Pseudomonas aeruginosa | 分子名称: | Hypothetical protein PA0269 | 著者 | McGrath, T.E, Battaile, K, Kisselman, G, Romanov, V, Wu-Brown, J, Virag, C, Ng, I, Kimber, M, Edwards, A.M, Pai, E.F, Chirgadze, N.Y. | 登録日 | 2006-12-04 | 公開日 | 2007-01-30 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Crystal Structure of a hypothetical protein from Pseudomonas aeruginosa To be Published
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2OBA
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![BU of 2oba by Molmil](/molmil-images/mine/2oba) | Pseudomonas aeruginosa 6-pyruvoyl tetrahydrobiopterin synthase | 分子名称: | Probable 6-pyruvoyl tetrahydrobiopterin synthase, ZINC ION | 著者 | McGrath, T.E, Kisselman, G, Battaile, K, Romanov, V, Wu-Brown, J, Guthrie, J, Virag, C, Mansoury, K, Edwards, A.M, Pai, E.F, Chirgadze, N.Y. | 登録日 | 2006-12-18 | 公開日 | 2007-01-30 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.33 Å) | 主引用文献 | Pseudomonas aeruginosa 6-pyruvoyl tetrahydrobiopterin synthase TO BE PUBLISHED
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2PR4
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![BU of 2pr4 by Molmil](/molmil-images/mine/2pr4) | Crystal Structure of Fab' from the HIV-1 Neutralizing Antibody 2F5 | 分子名称: | nmAb 2F5 Fab' Heavy Chain, nmAb 2F5 Fab' light Chain | 著者 | Bryson, S, Julien, J.-P, Pai, E.F. | 登録日 | 2007-05-03 | 公開日 | 2007-05-15 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (2.05 Å) | 主引用文献 | Structural details of HIV-1 recognition by the broadly neutralizing monoclonal antibody 2F5: epitope conformation, antigen-recognition loop mobility, and anion-binding site. J.Mol.Biol., 384, 2008
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2PW2
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![BU of 2pw2 by Molmil](/molmil-images/mine/2pw2) | Crystal structure of the HIV-1 Cross Neutralizing Monoclonal Antibody 2F5 in complex with gp41 Peptide ELDKWKSL | 分子名称: | 2F5 Fab' heavy chain, 2F5 Fab' light chain, peptide epitope | 著者 | Bryson, S, Julien, J.-P, Hynes, R.C, Pai, E.F. | 登録日 | 2007-05-10 | 公開日 | 2007-05-22 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (2.55 Å) | 主引用文献 | Crystallographic definition of the epitope promiscuity of the broadly neutralizing anti-human immunodeficiency virus type 1 antibody 2F5: vaccine design implications. J.Virol., 83, 2009
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2PG7
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![BU of 2pg7 by Molmil](/molmil-images/mine/2pg7) | Crystal Structure of Human Microsomal P450 2A6 N297Q/I300V | 分子名称: | Cytochrome P450 2A6, PROTOPORPHYRIN IX CONTAINING FE | 著者 | Sansen, S, Hsu, M.H, Stout, C.D, Johnson, E.F. | 登録日 | 2007-04-06 | 公開日 | 2007-07-24 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Structural insight into the altered substrate specificity of human cytochrome P450 2A6 mutants. Arch.Biochem.Biophys., 464, 2007
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3R3W
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![BU of 3r3w by Molmil](/molmil-images/mine/3r3w) | Crystal Structure of the Fluoroacetate Dehalogenase RPA1163 - Asp110Asn/Chloroacetate | 分子名称: | CALCIUM ION, CHLORIDE ION, Fluoroacetate dehalogenase, ... | 著者 | Chan, P.W.Y, Yakunin, A.F, Edwards, E.A, Pai, E.F. | 登録日 | 2011-03-16 | 公開日 | 2011-05-04 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Mapping the reaction coordinates of enzymatic defluorination. J.Am.Chem.Soc., 133, 2011
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3SGU
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2PG5
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![BU of 2pg5 by Molmil](/molmil-images/mine/2pg5) | Crystal Structure of Human Microsomal P450 2A6 N297Q | 分子名称: | 1,2-ETHANEDIOL, Cytochrome P450 2A6, PROTOPORPHYRIN IX CONTAINING FE | 著者 | Sansen, S, Hsu, M.H, Stout, C.D, Johnson, E.F. | 登録日 | 2007-04-06 | 公開日 | 2007-07-24 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Structural insight into the altered substrate specificity of human cytochrome P450 2A6 mutants. Arch.Biochem.Biophys., 464, 2007
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2Q8Z
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![BU of 2q8z by Molmil](/molmil-images/mine/2q8z) | Crystal structure of Plasmodium falciparum orotidine 5'-phosphate decarboxylase complexed with 6-amino-UMP | 分子名称: | 2-(2-(2-(2-(2-(2-ETHOXYETHOXY)ETHOXY)ETHOXY)ETHOXY)ETHOXY)ETHANOL, 6-AMINOURIDINE 5'-MONOPHOSPHATE, DI(HYDROXYETHYL)ETHER, ... | 著者 | Liu, Y, Lau, W, Bello, A.M, Kotra, L.P, Hui, R, Pai, E.F. | 登録日 | 2007-06-12 | 公開日 | 2008-01-29 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Structure-Activity Relationships of C6-Uridine Derivatives Targeting Plasmodia Orotidine Monophosphate Decarboxylase. J.Med.Chem., 51, 2008
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3R3V
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![BU of 3r3v by Molmil](/molmil-images/mine/3r3v) | Crystal Structure of the Fluoroacetate Dehalogenase RPA1163 - Asp110Asn/Fluoroacetate | 分子名称: | CALCIUM ION, CHLORIDE ION, Fluoroacetate dehalogenase, ... | 著者 | Chan, P.W.Y, Yakunin, A.F, Edwards, E.A, Pai, E.F. | 登録日 | 2011-03-16 | 公開日 | 2011-05-04 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Mapping the reaction coordinates of enzymatic defluorination. J.Am.Chem.Soc., 133, 2011
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2PG6
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![BU of 2pg6 by Molmil](/molmil-images/mine/2pg6) | Crystal Structure of Human Microsomal P450 2A6 L240C/N297Q | 分子名称: | Cytochrome P450 2A6, PROTOPORPHYRIN IX CONTAINING FE | 著者 | Sansen, S, Hsu, M.H, Stout, C.D, Johnson, E.F. | 登録日 | 2007-04-06 | 公開日 | 2007-07-24 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2.53 Å) | 主引用文献 | Structural insight into the altered substrate specificity of human cytochrome P450 2A6 mutants. Arch.Biochem.Biophys., 464, 2007
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