7VSG
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![BU of 7vsg by Molmil](/molmil-images/mine/7vsg) | |
7VSH
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7BSS
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![BU of 7bss by Molmil](/molmil-images/mine/7bss) | Cryo-EM structure of a human ATP11C-CDC50A flippase in E1AlF state | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, ATP11C, CDC50A, ... | 著者 | Abe, K, Nishizawa, T, Nakanishi, H. | 登録日 | 2020-03-31 | 公開日 | 2020-09-30 | 最終更新日 | 2020-10-14 | 実験手法 | ELECTRON MICROSCOPY (3.3 Å) | 主引用文献 | Transport Cycle of Plasma Membrane Flippase ATP11C by Cryo-EM. Cell Rep, 32, 2020
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7BSP
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![BU of 7bsp by Molmil](/molmil-images/mine/7bsp) | Cryo-EM structure of a human ATP11C-CDC50A flippase in E1-AMPPCP state | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-3)-2-acetamido-2-deoxy-beta-D-glucopyranose, ATP11C, ... | 著者 | Abe, K, Nishizawa, T, Nakanishi, H. | 登録日 | 2020-03-31 | 公開日 | 2020-09-30 | 最終更新日 | 2020-10-14 | 実験手法 | ELECTRON MICROSCOPY (4 Å) | 主引用文献 | Transport Cycle of Plasma Membrane Flippase ATP11C by Cryo-EM. Cell Rep, 32, 2020
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7BSV
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![BU of 7bsv by Molmil](/molmil-images/mine/7bsv) | Cryo-EM structure of a human ATP11C-CDC50A flippase in PtdSer-occluded E2-AlF state | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, ATP11C, CDC50A, ... | 著者 | Abe, K, Nishizawa, T, Nakanishi, H. | 登録日 | 2020-03-31 | 公開日 | 2020-09-30 | 最終更新日 | 2020-10-14 | 実験手法 | ELECTRON MICROSCOPY (3 Å) | 主引用文献 | Transport Cycle of Plasma Membrane Flippase ATP11C by Cryo-EM. Cell Rep, 32, 2020
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7BSW
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![BU of 7bsw by Molmil](/molmil-images/mine/7bsw) | Cryo-EM structure of a human ATP11C-CDC50A flippase in PtdEtn-occluded E2-AlF state | 分子名称: | 1,2-Dioleoyl-sn-glycero-3-phosphoethanolamine, 2-acetamido-2-deoxy-beta-D-glucopyranose, ATP11C, ... | 著者 | Abe, K, Nishizawa, T, Nakanishi, H. | 登録日 | 2020-03-31 | 公開日 | 2020-09-30 | 最終更新日 | 2020-10-14 | 実験手法 | ELECTRON MICROSCOPY (3.9 Å) | 主引用文献 | Transport Cycle of Plasma Membrane Flippase ATP11C by Cryo-EM. Cell Rep, 32, 2020
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7BSQ
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![BU of 7bsq by Molmil](/molmil-images/mine/7bsq) | Cryo-EM structure of a human ATP11C-CDC50A flippase in E1AlF-ADP state | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, ADENOSINE-5'-DIPHOSPHATE, ATP11C, ... | 著者 | Abe, K, Nishizawa, T, Nakanishi, H. | 登録日 | 2020-03-31 | 公開日 | 2020-09-30 | 最終更新日 | 2020-10-14 | 実験手法 | ELECTRON MICROSCOPY (3.2 Å) | 主引用文献 | Transport Cycle of Plasma Membrane Flippase ATP11C by Cryo-EM. Cell Rep, 32, 2020
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7BSU
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![BU of 7bsu by Molmil](/molmil-images/mine/7bsu) | Cryo-EM structure of a human ATP11C-CDC50A flippase in PtdSer-bound E2BeF state | 分子名称: | 1-deoxy-alpha-D-mannopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose, ATP11C, ... | 著者 | Abe, K, Nishizawa, T, Nakanishi, H. | 登録日 | 2020-03-31 | 公開日 | 2020-09-30 | 最終更新日 | 2020-10-14 | 実験手法 | ELECTRON MICROSCOPY (3.2 Å) | 主引用文献 | Transport Cycle of Plasma Membrane Flippase ATP11C by Cryo-EM. Cell Rep, 32, 2020
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6LKN
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![BU of 6lkn by Molmil](/molmil-images/mine/6lkn) | Crystal structure of ATP11C-CDC50A in PtdSer-bound E2P state | 分子名称: | 1-deoxy-alpha-D-mannopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose, Cell cycle control protein 50A, ... | 著者 | Abe, K, Irie, K, Nakanishi, H, Hasegawa, K. | 登録日 | 2019-12-19 | 公開日 | 2020-06-10 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (3.9 Å) | 主引用文献 | Crystal structure of a human plasma membrane phospholipid flippase. J.Biol.Chem., 295, 2020
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7X22
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![BU of 7x22 by Molmil](/molmil-images/mine/7x22) | Cryo-EM structure of non gastric H,K-ATPase alpha2 K794S in (2K+)E2-AlF state | 分子名称: | 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 2-acetamido-2-deoxy-beta-D-glucopyranose, CHOLESTEROL, ... | 著者 | Nakanishi, H, Abe, K. | 登録日 | 2022-02-25 | 公開日 | 2022-10-05 | 実験手法 | ELECTRON MICROSCOPY (3 Å) | 主引用文献 | Structure and function of H + /K + pump mutants reveal Na + /K + pump mechanisms. Nat Commun, 13, 2022
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7X20
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7X21
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![BU of 7x21 by Molmil](/molmil-images/mine/7x21) | Cryo-EM structure of non gastric H,K-ATPase alpha2 K794A in (K+)E2-AlF state | 分子名称: | 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 2-acetamido-2-deoxy-beta-D-glucopyranose, CHOLESTEROL, ... | 著者 | Nakanishi, H, Abe, K. | 登録日 | 2022-02-25 | 公開日 | 2022-10-05 | 実験手法 | ELECTRON MICROSCOPY (2.8 Å) | 主引用文献 | Structure and function of H + /K + pump mutants reveal Na + /K + pump mechanisms. Nat Commun, 13, 2022
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5YLU
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![BU of 5ylu by Molmil](/molmil-images/mine/5ylu) | Crystal structure of the gastric proton pump complexed with vonoprazan | 分子名称: | 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 1-[5-(2-fluorophenyl)-1-pyridin-3-ylsulfonyl-pyrrol-3-yl]-~{N}-methyl-methanamine, 2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Abe, K, Irie, K, Nakanishi, H, Fujiyoshi, Y. | 登録日 | 2017-10-19 | 公開日 | 2018-04-11 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.79988956 Å) | 主引用文献 | Crystal structures of the gastric proton pump Nature, 556, 2018
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5YLV
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![BU of 5ylv by Molmil](/molmil-images/mine/5ylv) | Crystal structure of the gastric proton pump complexed with SCH28080 | 分子名称: | 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 2-(2-methyl-8-phenylmethoxy-imidazo[1,2-a]pyridin-3-yl)ethanenitrile, 2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Abe, K, Irie, K, Nakanishi, H, Fujiyoshi, Y. | 登録日 | 2017-10-19 | 公開日 | 2018-04-11 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.79977775 Å) | 主引用文献 | Crystal structures of the gastric proton pump Nature, 556, 2018
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7X24
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![BU of 7x24 by Molmil](/molmil-images/mine/7x24) | Cryo-EM structure of non gastric H,K-ATPase alpha2 SPWC mutant in (2K+)E2-AlF state | 分子名称: | 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 2-acetamido-2-deoxy-beta-D-glucopyranose, CHOLESTEROL, ... | 著者 | Abe, K, Nakanishi, H, Young, V, Artigas, P. | 登録日 | 2022-02-25 | 公開日 | 2022-10-05 | 実験手法 | ELECTRON MICROSCOPY (3.4 Å) | 主引用文献 | Structure and function of H + /K + pump mutants reveal Na + /K + pump mechanisms. Nat Commun, 13, 2022
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7X23
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![BU of 7x23 by Molmil](/molmil-images/mine/7x23) | Cryo-EM structure of non gastric H,K-ATPase alpha2 SPWC mutant in 3Na+E1-AMPPCPF state | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, PHOSPHOMETHYLPHOSPHONIC ACID ADENYLATE ESTER, Potassium-transporting ATPase alpha chain 2, ... | 著者 | Abe, K, Nakanishi, H, Young, V, Artigas, P. | 登録日 | 2022-02-25 | 公開日 | 2022-10-05 | 実験手法 | ELECTRON MICROSCOPY (3.2 Å) | 主引用文献 | Structure and function of H + /K + pump mutants reveal Na + /K + pump mechanisms. Nat Commun, 13, 2022
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8K1L
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![BU of 8k1l by Molmil](/molmil-images/mine/8k1l) | Cryo-EM structure of Na+,K+-ATPase alpha2 from Artemia salina in cation-free E2P form | 分子名称: | Na+,K+-ATPase alpha2KK, Na+,K+-ATPase beta2, TETRAFLUOROALUMINATE ION | 著者 | Abe, K, Artigas, P. | 登録日 | 2023-07-11 | 公開日 | 2023-11-29 | 最終更新日 | 2024-01-31 | 実験手法 | ELECTRON MICROSCOPY (3.44 Å) | 主引用文献 | A Na pump with reduced stoichiometry is up-regulated by brine shrimp in extreme salinities. Proc.Natl.Acad.Sci.USA, 120, 2023
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1RKR
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![BU of 1rkr by Molmil](/molmil-images/mine/1rkr) | CRYSTAL STRUCTURE OF AZURIN-I FROM ALCALIGENES XYLOSOXIDANS NCIMB 11015 | 分子名称: | AZURIN-I, COPPER (II) ION | 著者 | Li, C, Inoue, T, Gotowda, M, Suzuki, S, Yamaguchi, K, Kataoka, K, Kai, Y. | 登録日 | 1997-05-17 | 公開日 | 1998-05-20 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.45 Å) | 主引用文献 | Structure of azurin I from the denitrifying bacterium Alcaligenes xylosoxidans NCIMB 11015 at 2.45 A resolution. Acta Crystallogr.,Sect.D, 54, 1998
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3HAT
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6JXK
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![BU of 6jxk by Molmil](/molmil-images/mine/6jxk) | Rb+-bound E2-MgF state of the gastric proton pump (Wild-type) | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, CHOLESTEROL, MAGNESIUM ION, ... | 著者 | Abe, K, Irie, K, Yamamoto, K. | 登録日 | 2019-04-23 | 公開日 | 2019-08-14 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (4.3 Å) | 主引用文献 | A single K + -binding site in the crystal structure of the gastric proton pump. Elife, 8, 2019
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6JXI
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6JXH
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6JXJ
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1FPC
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![BU of 1fpc by Molmil](/molmil-images/mine/1fpc) | ACTIVE SITE MIMETIC INHIBITION OF THROMBIN | 分子名称: | Hirudin, amino{[(4S)-4-({[5-(dimethylamino)naphthalen-1-yl]sulfonyl}amino)-5-(4-ethylpiperidin-1-yl)-5-oxopentyl]amino}methaniminium, thrombin | 著者 | Tulinsky, A, Mathews, I.I. | 登録日 | 1994-10-16 | 公開日 | 1995-02-27 | 最終更新日 | 2024-06-05 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Active-site mimetic inhibition of thrombin. Acta Crystallogr.,Sect.D, 51, 1995
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1A61
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![BU of 1a61 by Molmil](/molmil-images/mine/1a61) | THROMBIN COMPLEXED WITH A BETA-MIMETIC THIAZOLE-CONTAINING INHIBITOR | 分子名称: | (1S,7S)-7-amino-7-benzyl-N-{(1S)-4-carbamimidamido-1-[(S)-hydroxy(1,3-thiazol-2-yl)methyl]butyl}-8-oxohexahydro-1H-pyra zolo[1,2-a]pyridazine-1-carboxamide, ALPHA-THROMBIN (LARGE SUBUNIT), ALPHA-THROMBIN (SMALL SUBUNIT), ... | 著者 | St Charles, R, Matthews, J.H, Zhang, E, Tulinsky, A, Kahn, M. | 登録日 | 1998-03-05 | 公開日 | 1998-06-17 | 最終更新日 | 2024-06-05 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Bound structures of novel P3-P1' beta-strand mimetic inhibitors of thrombin. J.Med.Chem., 42, 1999
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