5XIG
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![BU of 5xig by Molmil](/molmil-images/mine/5xig) | Crystal Structure of Toxoplasma gondii Prolyl-tRNA Synthetase (TgPRS) in complex with Inhibitor 1 | 分子名称: | 3-[3-[(2R)-3-oxidanylidenepiperidin-2-yl]propyl]quinazolin-4-one, MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, ... | 著者 | Jain, V, Manickam, Y, Sharma, A. | 登録日 | 2017-04-26 | 公開日 | 2018-03-07 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.41 Å) | 主引用文献 | Targeting Prolyl-tRNA Synthetase to Accelerate Drug Discovery against Malaria, Leishmaniasis, Toxoplasmosis, Cryptosporidiosis, and Coccidiosis Structure, 25, 2017
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5XIP
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![BU of 5xip by Molmil](/molmil-images/mine/5xip) | Crystal Structure of Eimeria tenella Prolyl-tRNA Synthetase (EtPRS) in complex with Halofuginone | 分子名称: | 7-bromo-6-chloro-3-{3-[(2R,3S)-3-hydroxypiperidin-2-yl]-2-oxopropyl}quinazolin-4(3H)-one, MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, ... | 著者 | Jain, V, Manickam, Y, Sharma, A. | 登録日 | 2017-04-26 | 公開日 | 2018-03-07 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Targeting Prolyl-tRNA Synthetase to Accelerate Drug Discovery against Malaria, Leishmaniasis, Toxoplasmosis, Cryptosporidiosis, and Coccidiosis Structure, 25, 2017
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7ZM6
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![BU of 7zm6 by Molmil](/molmil-images/mine/7zm6) | Nariva virus receptor binding protein | 分子名称: | Attachment protein | 著者 | Stelfox, A.J, Rissanen, I, Rambo, R, Lee, B, Bowden, T.A. | 登録日 | 2022-04-19 | 公開日 | 2023-09-13 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.07 Å) | 主引用文献 | Crystal structure and solution state of the C-terminal head region of the narmovirus receptor binding protein. Mbio, 14, 2023
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7P4B
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![BU of 7p4b by Molmil](/molmil-images/mine/7p4b) | HLA-E*01:03 in complex with IL9 | 分子名称: | Beta-2-microglobulin, ESAT-6-like protein EsxH, GLYCEROL, ... | 著者 | Walters, L.C, Gillespie, G.M. | 登録日 | 2021-07-10 | 公開日 | 2022-07-27 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.72 Å) | 主引用文献 | Primary and secondary functions of HLA-E are determined by stability and conformation of the peptide-bound complexes. Cell Rep, 39, 2022
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7P49
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![BU of 7p49 by Molmil](/molmil-images/mine/7p49) | HLA-E*01:03 in complex with Mtb14 | 分子名称: | Beta-2-microglobulin, GLYCEROL, HLA class I histocompatibility antigen, ... | 著者 | Walters, L.C, Gillespie, G.M. | 登録日 | 2021-07-10 | 公開日 | 2022-06-22 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2.05 Å) | 主引用文献 | Primary and secondary functions of HLA-E are determined by stability and conformation of the peptide-bound complexes. Cell Rep, 39, 2022
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6I7R
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![BU of 6i7r by Molmil](/molmil-images/mine/6i7r) | |
6YJP
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![BU of 6yjp by Molmil](/molmil-images/mine/6yjp) | Crystal structure of a complex between glycosylated NKp30 and its deglycosylated tumour ligand B7-H6 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Natural cytotoxicity triggering receptor 3, Natural cytotoxicity triggering receptor 3 ligand 1 | 著者 | Skalova, T, Dohnalek, J, Skorepa, O, Kalouskova, B, Pazicky, S, Blaha, J, Vanek, O. | 登録日 | 2020-04-04 | 公開日 | 2020-07-29 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Natural Killer Cell Activation Receptor NKp30 Oligomerization Depends on Its N -Glycosylation. Cancers (Basel), 12, 2020
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6Z30
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![BU of 6z30 by Molmil](/molmil-images/mine/6z30) | Human cation-independent mannose 6-phosphate/ IGF2 receptor domains 9-10 | 分子名称: | Cation-independent mannose-6-phosphate receptor, alpha-D-mannopyranose-(1-3)-alpha-D-mannopyranose-(1-6)-[alpha-D-mannopyranose-(1-3)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose | 著者 | Bochel, A.J, Williams, C, Crump, M.P. | 登録日 | 2020-05-19 | 公開日 | 2020-08-19 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Structure of the Human Cation-Independent Mannose 6-Phosphate/IGF2 Receptor Domains 7-11 Uncovers the Mannose 6-Phosphate Binding Site of Domain 9. Structure, 28, 2020
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6Z31
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![BU of 6z31 by Molmil](/molmil-images/mine/6z31) | |
5JQ3
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![BU of 5jq3 by Molmil](/molmil-images/mine/5jq3) | Crystal structure of Ebola glycoprotein | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Envelope glycoprotein 1,Envelope glycoprotein 1,Envelope glycoprotein 1, Envelope glycoprotein 2, ... | 著者 | Zhao, Y, Ren, J, Stuart, D.I. | 登録日 | 2016-05-04 | 公開日 | 2016-06-29 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.23 Å) | 主引用文献 | Toremifene interacts with and destabilizes the Ebola virus glycoprotein. Nature, 535, 2016
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5JQB
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![BU of 5jqb by Molmil](/molmil-images/mine/5jqb) | Crystal structure of Ebola glycoprotein in complex with ibuprofen | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Envelope glycoprotein 1,Envelope glycoprotein 1,Envelope glycoprotein 1, Envelope glycoprotein 2, ... | 著者 | Zhao, Y, Ren, J, Stuart, D.I. | 登録日 | 2016-05-04 | 公開日 | 2016-06-29 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.68 Å) | 主引用文献 | Toremifene interacts with and destabilizes the Ebola virus glycoprotein. Nature, 535, 2016
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5JQ7
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![BU of 5jq7 by Molmil](/molmil-images/mine/5jq7) | Crystal structure of Ebola glycoprotein in complex with toremifene | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, DIMETHYL SULFOXIDE, Envelope glycoprotein 1,Envelope glycoprotein 1,Envelope glycoprotein 1, ... | 著者 | Zhao, Y, Ren, J, Stuart, D.I. | 登録日 | 2016-05-04 | 公開日 | 2016-06-29 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.69 Å) | 主引用文献 | Toremifene interacts with and destabilizes the Ebola virus glycoprotein. Nature, 535, 2016
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4QKJ
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![BU of 4qkj by Molmil](/molmil-images/mine/4qkj) | Glycosylated form of human LLT1, a ligand for NKR-P1, in this structure forming hexamers | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, C-type lectin domain family 2 member D | 著者 | Skalova, T, Blaha, J, Duskova, J, Koval, T, Stransky, J, Hasek, J, Vanek, O, Dohnalek, J. | 登録日 | 2014-06-06 | 公開日 | 2015-03-11 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.75 Å) | 主引用文献 | Four crystal structures of human LLT1, a ligand of human NKR-P1, in varied glycosylation and oligomerization states Acta Crystallogr.,Sect.D, 71, 2015
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6J7V
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![BU of 6j7v by Molmil](/molmil-images/mine/6j7v) | |
6IAK
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![BU of 6iak by Molmil](/molmil-images/mine/6iak) | The crystal structure of the chicken CREB3 bZIP | 分子名称: | Uncharacterized protein | 著者 | Sabaratnam, K, Renner, M. | 登録日 | 2018-11-26 | 公開日 | 2019-12-11 | 最終更新日 | 2020-06-24 | 実験手法 | X-RAY DIFFRACTION (3.95 Å) | 主引用文献 | Insights from the crystal structure of the chicken CREB3 bZIP suggest that members of the CREB3 subfamily transcription factors may be activated in response to oxidative stress. Protein Sci., 28, 2019
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7VC1
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![BU of 7vc1 by Molmil](/molmil-images/mine/7vc1) | Toxoplasma gondii Prolyl-tRNA Synthetase (TgPRS) in Complex with inhibitor L95 and L-proline in space group P21 | 分子名称: | 1,2-ETHANEDIOL, CHLORIDE ION, GLYCEROL, ... | 著者 | Yogavel, M, Malhotra, N, Sharma, A. | 登録日 | 2021-09-01 | 公開日 | 2022-09-07 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.892 Å) | 主引用文献 | Targeting prolyl-tRNA synthetase via a series of ATP-mimetics to accelerate drug discovery against toxoplasmosis. Plos Pathog., 19, 2023
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7VC2
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![BU of 7vc2 by Molmil](/molmil-images/mine/7vc2) | Toxoplasma gondii Prolyl-tRNA Synthetase (TgPRS) in Complex with inhibitor L96 and L-proline in space group P21 | 分子名称: | 1,2-ETHANEDIOL, 4-[(3S)-3-cyano-3-cyclopropyl-2-oxidanylidene-pyrrolidin-1-yl]-N-[[3-fluoranyl-5-(5-methoxypyridin-3-yl)phenyl]methyl]-6-methyl-pyridine-2-carboxamide, CHLORIDE ION, ... | 著者 | Yogavel, M, Malhotra, N, Sharma, A. | 登録日 | 2021-09-01 | 公開日 | 2022-09-07 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.096 Å) | 主引用文献 | Targeting prolyl-tRNA synthetase via a series of ATP-mimetics to accelerate drug discovery against toxoplasmosis. Plos Pathog., 19, 2023
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7VC3
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![BU of 7vc3 by Molmil](/molmil-images/mine/7vc3) | Toxoplasma gondii Prolyl-tRNA Synthetase (TgPRS) in Complex with inhibitor L97 and L-proline at 1.97 A resolution | 分子名称: | 4-[(3S)-3-cyclopropyl-3-(hydroxymethyl)-2-oxidanylidene-pyrrolidin-1-yl]-N-[[3-fluoranyl-5-(1-methylpyrazol-4-yl)phenyl]methyl]-6-methyl-pyridine-2-carboxamide, CHLORIDE ION, ETHANOLAMINE, ... | 著者 | Malhotra, N, Yogavel, M, Sharma, A. | 登録日 | 2021-09-01 | 公開日 | 2022-09-07 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.973 Å) | 主引用文献 | Targeting prolyl-tRNA synthetase via a series of ATP-mimetics to accelerate drug discovery against toxoplasmosis. Plos Pathog., 19, 2023
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2C6U
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![BU of 2c6u by Molmil](/molmil-images/mine/2c6u) | |
1POP
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![BU of 1pop by Molmil](/molmil-images/mine/1pop) | |
6I9I
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![BU of 6i9i by Molmil](/molmil-images/mine/6i9i) | |
2XR9
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![BU of 2xr9 by Molmil](/molmil-images/mine/2xr9) | Crystal structure of Autotaxin (ENPP2) | 分子名称: | CALCIUM ION, ECTONUCLEOTIDE PYROPHOSPHATASE/PHOSPHODIESTERASE FAMILY MEMBER 2, IODIDE ION, ... | 著者 | Kamtekar, S, Hausmann, J, Day, J.E, Christodoulou, E, Perrakis, A. | 登録日 | 2010-09-13 | 公開日 | 2011-01-19 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.05 Å) | 主引用文献 | Structural basis of substrate discrimination and integrin binding by autotaxin. Nat. Struct. Mol. Biol., 18, 2011
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2XRG
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![BU of 2xrg by Molmil](/molmil-images/mine/2xrg) | Crystal structure of Autotaxin (ENPP2) in complex with the HA155 boronic acid inhibitor | 分子名称: | CALCIUM ION, ECTONUCLEOTIDE PYROPHOSPHATASE/PHOSPHODIESTERASE FAMILY MEMBER 2, IODIDE ION, ... | 著者 | Hausmann, J, Albers, H.M.H.G, Perrakis, A. | 登録日 | 2010-09-14 | 公開日 | 2011-01-19 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (3.2 Å) | 主引用文献 | Structural Basis of Substrate Discrimination and Integrin Binding by Autotaxin. Nat.Struct.Mol.Biol., 18, 2011
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1UNS
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![BU of 1uns by Molmil](/molmil-images/mine/1uns) | IDENTIFICATION OF A SECONDARY ZINC-BINDING SITE IN STAPHYLOCOCCAL ENTEROTOXIN C2: IMPLICATIONS FOR SUPERANTIGEN RECOGNITION | 分子名称: | ENTEROTOXIN TYPE C-2, ZINC ION | 著者 | Papageorgiou, A.C, Baker, M.D, McLeod, J.D, Goda, S, Sansom, D.M, Tranter, H.S, Acharya, K.R. | 登録日 | 2003-09-15 | 公開日 | 2003-11-13 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Identification of a Secondary Zinc-Binding Site in Staphylococcal Enterotoxin C2: Implications for Superantigen Recognition J.Biol.Chem., 279, 2004
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5XIO
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![BU of 5xio by Molmil](/molmil-images/mine/5xio) | Crystal Structure of Cryptosporidium parvum Prolyl-tRNA Synthetase (CpPRS) in complex with Halofuginone | 分子名称: | 7-bromo-6-chloro-3-{3-[(2R,3S)-3-hydroxypiperidin-2-yl]-2-oxopropyl}quinazolin-4(3H)-one, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, Proline-tRNA synthetase class II aaRS (Ybak RNA binding domain plus tRNA synthetase), ... | 著者 | Jain, V, Manickam, Y, Sharma, A. | 登録日 | 2017-04-26 | 公開日 | 2018-03-07 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.46 Å) | 主引用文献 | Targeting Prolyl-tRNA Synthetase to Accelerate Drug Discovery against Malaria, Leishmaniasis, Toxoplasmosis, Cryptosporidiosis, and Coccidiosis Structure, 25, 2017
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