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7V3L
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MERS S ectodomain trimer in complex with neutralizing antibody 6516
分子名称: Spike glycoprotein, antibody H, antibody L
著者Wang, X, Zhao, J, Wang, Z, Wang, Y, Zeng, J.
登録日2021-08-10
公開日2022-08-17
実験手法ELECTRON MICROSCOPY (3.47 Å)
主引用文献MERS S ectodomain trimer in complex with neutralizing antibody 6516
to be published
6P05
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Bromodomain-containing protein 4 (BRD4) bromodomain 1 (BD1) complexed with compound 27
分子名称: Bromodomain-containing protein 4, GLYCEROL, N-{1-[1,1-di(pyridin-2-yl)ethyl]-6-(1-methyl-7-oxo-6,7-dihydro-1H-pyrrolo[2,3-c]pyridin-3-yl)-1H-indol-4-yl}ethanesulfonamide
著者Ratia, K.M, Xiong, R, Li, Y, Zhao, J, Gutgesell, L.M, Shen, Z, Dye, K, Dubrovyskyii, O, Zhao, H, Huang, F, Tonetti, D.A, Thatcher, G.R.
登録日2019-05-16
公開日2020-05-20
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (1.54 Å)
主引用文献Novel Pyrrolopyridone Bromodomain and Extra-Terminal Motif (BET) Inhibitors Effective in Endocrine-Resistant ER+ Breast Cancer with Acquired Resistance to Fulvestrant and Palbociclib.
J.Med.Chem., 63, 2020
1LPL
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Structural Genomics of Caenorhabditis elegans: CAP-Gly domain of F53F4.3
分子名称: Hypothetical 25.4 kDa protein F53F4.3 in chromosome V
著者Li, S, Finley, J, Liu, Z.-J, Qiu, S.H, Luan, C.H, Carson, M, Tsao, J, Johnson, D, Lin, G, Zhao, J, Thomas, W, Nagy, L.A, Sha, B, DeLucas, L.J, Wang, B.-C, Luo, M, Southeast Collaboratory for Structural Genomics (SECSG)
登録日2002-05-08
公開日2002-05-22
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.77 Å)
主引用文献Crystal Structure of the Cytoskeleton-associated Protein Glycine-rich (CAP-Gly) Domain
J.Biol.Chem., 277, 2002
6QRZ
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Crystal structure of R2-like ligand-binding oxidase from Sulfolobus acidocaldarius solved by 3D micro-crystal electron diffraction
分子名称: FE (III) ION, MANGANESE (III) ION, Ribonucleoside-diphosphate reductase
著者Xu, H, Lebrette, H, Clabbers, M.T.B, Zhao, J, Griese, J.J, Zou, X, Hogbom, M.
登録日2019-02-20
公開日2019-04-24
最終更新日2024-05-15
実験手法ELECTRON CRYSTALLOGRAPHY (3 Å)
主引用文献Solving a new R2lox protein structure by microcrystal electron diffraction.
Sci Adv, 5, 2019
7JKY
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Bromodomain-containing protein 4 (BRD4) bromodomain 1 (BD1) complexed with YF3-126
分子名称: Bromodomain-containing protein 4, N-(1-[1,1-di(pyridin-2-yl)ethyl]-6-{1-methyl-6-oxo-5-[(piperidin-4-yl)amino]-1,6-dihydropyridin-3-yl}-1H-indol-4-yl)ethanesulfonamide, SODIUM ION
著者Ratia, K.M, Xiong, R, Li, Y, Shen, Z, Zhao, J, Huang, F, Dubrovyskyii, O, Thatcher, G.R.
登録日2020-07-29
公開日2021-08-25
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.16 Å)
主引用文献Novel Pyrrolopyridone Bromodomain and Extra-Terminal Motif (BET) Inhibitors Effective in Endocrine-Resistant ER+ Breast Cancer with Acquired Resistance to Fulvestrant and Palbociclib.
J.Med.Chem., 63, 2020
7JKW
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Bromodomain-containing protein 4 (BRD4) bromodomain 1 (BD1) complexed with ZN1-99
分子名称: Bromodomain-containing protein 4, N-(6-{5-[(azetidin-3-yl)amino]-1-methyl-6-oxo-1,6-dihydropyridin-3-yl}-1-[1,1-di(pyridin-2-yl)ethyl]-1H-indol-4-yl)ethanesulfonamide
著者Ratia, K.M, Xiong, R, Li, Y, Shen, Z, Zhao, J, Huang, F, Dubrovyskyii, O, Thatcher, G.R.
登録日2020-07-29
公開日2021-08-25
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.2 Å)
主引用文献Novel Pyrrolopyridone Bromodomain and Extra-Terminal Motif (BET) Inhibitors Effective in Endocrine-Resistant ER+ Breast Cancer with Acquired Resistance to Fulvestrant and Palbociclib.
J.Med.Chem., 63, 2020
7JKZ
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Bromodomain-containing protein 4 (BRD4) bromodomain 2 (BD2) complexed with YF3-126
分子名称: 1,2-ETHANEDIOL, Bromodomain-containing protein 4, GLYCEROL, ...
著者Ratia, K.M, Xiong, R, Li, Y, Shen, Z, Zhao, J, Huang, F, Dubrovyskyii, O, Thatcher, G.R.
登録日2020-07-29
公開日2021-08-25
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.49 Å)
主引用文献Novel Pyrrolopyridone Bromodomain and Extra-Terminal Motif (BET) Inhibitors Effective in Endocrine-Resistant ER+ Breast Cancer with Acquired Resistance to Fulvestrant and Palbociclib.
J.Med.Chem., 63, 2020
5DO2
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Complex structure of MERS-RBD bound with 4C2 antibody
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 4C2 heavy chain, 4C2 light chain, ...
著者Li, Y, Wan, Y, Liu, P, Zhao, J, Lu, G, Qi, J, Wang, Q, Lu, X, Wu, Y, Liu, W, Yuen, K.Y, Perlman, S, Gao, G.F, Yan, J.
登録日2015-09-10
公開日2015-10-14
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.409 Å)
主引用文献A humanized neutralizing antibody against MERS-CoV targeting the receptor-binding domain of the spike protein.
Cell Res., 25, 2015
1TOV
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Structural genomics of Caenorhabditis elegans: CAP-GLY domain of F53F4.3
分子名称: Hypothetical protein F53F4.3 in chromosome V, SULFATE ION
著者Li, S, Finley, J, Liu, Z.J, Qiu, S.H, Luan, C.H, Carson, M, Tsao, J, Johnson, D, Lin, G, Zhao, J, Thomas, W, Nagy, L.A, Sha, B, Delucas, L.J, Richardson, D, Richardson, J, Wang, B.C, Luo, M, Southeast Collaboratory for Structural Genomics (SECSG)
登録日2004-06-15
公開日2004-07-27
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.77 Å)
主引用文献Crystal Structure of the Cytoskeleton-Associated Protein Glycine-Rich (CAP-Gly) Domain
J.Biol.Chem., 277, 2002
7RUH
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Bromodomain-containing protein 4 (BRD4) bromodomain 2 (BD2) complexed with XR844
分子名称: Bromodomain-containing protein 4, N-{1-[1,1-di(pyridin-2-yl)ethyl]-6-(5-{[(2-fluorophenyl)carbamoyl]amino}-1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-1H-indol-4-yl}-2,2,2-trifluoroethane-1-sulfonamide
著者Ratia, K.M, Xiong, R, Li, Y, Shen, Z, Zhao, J, Huang, F, Dubrovyskyii, O, Thatcher, G.R.
登録日2021-08-17
公開日2022-08-24
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Bromodomain-containing protein 4 (BRD4) bromodomain 2 (BD2) complexed with XR844
To Be Published
7RUI
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Bromodomain-containing protein 4 (BRD4) bromodomain 1 (BD1) complexed with XR844
分子名称: Bromodomain-containing protein 4, N-{1-[1,1-di(pyridin-2-yl)ethyl]-6-(5-{[(2-fluorophenyl)carbamoyl]amino}-1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-1H-indol-4-yl}-2,2,2-trifluoroethane-1-sulfonamide
著者Ratia, K.M, Xiong, R, Li, Y, Shen, Z, Zhao, J, Huang, F, Dubrovyskyii, O, Thatcher, G.R.
登録日2021-08-17
公開日2022-08-24
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.35 Å)
主引用文献Bromodomain-containing protein 4 (BRD4) bromodomain 1 (BD1) complexed with XR844
To Be Published
1JXF
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SOLUTION STRUCTURE OF REDUCED CU(I) PLASTOCYANIN FROM SYNECHOCYSTIS PCC6803
分子名称: COPPER (II) ION, PLASTOCYANIN
著者Bertini, I, Bryant, D.A, Ciurli, S, Dikiy, A, Fernandez, C.O, Luchinat, C, Safarov, N, Vila, A.J, Zhao, J.
登録日2001-09-07
公開日2001-09-26
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Backbone dynamics of plastocyanin in both oxidation states. Solution structure of the reduced form and comparison with the oxidized state.
J.Biol.Chem., 276, 2001
1JXD
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SOLUTION STRUCTURE OF REDUCED CU(I) PLASTOCYANIN FROM SYNECHOCYSTIS PCC6803
分子名称: COPPER (II) ION, PLASTOCYANIN
著者Bertini, I, Bryant, D.A, Ciurli, S, Dikiy, A, Fernandez, C.O, Luchinat, C, Safarov, N, Vila, A.J, Zhao, J.
登録日2001-09-07
公開日2001-09-26
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Backbone dynamics of plastocyanin in both oxidation states. Solution structure of the reduced form and comparison with the oxidized state.
J.Biol.Chem., 276, 2001
6BGI
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Cryo-EM structure of the TMEM16A calcium-activated chloride channel in nanodisc
分子名称: Anoctamin-1, CALCIUM ION
著者Dang, S, Feng, S, Tien, J, Peters, C.J, Bulkley, D, Lolicato, M, Zhao, J, Zuberbuhler, K, Ye, W, Qi, J, Chen, T, Craik, C.S, Jan, Y.N, Minor Jr, D.L, Cheng, Y, Jan, L.Y.
登録日2017-10-28
公開日2017-12-27
最終更新日2024-03-13
実験手法ELECTRON MICROSCOPY (3.8 Å)
主引用文献Cryo-EM structures of the TMEM16A calcium-activated chloride channel.
Nature, 552, 2017
1T0L
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Crystal structure of human cytosolic NADP(+)-dependent isocitrate dehydrogenase in complex with NADP, isocitrate, and calcium(2+)
分子名称: CALCIUM ION, ISOCITRIC ACID, Isocitrate dehydrogenase [NADP] cytoplasmic, ...
著者Xu, X, Zhao, J, Peng, B, Huang, Q, Arnold, E, Ding, J.
登録日2004-04-10
公開日2004-06-15
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.41 Å)
主引用文献Structures of human cytosolic NADP-dependent isocitrate dehydrogenase reveal a novel self-regulatory mechanism of activity
J.Biol.Chem., 279, 2004
1T09
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Crystal structure of human cytosolic NADP(+)-dependent isocitrate dehydrogenase in complex NADP
分子名称: Isocitrate dehydrogenase [NADP] cytoplasmic, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE
著者Xu, X, Zhao, J, Peng, B, Huang, Q, Arnold, E, Ding, J.
登録日2004-04-08
公開日2004-06-15
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Structures of human cytosolic NADP-dependent isocitrate dehydrogenase reveal a novel self-regulatory mechanism of activity
J.Biol.Chem., 279, 2004
6BGJ
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Cryo-EM structure of the TMEM16A calcium-activated chloride channel in LMNG
分子名称: Anoctamin-1, CALCIUM ION
著者Dang, S, Feng, S, Tien, J, Peters, C.J, Bulkley, D, Lolicato, M, Zhao, J, Zuberbuhler, K, Ye, W, Qi, L, Chen, T, Craik, C.S, Jan, Y.N, Minor Jr, D.L, Cheng, Y, Jan, L.Y.
登録日2017-10-28
公開日2017-12-27
最終更新日2024-03-13
実験手法ELECTRON MICROSCOPY (3.8 Å)
主引用文献Cryo-EM structures of the TMEM16A calcium-activated chloride channel.
Nature, 552, 2017
8GXI
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The crystal structure of SARS-CoV-2 main protease in complex with 14c
分子名称: 3C-like proteinase nsp5, N-[(2S)-3-cyclohexyl-1-[[(2S,3R)-4-(cyclopropylamino)-3-oxidanyl-4-oxidanylidene-1-[(3S)-2-oxidanylidenepiperidin-3-yl]butan-2-yl]amino]-1-oxidanylidene-propan-2-yl]-1-benzofuran-2-carboxamide
著者Zhao, Y, Zhao, J, Shao, M, Yang, H, Rao, Z.
登録日2022-09-20
公開日2023-09-27
実験手法X-RAY DIFFRACTION (1.69 Å)
主引用文献The crystal structure of SARS-CoV-2 main protease in complex with 14c
To Be Published
8GXH
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The crystal structure of SARS-CoV-2 main protease in complex with 14b
分子名称: 3C-like proteinase nsp5, N-[(2S)-3-cyclohexyl-1-oxidanylidene-1-[[(2S,3R)-3-oxidanyl-4-oxidanylidene-1-[(3S)-2-oxidanylidenepiperidin-3-yl]-4-[(phenylmethyl)amino]butan-2-yl]amino]propan-2-yl]-1-benzofuran-2-carboxamide
著者Zhao, Y, Zhao, J, Shao, M, Yang, H, Rao, Z.
登録日2022-09-20
公開日2023-09-27
実験手法X-RAY DIFFRACTION (1.59 Å)
主引用文献The crystal structure of SARS-CoV-2 main protease in complex with 14b
To Be Published
8GX3
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The crystal structure of human Calpain-1 protease core in complex with 14c
分子名称: CALCIUM ION, Calpain-1 catalytic subunit, N-[(2S)-3-cyclohexyl-1-[[(2S,3S)-4-(cyclopropylamino)-3-oxidanyl-4-oxidanylidene-1-[(3S)-2-oxidanylidenepiperidin-3-yl]butan-2-yl]amino]-1-oxidanylidene-propan-2-yl]-1-benzofuran-2-carboxamide
著者Zhao, Y, Zhao, J, Shao, M, Yang, H, Rao, Z.
登録日2022-09-18
公開日2023-09-20
実験手法X-RAY DIFFRACTION (1.99 Å)
主引用文献The crystal structure of human Calpain-1 protease core in complex with 14c
To Be Published
8GX2
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The crystal structure of human CtsL in complex with 14c
分子名称: DIMETHYL SULFOXIDE, N-[(2S)-3-cyclohexyl-1-[[(2S,3S)-4-(cyclopropylamino)-3-oxidanyl-4-oxidanylidene-1-[(3S)-2-oxidanylidenepiperidin-3-yl]butan-2-yl]amino]-1-oxidanylidene-propan-2-yl]-1-benzofuran-2-carboxamide, Procathepsin L
著者Zhao, Y, Shao, M, Zhao, J, Yang, H, Rao, Z.
登録日2022-09-18
公開日2023-09-20
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献The crystal structure of human CtsL in complex with 14a
To Be Published
8GXG
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The crystal structure of SARS-CoV-2 main protease in complex with 14a
分子名称: 3C-like proteinase nsp5, N-[(2S)-3-(4-fluorophenyl)-1-oxidanylidene-1-[[(2S,3S)-3-oxidanyl-4-oxidanylidene-1-[(3S)-2-oxidanylidenepiperidin-3-yl]-4-[(phenylmethyl)amino]butan-2-yl]amino]propan-2-yl]-1-benzofuran-2-carboxamide
著者Zhao, Y, Zhao, J, Shao, M, Yang, H, Rao, Z.
登録日2022-09-20
公開日2023-09-27
実験手法X-RAY DIFFRACTION (1.69 Å)
主引用文献The crystal structure of SARS-CoV-2 main protease in complex with 14a
To Be Published
6WK7
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Crystal Structure Analysis of a poly(thymine) DNA duplex
分子名称: 1,3,5-triazine-2,4,6-triamine, DNA (5'-D(*TP*TP*TP*TP*TP*T)-3')
著者Li, Q, Zhao, J, Liu, L, Mandal, S, Rizzuto, F.J, He, H, Wei, S, Jonchhe, S, Sleiman, H.F, Mao, H, Mao, C.
登録日2020-04-15
公開日2020-07-22
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.423 Å)
主引用文献A poly(thymine)-melamine duplex for the assembly of DNA nanomaterials.
Nat Mater, 19, 2020
1PSE
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THE THREE-DIMENSIONAL SOLUTION STRUCTURE OF PSAE FROM THE CYANOBACTERIUM SYNECHOCOCCUS SP. STRAIN PCC 7002: A PHOTOSYSTEM I PROTEIN THAT SHOWS STRUCTURAL HOMOLOGY WITH SH3 DOMAINS
分子名称: PHOTOSYSTEM I ACCESSORY PROTEIN E
著者Falzone, C.J, Kao, Y.-H, Zhao, J, Bryant, D.A, Lecomte, J.T.J.
登録日1994-04-13
公開日1995-04-20
最終更新日2024-05-01
実験手法SOLUTION NMR
主引用文献Three-dimensional solution structure of PsaE from the cyanobacterium Synechococcus sp. strain PCC 7002, a photosystem I protein that shows structural homology with SH3 domains.
Biochemistry, 33, 1994
1PSF
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THE THREE-DIMENSIONAL SOLUTION STRUCTURE OF PSAE FROM THE CYANOBACTERIUM SYNECHOCOCCUS SP. STRAIN PCC 7002: A PHOTOSYSTEM I PROTEIN THAT SHOWS STRUCTURAL HOMOLOGY WITH SH3 DOMAINS
分子名称: PHOTOSYSTEM I ACCESSORY PROTEIN E
著者Falzone, C.J, Kao, Y.-H, Zhao, J, Bryant, D.A, Lecomte, J.T.J.
登録日1994-04-13
公開日1995-04-20
最終更新日2024-05-01
実験手法SOLUTION NMR
主引用文献Three-dimensional solution structure of PsaE from the cyanobacterium Synechococcus sp. strain PCC 7002, a photosystem I protein that shows structural homology with SH3 domains.
Biochemistry, 33, 1994

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