8BG0
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![BU of 8bg0 by Molmil](/molmil-images/mine/8bg0) | Amyloid-beta tetrameric filaments with the Arctic mutation (E22G) from Alzheimer's disease brains | ABeta40 | 分子名称: | Amyloid-beta precursor protein | 著者 | Yang, Y, Zhang, W.J, Murzin, A.G, Schweighauser, M, Huang, M, Lovestam, S.K.A, Peak-Chew, S.Y, Macdonald, J, Lavenir, I, Ghetti, B, Graff, C, Kumar, A, Nordber, A, Goedert, M, Scheres, S.H.W. | 登録日 | 2022-10-27 | 公開日 | 2023-01-18 | 最終更新日 | 2023-02-22 | 実験手法 | ELECTRON MICROSCOPY (1.9 Å) | 主引用文献 | Cryo-EM structures of amyloid-beta filaments with the Arctic mutation (E22G) from human and mouse brains. Acta Neuropathol, 145, 2023
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8BFZ
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![BU of 8bfz by Molmil](/molmil-images/mine/8bfz) | Amyloid-beta 42 filaments extracted from the human brain with Arctic mutation (E22G) of Alzheimer's disease | ABeta42 | 分子名称: | Amyloid-beta precursor protein | 著者 | Yang, Y, Zhang, W.J, Murzin, A.G, Schweighauser, M, Huang, M, Lovestam, S.K.A, Peak-Chew, S.Y, Macdonald, J, Lavenir, I, Ghetti, B, Graff, C, Kumar, A, Nordberg, A, Goedert, M, Scheres, S.H.W. | 登録日 | 2022-10-27 | 公開日 | 2023-01-18 | 最終更新日 | 2024-01-31 | 実験手法 | ELECTRON MICROSCOPY (2.8 Å) | 主引用文献 | Cryo-EM structures of amyloid-beta filaments with the Arctic mutation (E22G) from human and mouse brains. Acta Neuropathol, 145, 2023
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3K37
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3K38
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![BU of 3k38 by Molmil](/molmil-images/mine/3k38) | |
3K3A
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8HUB
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![BU of 8hub by Molmil](/molmil-images/mine/8hub) | AMP deaminase 2 in complex with an inhibitor | 分子名称: | 3,3-dimethyl-4-(phenylmethyl)-2~{H}-quinoxaline-1-carboxamide, AMP deaminase 2, ZINC ION | 著者 | Adachi, T, Doi, S. | 登録日 | 2022-12-23 | 公開日 | 2023-01-18 | 最終更新日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (3.25 Å) | 主引用文献 | The discovery of 3,3-dimethyl-1,2,3,4-tetrahydroquinoxaline-1-carboxamides as AMPD2 inhibitors with a novel mechanism of action. Bioorg.Med.Chem.Lett., 80, 2023
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8HU6
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![BU of 8hu6 by Molmil](/molmil-images/mine/8hu6) | AMP deaminase 2 in complex with AMP | 分子名称: | ADENOSINE MONOPHOSPHATE, AMP deaminase 2, SULFATE ION, ... | 著者 | Adachi, T, Doi, S. | 登録日 | 2022-12-22 | 公開日 | 2023-01-18 | 最終更新日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (2.33 Å) | 主引用文献 | The discovery of 3,3-dimethyl-1,2,3,4-tetrahydroquinoxaline-1-carboxamides as AMPD2 inhibitors with a novel mechanism of action. Bioorg.Med.Chem.Lett., 80, 2023
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3AUJ
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![BU of 3auj by Molmil](/molmil-images/mine/3auj) | Structure of diol dehydratase complexed with glycerol | 分子名称: | CALCIUM ION, COBALAMIN, Diol dehydrase alpha subunit, ... | 著者 | Yamanishi, M, Kinoshita, K, Fukuoka, M, Shibata, T, Tobimatsu, T, Toraya, T. | 登録日 | 2011-02-07 | 公開日 | 2012-02-22 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Redesign of coenzyme B(12) dependent diol dehydratase to be resistant to the mechanism-based inactivation by glycerol and act on longer chain 1,2-diols Febs J., 279, 2012
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5AZV
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![BU of 5azv by Molmil](/molmil-images/mine/5azv) | Crystal structure of hPPARgamma ligand binding domain complexed with 17-oxoDHA | 分子名称: | (4~{Z},7~{Z},10~{Z},13~{Z},19~{Z})-17-oxidanylidenedocosa-4,7,10,13,19-pentaenoic acid, Peroxisome proliferator-activated receptor gamma | 著者 | Egawa, D, Itoh, T, Yamamoto, K. | 登録日 | 2015-10-23 | 公開日 | 2016-07-06 | 最終更新日 | 2020-02-26 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | 17-OxoDHA Is a PPAR alpha/gamma Dual Covalent Modifier and Agonist Acs Chem.Biol., 2016
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5AZT
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![BU of 5azt by Molmil](/molmil-images/mine/5azt) | Ternary complex of hPPARalpha ligand binding domain, 17-oxoDHA and a SRC1 peptide | 分子名称: | (4~{Z},7~{Z},10~{Z},13~{Z},19~{Z})-17-oxidanylidenedocosa-4,7,10,13,19-pentaenoic acid, 15-meric peptide from Nuclear receptor coactivator 1, Peroxisome proliferator-activated receptor alpha | 著者 | Egawa, D, Itoh, T, Yamamoto, K. | 登録日 | 2015-10-23 | 公開日 | 2016-07-06 | 最終更新日 | 2020-02-26 | 実験手法 | X-RAY DIFFRACTION (3.45 Å) | 主引用文献 | 17-OxoDHA Is a PPAR alpha/gamma Dual Covalent Modifier and Agonist Acs Chem.Biol., 2016
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3K39
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3K36
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3WDZ
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![BU of 3wdz by Molmil](/molmil-images/mine/3wdz) | Crystal Structure of Keap1 in Complex with phosphorylated p62 | 分子名称: | Kelch-like ECH-associated protein 1, Peptide from Sequestosome-1 | 著者 | Fukutomi, T, Takagi, K, Mizushima, T, Tanaka, K, Komatsu, M, Yamamoto, M. | 登録日 | 2013-06-26 | 公開日 | 2013-09-04 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Phosphorylation of p62 activates the Keap1-Nrf2 pathway during selective autophagy. Mol.Cell, 51, 2013
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7E5P
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![BU of 7e5p by Molmil](/molmil-images/mine/7e5p) | Aptamer enhancing peroxidase activity of myoglobin | 分子名称: | DNA (5'-D(*GP*GP*GP*TP*GP*GP*GP*TP*TP*GP*GP*GP*AP*GP*GP*G)-3') | 著者 | Tsukakoshi, K, Matsugami, A, Khunathai, K, Kanazashi, M, Yamagishi, Y, Nakama, K, Oshikawa, D, Hayashi, F, Kuno, H, Ikebukuro, K. | 登録日 | 2021-02-19 | 公開日 | 2021-06-16 | 最終更新日 | 2024-05-15 | 実験手法 | SOLUTION NMR | 主引用文献 | G-quadruplex-forming aptamer enhances the peroxidase activity of myoglobin against luminol. Nucleic Acids Res., 49, 2021
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5Z8Y
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![BU of 5z8y by Molmil](/molmil-images/mine/5z8y) | Crystal structure of human LRRTM2 in complex with Neurexin 1beta | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ... | 著者 | Yamagata, A, Fukai, S. | 登録日 | 2018-02-01 | 公開日 | 2018-10-10 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (3.4 Å) | 主引用文献 | Structural insights into modulation and selectivity of transsynaptic neurexin-LRRTM interaction. Nat Commun, 9, 2018
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5Z8X
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![BU of 5z8x by Molmil](/molmil-images/mine/5z8x) | Crystal structure of human LRRTM2 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Leucine-rich repeat transmembrane neuronal protein 2 | 著者 | Yamagata, A, Fukai, S. | 登録日 | 2018-02-01 | 公開日 | 2018-10-10 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (3.15 Å) | 主引用文献 | Structural insights into modulation and selectivity of transsynaptic neurexin-LRRTM interaction. Nat Commun, 9, 2018
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7CEG
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![BU of 7ceg by Molmil](/molmil-images/mine/7ceg) | Crystal structure of the complex between mouse PTP delta and neuroligin-3 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Isoform C of Receptor-type tyrosine-protein phosphatase delta, Neuroligin-3 | 著者 | Yamagata, A, Yoshida, T, Shiroshima, T, Maeda, A, Fukai, S. | 登録日 | 2020-06-23 | 公開日 | 2021-02-24 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (3.85 Å) | 主引用文献 | Canonical versus non-canonical transsynaptic signaling of neuroligin 3 tunes development of sociality in mice. Nat Commun, 12, 2021
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7CEE
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![BU of 7cee by Molmil](/molmil-images/mine/7cee) | Crystal structure of mouse neuroligin-3 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Neuroligin-3 | 著者 | Yamagata, A, Yoshida, T, Shiroshima, T, Maeda, A, Fukai, S. | 登録日 | 2020-06-23 | 公開日 | 2021-02-24 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.763 Å) | 主引用文献 | Canonical versus non-canonical transsynaptic signaling of neuroligin 3 tunes development of sociality in mice. Nat Commun, 12, 2021
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3B2G
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![BU of 3b2g by Molmil](/molmil-images/mine/3b2g) | Leptolyngbya boryana Ferredoxin | 分子名称: | FE2/S2 (INORGANIC) CLUSTER, Ferredoxin-1 | 著者 | Kurisu, G, Hase, T. | 登録日 | 2011-08-01 | 公開日 | 2012-06-13 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (1.76 Å) | 主引用文献 | A new structural insight into differential interaction of cyanobacterial and plant ferredoxins with nitrite reductase as revealed by NMR and X-ray crystallographic studies J.Biochem., 151, 2012
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3B2F
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![BU of 3b2f by Molmil](/molmil-images/mine/3b2f) | Maize Ferredoxin 1 | 分子名称: | FE2/S2 (INORGANIC) CLUSTER, Ferredoxin-1, chloroplastic | 著者 | Kurisu, G, Hase, T. | 登録日 | 2011-08-01 | 公開日 | 2012-06-13 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | A new structural insight into differential interaction of cyanobacterial and plant ferredoxins with nitrite reductase as revealed by NMR and X-ray crystallographic studies J.Biochem., 151, 2012
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