2BFX
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![BU of 2bfx by Molmil](/molmil-images/mine/2bfx) | Mechanism of Aurora-B activation by INCENP and inhibition by Hesperadin. | 分子名称: | AURORA KINASE B-A, INNER CENTROMERE PROTEIN A | 著者 | Sessa, F, Mapelli, M, Ciferri, C, Tarricone, C, Areces, L.B, Schneider, T.R, Stukenberg, P.T, Musacchio, A. | 登録日 | 2004-12-15 | 公開日 | 2005-05-03 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Mechanism of Aurora B Activation by Incenp and Inhibition by Hesperadin Mol.Cell, 18, 2005
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2VE7
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![BU of 2ve7 by Molmil](/molmil-images/mine/2ve7) | Crystal structure of a bonsai version of the human Ndc80 complex | 分子名称: | GLYCEROL, KINETOCHORE PROTEIN HEC1, KINETOCHORE PROTEIN SPC25, ... | 著者 | Ciferri, C, Pasqualato, S, Dos Reis, G, Screpanti, E, Maiolica, A, Polka, J, De Luca, J.G, De Wulf, P, Salek, M, Rappsilber, J, Moores, C.A, Salmon, E.D, Musacchio, A. | 登録日 | 2007-10-17 | 公開日 | 2008-05-13 | 最終更新日 | 2024-06-19 | 実験手法 | X-RAY DIFFRACTION (2.88 Å) | 主引用文献 | Implications for Kinetochore-Microtubule Attachment from the Structure of an Engineered Ndc80 Complex Cell(Cambridge,Mass.), 133, 2008
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2XBB
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![BU of 2xbb by Molmil](/molmil-images/mine/2xbb) | Nedd4 HECT:Ub complex | 分子名称: | E3 UBIQUITIN-PROTEIN LIGASE NEDD4, GLYCEROL, UBIQUITIN | 著者 | Maspero, E, Cecatiello, V, Musacchio, A, Polo, S, Pasqualato, S. | 登録日 | 2010-04-08 | 公開日 | 2011-03-23 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.68 Å) | 主引用文献 | Structure of the Hect:Ubiquitin Complex and its Role in Ubiquitin Chain Elongation Embo Rep., 12, 2011
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2V66
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![BU of 2v66 by Molmil](/molmil-images/mine/2v66) | |
2XBF
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![BU of 2xbf by Molmil](/molmil-images/mine/2xbf) | Nedd4 HECT structure | 分子名称: | 1,2-ETHANEDIOL, CALCIUM ION, E3 UBIQUITIN-PROTEIN LIGASE NEDD4 | 著者 | Maspero, E, Cecatiello, V, Musacchio, A, Polo, S, Pasqualato, S. | 登録日 | 2010-04-09 | 公開日 | 2011-03-23 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.503 Å) | 主引用文献 | Structure of the Hect:Ubiquitin Complex and its Role in Ubiquitin Chain Elongation Embo Rep., 12, 2011
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1RGP
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![BU of 1rgp by Molmil](/molmil-images/mine/1rgp) | GTPASE-ACTIVATION DOMAIN FROM RHOGAP | 分子名称: | RHOGAP | 著者 | Barrett, T, Xiao, B, Dodson, E.J, Dodson, G, Ludbrook, S.B, Nurmahomed, K, Gamblin, S.J, Musacchio, A, Smerdon, S.J, Eccleston, J.F. | 登録日 | 1996-12-05 | 公開日 | 1997-10-15 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | The structure of the GTPase-activating domain from p50rhoGAP. Nature, 385, 1997
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1UNL
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![BU of 1unl by Molmil](/molmil-images/mine/1unl) | Structural mechanism for the inhibition of CD5-p25 from the roscovitine, aloisine and indirubin. | 分子名称: | CYCLIN-DEPENDENT KINASE 5, CYCLIN-DEPENDENT KINASE 5 ACTIVATOR 1, R-ROSCOVITINE | 著者 | Mapelli, M, Crovace, C, Massimiliano, L, Musacchio, A. | 登録日 | 2003-09-10 | 公開日 | 2004-11-10 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Mechanism of Cdk5/P25 Binding by Cdk Inhibitors J.Med.Chem., 48, 2005
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1UNG
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![BU of 1ung by Molmil](/molmil-images/mine/1ung) | Structural mechanism for the inhibition of CDK5-p25 by roscovitine, aloisine and indirubin. | 分子名称: | 6-PHENYL[5H]PYRROLO[2,3-B]PYRAZINE, CELL DIVISION PROTEIN KINASE 5, CYCLIN-DEPENDENT KINASE 5 ACTIVATOR 1 | 著者 | Mapelli, M, Crovace, C, Massimiliano, L, Musacchio, A. | 登録日 | 2003-09-10 | 公開日 | 2004-11-10 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Mechanism of Cdk5/P25 Binding by Cdk Inhibitors J.Med.Chem., 48, 2005
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1UNH
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![BU of 1unh by Molmil](/molmil-images/mine/1unh) | Structural mechanism for the inhibition of CDK5-p25 by roscovitine, aloisine and indirubin. | 分子名称: | (Z)-1H,1'H-[2,3']BIINDOLYLIDENE-3,2'-DIONE-3-OXIME, CYCLIN-DEPENDENT KINASE 5, CYCLIN-DEPENDENT KINASE 5 ACTIVATOR 1 | 著者 | Mapelli, M, Crovace, C, Massimiliano, L, Musacchio, A. | 登録日 | 2003-09-10 | 公開日 | 2004-11-10 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (2.35 Å) | 主引用文献 | Mechanism of Cdk5/P25 Binding by Cdk Inhibitors J.Med.Chem., 48, 2005
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1SHF
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![BU of 1shf by Molmil](/molmil-images/mine/1shf) | |
2VGP
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![BU of 2vgp by Molmil](/molmil-images/mine/2vgp) | Crystal structure of Aurora B kinase in complex with a aminothiazole inhibitor | 分子名称: | 4-[(5-bromo-1,3-thiazol-2-yl)amino]-N-methylbenzamide, INNER CENTROMERE PROTEIN A, SERINE/THREONINE-PROTEIN KINASE 12-A | 著者 | Andersen, C.B, Wan, Y, Chang, J.W, Lee, C, Liu, Y, Sessa, F, Villa, F, Nallan, L, Musacchio, A, Gray, N.S. | 登録日 | 2007-11-15 | 公開日 | 2008-02-26 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Discovery of Selective Aminothiazole Aurora Kinase Inhibitors Acs Chem.Biol., 3, 2008
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2VRX
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![BU of 2vrx by Molmil](/molmil-images/mine/2vrx) | Structure of Aurora B kinase in complex with ZM447439 | 分子名称: | INNER CENTROMERE PROTEIN A, N-(4-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinazolin-4-yl]amino}phenyl)benzamide, SERINE/THREONINE-PROTEIN KINASE 12-A | 著者 | Girdler, F, Sessa, F, Patercoli, S, Villa, F, Ridgway, E, Musacchio, A, Taylor, S.S. | 登録日 | 2008-04-16 | 公開日 | 2008-07-01 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (1.86 Å) | 主引用文献 | Molecular Basis of Drug Resistance in Aurora Kinases. Chem.Biol., 15, 2008
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2VGO
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![BU of 2vgo by Molmil](/molmil-images/mine/2vgo) | Crystal structure of Aurora B kinase in complex with Reversine inhibitor | 分子名称: | INNER CENTROMERE PROTEIN A, N~6~-cyclohexyl-N~2~-(4-morpholin-4-ylphenyl)-9H-purine-2,6-diamine, SERINE/THREONINE-PROTEIN KINASE 12-A | 著者 | D'Alise, A.M, Amabile, G, Iovino, M, Di Giorgio, F.P, Bartiromo, M, Sessa, F, Villa, F, Musacchio, A, Cortese, R. | 登録日 | 2007-11-15 | 公開日 | 2008-10-28 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Reversine, a Novel Aurora Kinases Inhibitor, Inhibits Colony Formation of Human Acute Myeloid Leukemia Cells. Mol.Cancer Ther., 7, 2008
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2V64
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![BU of 2v64 by Molmil](/molmil-images/mine/2v64) | Crystallographic structure of the conformational dimer of the Spindle Assembly Checkpoint protein Mad2. | 分子名称: | MBP1, MITOTIC SPINDLE ASSEMBLY CHECKPOINT PROTEIN MAD2A | 著者 | Mapelli, M, Massimiliano, L, Santaguida, S, Musacchio, A. | 登録日 | 2007-07-13 | 公開日 | 2007-11-27 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | The MAD2 Conformational Dimer: Structure and Implications for the Spindle Assembly Checkpoint Cell(Cambridge,Mass.), 131, 2007
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1BPO
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![BU of 1bpo by Molmil](/molmil-images/mine/1bpo) | CLATHRIN HEAVY-CHAIN TERMINAL DOMAIN AND LINKER | 分子名称: | PROTEIN (CLATHRIN) | 著者 | Harr, E.T, Musacchio, A, Harrison, S.C, Kirchhausen, T. | 登録日 | 1998-08-11 | 公開日 | 1998-12-16 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Atomic structure of clathrin: a beta propeller terminal domain joins an alpha zigzag linker. Cell(Cambridge,Mass.), 95, 1998
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8ARF
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![BU of 8arf by Molmil](/molmil-images/mine/8arf) | |
1E7O
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![BU of 1e7o by Molmil](/molmil-images/mine/1e7o) | A-SPECTRIN SH3 DOMAIN A11V, V23L, M25V, V44I, V58L MUTATIONS | 分子名称: | GLYCEROL, SPECTRIN ALPHA CHAIN | 著者 | Vega, M.C, Serrano, L. | 登録日 | 2000-08-31 | 公開日 | 2003-05-21 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (3.2 Å) | 主引用文献 | A Thermodynamic and Kinetic Analysis of the Folding Pathway of an SH3 Domain Entropically Stabilised by a Redesigned Hydrophobic Core J.Mol.Biol., 328, 2003
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3O0G
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![BU of 3o0g by Molmil](/molmil-images/mine/3o0g) | Crystal Structure of Cdk5:p25 in complex with an ATP analogue | 分子名称: | Cell division protein kinase 5, Cyclin-dependent kinase 5 activator 1, {4-amino-2-[(4-chlorophenyl)amino]-1,3-thiazol-5-yl}(3-nitrophenyl)methanone | 著者 | Mapelli, M. | 登録日 | 2010-07-19 | 公開日 | 2011-01-26 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Defining Cdk5 ligand chemical space with small molecule inhibitors of Tau phosphorylation Chem.Biol., 12, 2005
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1AWO
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![BU of 1awo by Molmil](/molmil-images/mine/1awo) | |
5LSI
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![BU of 5lsi by Molmil](/molmil-images/mine/5lsi) | CRYSTAL STRUCTURE OF THE KINETOCHORE MIS12 COMPLEX HEAD2 SUBDOMAIN CONTAINING DSN1 AND NSL1 FRAGMENTS | 分子名称: | Kinetochore-associated protein DSN1 homolog, Kinetochore-associated protein NSL1 homolog, SULFATE ION | 著者 | Vetter, I.R, Petrovic, A, Keller, J, Liu, Y. | 登録日 | 2016-09-02 | 公開日 | 2016-11-16 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (2.002 Å) | 主引用文献 | Structure of the MIS12 Complex and Molecular Basis of Its Interaction with CENP-C at Human Kinetochores. Cell, 167, 2016
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5LSK
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![BU of 5lsk by Molmil](/molmil-images/mine/5lsk) | CRYSTAL STRUCTURE OF THE HUMAN KINETOCHORE MIS12-CENP-C COMPLEX | 分子名称: | Centromere protein C, Kinetochore-associated protein DSN1 homolog, Kinetochore-associated protein NSL1 homolog, ... | 著者 | Vetter, I.R, Petrovic, A, Keller, J, Liu, Y. | 登録日 | 2016-09-02 | 公開日 | 2016-11-16 | 最終更新日 | 2017-10-11 | 実験手法 | X-RAY DIFFRACTION (3.502 Å) | 主引用文献 | Structure of the MIS12 Complex and Molecular Basis of Its Interaction with CENP-C at Human Kinetochores. Cell, 167, 2016
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5LSJ
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![BU of 5lsj by Molmil](/molmil-images/mine/5lsj) | CRYSTAL STRUCTURE OF THE HUMAN KINETOCHORE MIS12-CENP-C delta-HEAD2 COMPLEX | 分子名称: | Centromere protein C, Kinetochore-associated protein DSN1 homolog, Kinetochore-associated protein NSL1 homolog, ... | 著者 | Vetter, I.R, Petrovic, A, Keller, J, Liu, Y. | 登録日 | 2016-09-02 | 公開日 | 2016-11-16 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (3.25 Å) | 主引用文献 | Structure of the MIS12 Complex and Molecular Basis of Its Interaction with CENP-C at Human Kinetochores. Cell, 167, 2016
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7QOO
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![BU of 7qoo by Molmil](/molmil-images/mine/7qoo) | Structure of the human inner kinetochore CCAN complex | 分子名称: | Centromere protein C, Centromere protein H, Centromere protein I, ... | 著者 | Vetter, I.R, Pesenti, M, Raisch, T. | 登録日 | 2021-12-24 | 公開日 | 2022-06-08 | 最終更新日 | 2024-07-17 | 実験手法 | ELECTRON MICROSCOPY (4.6 Å) | 主引用文献 | Structure of the human inner kinetochore CCAN complex and its significance for human centromere organization. Mol.Cell, 82, 2022
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4AF3
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![BU of 4af3 by Molmil](/molmil-images/mine/4af3) | Human Aurora B Kinase in complex with INCENP and VX-680 | 分子名称: | AURORA KINASE B, CYCLOPROPANECARBOXYLIC ACID {4-[4-(4-METHYL-PIPERAZIN-1-YL)-6-(5-METHYL-2H-PYRAZOL-3-YLAMINO)-PYRIMIDIN-2-YLSULFANYL]-PHENYL}-AMIDE, INNER CENTROMERE PROTEIN | 著者 | Elkins, J.M, Vollmar, M, Wang, J, Picaud, S, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Knapp, S. | 登録日 | 2012-01-16 | 公開日 | 2012-04-11 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.75 Å) | 主引用文献 | Crystal Structure of Human Aurora B in Complex with Incenp and Vx-680. J.Med.Chem., 55, 2012
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1CYW
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![BU of 1cyw by Molmil](/molmil-images/mine/1cyw) | QUINOL OXIDASE (PERIPLASMIC FRAGMENT OF SUBUNIT II) (CYOA) | 分子名称: | CYOA | 著者 | Wilmanns, M, Lappalainen, P, Kelly, M, Sauer-Eriksson, E, Saraste, M. | 登録日 | 1995-08-22 | 公開日 | 1996-03-08 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Crystal structure of the membrane-exposed domain from a respiratory quinol oxidase complex with an engineered dinuclear copper center. Proc.Natl.Acad.Sci.USA, 92, 1995
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