7QBE
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![BU of 7qbe by Molmil](/molmil-images/mine/7qbe) | TC:CD320 in complex with nanobody TC-Nb11 | 分子名称: | Anti-transcobalamin-2 nanobody TC-Nb11, CALCIUM ION, CD320 antigen, ... | 著者 | Bloch, J.S, Locher, K.P. | 登録日 | 2021-11-19 | 公開日 | 2022-03-16 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Generation of nanobodies targeting the human, transcobalamin-mediated vitamin B 12 uptake route. Faseb J., 36, 2022
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5M3B
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![BU of 5m3b by Molmil](/molmil-images/mine/5m3b) | Structure of cobinamide-bound BtuF mutant W66L, the periplasmic vitamin B12 binding protein in E.coli | 分子名称: | COB(II)INAMIDE, CYANIDE ION, GLYCEROL, ... | 著者 | Mireku, S.A, Ruetz, M, Zhou, T, Korkhov, V.M, Kraeutler, B, Locher, K.P. | 登録日 | 2016-10-14 | 公開日 | 2017-03-01 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Conformational Change of a Tryptophan Residue in BtuF Facilitates Binding and Transport of Cobinamide by the Vitamin B12 Transporter BtuCD-F. Sci Rep, 7, 2017
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5M34
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![BU of 5m34 by Molmil](/molmil-images/mine/5m34) | Structure of cobinamide-bound BtuF mutant W66Y, the periplasmic vitamin B12 binding protein in E.coli | 分子名称: | COB(II)INAMIDE, CYANIDE ION, GLYCEROL, ... | 著者 | Mireku, S.A, Ruetz, M, Zhou, T, Korkhov, V.M, Kraeutler, B, Locher, K.P. | 登録日 | 2016-10-14 | 公開日 | 2017-03-01 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Conformational Change of a Tryptophan Residue in BtuF Facilitates Binding and Transport of Cobinamide by the Vitamin B12 Transporter BtuCD-F. Sci Rep, 7, 2017
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5M29
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![BU of 5m29 by Molmil](/molmil-images/mine/5m29) | Structure of cobinamide-bound BtuF, the periplasmic vitamin B12 binding protein in E.coli | 分子名称: | COB(II)INAMIDE, CYANIDE ION, GLYCEROL, ... | 著者 | Mireku, S.A, Ruetz, M, Zhou, T, Korkhov, V.M, Kraeutler, B, Locher, K.P. | 登録日 | 2016-10-12 | 公開日 | 2017-02-08 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Conformational Change of a Tryptophan Residue in BtuF Facilitates Binding and Transport of Cobinamide by the Vitamin B12 Transporter BtuCD-F. Sci Rep, 7, 2017
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5M2Q
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![BU of 5m2q by Molmil](/molmil-images/mine/5m2q) | Structure of cobinamide-bound BtuF mutant W66F, the periplasmic vitamin B12 binding protein in E.coli | 分子名称: | COB(II)INAMIDE, CYANIDE ION, GLYCEROL, ... | 著者 | Mireku, S.A, Ruetz, M, Zhou, T, Korkhov, V.M, Kraeutler, B, Locher, K.P. | 登録日 | 2016-10-13 | 公開日 | 2017-03-01 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Conformational Change of a Tryptophan Residue in BtuF Facilitates Binding and Transport of Cobinamide by the Vitamin B12 Transporter BtuCD-F. Sci Rep, 7, 2017
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2ONJ
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2ONK
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![BU of 2onk by Molmil](/molmil-images/mine/2onk) | ABC transporter ModBC in complex with its binding protein ModA | 分子名称: | MAGNESIUM ION, Molybdate/tungstate ABC transporter, ATP-binding protein, ... | 著者 | Hollenstein, K, Frei, D.C, Locher, K.P. | 登録日 | 2007-01-24 | 公開日 | 2007-03-06 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Structure of an ABC transporter in complex with its binding protein. Nature, 446, 2007
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8P8J
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![BU of 8p8j by Molmil](/molmil-images/mine/8p8j) | Structure of 5D3-Fab and nanobody(Nb96)-bound ABCG2 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 5D3(Fab) heavy chain variable domain, 5D3(Fab) light chain variable domain, ... | 著者 | Irobalieva, R.N, Manolaridis, I, Jackson, S.M, Ni, D, Pardon, E, Stahlberg, H, Steyaert, J, Locher, K.P. | 登録日 | 2023-06-01 | 公開日 | 2023-08-30 | 最終更新日 | 2023-09-13 | 実験手法 | ELECTRON MICROSCOPY (3.49 Å) | 主引用文献 | Structural Basis of the Allosteric Inhibition of Human ABCG2 by Nanobodies. J.Mol.Biol., 435, 2023
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8P7W
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![BU of 8p7w by Molmil](/molmil-images/mine/8p7w) | Structure of 5D3-Fab and nanobody(Nb8)-bound ABCG2 | 分子名称: | 5D3(Fab) heavy chain variable domain, 5D3(Fab) light chain variable domain, ATP-binding cassette sub-family G member 2, ... | 著者 | Irobalieva, R.N, Manolaridis, I, Jackson, S.M, Ni, D, Pardon, E, Stahlberg, H, Steyaert, J, Locher, K.P. | 登録日 | 2023-05-31 | 公開日 | 2023-08-30 | 最終更新日 | 2023-09-13 | 実験手法 | ELECTRON MICROSCOPY (3.04 Å) | 主引用文献 | Structural Basis of the Allosteric Inhibition of Human ABCG2 by Nanobodies. J.Mol.Biol., 435, 2023
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8P8A
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![BU of 8p8a by Molmil](/molmil-images/mine/8p8a) | Structure of 5D3-Fab and nanobody(Nb17)-bound ABCG2 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 5D3(Fab) heavy chain variable domain, 5D3(Fab) light chain variable domain, ... | 著者 | Irobalieva, R.N, Manolaridis, I, Jackson, S.M, Ni, D, Pardon, E, Stahlberg, H, Steyaert, J, Locher, K.P. | 登録日 | 2023-05-31 | 公開日 | 2023-08-30 | 最終更新日 | 2023-09-13 | 実験手法 | ELECTRON MICROSCOPY (3.2 Å) | 主引用文献 | Structural Basis of the Allosteric Inhibition of Human ABCG2 by Nanobodies. J.Mol.Biol., 435, 2023
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8PG0
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![BU of 8pg0 by Molmil](/molmil-images/mine/8pg0) | Human OATP1B3 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, BICARBONATE ION, CHOLESTEROL, ... | 著者 | Ciuta, A.-D, Nosol, K, Kowal, J, Mukherjee, S, Ramirez, A.S, Stieger, B, Kossiakoff, A.A, Locher, K.P. | 登録日 | 2023-06-17 | 公開日 | 2023-09-27 | 実験手法 | ELECTRON MICROSCOPY (2.97 Å) | 主引用文献 | Structure of human drug transporters OATP1B1 and OATP1B3. Nat Commun, 14, 2023
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8PHW
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![BU of 8phw by Molmil](/molmil-images/mine/8phw) | Human OATP1B1 | 分子名称: | CHOLESTEROL HEMISUCCINATE, Fab18 (heavy chain, variable region), ... | 著者 | Ciuta, A.-D, Nosol, K, Kowal, J, Mukherjee, S, Ramirez, A.S, Stieger, B, Kossiakoff, A.A, Locher, K.P. | 登録日 | 2023-06-20 | 公開日 | 2023-09-27 | 最終更新日 | 2024-03-20 | 実験手法 | ELECTRON MICROSCOPY (3.6 Å) | 主引用文献 | Structure of human drug transporters OATP1B1 and OATP1B3. Nat Commun, 14, 2023
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8PMJ
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![BU of 8pmj by Molmil](/molmil-images/mine/8pmj) | Vanadate-trapped BSEP in nanodiscs | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, ADENOSINE-5'-TRIPHOSPHATE, Bile salt export pump, ... | 著者 | Liu, H, Irobalieva, R.N, Kowal, J, Ni, D, Nosol, K, Bang-Sorensen, R, Lancien, L, Stahlberg, H, Stieger, B, Locher, K.P. | 登録日 | 2023-06-28 | 公開日 | 2023-11-29 | 実験手法 | ELECTRON MICROSCOPY (2.81 Å) | 主引用文献 | Structural basis of bile salt extrusion and small-molecule inhibition in human BSEP. Nat Commun, 14, 2023
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8PMD
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![BU of 8pmd by Molmil](/molmil-images/mine/8pmd) | Nucleotide-bound BSEP in nanodiscs | 分子名称: | ADENOSINE-5'-TRIPHOSPHATE, Bile salt export pump, MAGNESIUM ION | 著者 | Liu, H, Irobalieva, R.N, Kowal, J, Ni, D, Nosol, K, Bang-Sorensen, R, Lancien, L, Stahlberg, H, Stieger, B, Locher, K.P. | 登録日 | 2023-06-28 | 公開日 | 2023-11-22 | 実験手法 | ELECTRON MICROSCOPY (2.95 Å) | 主引用文献 | Structural basis of bile salt extrusion and small-molecule inhibition in human BSEP. Nat Commun, 14, 2023
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8PM6
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![BU of 8pm6 by Molmil](/molmil-images/mine/8pm6) | Human bile salt export pump (BSEP) in complex with inhibitor GBM in nanodiscs | 分子名称: | 5-chloro-N-(2-{4-[(cyclohexylcarbamoyl)sulfamoyl]phenyl}ethyl)-2-methoxybenzamide, Bile salt export pump, CHOLESTEROL | 著者 | Liu, H, Irobalieva, R.N, Kowal, J, Ni, D, Nosol, K, Bang-Sorensen, R, Lancien, L, Stahlberg, H, Stieger, B, Locher, K.P. | 登録日 | 2023-06-28 | 公開日 | 2023-11-22 | 実験手法 | ELECTRON MICROSCOPY (3.22 Å) | 主引用文献 | Structural basis of bile salt extrusion and small-molecule inhibition in human BSEP. Nat Commun, 14, 2023
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8PN9
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![BU of 8pn9 by Molmil](/molmil-images/mine/8pn9) | Structure of human oligosaccharyltransferase OST-A complex bound to NGI-1 | 分子名称: | (2E,6E,10E,14E,18E,22E,26E)-3,7,11,15,19,23,27,31-OCTAMETHYLDOTRIACONTA-2,6,10,14,18,22,26,30-OCTAENYL TRIHYDROGEN DIPHOSPHATE, (2~{S},3~{R},4~{R},5~{S},6~{S})-2-(hydroxymethyl)-6-[(1~{S},2~{R},3~{R},4~{R},5'~{S},6~{S},7~{R},8~{S},9~{R},12~{R},13~{R},15~{S},16~{S},18~{R})-5',7,9,13-tetramethyl-3,15-bis(oxidanyl)spiro[5-oxapentacyclo[10.8.0.0^{2,9}.0^{4,8}.0^{13,18}]icosane-6,2'-oxane]-16-yl]oxy-oxane-3,4,5-triol, (4R,7R)-4-hydroxy-N,N,N-trimethyl-4,9-dioxo-7-[(undecanoyloxy)methyl]-3,5,8-trioxa-4lambda~5~-phosphadocosan-1-aminium, ... | 著者 | Ramirez, A.S, Kowal, J, Locher, K.P. | 登録日 | 2023-06-30 | 公開日 | 2024-05-08 | 実験手法 | ELECTRON MICROSCOPY (3.61 Å) | 主引用文献 | Positive selection CRISPR screens reveal a druggable pocket in an oligosaccharyltransferase required for inflammatory signaling to NF-kappa B. Cell, 187, 2024
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2QI9
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![BU of 2qi9 by Molmil](/molmil-images/mine/2qi9) | ABC-transporter BtuCD in complex with its periplasmic binding protein BtuF | 分子名称: | DI(HYDROXYETHYL)ETHER, PENTAETHYLENE GLYCOL, PHOSPHATE ION, ... | 著者 | Hvorup, R.N, Goetz, B.A, Niederer, M, Hollenstein, K, Perozo, E, Locher, K.P. | 登録日 | 2007-07-03 | 公開日 | 2007-08-14 | 最終更新日 | 2021-10-20 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Asymmetry in the structure of the ABC transporter-binding protein complex BtuCD-BtuF. Science, 317, 2007
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2ONR
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![BU of 2onr by Molmil](/molmil-images/mine/2onr) | Crystal structure of A. fulgidus periplasmic binding protein ModA with bound molybdate | 分子名称: | MAGNESIUM ION, MOLYBDATE ION, NITRATE ION, ... | 著者 | Hollenstein, K, Frei, D.C, Locher, K.P. | 登録日 | 2007-01-24 | 公開日 | 2007-03-06 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Structure of an ABC transporter in complex with its binding protein. Nature, 446, 2007
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2ONS
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![BU of 2ons by Molmil](/molmil-images/mine/2ons) | Crystal structure of A. fulgidus periplasmic binding protein ModA with bound tungstate | 分子名称: | MAGNESIUM ION, NITRATE ION, TUNGSTATE(VI)ION, ... | 著者 | Hollenstein, K, Frei, D.C, Locher, K.P. | 登録日 | 2007-01-24 | 公開日 | 2007-03-06 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Structure of an ABC transporter in complex with its binding protein. Nature, 446, 2007
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3NU1
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![BU of 3nu1 by Molmil](/molmil-images/mine/3nu1) | Structure of holo form of a periplasmic heme binding protein | 分子名称: | Hemin-binding periplasmic protein, PROTOPORPHYRIN IX CONTAINING FE | 著者 | Mattle, D, Goetz, B.A, Woo, J.S, Locher, K.P. | 登録日 | 2010-07-06 | 公開日 | 2010-10-13 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Two stacked heme molecules in the binding pocket of the periplasmic heme-binding protein HmuT from Yersinia pestis. J.Mol.Biol., 404, 2010
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3RCE
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![BU of 3rce by Molmil](/molmil-images/mine/3rce) | Bacterial oligosaccharyltransferase PglB | 分子名称: | MAGNESIUM ION, Oligosaccharide transferase to N-glycosylate proteins, Substrate Mimic Peptide | 著者 | Lizak, C, Gerber, S, Numao, S, Aebi, M, Locher, K.P. | 登録日 | 2011-03-31 | 公開日 | 2011-06-15 | 最終更新日 | 2017-11-08 | 実験手法 | X-RAY DIFFRACTION (3.4 Å) | 主引用文献 | X-ray structure of a bacterial oligosaccharyltransferase. Nature, 474, 2011
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7A65
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7A6E
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![BU of 7a6e by Molmil](/molmil-images/mine/7a6e) | |
7A6C
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![BU of 7a6c by Molmil](/molmil-images/mine/7a6c) | |
7A69
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![BU of 7a69 by Molmil](/molmil-images/mine/7a69) | |