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6ULA
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BU of 6ula by Molmil
Crystal structure of human GAC in complex with inhibitor UPGL00012
分子名称: 2-cyclopropyl-N-{5-[4-({5-[(cyclopropylacetyl)amino]-1,3,4-thiadiazol-2-yl}oxy)piperidin-1-yl]-1,3,4-thiadiazol-2-yl}acetamide, Glutaminase kidney isoform, mitochondrial
著者Huang, Q, Cerione, R.A.
登録日2019-10-07
公開日2020-10-14
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.95 Å)
主引用文献Crystal structure of human GAC in complex with inhibitor UPGL00030
To Be Published
6UJM
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BU of 6ujm by Molmil
Crystal structure of human GAC in complex with inhibitor UPGL00013
分子名称: Glutaminase kidney isoform, mitochondrial, N-{5-[(3R)-3-{[5-(acetylamino)-1,3,4-thiadiazol-2-yl]amino}pyrrolidin-1-yl]-1,3,4-thiadiazol-2-yl}acetamide
著者Huang, Q, Cerione, R.A.
登録日2019-10-03
公開日2020-10-07
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Crystal structure of human GAC in complex with inhibitor UPGL00013
To Be Published
1MRH
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BU of 1mrh by Molmil
STUDIES ON CRYSTAL STRUCTURES ACTIVE CENTER GEOMETRY AND DEPURINE MECHANISM OF TWO RIBOSOME-INACTIVATING PROTEINS
分子名称: (1S)-1-(7-amino-1H-pyrazolo[4,3-d]pyrimidin-3-yl)-1,4-anhydro-D-ribitol, ALPHA-MOMORCHARIN
著者Huang, Q, Liu, S, Tang, Y, Jin, S, Wang, Y.
登録日1994-07-01
公開日1995-02-07
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Studies on crystal structures, active-centre geometry and depurinating mechanism of two ribosome-inactivating proteins.
Biochem.J., 309, 1995
1MRK
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BU of 1mrk by Molmil
STUDIES ON CRYSTAL STRUCTURES ACTIVE CENTER GEOMETRY AND DEPURINE MECHANISM OF TWO RIBOSOME-INACTIVATING PROTEINS
分子名称: (1S)-1-(7-amino-1H-pyrazolo[4,3-d]pyrimidin-3-yl)-1,4-anhydro-D-ribitol, ALPHA-TRICHOSANTHIN
著者Huang, Q, Liu, S, Tang, Y, Jin, S, Wang, Y.
登録日1994-07-01
公開日1995-02-07
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Studies on crystal structures, active-centre geometry and depurinating mechanism of two ribosome-inactivating proteins.
Biochem.J., 309, 1995
1MRJ
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BU of 1mrj by Molmil
STUDIES ON CRYSTAL STRUCTURES ACTIVE CENTER GEOMETRY AND DEPURINE MECHANISM OF TWO RIBOSOME-INACTIVATING PROTEINS
分子名称: ADENOSINE, ALPHA-TRICHOSANTHIN
著者Huang, Q, Liu, S, Tang, Y, Jin, S, Wang, Y.
登録日1994-07-01
公開日1995-02-07
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Studies on crystal structures, active-centre geometry and depurinating mechanism of two ribosome-inactivating proteins.
Biochem.J., 309, 1995
1MRI
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BU of 1mri by Molmil
STUDIES ON CRYSTAL STRUCTURES ACTIVE CENTER GEOMETRY AND DEPURINE MECHANISM OF TWO RIBOSOME-INACTIVATING PROTEINS
分子名称: ALPHA-MOMORCHARIN
著者Huang, Q, Liu, S, Tang, Y, Jin, S, Wang, Y.
登録日1994-07-01
公開日1995-02-07
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Studies on crystal structures, active-centre geometry and depurinating mechanism of two ribosome-inactivating proteins.
Biochem.J., 309, 1995
1MRG
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BU of 1mrg by Molmil
STUDIES ON CRYSTAL STRUCTURES ACTIVE CENTER GEOMETRY AND DEPURINE MECHANISM OF TWO RIBOSOME-INACTIVATING PROTEINS
分子名称: ADENOSINE, ALPHA-MOMORCHARIN
著者Huang, Q, Liu, S, Tang, Y, Jin, S, Wang, Y.
登録日1994-07-01
公開日1995-02-07
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Studies on crystal structures, active-centre geometry and depurinating mechanism of two ribosome-inactivating proteins.
Biochem.J., 309, 1995
1K3K
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BU of 1k3k by Molmil
Solution Structure of a Bcl-2 Homolog from Kaposi's Sarcoma Virus
分子名称: functional anti-apoptotic factor vBCL-2 homolog
著者Huang, Q, Petros, A.M, Virgin, H.W, Fesik, S.W, Olejniczak, E.T.
登録日2001-10-03
公開日2002-04-10
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Solution structure of a Bcl-2 homolog from Kaposi sarcoma virus.
Proc.Natl.Acad.Sci.USA, 99, 2002
1MG6
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BU of 1mg6 by Molmil
The Crystal Structure of a K49 PLA2 from the Snake Venom of Agkistrodon acutus
分子名称: PHOSPHOLIPASE A2
著者Huang, Q, Teng, M, Niu, L.
登録日2002-08-14
公開日2002-09-04
最終更新日2018-04-04
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献The Crystal Structure of a K49 PLA2 from the Snake Venom of Agkistrodon acutus
TO BE PUBLISHED
1IAY
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BU of 1iay by Molmil
CRYSTAL STRUCTURE OF ACC SYNTHASE COMPLEXED WITH COFACTOR PLP AND INHIBITOR AVG
分子名称: 1-AMINOCYCLOPROPANE-1-CARBOXYLATE SYNTHASE 2, 2-AMINO-4-(2-AMINO-ETHOXY)-BUTYRIC ACID, PYRIDOXAL-5'-PHOSPHATE
著者Huai, Q, Xia, Y, Chen, Y, Callahan, B, Li, N, Ke, H.
登録日2001-03-24
公開日2001-04-04
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Crystal structures of 1-aminocyclopropane-1-carboxylate (ACC) synthase in complex with aminoethoxyvinylglycine and pyridoxal-5'-phosphate provide new insight into catalytic mechanisms
J.Biol.Chem., 276, 2001
1IAW
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BU of 1iaw by Molmil
CRYSTAL STRUCTURE OF NAEI COMPLEXED WITH 17MER DNA
分子名称: 5'-D(*TP*GP*CP*CP*AP*CP*GP*CP*CP*GP*GP*CP*GP*TP*GP*GP*C)-3', TYPE II RESTRICTION ENZYME NAEI
著者Huai, Q, Colandene, J.D, Topal, M.D, Ke, H.
登録日2001-03-23
公開日2001-08-03
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structure of NaeI-DNA complex reveals dual-mode DNA recognition and complete dimer rearrangement.
Nat.Struct.Biol., 8, 2001
1IAX
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BU of 1iax by Molmil
CRYSTAL STRUCTURE OF ACC SYNTHASE COMPLEXED WITH PLP
分子名称: 1-AMINOCYCLOPROPANE-1-CARBOXYLATE SYNTHASE 2, PYRIDOXAL-5'-PHOSPHATE, SULFATE ION
著者Huai, Q, Xia, Y, Chen, Y, Callahan, B, Li, N, Ke, H.
登録日2001-03-24
公開日2001-04-04
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Crystal structures of 1-aminocyclopropane-1-carboxylate (ACC) synthase in complex with aminoethoxyvinylglycine and pyridoxal-5'-phosphate provide new insight into catalytic mechanisms
J.Biol.Chem., 276, 2001
1M63
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BU of 1m63 by Molmil
Crystal structure of calcineurin-cyclophilin-cyclosporin shows common but distinct recognition of immunophilin-drug complexes
分子名称: CALCINEURIN B SUBUNIT ISOFORM 1, CALCIUM ION, CYCLOSPORIN A, ...
著者Huai, Q, Kim, H.-Y, Liu, Y, Zhao, Y, Mondragon, A, Liu, J.O, Ke, H.
登録日2002-07-12
公開日2002-09-25
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Crystal Structure of Calcineurin-Cyclophilin-Cyclosporin Shows Common But Distinct Recognition of Immunophilin-Drug Complexes
Proc.Natl.Acad.Sci.USA, 99, 2002
3CN8
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BU of 3cn8 by Molmil
Crystal structure of fms1 in complex with spermidine
分子名称: FLAVIN-ADENINE DINUCLEOTIDE, Polyamine oxidase FMS1, SPERMIDINE
著者Huang, Q, Hao, Q.
登録日2008-03-25
公開日2008-04-22
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Crystal structure of fms1 in complex with spermidine
TO BE PUBLISHED
3CNS
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BU of 3cns by Molmil
Crystal structure of fms1 in complex with S-Bz-MeSpermidine
分子名称: FLAVIN-ADENINE DINUCLEOTIDE, N-{(1S)-3-[(4-aminobutyl)amino]-1-methylpropyl}benzamide, fms1
著者Huang, Q, Hao, H.
登録日2008-03-26
公開日2008-04-22
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Crystal structure of fms1 in complex with S-Bz-MeSpermidine
TO BE PUBLISHED
1RKP
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BU of 1rkp by Molmil
Crystal structure of PDE5A1-IBMX
分子名称: 3-ISOBUTYL-1-METHYLXANTHINE, MAGNESIUM ION, ZINC ION, ...
著者Huai, Q, Liu, Y, Francis, S.H, Corbin, J.D, Ke, H.
登録日2003-11-22
公開日2004-03-30
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献Crystal structures of phosphodiesterases 4 and 5 in complex with inhibitor IBMX suggest a conformation determinant of inhibitor selectivity
J.Biol.Chem., 279, 2004
1SSK
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BU of 1ssk by Molmil
Structure of the N-terminal RNA-binding Domain of the SARS CoV Nucleocapsid Protein
分子名称: Nucleocapsid protein
著者Huang, Q, Yu, L, Petros, A.M, Gunasekera, A, Liu, Z, Xu, N, Hajduk, P, Mack, J, Fesik, S.W, Olejniczak, E.T.
登録日2004-03-24
公開日2004-06-08
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Structure of the N-Terminal RNA-Binding Domain of the SARS CoV Nucleocapsid Protein.
Biochemistry, 43, 2004
1Q59
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BU of 1q59 by Molmil
Solution Structure of the BHRF1 Protein From Epstein-Barr Virus, a Homolog of Human Bcl-2
分子名称: Early antigen protein R
著者Huang, Q, Petros, A.M, Virgin, H.W, Fesik, S.W, Olejniczak, E.T.
登録日2003-08-06
公開日2003-09-23
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Solution Structure of the BHRF1 Protein From Epstein-Barr Virus, a Homolog of Human Bcl-2
J.Mol.Biol., 332, 2003
5T8B
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BU of 5t8b by Molmil
Crystal structure of lpg1496 under 350 MPa
分子名称: lpg1496
著者Huang, Q, Szebenyi, D.
登録日2016-09-07
公開日2017-08-16
最終更新日2019-12-25
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Crystal structure of lpg1496 under 350 MPa
To Be Published
5T8C
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BU of 5t8c by Molmil
Crystal structure of lpg1496 under 300 MPa
分子名称: lpg1496
著者Huang, Q, Szebenyi, D.
登録日2016-09-07
公開日2017-08-16
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.481 Å)
主引用文献Crystal structure of lpg1496 under 300 MPa
To Be Published
1Q2U
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BU of 1q2u by Molmil
Crystal structure of DJ-1/RS and implication on familial Parkinson's disease
分子名称: RNA-binding protein regulatory subunit
著者Huai, Q, Sun, Y, Wang, H, Chin, L.S, Li, L, Robinson, H, Ke, H.
登録日2003-07-26
公開日2003-10-07
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Crystal structure of DJ-1/RS and implication on familial Parkinson's disease
Febs Lett., 549, 2003
1PTW
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BU of 1ptw by Molmil
The Crystal Structure of AMP-Bound PDE4 Suggests a Mechanism for Phosphodiesterase Catalysis
分子名称: ADENOSINE MONOPHOSPHATE, ZINC ION, cAMP-specific phosphodiesterase PDE4D2
著者Huai, Q, Colicelli, J, Ke, H.
登録日2003-06-23
公開日2003-11-11
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献The crystal structure of AMP-bound PDE4 suggests a mechanism for phosphodiesterase catalysis
Biochemistry, 42, 2003
3M7F
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BU of 3m7f by Molmil
Crystal structure of the Nedd4 C2/Grb10 SH2 complex
分子名称: E3 ubiquitin-protein ligase NEDD4, Growth factor receptor-bound protein 10
著者Huang, Q, Szebenyi, M.
登録日2010-03-16
公開日2010-10-27
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural Basis for the Interaction between the Growth Factor-binding Protein GRB10 and the E3 Ubiquitin Ligase NEDD4.
J.Biol.Chem., 285, 2010
1Q9M
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BU of 1q9m by Molmil
Three dimensional structures of PDE4D in complex with roliprams and implication on inhibitor selectivity
分子名称: ROLIPRAM, ZINC ION, cAMP-specific phosphodiesterase PDE4D2
著者Huai, Q, Wang, H, Sun, Y, Kim, H.Y, Liu, Y, Ke, H.
登録日2003-08-25
公開日2003-09-02
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Three dimensional structures of PDE4D in complex with roliprams and implication on inhibitor selectivity
Structure, 11, 2003
1OYN
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BU of 1oyn by Molmil
Crystal structure of PDE4D2 in complex with (R,S)-rolipram
分子名称: ROLIPRAM, ZINC ION, cAMP-specific phosphodiesterase PDE4D2
著者Huai, Q, Wang, H, Sun, Y, Kim, H.Y, Liu, Y, Ke, H.
登録日2003-04-05
公開日2003-07-15
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Three-dimensional structures of PDE4D in complex with roliprams and implication on inhibitor selectivity
Structure, 11, 2003

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