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1RKP

Crystal structure of PDE5A1-IBMX

Summary for 1RKP
Entry DOI10.2210/pdb1rkp/pdb
Related1RKO
DescriptorcGMP-specific 3',5'-cyclic phosphodiesterase, ZINC ION, MAGNESIUM ION, ... (5 entities in total)
Functional Keywordspde5a, viagra, ibmx, hydrolase
Biological sourceHomo sapiens (human)
Total number of polymer chains1
Total formula weight38100.49
Authors
Huai, Q.,Liu, Y.,Francis, S.H.,Corbin, J.D.,Ke, H. (deposition date: 2003-11-22, release date: 2004-03-30, Last modification date: 2024-02-14)
Primary citationHuai, Q.,Liu, Y.,Francis, S.H.,Corbin, J.D.,Ke, H.
Crystal structures of phosphodiesterases 4 and 5 in complex with inhibitor IBMX suggest a conformation determinant of inhibitor selectivity
J.Biol.Chem., 279:13095-13101, 2004
Cited by
PubMed: 14668322
DOI: 10.1074/jbc.M311556200
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.05 Å)
Structure validation

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