4JSQ
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![BU of 4jsq by Molmil](/molmil-images/mine/4jsq) | Yeast 20S proteasome in complex with the dimerized linear mimetic of TMC-95A - yCP:4e | 分子名称: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, Probable proteasome subunit alpha type-7, Proteasome subunit alpha type-1, ... | 著者 | Desvergne, A, Genin, E, Marechal, X, Gallastegui, N, Dufau, L, Richy, N, Groll, M, Vidal, J, Reboud-Ravaux, M. | 登録日 | 2013-03-22 | 公開日 | 2013-05-01 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Dimerized linear mimics of a natural cyclopeptide (TMC-95A) are potent noncovalent inhibitors of the eukaryotic 20S proteasome J.Med.Chem., 56, 2013
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4LQI
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![BU of 4lqi by Molmil](/molmil-images/mine/4lqi) | Yeast 20S Proteasome in complex with Vibralactone | 分子名称: | Proteasome subunit alpha type-1, Proteasome subunit alpha type-2, Proteasome subunit alpha type-3, ... | 著者 | List, A, Zeiler, E, Gallastegui, N, Rusch, M, Hedberg, C, Sieber, S.A, Groll, M. | 登録日 | 2013-07-18 | 公開日 | 2013-12-25 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Omuralide and Vibralactone: Differences in the Proteasome-beta-Lactone-gamma-Lactam Binding Scaffold Alter Target Preferences. Angew.Chem.Int.Ed.Engl., 53, 2014
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4JSU
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![BU of 4jsu by Molmil](/molmil-images/mine/4jsu) | Yeast 20S proteasome in complex with the dimerized linear mimetic of TMC-95A - yCP:3a | 分子名称: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, Probable proteasome subunit alpha type-7, Proteasome subunit alpha type-1, ... | 著者 | Desvergne, A, Genin, E, Marechal, X, Gallastegui, N, Dufau, L, Richy, N, Groll, M, Vidal, J, Reboud-Ravaux, M. | 登録日 | 2013-03-22 | 公開日 | 2013-05-01 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Dimerized linear mimics of a natural cyclopeptide (TMC-95A) are potent noncovalent inhibitors of the eukaryotic 20S proteasome J.Med.Chem., 56, 2013
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4JVW
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![BU of 4jvw by Molmil](/molmil-images/mine/4jvw) | IgM C4-domain from mouse | 分子名称: | Ig mu chain C region secreted form | 著者 | Mueller, R, Graewert, A.M, Kern, T, Madl, T, Peschek, J, Sattler, M, Groll, M, Buchner, J. | 登録日 | 2013-03-26 | 公開日 | 2013-06-12 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | High-resolution structures of the IgM Fc domains reveal principles of its hexamer formation. Proc.Natl.Acad.Sci.USA, 110, 2013
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4YDZ
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![BU of 4ydz by Molmil](/molmil-images/mine/4ydz) | Stress-induced protein 1 from Caenorhabditis elegans | 分子名称: | Stress-induced protein 1 | 著者 | Fleckenstein, T, Kastenmueller, A, Stein, M.L, Peters, C, Daake, M, Krause, M, Weinfurtner, D, Haslbeck, M, Weinkauf, S, Groll, M, Buchner, J. | 登録日 | 2015-02-23 | 公開日 | 2015-06-10 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (3.6 Å) | 主引用文献 | The Chaperone Activity of the Developmental Small Heat Shock Protein Sip1 Is Regulated by pH-Dependent Conformational Changes. Mol.Cell, 58, 2015
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8A7L
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![BU of 8a7l by Molmil](/molmil-images/mine/8a7l) | PcIDS1 in complex with Mg2+, GPP, and ZOL | 分子名称: | GERANYL DIPHOSPHATE, GLYCEROL, Isoprenyl diphosphate synthase, ... | 著者 | Ecker, F, Boland, W, Groll, M. | 登録日 | 2022-06-21 | 公開日 | 2023-05-31 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Metal-dependent enzyme symmetry guides the biosynthetic flux of terpene precursors. Nat.Chem., 15, 2023
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8A7C
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![BU of 8a7c by Molmil](/molmil-images/mine/8a7c) | PcIDS1 in complex with Mg2+, IPP, and ZOL | 分子名称: | 3-METHYLBUT-3-ENYL TRIHYDROGEN DIPHOSPHATE, GLYCEROL, Isoprenyl diphosphate synthase, ... | 著者 | Ecker, F, Boland, W, Groll, M. | 登録日 | 2022-06-20 | 公開日 | 2023-05-31 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.2 Å) | 主引用文献 | Metal-dependent enzyme symmetry guides the biosynthetic flux of terpene precursors. Nat.Chem., 15, 2023
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8A7K
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![BU of 8a7k by Molmil](/molmil-images/mine/8a7k) | PcIDS1 in complex with Mg2+/Mn2+, IPP, and ZOL | 分子名称: | 3-METHYLBUT-3-ENYL TRIHYDROGEN DIPHOSPHATE, GLYCEROL, Isoprenyl diphosphate synthase, ... | 著者 | Ecker, F, Boland, W, Groll, M. | 登録日 | 2022-06-21 | 公開日 | 2023-05-31 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.3 Å) | 主引用文献 | Metal-dependent enzyme symmetry guides the biosynthetic flux of terpene precursors. Nat.Chem., 15, 2023
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8A7U
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![BU of 8a7u by Molmil](/molmil-images/mine/8a7u) | PcIDS1_F315D in complex with Mg2+ and GPP | 分子名称: | GERANYL DIPHOSPHATE, GLYCEROL, Isoprenyl diphosphate synthase, ... | 著者 | Ecker, F, Boland, F, Groll, M. | 登録日 | 2022-06-21 | 公開日 | 2023-05-31 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Metal-dependent enzyme symmetry guides the biosynthetic flux of terpene precursors. Nat.Chem., 15, 2023
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8A7R
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![BU of 8a7r by Molmil](/molmil-images/mine/8a7r) | PcIDS1_I420A in complex with Mg2+ and GPP | 分子名称: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, GERANYL DIPHOSPHATE, GLYCEROL, ... | 著者 | Ecker, F, Boland, W, Groll, M. | 登録日 | 2022-06-21 | 公開日 | 2023-05-31 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Metal-dependent enzyme symmetry guides the biosynthetic flux of terpene precursors. Nat.Chem., 15, 2023
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8A7A
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![BU of 8a7a by Molmil](/molmil-images/mine/8a7a) | PcIDS1 in complex with Mg2+ and 3-Br-GPP | 分子名称: | Isoprenyl diphosphate synthase, MAGNESIUM ION, [(2Z)-3-bromanyl-7-methyl-octa-2,6-dienyl] phosphono hydrogen phosphate | 著者 | Ecker, F, Boland, W, Groll, M. | 登録日 | 2022-06-20 | 公開日 | 2023-05-31 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Metal-dependent enzyme symmetry guides the biosynthetic flux of terpene precursors. Nat.Chem., 15, 2023
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8A78
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![BU of 8a78 by Molmil](/molmil-images/mine/8a78) | PcIDS1_F315A in complex with Mg2+/Mn2+ and GPP | 分子名称: | GERANYL DIPHOSPHATE, GLYCEROL, Isoprenyl diphosphate synthase, ... | 著者 | Ecker, F, Boland, W, Groll, M. | 登録日 | 2022-06-20 | 公開日 | 2023-05-31 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Metal-dependent enzyme symmetry guides the biosynthetic flux of terpene precursors. Nat.Chem., 15, 2023
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8A7B
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![BU of 8a7b by Molmil](/molmil-images/mine/8a7b) | PcIDS1_D319N in complex with Mg2+ and 3-Br-GPP | 分子名称: | CARBONATE ION, GLYCEROL, Isoprenyl diphosphate synthase, ... | 著者 | Ecker, F, Boland, W, Groll, M. | 登録日 | 2022-06-20 | 公開日 | 2023-05-31 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.65 Å) | 主引用文献 | Metal-dependent enzyme symmetry guides the biosynthetic flux of terpene precursors. Nat.Chem., 15, 2023
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8A7J
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![BU of 8a7j by Molmil](/molmil-images/mine/8a7j) | PcIDS1 in complex with Mn2+, IPP, and ZOL | 分子名称: | 3-METHYLBUT-3-ENYL TRIHYDROGEN DIPHOSPHATE, GLYCEROL, Isoprenyl diphosphate synthase, ... | 著者 | Ecker, F, Boland, W, Groll, M. | 登録日 | 2022-06-21 | 公開日 | 2023-05-31 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.2 Å) | 主引用文献 | Metal-dependent enzyme symmetry guides the biosynthetic flux of terpene precursors. Nat.Chem., 15, 2023
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8ANP
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![BU of 8anp by Molmil](/molmil-images/mine/8anp) | Legionella effector Lem3 mutant D190A in complex with Mg2+ | 分子名称: | MAGNESIUM ION, Phosphocholine hydrolase Lem3, SULFATE ION, ... | 著者 | Kaspers, M.S, Pogenberg, V, Ernst, S, Ecker, F, Pett, C, Ochtrop, P, Hedberg, C, Groll, M, Itzen, A. | 登録日 | 2022-08-05 | 公開日 | 2023-04-12 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Dephosphocholination by Legionella effector Lem3 functions through remodelling of the switch II region of Rab1b. Nat Commun, 14, 2023
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4YE0
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![BU of 4ye0 by Molmil](/molmil-images/mine/4ye0) | Stress-induced protein 1 truncation mutant (43 - 140) from Caenorhabditis elegans | 分子名称: | SULFATE ION, Stress-induced protein 1 | 著者 | Fleckenstein, T, Kastenmueller, A, Stein, M.L, Peters, C, Daake, M, Krause, M, Weinfurtner, D, Haslbeck, M, Weinkauf, S, Groll, M, Buchner, J. | 登録日 | 2015-02-23 | 公開日 | 2015-06-10 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | The Chaperone Activity of the Developmental Small Heat Shock Protein Sip1 Is Regulated by pH-Dependent Conformational Changes. Mol.Cell, 58, 2015
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5EGP
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![BU of 5egp by Molmil](/molmil-images/mine/5egp) | Crystal structure of the S-methyltransferase TmtA | 分子名称: | ACETATE ION, S-ADENOSYL-L-HOMOCYSTEINE, SULFATE ION, ... | 著者 | Duell, E.R, Glaser, M, Antes, I, Groll, M, Huber, E.M. | 登録日 | 2015-10-27 | 公開日 | 2016-02-03 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Sequential Inactivation of Gliotoxin by the S-Methyltransferase TmtA. Acs Chem.Biol., 11, 2016
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5CZ6
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![BU of 5cz6 by Molmil](/molmil-images/mine/5cz6) | Yeast 20S proteasome beta5-T1A mutant in complex with Syringolin A, propeptide expressed in trans | 分子名称: | (2S)-2-[[(2S)-1-[[(5S,8S,9E)-2,7-dioxo-5-propan-2-yl-1,6-diazacyclododeca-3,9-dien-8-yl]amino]-3-methyl-1-oxo-butan-2-yl]carbamoylamino]-3-methyl-butanoic acid, CHLORIDE ION, MAGNESIUM ION, ... | 著者 | Huber, E.M, Groll, M. | 登録日 | 2015-07-31 | 公開日 | 2016-03-23 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | A unified mechanism for proteolysis and autocatalytic activation in the 20S proteasome. Nat Commun, 7, 2016
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5D0T
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![BU of 5d0t by Molmil](/molmil-images/mine/5d0t) | |
5CZ8
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![BU of 5cz8 by Molmil](/molmil-images/mine/5cz8) | |
5D0Z
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![BU of 5d0z by Molmil](/molmil-images/mine/5d0z) | |
6SKU
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![BU of 6sku by Molmil](/molmil-images/mine/6sku) | Legionella effector AnkX in complex with human Rab1b | 分子名称: | GUANOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, Phosphocholine transferase AnkX, ... | 著者 | Ernst, S, Ecker, F, Kaspers, M, Ochtrop, P, Hedberg, C, Groll, M, Itzen, A. | 登録日 | 2019-08-16 | 公開日 | 2020-06-10 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (3.2 Å) | 主引用文献 | Legionellaeffector AnkX displaces the switch II region for Rab1b phosphocholination. Sci Adv, 6, 2020
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5CZ7
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![BU of 5cz7 by Molmil](/molmil-images/mine/5cz7) | |
5D0X
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![BU of 5d0x by Molmil](/molmil-images/mine/5d0x) | |
5D0S
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![BU of 5d0s by Molmil](/molmil-images/mine/5d0s) | |