6CCY
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![BU of 6ccy by Molmil](/molmil-images/mine/6ccy) | Crystal structure of Akt1 in complex with a selective inhibitor | 分子名称: | (5R)-4-(4-{4-[4-fluoro-3-(trifluoromethyl)phenyl]-1-[2-(pyrrolidin-1-yl)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-5-methyl-5,8-dihydropyrido[2,3-d]pyrimidin-7(6H)-one, RAC-alpha serine/threonine-protein kinase,PIFtide | 著者 | Wang, Y, Stout, S. | 登録日 | 2018-02-07 | 公開日 | 2018-05-02 | 最終更新日 | 2018-05-16 | 実験手法 | X-RAY DIFFRACTION (2.18 Å) | 主引用文献 | Discovery of chiral dihydropyridopyrimidinones as potent, selective and orally bioavailable inhibitors of AKT. Bioorg. Med. Chem. Lett., 28, 2018
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2I0J
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![BU of 2i0j by Molmil](/molmil-images/mine/2i0j) | Benzopyrans are Selective Estrogen Receptor beta Agonists (SERBAs) with Novel Activity in Models of Benign Prostatic Hyperplasia | 分子名称: | (3AS,4R,9BR)-4-(4-HYDROXYPHENYL)-1,2,3,3A,4,9B-HEXAHYDROCYCLOPENTA[C]CHROMEN-8-OL, Estrogen receptor alpha | 著者 | Wang, Y. | 登録日 | 2006-08-10 | 公開日 | 2006-10-24 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Benzopyrans are selective estrogen receptor Beta agonists with novel activity in models of benign prostatic hyperplasia. J.Med.Chem., 49, 2006
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8HJ4
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![BU of 8hj4 by Molmil](/molmil-images/mine/8hj4) | |
6LYH
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![BU of 6lyh by Molmil](/molmil-images/mine/6lyh) | Crystal structure of tea N9-methyltransferase CkTcS in complex with SAH and 1,3,7-trimethyluric acid | 分子名称: | 1,3,7-trimethyl-9H-purine-2,6,8-trione, N-methyltransferase CkTcS, S-ADENOSYL-L-HOMOCYSTEINE | 著者 | Wang, Y, Zhang, Z.-M. | 登録日 | 2020-02-14 | 公開日 | 2020-03-04 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (3.15000319 Å) | 主引用文献 | Identification and characterization of N9-methyltransferase involved in converting caffeine into non-stimulatory theacrine in tea. Nat Commun, 11, 2020
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6LYI
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6NOD
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![BU of 6nod by Molmil](/molmil-images/mine/6nod) | Crystal structure of C. elegans PUF-8 in complex with RNA | 分子名称: | PUF (Pumilio/FBF) domain-containing, RNA (5'-R(P*UP*GP*UP*AP*UP*AP*UP*A)-3') | 著者 | Wang, Y, McCann, K.L, Qiu, C, Hall, T.M.T. | 登録日 | 2019-01-16 | 公開日 | 2019-01-30 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2.547 Å) | 主引用文献 | Engineering a conserved RNA regulatory protein repurposes its biological function in vivo . Elife, 8, 2019
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5XG8
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![BU of 5xg8 by Molmil](/molmil-images/mine/5xg8) | |
5Y03
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![BU of 5y03 by Molmil](/molmil-images/mine/5y03) | |
7CE2
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![BU of 7ce2 by Molmil](/molmil-images/mine/7ce2) | The Crystal structure of TeNT Hc complexed with neutralizing antibody | 分子名称: | Tetanus toxin, neutralizing antibody heavy chain, neutralizing antibody light chain | 著者 | Wang, X, Wang, Y, Wu, C, Yu, J, Liao, H. | 登録日 | 2020-06-21 | 公開日 | 2021-04-07 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.01 Å) | 主引用文献 | Structural basis of tetanus toxin neutralization by native human monoclonal antibodies. Cell Rep, 35, 2021
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6ISO
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![BU of 6iso by Molmil](/molmil-images/mine/6iso) | Human SIRT3 Recognizing H3K4cr | 分子名称: | (2E)-BUT-2-ENAL, ARG-THR-LYS-GLN-THR-ALA-ARG, GLYCEROL, ... | 著者 | Wang, Y, Hao, Q. | 登録日 | 2018-11-17 | 公開日 | 2019-01-23 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.95 Å) | 主引用文献 | Identification of 'erasers' for lysine crotonylated histone marks using a chemical proteomics approach. Elife, 3, 2014
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7X7E
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![BU of 7x7e by Molmil](/molmil-images/mine/7x7e) | SARS-CoV-2 RBD and Nb22 | 分子名称: | Nb22, Spike protein S1, TETRAETHYLENE GLYCOL | 著者 | Wang, Y, Ye, S. | 登録日 | 2022-03-09 | 公開日 | 2022-04-20 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.67 Å) | 主引用文献 | Short-Term Instantaneous Prophylaxis and Efficient Treatment Against SARS-CoV-2 in hACE2 Mice Conferred by an Intranasal Nanobody (Nb22). Front Immunol, 13, 2022
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7X7D
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![BU of 7x7d by Molmil](/molmil-images/mine/7x7d) | SARS-CoV-2 Delta RBD and Nb22 | 分子名称: | Nb22, Spike protein S1 | 著者 | Wang, Y, Ye, S. | 登録日 | 2022-03-09 | 公開日 | 2022-04-13 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.92 Å) | 主引用文献 | Short-Term Instantaneous Prophylaxis and Efficient Treatment Against SARS-CoV-2 in hACE2 Mice Conferred by an Intranasal Nanobody (Nb22). Front Immunol, 13, 2022
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6K1M
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![BU of 6k1m by Molmil](/molmil-images/mine/6k1m) | Engineered form of a putative cystathionine gamma-lyase | 分子名称: | Cystathionine gamma-lyase, PYRIDOXAL-5'-PHOSPHATE, PYRUVIC ACID | 著者 | Chen, S, Wang, Y. | 登録日 | 2019-05-10 | 公開日 | 2020-05-13 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.32 Å) | 主引用文献 | Structural characterization of cystathionine gamma-lyase smCSE enables aqueous metal quantum dot biosynthesis. Int.J.Biol.Macromol., 174, 2021
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6K1O
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![BU of 6k1o by Molmil](/molmil-images/mine/6k1o) | Apo form of a putative cystathionine gamma-lyase | 分子名称: | Cystathionine gamma-lyase | 著者 | Chen, S, Wang, Y. | 登録日 | 2019-05-10 | 公開日 | 2020-05-13 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.033 Å) | 主引用文献 | Structural characterization of cystathionine gamma-lyase smCSE enables aqueous metal quantum dot biosynthesis. Int.J.Biol.Macromol., 174, 2021
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6K1L
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![BU of 6k1l by Molmil](/molmil-images/mine/6k1l) | E53A mutant of a putative cystathionine gamma-lyase | 分子名称: | Cystathionine gamma-lyase, PYRIDOXAL-5'-PHOSPHATE, PYRUVIC ACID | 著者 | Chen, S, Wang, Y. | 登録日 | 2019-05-10 | 公開日 | 2020-05-13 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.46 Å) | 主引用文献 | Structural characterization of cystathionine gamma-lyase smCSE enables aqueous metal quantum dot biosynthesis. Int.J.Biol.Macromol., 174, 2021
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5ZED
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![BU of 5zed by Molmil](/molmil-images/mine/5zed) | Crystal structure of Kluyveromyces polyspora ADH (KpADH) mutant (E214V/T215S) | 分子名称: | NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, Uncharacterized protein ADH | 著者 | Wang, Y, Zhou, J.Y, Hou, X.D, Xu, G.C, Wu, L, Rao, Y.J, ZHou, J.H, Ni, Y. | 登録日 | 2018-02-27 | 公開日 | 2019-01-02 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.199 Å) | 主引用文献 | Structural Insight into Enantioselective Inversion of an Alcohol Dehydrogenase Reveals a "Polar Gate" in Stereorecognition of Diaryl Ketones. J. Am. Chem. Soc., 140, 2018
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5Z2X
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![BU of 5z2x by Molmil](/molmil-images/mine/5z2x) | Structure of Alcohol dehydrogenase from Kluyveromyces polyspora(KpADH) | 分子名称: | 1,2-ETHANEDIOL, Alcohol dehydrogenase, DI(HYDROXYETHYL)ETHER, ... | 著者 | Wang, Y, Zhou, J.Y, Hou, X.D, Xu, G.C, Wu, L, Rao, Y.J, ZHou, J.H, Ni, Y. | 登録日 | 2018-01-04 | 公開日 | 2019-01-02 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.98 Å) | 主引用文献 | Structural Insight into Enantioselective Inversion of an Alcohol Dehydrogenase Reveals a "Polar Gate" in Stereorecognition of Diaryl Ketones. J. Am. Chem. Soc., 140, 2018
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5ZEC
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![BU of 5zec by Molmil](/molmil-images/mine/5zec) | Crystal structure of Kluyveromyces polyspora ADH (KpADH) mutant (Q136N/F161V/S196G/E214G/S237C) | 分子名称: | 1,2-ETHANEDIOL, DI(HYDROXYETHYL)ETHER, ETHANOL, ... | 著者 | Wang, Y, ZHou, J.Y, Hou, X.D, Xu, G.C, Rao, Y.J, Wu, L, Zhou, J.H, Ni, Y. | 登録日 | 2018-02-27 | 公開日 | 2019-01-02 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.779 Å) | 主引用文献 | Structural Insight into Enantioselective Inversion of an Alcohol Dehydrogenase Reveals a "Polar Gate" in Stereorecognition of Diaryl Ketones. J. Am. Chem. Soc., 140, 2018
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7ESI
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![BU of 7esi by Molmil](/molmil-images/mine/7esi) | Crystal structure of the collagenase unit of a Vibrio collagenase from Vibrio harveyi VHJR7 at 1. 8 angstrom resolution. | 分子名称: | CALCIUM ION, Collagenase unit (CU), Peptide P1, ... | 著者 | Cao, H.Y, Wang, Y, Peng, M, Zhang, Y.Z. | 登録日 | 2021-05-11 | 公開日 | 2022-02-09 | 最終更新日 | 2023-02-22 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Structure of Vibrio collagenase VhaC provides insight into the mechanism of bacterial collagenolysis. Nat Commun, 13, 2022
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8HXB
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![BU of 8hxb by Molmil](/molmil-images/mine/8hxb) | Cryo-EM structure of MPXV M2 hexamer in complex with human B7.2 | 分子名称: | NFkB inhibitor, T-lymphocyte activation antigen CD86 | 著者 | Wang, Y, Yang, S, Zhao, H, Deng, Z. | 登録日 | 2023-01-04 | 公開日 | 2023-08-30 | 最終更新日 | 2023-12-13 | 実験手法 | ELECTRON MICROSCOPY (2.7 Å) | 主引用文献 | Structural and functional insights into the modulation of T cell costimulation by monkeypox virus protein M2. Nat Commun, 14, 2023
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8HXC
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![BU of 8hxc by Molmil](/molmil-images/mine/8hxc) | Cryo-EM structure of MPXV M2 heptamer in complex with human B7.2 | 分子名称: | NFkB inhibitor, T-lymphocyte activation antigen CD86 | 著者 | Wang, Y, Yang, S, Zhao, H, Deng, Z. | 登録日 | 2023-01-04 | 公開日 | 2023-08-30 | 最終更新日 | 2023-12-13 | 実験手法 | ELECTRON MICROSCOPY (3.12 Å) | 主引用文献 | Structural and functional insights into the modulation of T cell costimulation by monkeypox virus protein M2. Nat Commun, 14, 2023
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8HXA
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![BU of 8hxa by Molmil](/molmil-images/mine/8hxa) | Cryo-EM structure of MPXV M2 in complex with human B7.1 | 分子名称: | NFkB inhibitor, T-lymphocyte activation antigen CD80 | 著者 | Wang, Y, Yang, S, Zhao, H, Deng, Z. | 登録日 | 2023-01-04 | 公開日 | 2023-08-30 | 最終更新日 | 2023-12-13 | 実験手法 | ELECTRON MICROSCOPY (3.04 Å) | 主引用文献 | Structural and functional insights into the modulation of T cell costimulation by monkeypox virus protein M2. Nat Commun, 14, 2023
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7EN3
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![BU of 7en3 by Molmil](/molmil-images/mine/7en3) | Crystal structure of tubulin in complex with Tubulysin analogue TGL | 分子名称: | (2S,4R)-5-(4-fluorophenyl)-2-methyl-4-[[2-[(1R,3R)-4-methyl-3-[5-methylhexyl-[(2S,3S)-3-methyl-2-[[(2R)-1-methylpiperidin-2-yl]carbonylamino]pentanoyl]amino]-1-oxidanyl-pentyl]-1,3-thiazol-4-yl]carbonylamino]pentanoic acid, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, ... | 著者 | Wang, Y, Li, W. | 登録日 | 2021-04-15 | 公開日 | 2022-04-27 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.643 Å) | 主引用文献 | The X-ray structure of tubulysin analogue TGL in complex with tubulin and three possible routes for the development of next-generation tubulysin analogues. Biochem.Biophys.Res.Commun., 565, 2021
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7WA8
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![BU of 7wa8 by Molmil](/molmil-images/mine/7wa8) | Strigolactone receptors in Striga ShHTL7 | 分子名称: | Hyposensitive to light 7 | 著者 | Wang, Y, Yao, R. | 登録日 | 2021-12-12 | 公開日 | 2022-01-05 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.33 Å) | 主引用文献 | Molecular basis for high ligand sensitivity and selectivity of strigolactone receptors in Striga. Plant Physiology, Volume 185, 2021
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7VLZ
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![BU of 7vlz by Molmil](/molmil-images/mine/7vlz) | Crystal structure of the collagenase unit of a Vibrio collagenase from Vibrio harveyi VHJR7 | 分子名称: | CALCIUM ION, Peptide P1, Peptide P2, ... | 著者 | Cao, H.Y, Wang, Y, Peng, M, Zhang, Y.Z. | 登録日 | 2021-10-05 | 公開日 | 2022-10-19 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Crystal structure of the collagenase unit of a Vibrio collagenase from Vibrio harveyi VHJR7 To Be Published
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