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3ZID
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BU of 3zid by Molmil
CetZ from Methanosaeta thermophila strain DSM 6194
Descriptor: GUANOSINE-5'-DIPHOSPHATE, TUBULIN/FTSZ, GTPASE
Authors:Aylett, C.H.S, Amos, L.A, Lowe, J.
Deposit date:2013-01-08
Release date:2013-08-14
Last modified:2024-05-01
Method:X-RAY DIFFRACTION (2 Å)
Cite:Cetz Tubulin-Like Proteins Control Archaeal Cell Shape
Nature, 519, 2015
2HXH
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BU of 2hxh by Molmil
KIF1A head-microtubule complex structure in adp-form
Descriptor: ADENOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, ...
Authors:Kikkawa, M, Hirokawa, N.
Deposit date:2006-08-03
Release date:2006-10-10
Last modified:2024-06-05
Method:ELECTRON MICROSCOPY (11 Å)
Cite:High-resolution cryo-EM maps show the nucleotide binding pocket of KIF1A in open and closed conformations
Embo J., 25, 2006
5JH7
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BU of 5jh7 by Molmil
Tubulin-Eribulin complex
Descriptor: (1S,3S,6S,9S,12S,14R,16R,18S,20R,21R,22S,26R,29S,31R,32S,33R,35R,36S)-20-[(2S)-3-amino-2-hydroxypropyl]-21-methoxy-14-methyl-8,15-dimethylidene-2,19,30,34,37,39,40,41-octaoxanonacyclo[24.9.2.1~3,32~.1~3,33~.1~6,9~.1~12,16~.0~18,22~.0~29,36~.0~31,35~]hentetracontan-24-one (non-preferred name), 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, ...
Authors:Doodhi, H, Prota, A.E, Rodriguez-Garcia, R, Xiao, H, Custar, D.W, Bargsten, K, Katrukha, E.A, Hilbert, M, Hua, S, Jiang, K, Grigoriev, I, Yang, C.-P.H, Cox, D, Band Horwitz, S, Kapitein, L.C, Akhmanova, A, Steinmetz, M.O.
Deposit date:2016-04-20
Release date:2016-06-29
Last modified:2024-01-10
Method:X-RAY DIFFRACTION (2.25 Å)
Cite:Termination of Protofilament Elongation by Eribulin Induces Lattice Defects that Promote Microtubule Catastrophes.
Curr.Biol., 26, 2016
7EXC
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BU of 7exc by Molmil
Crystal structure of T2R-TTL-1129A2 complex
Descriptor: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, GLYCEROL, ...
Authors:Yang, J.H, Yan, W.
Deposit date:2021-05-26
Release date:2022-06-01
Last modified:2023-11-29
Method:X-RAY DIFFRACTION (2.39 Å)
Cite:Structure-Based Design and Synthesis of N-Substituted 3-Amino-beta-Carboline Derivatives as Potent alpha beta-Tubulin Degradation Agents
J.Med.Chem., 65, 2022
7RRO
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BU of 7rro by Molmil
Structure of the 48-nm repeat doublet microtubule from bovine tracheal cilia
Descriptor: Armadillo repeat containing 4, Chromosome 3 C1orf194 homolog, Cilia and flagella associated protein 161, ...
Authors:Gui, M, Anderson, J.R, Botsch, J.J, Meleppattu, S, Singh, S.K, Zhang, Q, Brown, A.
Deposit date:2021-08-10
Release date:2021-10-27
Last modified:2024-06-05
Method:ELECTRON MICROSCOPY (3.4 Å)
Cite:De novo identification of mammalian ciliary motility proteins using cryo-EM.
Cell, 184, 2021
9BP6
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BU of 9bp6 by Molmil
Structure of alpha1B and betaI/IVb microtubule bound to GMPCPP
Descriptor: GUANOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, PHOSPHOMETHYLPHOSPHONIC ACID GUANYLATE ESTER, ...
Authors:Zehr, E.A, Roll-Mecak, A.
Deposit date:2024-05-07
Release date:2024-06-12
Last modified:2025-06-11
Method:ELECTRON MICROSCOPY (3.1 Å)
Cite:Cryo-EM structures of human alpha1B/betaI+betaIVb microtubules shed light on isoform specific assembly
Biorxiv, 2023
1TVK
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BU of 1tvk by Molmil
The binding mode of epothilone A on a,b-tubulin by electron crystallography
Descriptor: EPOTHILONE A, GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, ...
Authors:Nettles, J.H, Li, H, Cornett, B, Krahn, J.M, Snyder, J.P, Downing, K.H.
Deposit date:2004-06-29
Release date:2004-09-14
Last modified:2023-08-23
Method:ELECTRON CRYSTALLOGRAPHY (2.89 Å)
Cite:The binding mode of epothilone A on alpha,beta-tubulin by electron crystallography
Science, 305, 2004
3CB2
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BU of 3cb2 by Molmil
Crystal structure of human gamma-tubulin bound to GDP
Descriptor: GUANOSINE-5'-DIPHOSPHATE, tubulin gamma-1 chain
Authors:Rice, L.M, Montabana, E.A, Agard, D.A.
Deposit date:2008-02-21
Release date:2008-06-10
Last modified:2023-08-30
Method:X-RAY DIFFRACTION (2.303 Å)
Cite:The lattice as allosteric effector: structural studies of alphabeta- and gamma-tubulin clarify the role of GTP in microtubule assembly
Proc.Natl.Acad.Sci.Usa, 105, 2008
2HXF
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BU of 2hxf by Molmil
KIF1A head-microtubule complex structure in amppnp-form
Descriptor: GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, Kinesin-like protein KIF1A, ...
Authors:Kikkawa, M, Hirokawa, N.
Deposit date:2006-08-03
Release date:2006-10-10
Last modified:2024-06-05
Method:ELECTRON MICROSCOPY (10 Å)
Cite:High-resolution cryo-EM maps show the nucleotide binding pocket of KIF1A in open and closed conformations
Embo J., 25, 2006
6KVP
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BU of 6kvp by Molmil
S. aureus FtsZ in complex with 3-(1-(5-bromo-4-(4-(trifluoromethyl)phenyl)oxazol-2-yl)ethoxy)-2,6-difluorobenzamide (compound 2)
Descriptor: 3-[(1R)-1-[5-bromanyl-4-[4-(trifluoromethyl)phenyl]-1,3-oxazol-2-yl]ethoxy]-2,6-bis(fluoranyl)benzamide, CALCIUM ION, Cell division protein FtsZ, ...
Authors:Ferrer-Gonzalez, E, Fujita, J, Yoshizawa, T, Nelson, J.M, Pilch, A.J, Hillman, E, Ozawa, M, Kuroda, N, Parhi, A.K, LaVoie, E.J, Matsumura, H, Pilch, D.S.
Deposit date:2019-09-05
Release date:2020-01-15
Last modified:2023-11-22
Method:X-RAY DIFFRACTION (1.4 Å)
Cite:Structure-Guided Design of a Fluorescent Probe for the Visualization of FtsZ in Clinically Important Gram-Positive and Gram-Negative Bacterial Pathogens.
Sci Rep, 9, 2019
3RYH
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BU of 3ryh by Molmil
GMPCPP-Tubulin: RB3 Stathmin-like domain complex
Descriptor: GUANOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, PHOSPHOMETHYLPHOSPHONIC ACID GUANYLATE ESTER, ...
Authors:Nawrotek, A, Knossow, M, Gigant, B.
Deposit date:2011-05-11
Release date:2011-10-05
Last modified:2024-11-20
Method:X-RAY DIFFRACTION (2.8 Å)
Cite:The Determinants That Govern Microtubule Assembly from the Atomic Structure of GTP-Tubulin.
J.Mol.Biol., 412, 2011
4U3J
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BU of 4u3j by Molmil
TOG2:alpha/beta-tubulin complex
Descriptor: GUANOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, Protein STU2, ...
Authors:Ayaz, P, Rice, L.M.
Deposit date:2014-07-22
Release date:2014-08-20
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (2.81 Å)
Cite:A tethered delivery mechanism explains the catalytic action of a microtubule polymerase.
Elife, 3, 2014
4U39
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BU of 4u39 by Molmil
Crystal Structure of FtsZ:MciZ Complex from Bacillus subtilis
Descriptor: Cell division factor, Cell division protein FtsZ, PHOSPHATE ION
Authors:Bisson-Filho, A.W, Discola, K.F, Castellen, P, Blasios, V, Martins, A, Sforca, M.L, Garcia, W, Zeri, A.C, Erickson, H.P, Dessen, A, Gueiros-Filho, F.J.
Deposit date:2014-07-19
Release date:2015-03-18
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (3.194 Å)
Cite:Crystal Structure of FtsZ:MciZ Complex from Bacillus subtilis
To be Published
3RYF
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BU of 3ryf by Molmil
GTP-Tubulin: RB3 Stathmin-like domain complex
Descriptor: GUANOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, SULFATE ION, ...
Authors:Nawrotek, A, Knossow, M, Gigant, B.
Deposit date:2011-05-11
Release date:2011-10-05
Last modified:2024-11-20
Method:X-RAY DIFFRACTION (2.52 Å)
Cite:The Determinants That Govern Microtubule Assembly from the Atomic Structure of GTP-Tubulin.
J.Mol.Biol., 412, 2011
4TV8
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BU of 4tv8 by Molmil
Tubulin-Maytansine complex
Descriptor: (3beta,4beta,5beta,10beta,11E,13E)-maytansine, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, ...
Authors:Prota, A.E, Bargsten, K, Diaz, J.F, Marsh, M, Cuevas, C, Liniger, M, Neuhaus, C, Andreu, J.M, Altmann, K.H, Steinmetz, M.O.
Deposit date:2014-06-26
Release date:2014-08-27
Last modified:2023-12-20
Method:X-RAY DIFFRACTION (2.103 Å)
Cite:A new tubulin-binding site and pharmacophore for microtubule-destabilizing anticancer drugs.
Proc.Natl.Acad.Sci.USA, 111, 2014
2VAW
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BU of 2vaw by Molmil
FtsZ Pseudomonas aeruginosa GDP
Descriptor: CELL DIVISION PROTEIN FTSZ, GUANOSINE-5'-DIPHOSPHATE
Authors:Oliva, M.A, Lowe, J.
Deposit date:2007-09-04
Release date:2007-09-11
Last modified:2023-12-13
Method:X-RAY DIFFRACTION (2.9 Å)
Cite:Structural Insights Into the Conformational Variability of Ftsz
J.Mol.Biol., 373, 2007
7ZYW
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BU of 7zyw by Molmil
Crystal structure of T2R-TTL-PM534 complex
Descriptor: (4R)-N-[(1R)-1-[4-(cyclopropylmethoxy)-6-oxidanylidene-pyran-2-yl]butyl]-4-methyl-2-[(E)-C-methyl-N-oxidanyl-carbonimidoyl]-5H-1,3-thiazole-4-carboxamide, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, ...
Authors:Oliva, M.A, Diaz, J.F, Cuevas, C.
Deposit date:2022-05-25
Release date:2023-11-29
Last modified:2024-06-12
Method:X-RAY DIFFRACTION (2.45 Å)
Cite:PM534, an Optimized Target-Protein Interaction Strategy through the Colchicine Site of Tubulin.
J.Med.Chem., 67, 2024
8ASN
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BU of 8asn by Molmil
Crystal structure of the apo human TTL in complex with tubulin-stathmin
Descriptor: GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, ...
Authors:Vuillard, L, Miallau, L.
Deposit date:2022-08-19
Release date:2022-09-21
Last modified:2024-01-31
Method:X-RAY DIFFRACTION (2.571 Å)
Cite:Crystal structure of the apo human TTL in complex with tubulin-stathmin
To Be Published
2VAM
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BU of 2vam by Molmil
FtsZ B. subtilis
Descriptor: CELL DIVISION PROTEIN FTSZ, SULFATE ION
Authors:Oliva, M.A, Lowe, J.
Deposit date:2007-09-03
Release date:2007-09-11
Last modified:2023-12-13
Method:X-RAY DIFFRACTION (2.5 Å)
Cite:Structural Insights Into the Conformational Variability of Ftsz
J.Mol.Biol., 373, 2007
4UXT
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BU of 4uxt by Molmil
Conserved mechanisms of microtubule-stimulated ADP release, ATP binding, and force generation in transport kinesins
Descriptor: GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, KINESIN HEAVY CHAIN ISOFORM 5A, ...
Authors:Atherton, J, Farabella, I, Yu, I.M, Rosenfeld, S.S, Houdusse, A, Topf, M, Moores, C.
Deposit date:2014-08-27
Release date:2014-09-24
Last modified:2024-05-08
Method:ELECTRON MICROSCOPY (7.4 Å)
Cite:Conserved Mechanisms of Microtubule-Stimulated Adp Release, ATP Binding, and Force Generation in Transport Kinesins.
Elife, 3, 2014
6LS4
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BU of 6ls4 by Molmil
A novel anti-tumor agent S-40 in complex with tubulin
Descriptor: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 3-[(4-cyclopropylphenyl)sulfonylamino]-4-methyl-N-(pyridin-3-ylmethyl)benzamide, GLYCEROL, ...
Authors:Du, T, Lin, S, Ji, M, Xue, N, Liu, Y, Zhang, K, Lu, D, Chen, X, Xu, H.
Deposit date:2020-01-17
Release date:2021-01-20
Last modified:2023-11-29
Method:X-RAY DIFFRACTION (2.4 Å)
Cite:A novel orally active microtubule destabilizing agent S-40 targets the colchicine-binding site and shows potent antitumor activity.
Cancer Lett., 495, 2020
1IA0
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BU of 1ia0 by Molmil
KIF1A HEAD-MICROTUBULE COMPLEX STRUCTURE IN ATP-FORM
Descriptor: GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, KINESIN-LIKE PROTEIN KIF1A, ...
Authors:Kikkawa, M, Sablin, E.P, Okada, Y, Yajima, H, Fletterick, R.J, Hirokawa, N.
Deposit date:2001-03-22
Release date:2002-03-22
Last modified:2024-12-25
Method:ELECTRON MICROSCOPY (15 Å)
Cite:Switch-based Mechanism of Kinesin Motors
Nature, 411, 2001
3N2K
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BU of 3n2k by Molmil
TUBULIN-NSC 613862: RB3 Stathmin-like domain complex
Descriptor: GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, ...
Authors:Barbier, P, Dorleans, A, Devred, F, Sanz, L, Allegro, D, Alfonso, C, Knossow, M, Peyrot, V, Andreu, J.M.
Deposit date:2010-05-18
Release date:2010-07-28
Last modified:2023-09-06
Method:X-RAY DIFFRACTION (4 Å)
Cite:Stathmin and interfacial microtubule inhibitors recognize a naturally curved conformation of tubulin dimers.
J.Biol.Chem., 285, 2010
1FFX
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BU of 1ffx by Molmil
TUBULIN:STATHMIN-LIKE DOMAIN COMPLEX
Descriptor: GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, PROTEIN (STATHMIN-LIKE DOMAIN OF RB3), ...
Authors:Gigant, B, Martin-Barbey, C, Knossow, M.
Deposit date:2000-07-26
Release date:2000-09-27
Last modified:2023-08-09
Method:X-RAY DIFFRACTION (3.95 Å)
Cite:The 4 A X-ray structure of a tubulin:stathmin-like domain complex.
Cell(Cambridge,Mass.), 102, 2000
7JFR
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BU of 7jfr by Molmil
Auristatin bound to tubulin
Descriptor: Auristatin, CALCIUM ION, GUANOSINE-5'-DIPHOSPHATE, ...
Authors:Moquist, P.N, Waight, A.
Deposit date:2020-07-17
Release date:2020-09-16
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (2.35 Å)
Cite:Novel Auristatins with High Bystander and Cytotoxic Activities in Drug Efflux-positive Tumor Models.
Mol.Cancer Ther., 20, 2021

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