EMDB/PDB/SASBDBから引用されている文献のデータベース

キーワード
構造解析手法	All X線回折 NMR 電子顕微鏡小角散乱中性子線回折線維回折粉末回折赤外分光 EPR FRET 理論モデルハイブリッド
著者・登録者
ジャーナル
IF	>30 >20 >10 >5 all

タイトル	Development and characterization of novel indazole-based PPAR-gamma partial agonists
ジャーナル・号・ページ	To Be Published
掲載日	2024年8月12日 (構造データの登録日)
著者	Koops, A.A. / Oerlemans, G.J.M. / Brunsveld, L.
リンク	PubMedで検索
手法	X線回折
解像度	1.8 - 2.7 Å
構造データ	PDB-9gfu: Human PPAR-gamma ligand binding domain in complex with AKGO172 手法: X-RAY DIFFRACTION / 解像度: 2.1 Å PDB-9gvp: Human PPAR-gamma ligand binding domain in complex with WG115 手法: X-RAY DIFFRACTION / 解像度: 2.05 Å PDB-9gvs: Human PPAR-gamma ligand binding domain in complex with AK176_C 手法: X-RAY DIFFRACTION / 解像度: 2.1 Å PDB-9gw3: Human PPAR-gamma ligand binding domain in complex with LW56 手法: X-RAY DIFFRACTION / 解像度: 2 Å PDB-9gw4: Human PPAR-gamma ligand binding domain in complex with LW78 手法: X-RAY DIFFRACTION / 解像度: 2.2 Å PDB-9gw7: Human PPAR-gamma ligand binding domain in complex with LW76 手法: X-RAY DIFFRACTION / 解像度: 2.1 Å PDB-9gw8: Human PPAR-gamma ligand binding domain in complex with LW75 手法: X-RAY DIFFRACTION / 解像度: 2.2 Å PDB-9gwb: Human PPAR-gamma ligand binding domain in complex with LW69 手法: X-RAY DIFFRACTION / 解像度: 2.2 Å PDB-9gwc: Human PPAR-gamma ligand binding domain in complex with LW99 手法: X-RAY DIFFRACTION / 解像度: 2 Å PDB-9gwe: Human PPAR-gamma ligand binding domain in complex with LW87 手法: X-RAY DIFFRACTION / 解像度: 2.1 Å PDB-9gwf: Human PPAR-gamma ligand binding domain in complex with LW100 手法: X-RAY DIFFRACTION / 解像度: 2.4 Å PDB-9gwg: Human PPAR-gamma ligand binding domain in complex with LW88 手法: X-RAY DIFFRACTION / 解像度: 2.3 Å PDB-9gwh: Human PPAR-gamma ligand binding domain in complex with LW77 手法: X-RAY DIFFRACTION / 解像度: 2.1 Å PDB-9gwi: Human PPAR-gamma ligand binding domain in complex with LW23 手法: X-RAY DIFFRACTION / 解像度: 2.2 Å PDB-9gwk: Human PPAR-gamma ligand binding domain in complex with AKGO6A 手法: X-RAY DIFFRACTION / 解像度: 2.2 Å PDB-9gwl: Human PPAR-gamma ligand binding domain in complex with AKGO157 手法: X-RAY DIFFRACTION / 解像度: 2.2 Å PDB-9gwm: Human PPAR-gamma ligand binding domain in complex with AKGO108 手法: X-RAY DIFFRACTION / 解像度: 2.2 Å PDB-9gwn: Human PPAR-gamma ligand binding domain in complex with LW30 手法: X-RAY DIFFRACTION / 解像度: 2.2 Å PDB-9gwp: Human PPAR-gamma ligand binding domain in complex with MRL-871 with two distinct binding modes 手法: X-RAY DIFFRACTION / 解像度: 2.55 Å PDB-9gwq: Human PPAR-gamma ligand binding domain in complex with AKGO6D 手法: X-RAY DIFFRACTION / 解像度: 2.1 Å PDB-9gwr: Human PPAR-gamma ligand binding domain in complex with AKGO10 手法: X-RAY DIFFRACTION / 解像度: 2.1 Å PDB-9gws: Human PPAR-gamma ligand binding domain in complex with AKGO8 手法: X-RAY DIFFRACTION / 解像度: 2.2 Å PDB-9gwx: Human PPAR-gamma ligand binding domain in complex with AKGO141 手法: X-RAY DIFFRACTION / 解像度: 2.2 Å PDB-9gwy: Human PPAR-gamma ligand binding domain in complex with AKGO78 手法: X-RAY DIFFRACTION / 解像度: 2.09 Å PDB-9gx0: Human PPAR-gamma ligand binding domain in complex with AKGO79 手法: X-RAY DIFFRACTION / 解像度: 2.1 Å PDB-9gx1: Human PPAR-gamma ligand binding domain in complex with AKGO80 手法: X-RAY DIFFRACTION / 解像度: 2.1 Å PDB-9gx2: Human PPAR-gamma ligand binding domain in complex with AKGO82 手法: X-RAY DIFFRACTION / 解像度: 2.35 Å PDB-9gx3: Human PPAR-gamma ligand binding domain in complex with AKGO12 手法: X-RAY DIFFRACTION / 解像度: 1.9 Å PDB-9gx4: Human PPAR-gamma ligand binding domain in complex with AKGO156 手法: X-RAY DIFFRACTION / 解像度: 2.2 Å PDB-9gx5: Human PPAR-gamma ligand binding domain in complex with AKGO173 手法: X-RAY DIFFRACTION / 解像度: 2.45 Å PDB-9gx6: Human PPAR-gamma ligand binding domain in complex with AKGO166 手法: X-RAY DIFFRACTION / 解像度: 2.1 Å PDB-9gx7: Human PPAR-gamma ligand binding domain in complex with WG17 手法: X-RAY DIFFRACTION / 解像度: 2.2 Å PDB-9gxd: Human PPAR-gamma ligand binding domain in complex with AKGO27 手法: X-RAY DIFFRACTION / 解像度: 2.2 Å PDB-9gz7: Human PPAR-gamma ligand binding domain in complex with AKGO29 手法: X-RAY DIFFRACTION / 解像度: 1.8 Å PDB-9gz8: Human PPAR-gamma ligand binding domain in complex with AKGO46 手法: X-RAY DIFFRACTION / 解像度: 2.2 Å PDB-9gz9: Human PPAR-gamma ligand binding domain in complex with AKGO48 手法: X-RAY DIFFRACTION / 解像度: 2.1 Å PDB-9gza: Human PPAR-gamma ligand binding domain in complex with AKGO50 手法: X-RAY DIFFRACTION / 解像度: 1.9 Å PDB-9gzb: Human PPAR-gamma ligand binding domain in complex with AKGO52 手法: X-RAY DIFFRACTION / 解像度: 2.2 Å PDB-9gzc: Human PPAR-gamma ligand binding domain in complex with AKGO142 手法: X-RAY DIFFRACTION / 解像度: 2.3 Å PDB-9gze: Human PPAR-gamma ligand binding domain in complex with AKGO72 手法: X-RAY DIFFRACTION / 解像度: 2.2 Å PDB-9gzf: Human PPAR-gamma ligand binding domain in complex with AKGO88 手法: X-RAY DIFFRACTION / 解像度: 2.65 Å PDB-9gzi: Human PPAR-gamma ligand binding domain in complex with LW98 手法: X-RAY DIFFRACTION / 解像度: 2.7 Å
化合物	PDB-1ik6: 3D structure of the E1beta subunit of pyruvate dehydrogenase from the archeon Pyrobaculum aerophilum ChemComp-HOH: WATER PDB-1ipp: HOMING ENDONUCLEASE/DNA COMPLEX PDB-1ipr: Unknown entry PDB-1ipw: INORGANIC PYROPHOSPHATASE FROM ESCHERICHIA COLI WITH THREE MAGNESIUM IONS PDB-1ips: ISOPENICILLIN N SYNTHASE FROM ASPERGILLUS NIDULANS (MANGANESE COMPLEX) PDB-1ipu: Unknown entry PDB-1irg: INTERFERON REGULATORY FACTOR-2 DNA BINDING DOMAIN, NMR, 20 STRUCTURES PDB-1ipz: Unknown entry PDB-1ipx: Unknown entry PDB-1ipv: Unknown entry PDB-1ipt: Unknown entry PDB-1ip1: G37A HUMAN LYSOZYME PDB-1ip0: NMR STRUCTURE OF HUMAN BETACELLULIN-2 PDB-1ipy: Unknown entry PDB-1ip9: SOLUTION STRUCTURE OF THE PB1 DOMAIN OF BEM1P PDB-1ip7: G129A HUMAN LYSOZYME PDB-1ip6: G127A HUMAN LYSOZYME PDB-1ip4: G72A HUMAN LYSOZYME ChemComp-4F1: 4-{1-[2-chloro-6-(trifluoromethyl)benzoyl]-1H-indazol-3-yl}benzoic acid PDB-1iqa: CRYSTAL STRUCTURE OF THE EXTRACELLULAR DOMAIN OF MOUSE RANK LIGAND PDB-1ip3: G68A HUMAN LYSOZYME PDB-1iqb: Crystal Structure of Urtica dioica Agglutinin Isolectin I PDB-1ip8: Unknown entry PDB-1iqd: Human Factor VIII C2 Domain complexed to human monoclonal BO2C11 Fab. PDB-1iqg: Human coagulation factor Xa in complex with M55159 PDB-1iqi: Human coagulation factor Xa in complex with M55125 PDB-1ip5: G105A HUMAN LYSOZYME PDB-1iqe: Human coagulation factor Xa in complex with M55590 PDB-1iqc: Crystal structure of Di-Heme Peroxidase from Nitrosomonas europaea PDB-1iqj: Human coagulation factor Xa in complex with M55124 PDB-1iql: Human coagulation factor Xa in complex with M54476 PDB-1iqh: Human coagulation factor Xa in complex with M55143 PDB-1iqf: Human coagulation factor Xa in complex with M55165 PDB-1iq8: Crystal Structure of archaeosine tRNA-guanine transglycosylase from Pyrococcus horikoshii PDB-1iq7: Ovotransferrin, C-Terminal Lobe, Apo Form PDB-1iq6: (R)-HYDRATASE FROM A. CAVIAE INVOLVED IN PHA BIOSYNTHESIS PDB-1iq5: Calmodulin/nematode CA2+/Calmodulin dependent kinase kinase fragment PDB-1iq4: 5S-RRNA BINDING RIBOSOMAL PROTEIN L5 FROM BACILLUS STEAROTHERMOPHILUS PDB-1iq3: SOLUTION STRUCTURE OF THE EPS15 HOMOLOGY DOMAIN OF A HUMAN POB1 PDB-1ird: Crystal Structure of Human Carbonmonoxy-Haemoglobin at 1.25 A Resolution PDB 未公開エントリ PDB-1iq2: Unknown entry PDB-1ira: COMPLEX OF THE INTERLEUKIN-1 RECEPTOR WITH THE INTERLEUKIN-1 RECEPTOR ANTAGONIST (IL1RA)
由来	homo sapiens (ヒト)
キーワード	TRANSCRIPTION / PPAR / PPAR gamma / PPARg / peroxisome proliferator-activated receptor gamma / nuclear receptor / transcription factor / partial agonist / agonist