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PDB: 5552 件

5WB7
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Crystal structure of the epidermal growth factor receptor extracellular region in complex with epiregulin
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Epidermal growth factor receptor, ...
著者Freed, D.M, Bessman, N.J, Ferguson, K.M, Lemmon, M.A.
登録日2017-06-28
公開日2017-10-18
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.941 Å)
主引用文献EGFR Ligands Differentially Stabilize Receptor Dimers to Specify Signaling Kinetics.
Cell, 171, 2017
5WB8
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Crystal structure of the epidermal growth factor receptor extracellular region in complex with epigen
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Epidermal growth factor receptor, Epigen, ...
著者Bessman, N.J, Freed, D.M, Moore, J.O, Ferguson, K.M, Lemmon, M.A.
登録日2017-06-28
公開日2017-10-18
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献EGFR Ligands Differentially Stabilize Receptor Dimers to Specify Signaling Kinetics.
Cell, 171, 2017
5WBE
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COX-1:MOFEZOLAC COMPLEX STRUCTURE
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Mofezolac, PROTOPORPHYRIN IX CONTAINING FE, ...
著者Cingolani, G, Panella, A, Perrone, M.G, Vitale, P, Smith, W.L, Scilimati, A.
登録日2017-06-28
公開日2017-07-26
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.75 Å)
主引用文献Structural basis for selective inhibition of Cyclooxygenase-1 (COX-1) by diarylisoxazoles mofezolac and 3-(5-chlorofuran-2-yl)-5-methyl-4-phenylisoxazole (P6).
Eur J Med Chem, 138, 2017
5WDU
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HIV-1 Env BG505 SOSIP.664 H72C-H564C trimer in complex with bNAbs PGT122 Fab, 35O22 Fab and NIH45-46 scFv
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Envelope glycoprotein gp160, ...
著者Julien, J.-P, Torrents de la Pena, A, Sanders, R.W, Wilson, I.A.
登録日2017-07-06
公開日2018-04-04
最終更新日2022-11-30
実験手法X-RAY DIFFRACTION (7 Å)
主引用文献Improving the Immunogenicity of Native-like HIV-1 Envelope Trimers by Hyperstabilization.
Cell Rep, 20, 2017
5WEE
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Crystal structure of HpVAL4
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-3)]2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Asojo, O.A.
登録日2017-07-09
公開日2018-03-28
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.99 Å)
主引用文献Heligmosomoides polygyrus Venom Allergen-like Protein-4 (HpVAL-4) is a sterol binding protein.
Int. J. Parasitol., 48, 2018
5WKU
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Structure of an acid sensing ion channel in a resting state with barium
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Acid-sensing ion channel 1, ...
著者Yoder, N, Gouaux, E.
登録日2017-07-25
公開日2018-03-14
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.95 Å)
主引用文献Gating mechanisms of acid-sensing ion channels.
Nature, 555, 2018
5WKV
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Structure of an acid sensing ion channel in a resting state with calcium
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Acid-sensing ion channel 1, ...
著者Yoder, N, Gouaux, E.
登録日2017-07-25
公開日2018-03-14
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Gating mechanisms of acid-sensing ion channels.
Nature, 555, 2018
5WKX
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Barium sites in the structure of a resting acid sensing ion channel
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Acid-sensing ion channel 1, ...
著者Yoder, N, Gouaux, E.
登録日2017-07-25
公開日2018-08-08
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (4.034 Å)
主引用文献Divalent cation and chloride ion sites of chicken acid sensing ion channel 1a elucidated by x-ray crystallography.
PLoS ONE, 13, 2018
5WKY
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Bromide sites in the structure of an acid sensing ion channel in a resting state
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Acid-sensing ion channel 1, ...
著者Yoder, N, Gouaux, E.
登録日2017-07-25
公開日2018-08-08
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (4 Å)
主引用文献Divalent cation and chloride ion sites of chicken acid sensing ion channel 1a elucidated by x-ray crystallography.
PLoS ONE, 13, 2018
5WLS
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Crystal Structure of a Pollen Receptor Kinase 3
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Pollen receptor-like kinase 3
著者Xu, G, Chakraborty, S, Pan, H.
登録日2017-07-27
公開日2018-06-06
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.496 Å)
主引用文献The Extracellular Domain of Pollen Receptor Kinase 3 is structurally similar to the SERK family of co-receptors.
Sci Rep, 8, 2018
5WPQ
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Cryo-EM structure of mammalian endolysosomal TRPML1 channel in nanodiscs in closed I conformation at 3.64 Angstrom resolution
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Mucolipin-1, SODIUM ION
著者Chen, Q, She, J, Guo, J, Bai, X, Jiang, Y.
登録日2017-08-07
公開日2017-10-18
最終更新日2023-04-05
実験手法ELECTRON MICROSCOPY (3.64 Å)
主引用文献Structure of mammalian endolysosomal TRPML1 channel in nanodiscs.
Nature, 550, 2017
5WPT
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Cryo-EM structure of mammalian endolysosomal TRPML1 channel in nanodiscs in closed II conformation at 3.75 Angstrom resolution
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Mucolipin-1, SODIUM ION
著者Chen, Q, She, J, Guo, J, Bai, X, Jiang, Y.
登録日2017-08-07
公開日2017-10-18
最終更新日2023-04-05
実験手法ELECTRON MICROSCOPY (3.75 Å)
主引用文献Structure of mammalian endolysosomal TRPML1 channel in nanodiscs.
Nature, 550, 2017
5WPV
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Cryo-EM structure of mammalian endolysosomal TRPML1 channel in nanodiscs at 3.59 Angstrom resolution
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Mucolipin-1, SODIUM ION
著者Chen, Q, She, J, Guo, J, Bai, X, Jiang, Y.
登録日2017-08-07
公開日2017-10-18
最終更新日2023-04-05
実験手法ELECTRON MICROSCOPY (3.59 Å)
主引用文献Structure of mammalian endolysosomal TRPML1 channel in nanodiscs.
Nature, 550, 2017
5WRR
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BU of 5wrr by Molmil
Crystal structure of Fam20A
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Pseudokinase FAM20A
著者Zhu, Q.
登録日2016-12-03
公開日2017-05-03
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.506 Å)
主引用文献Structure of Fam20A reveals a pseudokinase featuring a unique disulfide pattern and inverted ATP-binding
Elife, 6, 2017
5WRS
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Crystal Structure of Fam20A in complex with ATP
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ADENOSINE-5'-TRIPHOSPHATE, ...
著者Zhu, Q.
登録日2016-12-03
公開日2017-05-03
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.75 Å)
主引用文献Structure of Fam20A reveals a pseudokinase featuring a unique disulfide pattern and inverted ATP-binding
Elife, 6, 2017
5WV3
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Crystal structure of bovine lactoperoxidase with a partial Glu258-heme linkage at 2.07 A resolution.
分子名称: 1-(OXIDOSULFANYL)METHANAMINE, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Singh, P.K, Sirohi, H.V, Kaur, P, Sharma, S, Singh, T.P.
登録日2016-12-21
公開日2017-02-15
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.07 Å)
主引用文献Structural basis of activation of mammalian heme peroxidases
Prog. Biophys. Mol. Biol., 133, 2018
5WY8
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Crystal structure of PTP delta Ig1-Ig3 in complex with IL1RAPL1 Ig1-Ig3
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Interleukin-1 receptor accessory protein-like 1, ...
著者Kim, H.M, Won, S.Y, Kim, D.
登録日2017-01-11
公開日2017-11-22
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (3.07 Å)
主引用文献LAR-RPTP Clustering Is Modulated by Competitive Binding between Synaptic Adhesion Partners and Heparan Sulfate
Front Mol Neurosci, 10, 2017
5WYX
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Crystal structure of human TLR8 in complex with CU-CPT8m
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 7-(3-methylphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide, ...
著者Tanji, H, Ohto, U, Shimizu, T.
登録日2017-01-16
公開日2017-12-13
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Small-molecule inhibition of TLR8 through stabilization of its resting state
Nat. Chem. Biol., 14, 2018
5WYZ
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Crystal structure of human TLR8 in complex with CU-CPT9b
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 4-(3-methyl-4-oxidanyl-phenyl)quinolin-7-ol, ...
著者Tanji, H, Ohto, U, Shimizu, T.
登録日2017-01-16
公開日2017-12-13
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Small-molecule inhibition of TLR8 through stabilization of its resting state
Nat. Chem. Biol., 14, 2018
5X0M
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Structure of a eukaryotic voltage-gated sodium channel at near atomic resolution
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Sodium channel protein, ...
著者Shen, H, Zhou, Q, Pan, X, Li, Z, Wu, J, Yan, N.
登録日2017-01-21
公開日2017-03-08
最終更新日2020-07-29
実験手法ELECTRON MICROSCOPY (3.8 Å)
主引用文献Structure of a eukaryotic voltage-gated sodium channel at near-atomic resolution.
Science, 355, 2017
5X2P
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Crystal structure of the medaka fish taste receptor T1r2a-T1r3 ligand binding domains in complex with L-glutamate
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ...
著者Nuemket, N, Yasui, N, Atsumi, N, Yamashita, A.
登録日2017-02-02
公開日2017-05-24
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.608 Å)
主引用文献Structural basis for perception of diverse chemical substances by T1r taste receptors
Nat Commun, 8, 2017
5X2Q
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Crystal structure of the medaka fish taste receptor T1r2a-T1r3 ligand binding domains in complex with glycine
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ...
著者Nuemket, N, Yasui, N, Atsumi, N, Yamashita, A.
登録日2017-02-02
公開日2017-05-24
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Structural basis for perception of diverse chemical substances by T1r taste receptors
Nat Commun, 8, 2017
5X4A
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SLL-2-Forssman antigen tetrasaccharides complex
分子名称: 2-acetamido-2-deoxy-alpha-D-galactopyranose-(1-3)-2-acetamido-2-deoxy-beta-D-galactopyranose-(1-3)-alpha-D-galactopyranose-(1-4)-beta-D-galactopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Galactose-binding lectin, ...
著者Kita, A, Miki, K.
登録日2017-02-11
公開日2017-09-20
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (3.4 Å)
主引用文献Crystal structure of octocoral lectin SLL-2 complexed with Forssman antigen tetrasaccharide.
Glycobiology, 2017
5X4R
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Structure of the N-terminal domain (NTD) of MERS-CoV spike protein
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, S protein
著者Yuan, Y, Zhang, Y, Qi, J, Shi, Y, Gao, G.F.
登録日2017-02-14
公開日2017-05-03
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Cryo-EM structures of MERS-CoV and SARS-CoV spike glycoproteins reveal the dynamic receptor binding domains
Nat Commun, 8, 2017
5X4S
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Structure of the N-terminal domain (NTD)of SARS-CoV spike protein
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Spike glycoprotein
著者Yuan, Y, Zhang, Y, Qi, J, Shi, Y, Gao, G.F.
登録日2017-02-14
公開日2017-05-03
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Cryo-EM structures of MERS-CoV and SARS-CoV spike glycoproteins reveal the dynamic receptor binding domains
Nat Commun, 8, 2017

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