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2AZN
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BU of 2azn by Molmil
X-RAY Structure of 2,5-diamino-6-ribosylamino-4(3h)-pyrimidinone 5-phosphate reductase
分子名称: 2-(6-(2-CYCLOHEXYLETHOXY)-TETRAHYDRO-4,5-DIHYDROXY-2(HYDROXYMETHYL)-2H-PYRAN-3-YLOXY)-TETRAHYDRO-6(HYDROXYMETHYL)-2H-PYRAN-3,4,5-TRIOL, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, ...
著者Chatwell, L, Bacher, A, Huber, R, Fischer, M, Krojer, T.
登録日2005-09-12
公開日2006-08-29
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Biosynthesis of riboflavin: structure and properties of 2,5-diamino-6-ribosylamino-4(3H)-pyrimidinone 5'-phosphate reductase of Methanocaldococcus jannaschii
J.Mol.Biol., 359, 2006
6WWB
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BU of 6wwb by Molmil
Crystal Structure of the second bromodomain of human BRD2 in complex with the compound 3b
分子名称: 1,2-ETHANEDIOL, 2-((S)-4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)-N-((1-(4-(2-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)amino)acetamido)butyl)-1H-1,2,3-triazol-4-yl)methyl)acetamide, Bromodomain-containing protein 2
著者White, S.W, Yun, M.
登録日2020-05-08
公開日2021-11-17
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.31 Å)
主引用文献Phenyl-Glutarimides: Alternative Cereblon Binders for the Design of PROTACs.
Angew.Chem.Int.Ed.Engl., 60, 2021
2B3V
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BU of 2b3v by Molmil
Spermine spermidine acetyltransferase in complex with acetylcoa, K26R mutant
分子名称: ACETYL COENZYME *A, Diamine acetyltransferase 1
著者Bewley, M.C, Graziano, V, Jiang, J.S, Matz, E, Studier, F.W, Pegg, A.P, Coleman, C.S, Flanagan, J.M, Burley, S.K, New York SGX Research Center for Structural Genomics (NYSGXRC)
登録日2005-09-21
公開日2006-01-17
最終更新日2021-02-03
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Structures of wild-type and mutant human spermidine/spermine N1-acetyltransferase, a potential therapeutic drug target.
Proc.Natl.Acad.Sci.USA, 103, 2006
2B0V
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BU of 2b0v by Molmil
NUDIX hydrolase from Nitrosomonas europaea.
分子名称: 1,2-ETHANEDIOL, CHLORIDE ION, NUDIX hydrolase, ...
著者Osipiuk, J, Skarina, T, Savchenko, A, Edwards, A, Joachimiak, A, MCSG, Midwest Center for Structural Genomics (MCSG)
登録日2005-09-14
公開日2005-09-27
最終更新日2018-01-24
実験手法X-RAY DIFFRACTION (1.55 Å)
主引用文献X-ray structure of NUDIX hydrolase from Nitrosomonas europaea.
To be Published
2BAL
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BU of 2bal by Molmil
p38alpha MAP kinase bound to pyrazoloamine
分子名称: Mitogen-activated protein kinase 14, [5-AMINO-1-(4-FLUOROPHENYL)-1H-PYRAZOL-4-YL][3-(PIPERIDIN-4-YLOXY)PHENYL]METHANONE
著者Gerhardt, S, Pauptit, R.A, Read, J, Tucker, J, Norman, R.A, Breed, J.
登録日2005-10-14
公開日2005-12-06
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Prevention of MKK6-Dependent Activation by Binding to p38alpha MAP Kinase.
Biochemistry, 44, 2005
2B5F
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BU of 2b5f by Molmil
Crystal structure of the spinach aquaporin SoPIP2;1 in an open conformation to 3.9 resolution
分子名称: aquaporin
著者Tornroth-Horsefield, S, Wang, Y, Hedfalk, K, Johanson, U, Karlsson, M, Tajkhorshid, E, Neutze, R, Kjellbom, P.
登録日2005-09-28
公開日2005-12-20
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (3.9 Å)
主引用文献Structural mechanism of plant aquaporin gating
Nature, 439, 2006
2B67
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BU of 2b67 by Molmil
Crystal structure of the Nitroreductase Family Protein from Streptococcus pneumoniae TIGR4
分子名称: ACETIC ACID, COG0778: Nitroreductase, FLAVIN MONONUCLEOTIDE
著者Kim, Y, Volkart, L, Abdullah, J, Collart, F, Joachimiak, A, Midwest Center for Structural Genomics (MCSG)
登録日2005-09-30
公開日2005-11-15
最終更新日2017-10-11
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献Crystal Structure of the Nitroreductase Family Protein from Streptococcus pneumoniae TIGR4
To be Published
2B7P
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BU of 2b7p by Molmil
Crystal structure of quinolinic acid phosphoribosyltransferase from Helicobacter pylori with phthalic acid
分子名称: PHTHALIC ACID, Probable nicotinate-nucleotide pyrophosphorylase, SULFATE ION
著者Kim, M.K, Im, Y.J, Lee, J.H, Eom, S.H.
登録日2005-10-05
公開日2006-02-14
最終更新日2018-09-19
実験手法X-RAY DIFFRACTION (2.51 Å)
主引用文献Crystal structure of quinolinic acid phosphoribosyltransferase from Helicobacter pylori
Proteins, 63, 2006
2B6C
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BU of 2b6c by Molmil
Predicted DNA alkylation repair enzyme from Enterococcus faecalis.
分子名称: BETA-MERCAPTOETHANOL, CHLORIDE ION, GLYCEROL, ...
著者Osipiuk, J, Hatzos, C, Moy, S, Collart, F, Joachimiak, A, Midwest Center for Structural Genomics (MCSG)
登録日2005-09-30
公開日2005-11-15
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Xray structure of predicted DNA alkylation repair enzyme from Enterococcus faecalis.
To be Published
6OFY
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BU of 6ofy by Molmil
Crystal Structure of Arachidonic Acid bound to V349I murine COX-2
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, ACRYLIC ACID, ARACHIDONIC ACID, ...
著者Malkowski, M.G.
登録日2019-04-01
公開日2020-02-05
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Arg-513 and Leu-531 Are Key Residues Governing Time-Dependent Inhibition of Cyclooxygenase-2 by Aspirin and Celebrex.
Biochemistry, 58, 2019
4UYK
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BU of 4uyk by Molmil
Crystal structure of a Signal Recognition Particle Alu domain in the elongation arrest conformation
分子名称: SIGNAL RECOGNITION PARTICLE 14 KDA PROTEIN, SIGNAL RECOGNITION PARTICLE 9 KDA PROTEIN, SRP RNA
著者Bousset, L, Mary, C, Brooks, M.A, Scherrer, A, Strub, K, Cusack, S.
登録日2014-09-01
公開日2014-11-05
最終更新日2014-12-03
実験手法X-RAY DIFFRACTION (3.22 Å)
主引用文献Crystal Structure of a Signal Recognition Particle Alu Domain in the Elongation Arrest Conformation.
RNA, 20, 2014
4UV2
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BU of 4uv2 by Molmil
Structure of the curli transport lipoprotein CsgG in a non-lipidated, pre-pore conformation
分子名称: CURLI PRODUCTION TRANSPORT COMPONENT CSGG
著者Goyal, P, Krasteva, P.V, Gerven, N.V, Gubellini, F, Broeck, I.V.D, Troupiotis-Tsailaki, A, Jonckheere, W, Pehau-Arnaudet, G, Pinkner, J.S, Chapman, M.R, Hultgren, S.J, Howorka, S, Fronzes, R, Remaut, H.
登録日2014-08-04
公開日2014-09-24
最終更新日2014-12-17
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Structural and Mechanistic Insights Into the Bacterial Amyloid Secretion Channel Csgg.
Nature, 516, 2014
4V2D
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BU of 4v2d by Molmil
FLRT2 LRR domain
分子名称: FIBRONECTIN LEUCINE RICH TRANSMEMBRANE PROTEIN 2
著者Seiradake, E, del Toro, D, Nagel, D, Cop, F, Haertl, R, Ruff, T, Seyit-Bremer, G, Harlos, K, Border, E.C, Acker-Palmer, A, Jones, E.Y, Klein, R.
登録日2014-10-08
公開日2014-11-05
最終更新日2015-07-22
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Flrt Structure: Balancing Repulsion and Cell Adhesion in Cortical and Vascular Development
Neuron, 84, 2014
6DS5
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BU of 6ds5 by Molmil
Cryo EM structure of human SEIPIN
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Seipin
著者Yan, R.H, Qian, H.W, Yan, N, Yang, H.Y.
登録日2018-06-13
公開日2018-10-24
最終更新日2020-07-29
実験手法ELECTRON MICROSCOPY (3.8 Å)
主引用文献Human SEIPIN Binds Anionic Phospholipids.
Dev. Cell, 47, 2018
4UW9
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BU of 4uw9 by Molmil
The crystal structural of archaeal beta-phosphoglucomutase from hyper-thermophilic Pyrococcus sp. Strain ST 04
分子名称: BETA-PHOSPHOGLUCOMUTASE, MAGNESIUM ION
著者Park, K.-H, Woo, E.-J.
登録日2014-08-09
公開日2014-10-29
最終更新日2015-09-23
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Structural Features of Archaeal Beta-Phosphoglucomutase from Hyper-Thermophilic Pyrococcus Sp. Strain St 04
To be Published
4V34
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BU of 4v34 by Molmil
The Structure of A-PGS from Pseudomonas aeruginosa (SeMet derivative)
分子名称: ALANYL-TRNA-DEPENDENT L-ALANYL- PHOPHATIDYLGLYCEROL SYNTHASE, CHLORIDE ION, SULFATE ION
著者Krausze, J, Hebecker, S, Hasenkampf, T, Heinz, D.W, Moser, J.
登録日2014-10-16
公開日2015-08-19
最終更新日2017-07-12
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Structures of Two Bacterial Resistance Factors Mediating tRNA-Dependent Aminoacylation of Phosphatidylglycerol with Lysine or Alanine.
Proc.Natl.Acad.Sci.USA, 112, 2015
4UYT
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BU of 4uyt by Molmil
X-ray structure of the N-terminal domain of the flocculin Flo11 from Saccharomyces cerevisiae
分子名称: ACETATE ION, FLOCCULATION PROTEIN FLO11, SODIUM ION
著者Kraushaar, T, Veelders, M, Brueckner, S, Rhinow, D, Moesch, H.U, Essen, L.O.
登録日2014-09-03
公開日2015-08-12
実験手法X-RAY DIFFRACTION (1.03 Å)
主引用文献Interactions by the Fungal Flo11 Adhesin Depend on a Fibronectin Type III-Like Adhesin Domain Girdled by Aromatic Bands.
Structure, 23, 2015
4V0N
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BU of 4v0n by Molmil
Crystal structure of BBS1N in complex with ARL6DN, soaked with mercury
分子名称: ARF-LIKE SMALL GTPASE, BARDET-BIEDL SYNDROME 1 PROTEIN, GUANOSINE-5'-TRIPHOSPHATE, ...
著者Mourao, A, Lorentzen, E.
登録日2014-09-17
公開日2014-11-19
最終更新日2019-04-03
実験手法X-RAY DIFFRACTION (3.131 Å)
主引用文献Structural Basis for Membrane Targeting of the Bbsome by Arl6
Nat.Struct.Mol.Biol., 21, 2014
4V2P
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BU of 4v2p by Molmil
Ketosynthase MxnB
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, CHLORIDE ION, KETOSYNTHASE, ...
著者Koehnke, J.
登録日2014-10-13
公開日2015-08-26
最終更新日2018-04-18
実験手法X-RAY DIFFRACTION (1.67 Å)
主引用文献In vitro reconstitution of alpha-pyrone ring formation in myxopyronin biosynthesis.
Chem Sci, 6, 2015
4UYR
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BU of 4uyr by Molmil
X-ray structure of the N-terminal domain of the flocculin Flo11 from Saccharomyces cerevisiae
分子名称: FLOCCULATION PROTEIN FLO11, MAGNESIUM ION, PHOSPHATE ION, ...
著者Veelders, M, Kraushaar, T, Brueckner, S, Rhinow, D, Moesch, H.U, Essen, L.O.
登録日2014-09-03
公開日2015-08-12
最終更新日2017-06-28
実験手法X-RAY DIFFRACTION (0.89 Å)
主引用文献Interactions by the Fungal Flo11 Adhesin Depend on a Fibronectin Type III-Like Adhesin Domain Girdled by Aromatic Bands.
Structure, 23, 2015
4UYS
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BU of 4uys by Molmil
X-ray structure of the N-terminal domain of the flocculin Flo11 from Saccharomyces cerevisiae
分子名称: FLOCCULATION PROTEIN FLO11, MAGNESIUM ION, SODIUM ION
著者Kraushaar, T, Veelders, M, Brueckner, S, Rhinow, D, Moesch, H.U, Essen, L.O.
登録日2014-09-03
公開日2015-08-12
実験手法X-RAY DIFFRACTION (1.05 Å)
主引用文献Interactions by the Fungal Flo11 Adhesin Depend on a Fibronectin Type III-Like Adhesin Domain Girdled by Aromatic Bands.
Structure, 23, 2015
6DMB
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BU of 6dmb by Molmil
Cryo-EM structure of human Ptch1
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CHOLESTEROL HEMISUCCINATE, ...
著者Yan, N, Gong, X, Qian, H.W.
登録日2018-06-04
公開日2018-07-11
最終更新日2020-07-29
実験手法ELECTRON MICROSCOPY (3.9 Å)
主引用文献Structural basis for the recognition of Sonic Hedgehog by human Patched1.
Science, 361, 2018
4WBG
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BU of 4wbg by Molmil
Crystal structure of class C beta-lactamase Mox-1 covalently complexed with aztorenam
分子名称: 2-({[(1Z)-1-(2-amino-1,3-thiazol-4-yl)-2-oxo-2-{[(2S,3S)-1-oxo-3-(sulfoamino)butan-2-yl]amino}ethylidene]amino}oxy)-2-methylpropanoic acid, ACETATE ION, Beta-lactamase, ...
著者Oguri, T, Shimizu-ibuka, A, Ishii, Y.
登録日2014-09-03
公開日2015-07-01
最終更新日2020-01-29
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Conformational Change Observed in the Active Site of Class C beta-Lactamase MOX-1 upon Binding to Aztreonam
Antimicrob.Agents Chemother., 59, 2015
6DG8
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BU of 6dg8 by Molmil
Full-length 5-HT3A receptor in a serotonin-bound conformation- State 2
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 5-hydroxytryptamine receptor 3A, SEROTONIN, ...
著者Basak, S, Chakrapani, S.
登録日2018-05-17
公開日2018-11-07
最終更新日2020-07-29
実験手法ELECTRON MICROSCOPY (3.89 Å)
主引用文献Cryo-EM reveals two distinct serotonin-bound conformations of full-length 5-HT3Areceptor.
Nature, 563, 2018
4WD3
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Crystal structure of an L-amino acid ligase RizA
分子名称: L-amino acid ligase
著者Kagawa, W, Arai, T, Kino, K, Kurumizaka, H.
登録日2014-09-06
公開日2015-09-09
最終更新日2020-01-01
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Structure of RizA, an L-amino-acid ligase from Bacillus subtilis.
Acta Crystallogr.,Sect.F, 71, 2015

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